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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[3-(2H-tetrazol-5-yl)phenyl]-2-(trifluoromethyl)benzenesulfonamide —— C14H10F3N5O2S
N-[3-(2H-tetrazol-5-yl)phenyl]-2-(trifluoromethyl)benzenesulfonamide
—— 2-[[4-amino-5-(2-bromophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C20H26BrN5OS
2-[[4-amino-5-(2-bromophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— (4S)-1-(4-fluorophenyl)-4-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H29FN4O3S
(4S)-1-(4-fluorophenyl)-4-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[[4-(4-fluorophenyl)-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C26H36FN5OS
2-[[4-(4-fluorophenyl)-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— (4S)-1-(4-fluorophenyl)-4-(2-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H29FN4O2S
(4S)-1-(4-fluorophenyl)-4-(2-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide —— C28H32F2N4O3S
2-[(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide
—— N-[[4-(dimethylamino)phenyl]methyl]-2-[1-(2-methylphenyl)tetrazol-5-yl]sulfanylacetamide —— C19H22N6OS
N-[[4-(dimethylamino)phenyl]methyl]-2-[1-(2-methylphenyl)tetrazol-5-yl]sulfanylacetamide
—— 2-chloro-N-[3-(1,2,3-triaza-4-azanidacyclopenta-2,5-dien-5-yl)phenyl]benzenesulfonamide —— C13H9ClN5O2S-
2-chloro-N-[3-(1,2,3-triaza-4-azanidacyclopenta-2,5-dien-5-yl)phenyl]benzenesulfonamide
—— 4-propyl-N-[3-(2H-tetrazol-5-yl)phenyl]benzenesulfonamide —— C16H17N5O2S
4-propyl-N-[3-(2H-tetrazol-5-yl)phenyl]benzenesulfonamide
—— 4-propyl-N-[3-(1,2,3-triaza-4-azanidacyclopenta-2,5-dien-5-yl)phenyl]benzenesulfonamide —— C16H16N5O2S-
4-propyl-N-[3-(1,2,3-triaza-4-azanidacyclopenta-2,5-dien-5-yl)phenyl]benzenesulfonamide
—— (2R)-2-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-(3-fluoro-4-methylphenyl)propanamide —— C19H20FN5OS
(2R)-2-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-(3-fluoro-4-methylphenyl)propanamide
—— (2R)-2-[[5-(4-methoxyphenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-prop-2-enylpropanamide —— C20H26N4O3S
(2R)-2-[[5-(4-methoxyphenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-prop-2-enylpropanamide
—— N-[3-(2H-tetrazol-5-yl)phenyl]-4-(trifluoromethoxy)benzenesulfonamide —— C14H10F3N5O3S
N-[3-(2H-tetrazol-5-yl)phenyl]-4-(trifluoromethoxy)benzenesulfonamide
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 5-nitro-1-benzothiophene-2-carboxylate —— C19H12N2O5S
(5-Phenyl-1,3-oxazol-2-yl)methyl 5-nitro-1-benzothiophene-2-carboxylate
—— (E)-2-phenyl-N-[3-(1,2,3-triaza-4-azanidacyclopenta-2,5-dien-5-yl)phenyl]ethenesulfonamide —— C15H12N5O2S-
(E)-2-phenyl-N-[3-(1,2,3-triaza-4-azanidacyclopenta-2,5-dien-5-yl)phenyl]ethenesulfonamide
—— N-[2-(N-ethyl-3-methylanilino)ethyl]-2-[5-(2-methylphenyl)tetrazol-2-yl]acetamide —— C21H26N6O
N-[2-(N-ethyl-3-methylanilino)ethyl]-2-[5-(2-methylphenyl)tetrazol-2-yl]acetamide
—— (2R)-N-(2,4-dimethylphenyl)-2-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C20H23N5OS
(2R)-N-(2,4-dimethylphenyl)-2-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— (2S)-2-[[5-(4-chlorophenyl)-4-propyl-1,2,4-triazol-3-yl]sulfanyl]-N-cycloheptylpropanamide —— C21H29ClN4OS
(2S)-2-[[5-(4-chlorophenyl)-4-propyl-1,2,4-triazol-3-yl]sulfanyl]-N-cycloheptylpropanamide
—— (3-Phenyl-1,2,4-oxadiazol-5-yl)methyl 3-methyl-1,2-oxazole-5-carboxylate —— C14H11N3O4
(3-Phenyl-1,2,4-oxadiazol-5-yl)methyl 3-methyl-1,2-oxazole-5-carboxylate
—— (2R)-N-(2-methoxyethyl)-2-[[5-(4-methoxyphenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C20H28N4O4S
(2R)-N-(2-methoxyethyl)-2-[[5-(4-methoxyphenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (2R)-2-[[5-(4-methoxyphenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-prop-2-enylpropanamide —— C20H26N4O3S
(2R)-2-[[5-(4-methoxyphenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-prop-2-enylpropanamide
—— (2S)-N-(2,6-dimethylphenyl)-2-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C20H23N5OS
(2S)-N-(2,6-dimethylphenyl)-2-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— 3-[5-[[3-(4-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-4-ethyl-1,2,4-triazol-3-yl]propanamide —— C16H17ClN6O2S
3-[5-[[3-(4-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-4-ethyl-1,2,4-triazol-3-yl]propanamide
—— (2S)-N-(3,4-difluorophenyl)-2-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C18H17F2N5OS
(2S)-N-(3,4-difluorophenyl)-2-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— [2-[[4-(3-chlorophenyl)-5-(furan-2-yl)-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-thiazol-4-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C27H28ClN5O2S2
[2-[[4-(3-chlorophenyl)-5-(furan-2-yl)-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-thiazol-4-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— (2R)-2-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanyl-N,N-di(propan-2-yl)propanamide —— C18H27N5OS
(2R)-2-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanyl-N,N-di(propan-2-yl)propanamide
—— 2-[6-[1-(2-methoxyphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2R)-4-phenylbutan-2-yl]acetamide —— C30H31N5O3S
