中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
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(4R)-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C32H32N4O4S |
|
—— |
2-[(4R)-1-(4-fluorophenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C32H31FN4O3S |
|
—— |
(4S)-4-(3-fluorophenyl)-1-(3-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H29FN4O2S |
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—— |
N-cyclopropyl-2-[(4R)-4-(2,4-difluorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C31H28F2N4O2S |
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—— |
2-[(4S)-1-(4-methylphenyl)-4-(3-methylthiophen-2-yl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide |
—— |
C29H30N4O2S2 |
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—— |
[2-[[(3R)-3-methyl-1,1-dioxothiolan-3-yl]amino]-2-oxoethyl] 5-cyclopropyl-2-phenylpyrazole-3-carboxylate |
—— |
C20H23N3O5S |
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—— |
2-[(4S)-1-(4-fluorophenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C32H31FN4O3S |
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—— |
2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C29H28F2N4O3S |
|
—— |
2-[(4S)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C29H28F2N4O3S |
|
—— |
2-oxopropyl (E)-3-[1-benzyl-3-(4-methylphenyl)pyrazol-4-yl]prop-2-enoate |
—— |
C23H22N2O3 |
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—— |
(4S)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H29FN4O4S |
|
—— |
(4S)-4-(2,5-dimethoxyphenyl)-1-(2,4-dimethylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C34H36N4O4S |
|
—— |
(4R)-1,4-bis(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C32H32N4O3S |
|
—— |
2-[(4S)-4-(2,5-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide |
—— |
C31H31FN4O4S |
|
—— |
(4R)-1-(4-fluorophenyl)-4-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H29FN4O3S |
|
—— |
2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide |
—— |
C28H32F2N4O3S |
|
—— |
(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(3-fluorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C30H35FN4O3S |
|
—— |
(4R)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H29FN4O3S |
|
—— |
2-[(4R)-3-tert-butyl-1-(2-chlorophenyl)-4-(3,4-dimethoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide |
—— |
C30H37ClN4O4S |
|
—— |
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(3-fluorophenyl)-1-(3-methylphenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C33H32FN5O3S |
|
—— |
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(3-fluorophenyl)-1-(3-methylphenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C33H32FN5O3S |
|
—— |
2-[(4S)-3-tert-butyl-1-(2-chlorophenyl)-4-(3,4-dimethoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide |
—— |
C30H37ClN4O4S |
|
—— |
(4S)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H29FN4O3S |
|
—— |
(4S)-1-(2,3-dimethylphenyl)-4-(3-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C33H34N4O2S |
|
—— |
(4R)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H29FN4O4S |
|
—— |
(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H38N4O4S |
|
—— |
(4S)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C34H36N4O3S |
|
—— |
(4S)-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C32H32N4O4S |
|
—— |
2-[(4R)-1-(4-methylphenyl)-4-(3-methylthiophen-2-yl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide |
—— |
C29H30N4O2S2 |
|
—— |
(4S)-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C32H32N4O5S |
|
—— |
(4R)-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C32H32N4O5S |
|
—— |
[(2S)-1-amino-1-oxopropan-2-yl] (E)-3-[1-benzyl-3-(4-methylphenyl)pyrazol-4-yl]prop-2-enoate |
—— |
C23H23N3O3 |
|
—— |
(4R)-1-(2,3-dimethylphenyl)-4-(3-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C33H34N4O2S |
|
—— |
(4R)-4-(3-fluorophenyl)-1-(3-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H29FN4O3S |
|
—— |
(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H38N4O4S |
|
—— |
(4S)-4-(3-fluorophenyl)-1-(3-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H29FN4O3S |
|
—— |
2-[(4S)-1-(4-fluorophenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C32H31FN4O3S |
|
—— |
(4R)-4-(2,5-dimethoxyphenyl)-1-(2,4-dimethylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C34H36N4O4S |
|
—— |
2-[[4-(4-fluorophenyl)-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide |
—— |
C26H36FN5OS |
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—— |
(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H38N4O3S |
|
—— |
2-[(4R)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide |
—— |
C31H31FN4O3S |
|
—— |
(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H38N4O3S |
|
—— |
(5-phenyl-1,3-oxazol-2-yl)methyl (3S)-5-oxo-1-[(1R)-1-phenylethyl]pyrrolidine-3-carboxylate |
—— |
C23H22N2O4 |
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—— |
(2R)-2-chloro-N-[[4-(5-chloro-2-methylphenyl)-5-[(3-methoxyphenyl)methylsulfanyl]-1,2,4-triazol-3-yl]methyl]-2-phenylacetamide |
—— |
C26H24Cl2N4O2S |
|
—— |
(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H38N4O3S |
|
—— |
(2S)-2-chloro-N-[[4-(5-chloro-2-methylphenyl)-5-[(3-methoxyphenyl)methylsulfanyl]-1,2,4-triazol-3-yl]methyl]-2-phenylacetamide |
—— |
C26H24Cl2N4O2S |
|
—— |
2-[(4S)-1-(2,4-dimethylphenyl)-4-(2-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide |
—— |
C31H31FN4O2S |
|
—— |
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-(4-fluorophenyl)-4-(2-methylphenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C33H32FN5O3S |
|
—— |
(4R)-4-(3-fluorophenyl)-1-(3-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H29FN4O2S |
|
—— |
2-[(4S)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide |
—— |
C30H29FN4O3S |
|