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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-chloro-2-[(Z)-2-(4-imidazol-1-ylphenyl)ethenyl]-1,3-benzoxazole —— C18H12ClN3O
5-chloro-2-[(Z)-2-(4-imidazol-1-ylphenyl)ethenyl]-1,3-benzoxazole
—— (Z)-N-(2-methoxyethyl)-3-(1-methylpyrazol-4-yl)prop-2-enamide —— C10H15N3O2
(Z)-N-(2-methoxyethyl)-3-(1-methylpyrazol-4-yl)prop-2-enamide
—— (Z)-3-(4-bromo-3-nitrophenyl)-N-[2-(4-bromophenyl)-1,3-benzoxazol-5-yl]prop-2-en-1-imine —— C22H13Br2N3O3
(Z)-3-(4-bromo-3-nitrophenyl)-N-[2-(4-bromophenyl)-1,3-benzoxazol-5-yl]prop-2-en-1-imine
—— (Z)-3-(4-bromo-3-nitrophenyl)-N-[2-(3-methoxyphenyl)-1,3-benzoxazol-5-yl]prop-2-en-1-imine —— C23H16BrN3O4
(Z)-3-(4-bromo-3-nitrophenyl)-N-[2-(3-methoxyphenyl)-1,3-benzoxazol-5-yl]prop-2-en-1-imine
—— (Z)-N-(3-methoxypropyl)-3-(1-methylpyrazol-4-yl)prop-2-enamide —— C11H17N3O2
(Z)-N-(3-methoxypropyl)-3-(1-methylpyrazol-4-yl)prop-2-enamide
—— (4S)-3-tert-butyl-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C30H36N4O5S
(4S)-3-tert-butyl-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4S)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C30H36N4O4S
(4S)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (Z)-N-(2-methylbutan-2-yl)-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide —— C14H23N3O
(Z)-N-(2-methylbutan-2-yl)-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide
—— 2-[(4R)-3-tert-butyl-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C30H33N5O2S2
2-[(4R)-3-tert-butyl-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— N-[2-[[4-(4-chlorophenyl)-1-(3-methoxyphenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]thiophene-2-carboxamide —— C28H27ClN4O4S
N-[2-[[4-(4-chlorophenyl)-1-(3-methoxyphenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]thiophene-2-carboxamide
—— (4S)-3-tert-butyl-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C30H36N4O4S
(4S)-3-tert-butyl-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— N-[2-[[1-(3-chlorophenyl)-4-(4-chlorophenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]thiophene-2-carboxamide —— C27H24Cl2N4O3S
N-[2-[[1-(3-chlorophenyl)-4-(4-chlorophenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]thiophene-2-carboxamide
—— (Z)-3-(4-bromo-3-nitrophenyl)-N-[2-(2-chlorophenyl)-1,3-benzoxazol-5-yl]prop-2-en-1-imine —— C22H13BrClN3O3
(Z)-3-(4-bromo-3-nitrophenyl)-N-[2-(2-chlorophenyl)-1,3-benzoxazol-5-yl]prop-2-en-1-imine
—— N-[2-[[1,4-bis(4-methoxyphenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]furan-2-carboxamide —— C29H30N4O6
N-[2-[[1,4-bis(4-methoxyphenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]furan-2-carboxamide
—— (4R)-3-tert-butyl-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C30H36N4O4S
(4R)-3-tert-butyl-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4S)-3-tert-butyl-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C30H39N5O4S
2-[(4S)-3-tert-butyl-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 2-[(4S)-4-(2-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C31H32ClN5O2S
2-[(4S)-4-(2-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— N-[2-[[1,4-bis(4-methoxyphenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]furan-2-carboxamide —— C29H30N4O6
N-[2-[[1,4-bis(4-methoxyphenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]furan-2-carboxamide
—— 2-[(4R)-4-(2-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C31H32ClN5O2S
2-[(4R)-4-(2-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— N-[2-[[4-(4-chlorophenyl)-1-(3-methoxyphenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]thiophene-2-carboxamide —— C28H27ClN4O4S
N-[2-[[4-(4-chlorophenyl)-1-(3-methoxyphenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]thiophene-2-carboxamide
—— N-[3-(3,5-dimethylpyrazol-1-yl)phenyl]-2-[(1R,2S,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetamide —— C22H22N4O3
N-[3-(3,5-dimethylpyrazol-1-yl)phenyl]-2-[(1R,2S,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C31H30FN5O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C30H37N5O4S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 2-[(4S)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C31H31F2N5O3S
2-[(4S)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— N-[3-(3,5-dimethylpyrazol-1-yl)phenyl]-2-[(1R,2R,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetamide —— C22H22N4O3
N-[3-(3,5-dimethylpyrazol-1-yl)phenyl]-2-[(1R,2R,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetamide
—— 2-[(4R)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C31H31F2N5O3S
