中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
N-butyl-N-[2-[(2S)-2-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]decanamide |
—— |
C29H43ClN4O3 |
|
—— |
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-(2,4-dimethylphenyl)-4-(2-fluorophenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C34H34FN5O3S |
|
—— |
N-(3-cyano-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl)-3-[5-(4-methylphenyl)tetrazol-2-yl]propanamide |
—— |
C21H22N6OS |
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—— |
4-methyl-5-[4-nitro-2-(propan-2-ylsulfamoyl)phenoxy]-N-[[(2S)-oxolan-2-yl]methyl]-1-phenylpyrazole-3-carboxamide |
—— |
C25H29N5O7S |
|
—— |
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide |
—— |
C34H29N5O4S |
|
—— |
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-(2,4-dimethylphenyl)-4-(4-fluorophenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C34H34FN5O3S |
|
—— |
5-(1-Ethyl-2-oxoindol-3-ylidene)-2-(4-pentoxyphenyl)-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one |
—— |
C25H24N4O3S |
|
—— |
N-butyl-N-[2-[(2S)-2-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]octanamide |
—— |
C27H39ClN4O3 |
|
—— |
2-[(4S)-1-(2,4-dimethylphenyl)-4-(2-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide |
—— |
C35H30F2N4O2S |
|
—— |
2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide |
—— |
C31H30ClN5O4S |
|
—— |
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-(2,4-dimethylphenyl)-4-(4-fluorophenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C34H34FN5O3S |
|
—— |
(3S)-1-[2-[[5-(4-chlorophenyl)-4-octyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]piperidine-3-carboxamide |
—— |
C24H34ClN5O2S |
|
—— |
N-butyl-N-[2-[(2S)-2-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]nonanamide |
—— |
C28H41ClN4O3 |
|
—— |
[2-[4-(Furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl] 2-(prop-2-enylamino)-1,3-thiazole-4-carboxylate |
—— |
C18H20N4O5S |
|
—— |
2-[(4S)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide |
—— |
C33H29FN4O2S2 |
|
—— |
N-butyl-2-(4-chlorophenoxy)-N-[2-[(2R)-2-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]acetamide |
—— |
C27H30Cl2N4O4 |
|
—— |
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(2,4-difluorophenyl)-1-(2,4-dimethylphenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C34H33F2N5O3S |
|
—— |
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-(propanoylamino)phenoxy]-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxylic acid |
—— |
C25H30N4O7S |
|
—— |
[(1R,2S,5S)-5-methyl-2-propan-2-ylcyclohexyl] 2-[[4-cyclopentyl-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetate |
—— |
C29H42N4O5S2 |
|
—— |
2-[(4R)-3-tert-butyl-1-(2-chlorophenyl)-4-(3,4-dimethoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C32H34ClN5O4S |
|
—— |
ethyl (4R)-6-[[4-cyclopentyl-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate |
—— |
C26H34N6O6S2 |
|
—— |
N-butyl-N-[2-[(2R)-2-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]decanamide |
—— |
C29H43ClN4O3 |
|
—— |
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(2,4-difluorophenyl)-1-(2,4-dimethylphenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C34H33F2N5O3S |
|
—— |
2-[(4S)-3-tert-butyl-4-(2-chlorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide |
—— |
C32H32ClFN4O2S |
|
—— |
4-methyl-5-[4-nitro-2-(propan-2-ylsulfamoyl)phenoxy]-N-[[(2R)-oxolan-2-yl]methyl]-1-phenylpyrazole-3-carboxamide |
—— |
C25H29N5O7S |
|
—— |
N-butyl-2-(4-chlorophenoxy)-N-[2-[(2S)-2-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]acetamide |
—— |
C27H30Cl2N4O4 |
|
—— |
1-[(3-bromophenyl)methyl]-4-N-[(E)-pyridin-4-ylmethylideneamino]-5-N-[(Z)-pyridin-4-ylmethylideneamino]imidazole-4,5-dicarboxamide |
—— |
C24H19BrN8O2 |
|
—— |
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-(2,4-dimethylphenyl)-4-(2-fluorophenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C34H34FN5O3S |
|
—— |
(1R,2S,3S,4R)-3-(1H-1,2,4-triazol-5-ylmethylcarbamoyl)bicyclo[2.2.1]hept-5-ene-2-carboxylic acid |
—— |
C12H14N4O3 |
|
—— |
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide |
—— |
C31H30ClN5O4S |
|
—— |
N-butyl-N-[2-[(2R)-2-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]octanamide |
—— |
C27H39ClN4O3 |
|
—— |
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide |
—— |
C35H31N5O4S |
|
—— |
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-(propanoylamino)phenoxy]-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxylic acid |
—— |
C25H30N4O7S |
|
—— |
(3R)-1-[2-[[5-(4-chlorophenyl)-4-octyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]piperidine-3-carboxamide |
—— |
C24H34ClN5O2S |
|
—— |
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide |
—— |
C35H31N5O4S |
|
—— |
2-[(4R)-3-tert-butyl-1-(2-chlorophenyl)-4-(3,4-dimethoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C30H37ClN4O5S |
|
—— |
N-[5-chloro-2-(1,2,4-triazol-1-yl)phenyl]-4-propylbenzenesulfonamide |
—— |
C17H17ClN4O2S |
|
—— |
2-[(4S)-4-(2-fluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide |
—— |
C30H29FN4O3S |
|
—— |
2-[[4-benzyl-5-(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]acetamide |
—— |
C26H29ClN4OS |
|
—— |
2-[[4-benzyl-5-(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]acetamide |
—— |
C26H29ClN4OS |
|
—— |
2-[(4R)-1-(2,3-dimethylphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide |
—— |
C32H34N4O2S |
|
—— |
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide |
—— |
C34H29N5O4S |
|
—— |
2-[(4R)-4-(2,5-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C34H32N4O5S |
|
—— |
(1R,2S,3R,4R)-3-(1H-1,2,4-triazol-5-ylmethylcarbamoyl)bicyclo[2.2.1]hept-5-ene-2-carboxylic acid |
—— |
C12H14N4O3 |
|
—— |
2-[(4R)-4-(2-fluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide |
—— |
C30H29FN4O3S |
|
—— |
2-[(4S)-4-(2-fluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide |
—— |
C34H28F2N4O3S |
|
—— |
2-[(4R)-4-(2-fluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide |
—— |
C34H28F2N4O3S |
|
—— |
2-[[4-benzyl-5-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[2-[(5E)-2,4-dioxo-5-(pyridin-3-ylmethylidene)-1,3-thiazolidin-3-yl]ethyl]acetamide |
—— |
C28H23FN6O3S2 |
|
—— |
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-[(2-methoxyacetyl)amino]phenoxy]-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxylic acid |
—— |
C25H30N4O8S |
|
—— |
2-[(4R)-3-tert-butyl-1-(2-chlorophenyl)-4-(3,4-dimethoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide |
—— |
C32H34ClN5O4S |
|