2-[6-[1-(2-methoxyphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2R)-4-phenylbutan-2-yl]acetamide
—— 2-[6-[1-(2-methoxyphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2S)-4-phenylbutan-2-yl]acetamide —— C30H31N5O3S
2-[6-[1-(2-methoxyphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2S)-4-phenylbutan-2-yl]acetamide
—— ethyl (3R)-1-[2-[6-[1-(4-fluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C27H28FN5O4S
ethyl (3R)-1-[2-[6-[1-(4-fluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate
—— 2-[[4-(4-chlorophenyl)-5-[(1R)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2S,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C24H34ClN5OS
2-[[4-(4-chlorophenyl)-5-[(1R)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2S,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— 2,2-dichloro-N-[[3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]phenyl]methyl]acetamide —— C18H14Cl2FN3O
2,2-dichloro-N-[[3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]phenyl]methyl]acetamide
—— 2-[[5-(4-ethylphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2S,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C22H30N4OS
2-[[5-(4-ethylphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2S,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— ethyl (3R)-1-[2-[6-[1-(2-fluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C27H28FN5O4S
ethyl (3R)-1-[2-[6-[1-(2-fluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[2-[6-[1-(2-fluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C27H28FN5O4S
ethyl (3S)-1-[2-[6-[1-(2-fluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate
—— 2-[[5-(4-ethylphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C22H30N4OS
2-[[5-(4-ethylphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— 2-[6-[1-(2-fluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2R)-4-phenylbutan-2-yl]acetamide —— C29H28FN5O2S
2-[6-[1-(2-fluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2R)-4-phenylbutan-2-yl]acetamide
—— [2-[cyclopentyl-[(3S)-1,1-dioxothiolan-3-yl]amino]-2-oxoethyl] 3-methyl-1,2-oxazole-5-carboxylate —— C16H22N2O6S
[2-[cyclopentyl-[(3S)-1,1-dioxothiolan-3-yl]amino]-2-oxoethyl] 3-methyl-1,2-oxazole-5-carboxylate
—— 3,5-dichloro-N-[3-(1,2,3-triaza-4-azanidacyclopenta-2,5-dien-5-yl)phenyl]benzenesulfonamide —— C13H8Cl2N5O2S-
3,5-dichloro-N-[3-(1,2,3-triaza-4-azanidacyclopenta-2,5-dien-5-yl)phenyl]benzenesulfonamide
—— [(2R)-1-(2,6-difluoroanilino)-1-oxopropan-2-yl] 2-(2,4-dimethylphenyl)-5-methyltriazole-4-carboxylate —— C21H20F2N4O3
[(2R)-1-(2,6-difluoroanilino)-1-oxopropan-2-yl] 2-(2,4-dimethylphenyl)-5-methyltriazole-4-carboxylate
—— 2-[[4-(4-chlorophenyl)-5-[(1S)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2S,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C24H34ClN5OS
2-[[4-(4-chlorophenyl)-5-[(1S)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2S,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— [3-(2-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl thiophene-3-carboxylate —— C14H9ClN2O3S
[3-(2-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl thiophene-3-carboxylate
—— (2S)-2-[[5-(4-chlorophenyl)-4-(3-methoxypropyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methoxyethyl)propanamide —— C18H25ClN4O3S
(2S)-2-[[5-(4-chlorophenyl)-4-(3-methoxypropyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methoxyethyl)propanamide
—— 2-[[4-(4-chlorophenyl)-5-[(1R)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C24H34ClN5OS
2-[[4-(4-chlorophenyl)-5-[(1R)-1-(dimethylamino)ethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— [(2R)-1-(2,4-difluoroanilino)-1-oxopropan-2-yl] 2-(2,4-dimethylphenyl)-5-methyltriazole-4-carboxylate —— C21H20F2N4O3
[(2R)-1-(2,4-difluoroanilino)-1-oxopropan-2-yl] 2-(2,4-dimethylphenyl)-5-methyltriazole-4-carboxylate
—— N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]propanamide —— C23H24N4O4
N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]propanamide
—— ethyl (3S)-1-[2-[7-methyl-6-[5-methyl-1-(3-methylphenyl)pyrazol-3-yl]-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C28H31N5O4S
ethyl (3S)-1-[2-[7-methyl-6-[5-methyl-1-(3-methylphenyl)pyrazol-3-yl]-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate
—— methyl N-[(2S)-2-[[4-butyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]carbamate —— C18H24N4O4S
methyl N-[(2S)-2-[[4-butyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]carbamate
—— ethyl (3S)-1-[2-[6-[1-(5-fluoro-2-methylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C28H30FN5O4S
ethyl (3S)-1-[2-[6-[1-(5-fluoro-2-methylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate
—— 2-[(4S)-3-tert-butyl-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C29H31N5O3S2
2-[(4S)-3-tert-butyl-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— [(2S)-1-(2,6-difluoroanilino)-1-oxopropan-2-yl] 2-(2,4-dimethylphenyl)-5-methyltriazole-4-carboxylate —— C21H20F2N4O3
[(2S)-1-(2,6-difluoroanilino)-1-oxopropan-2-yl] 2-(2,4-dimethylphenyl)-5-methyltriazole-4-carboxylate