2-[(4R)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C30H37N5O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— (2-phenyl-1,3-thiazol-4-yl)-[(5S)-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepan-4-yl]methanone —— C20H25N3OS2
(2-phenyl-1,3-thiazol-4-yl)-[(5S)-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepan-4-yl]methanone
—— 2-[(4S)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C32H35N5O3S
2-[(4S)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— (5-methyl-1-phenylpyrazol-4-yl)-[(5S)-5-(piperidin-1-ylmethyl)-1,4-thiazepan-4-yl]methanone —— C22H30N4OS
(5-methyl-1-phenylpyrazol-4-yl)-[(5S)-5-(piperidin-1-ylmethyl)-1,4-thiazepan-4-yl]methanone
—— (2-methyl-5-phenylpyrazol-3-yl)-[(5S)-5-(morpholin-4-ylmethyl)-1,4-thiazepan-4-yl]methanone —— C21H28N4O2S
(2-methyl-5-phenylpyrazol-3-yl)-[(5S)-5-(morpholin-4-ylmethyl)-1,4-thiazepan-4-yl]methanone
—— [(2S)-1-[[(3R)-1,1-dioxothiolan-3-yl]amino]-1-oxopropan-2-yl] 2-(2-thiophen-2-yl-1,3-thiazol-4-yl)acetate —— C16H18N2O5S3
[(2S)-1-[[(3R)-1,1-dioxothiolan-3-yl]amino]-1-oxopropan-2-yl] 2-(2-thiophen-2-yl-1,3-thiazol-4-yl)acetate
—— 2-[(4R)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C32H35N5O3S
2-[(4R)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 5-[[5-(4-Bromophenyl)tetrazol-2-yl]methyl]-3-thiophen-3-yl-1,2,4-oxadiazole —— C14H9BrN6OS
5-[[5-(4-Bromophenyl)tetrazol-2-yl]methyl]-3-thiophen-3-yl-1,2,4-oxadiazole
—— 2-[(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C29H35F2N5O3S
2-[(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— [(2S)-1-(3-fluoroanilino)-1-oxopropan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate —— C19H17FN4O3
[(2S)-1-(3-fluoroanilino)-1-oxopropan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate
—— [(2R)-1-[[(3R)-1,1-dioxothiolan-3-yl]amino]-1-oxopropan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate —— C17H20N4O5S
[(2R)-1-[[(3R)-1,1-dioxothiolan-3-yl]amino]-1-oxopropan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate
—— (2-phenyl-1,3-thiazol-4-yl)-[(5R)-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepan-4-yl]methanone —— C20H25N3OS2
(2-phenyl-1,3-thiazol-4-yl)-[(5R)-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepan-4-yl]methanone
—— 2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C29H35F2N5O3S
2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 2-[(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C28H30F2N4O3S
2-[(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— [(2S)-1-[[(3S)-1,1-dioxothiolan-3-yl]-methylamino]-1-oxopropan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate —— C18H22N4O5S
[(2S)-1-[[(3S)-1,1-dioxothiolan-3-yl]-methylamino]-1-oxopropan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate
—— (5-methyl-1-phenylpyrazol-4-yl)-[(5R)-5-(piperidin-1-ylmethyl)-1,4-thiazepan-4-yl]methanone —— C22H30N4OS
(5-methyl-1-phenylpyrazol-4-yl)-[(5R)-5-(piperidin-1-ylmethyl)-1,4-thiazepan-4-yl]methanone
—— [(2S)-1-oxo-1-(prop-2-enylamino)propan-2-yl] 2-(3-methylbutylamino)-1,3-thiazole-4-carboxylate —— C15H23N3O3S
[(2S)-1-oxo-1-(prop-2-enylamino)propan-2-yl] 2-(3-methylbutylamino)-1,3-thiazole-4-carboxylate
—— [(2S)-1-(3-chloro-2-methylanilino)-1-oxopropan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate —— C20H19ClN4O3
[(2S)-1-(3-chloro-2-methylanilino)-1-oxopropan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate
—— [(2R)-1-oxo-1-(prop-2-enylamino)propan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate —— C16H18N4O3
[(2R)-1-oxo-1-(prop-2-enylamino)propan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate
—— [(2R)-1-oxo-1-(3-oxo-2,4-dihydroquinoxalin-1-yl)propan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate —— C21H19N5O4
[(2R)-1-oxo-1-(3-oxo-2,4-dihydroquinoxalin-1-yl)propan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate
—— [(2R)-1-(2-methoxyethylamino)-1-oxopropan-2-yl] 1-benzyl-3-phenylpyrazole-4-carboxylate —— C23H25N3O4
[(2R)-1-(2-methoxyethylamino)-1-oxopropan-2-yl] 1-benzyl-3-phenylpyrazole-4-carboxylate
—— [(2S)-1-[(4-methylphenyl)methylamino]-1-oxopropan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate —— C21H22N4O3
[(2S)-1-[(4-methylphenyl)methylamino]-1-oxopropan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate
—— (3-methoxy-1-methylpyrazol-4-yl)-[(5S)-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepan-4-yl]methanone —— C16H26N4O2S
(3-methoxy-1-methylpyrazol-4-yl)-[(5S)-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepan-4-yl]methanone
—— 2-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C23H30FN3O
2-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide