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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2S)-2-[[4-amino-5-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(3S)-1,1-dioxothiolan-3-yl]propanamide —— C15H18FN5O3S2
(2S)-2-[[4-amino-5-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(3S)-1,1-dioxothiolan-3-yl]propanamide
—— (2R)-2-[[4-amino-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(4-fluorophenyl)methyl]propanamide —— C18H17F2N5OS
(2R)-2-[[4-amino-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(4-fluorophenyl)methyl]propanamide
—— N-[(2S)-butan-2-yl]-4-methyl-5-(2-morpholin-4-ylsulfonyl-4-nitrophenoxy)-1-phenylpyrazole-3-carboxamide —— C25H29N5O7S
N-[(2S)-butan-2-yl]-4-methyl-5-(2-morpholin-4-ylsulfonyl-4-nitrophenoxy)-1-phenylpyrazole-3-carboxamide
—— (2R)-2-[[4-amino-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,4-difluorophenyl)propanamide —— C17H14F3N5OS
(2R)-2-[[4-amino-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,4-difluorophenyl)propanamide
—— (4R)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C32H30N4O4S
(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 3-[(5-Chloro-2-methoxyphenyl)methylsulfanyl]-5-(2-fluorophenyl)-1,2,4-triazol-4-amine —— C16H14ClFN4OS
3-[(5-Chloro-2-methoxyphenyl)methylsulfanyl]-5-(2-fluorophenyl)-1,2,4-triazol-4-amine
—— (2R)-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]-N,N-di(propan-2-yl)propanamide —— C18H26N4OS
(2R)-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]-N,N-di(propan-2-yl)propanamide
—— 2-[(4R)-1-(2,3-dimethylphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C36H33FN4O2S
2-[(4R)-1-(2,3-dimethylphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— (2S)-2-[[4-amino-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-prop-2-enylpropanamide —— C14H16FN5OS
(2S)-2-[[4-amino-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-prop-2-enylpropanamide
—— (2R)-2-[[4-amino-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methylpropyl)propanamide —— C15H20FN5OS
(2R)-2-[[4-amino-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methylpropyl)propanamide
—— (2R)-2-[[4-amino-5-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(3,4-difluorophenyl)propanamide —— C17H14F3N5OS
(2R)-2-[[4-amino-5-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(3,4-difluorophenyl)propanamide
—— (2R)-2-[[4-(furan-2-ylmethyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methoxyethyl)propanamide —— C19H22N4O3S
(2R)-2-[[4-(furan-2-ylmethyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methoxyethyl)propanamide
—— (4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(3-fluorophenyl)-1-(4-methoxyphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H36FN5O4S
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(3-fluorophenyl)-1-(4-methoxyphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[tert-butylcarbamoyl-[[(2S)-oxolan-2-yl]methyl]amino]-N-[4-(4-chlorophenyl)-1-(3,4-dimethylphenyl)imidazol-2-yl]acetamide —— C29H36ClN5O3
2-[tert-butylcarbamoyl-[[(2S)-oxolan-2-yl]methyl]amino]-N-[4-(4-chlorophenyl)-1-(3,4-dimethylphenyl)imidazol-2-yl]acetamide
—— (2S)-2-[[4-amino-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[2-(4-methoxyphenyl)ethyl]propanamide —— C20H22FN5O2S
(2S)-2-[[4-amino-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[2-(4-methoxyphenyl)ethyl]propanamide
—— (2S)-2-[[4-amino-5-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(3R)-1,1-dioxothiolan-3-yl]-N-methylpropanamide —— C16H20FN5O3S2
(2S)-2-[[4-amino-5-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(3R)-1,1-dioxothiolan-3-yl]-N-methylpropanamide
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-propan-2-ylpyrazole-3-carboxamide —— C24H28FN5O6S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-propan-2-ylpyrazole-3-carboxamide
—— (4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(3-fluorophenyl)-1-(4-methoxyphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H36FN5O4S
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(3-fluorophenyl)-1-(4-methoxyphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C26H30FN5O7S
5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— N-[(2R)-butan-2-yl]-5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methylpyrazole-3-carboxamide —— C25H30FN5O6S
N-[(2R)-butan-2-yl]-5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methylpyrazole-3-carboxamide
—— 3-(2-fluorophenyl)-5-[(1R)-1-(3-nitrophenyl)ethyl]sulfanyl-1,2,4-triazol-4-amine —— C16H14FN5O2S
3-(2-fluorophenyl)-5-[(1R)-1-(3-nitrophenyl)ethyl]sulfanyl-1,2,4-triazol-4-amine
—— (2R)-2-[[4-amino-5-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(3-fluorophenyl)propanamide —— C17H15F2N5OS
(2R)-2-[[4-amino-5-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(3-fluorophenyl)propanamide
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-chlorophenyl)-N-(2-methoxyethyl)-4-methylpyrazole-3-carboxamide —— C24H28ClN5O7S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-chlorophenyl)-N-(2-methoxyethyl)-4-methylpyrazole-3-carboxamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C31H28N4O4S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C35H29FN4O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 1-(4-fluorophenyl)-4-methyl-5-(2-morpholin-4-ylsulfonyl-4-nitrophenoxy)-N-propylpyrazole-3-carboxamide —— C24H26FN5O7S
1-(4-fluorophenyl)-4-methyl-5-(2-morpholin-4-ylsulfonyl-4-nitrophenoxy)-N-propylpyrazole-3-carboxamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C33H28N4O5S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— (4S)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C33H32F2N4O3S
(4S)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— N-[(2R)-butan-2-yl]-5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methylpyrazole-3-carboxamide —— C25H30FN5O6S
N-[(2R)-butan-2-yl]-5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methylpyrazole-3-carboxamide
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-chlorophenyl)-4-methyl-N-(pyridin-3-ylmethyl)pyrazole-3-carboxamide —— C27H27ClN6O6S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-chlorophenyl)-4-methyl-N-(pyridin-3-ylmethyl)pyrazole-3-carboxamide
—— N-[(2R)-butan-2-yl]-4-methyl-5-(2-morpholin-4-ylsulfonyl-4-nitrophenoxy)-1-phenylpyrazole-3-carboxamide —— C25H29N5O7S
N-[(2R)-butan-2-yl]-4-methyl-5-(2-morpholin-4-ylsulfonyl-4-nitrophenoxy)-1-phenylpyrazole-3-carboxamide
—— 1-(4-fluorophenyl)-4-methyl-5-(2-morpholin-4-ylsulfonyl-4-nitrophenoxy)-N-propan-2-ylpyrazole-3-carboxamide —— C24H26FN5O7S
1-(4-fluorophenyl)-4-methyl-5-(2-morpholin-4-ylsulfonyl-4-nitrophenoxy)-N-propan-2-ylpyrazole-3-carboxamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C33H28N4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C31H28N4O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— 5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C26H30FN5O7S
5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— (4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C32H30N4O5S
(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4R)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C33H32F2N4O3S
(4R)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C27H31ClN4O3S2
2-[(4R)-3-tert-butyl-1-(3-chlorophenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— (4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-fluorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C28H30ClFN4O3S
(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-fluorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 1-(4-methoxyphenyl)-4-methyl-5-[4-[[(2S)-2-methylbutanoyl]amino]-2-(2-morpholin-4-ylethylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid —— C29H37N5O8S
1-(4-methoxyphenyl)-4-methyl-5-[4-[[(2S)-2-methylbutanoyl]amino]-2-(2-morpholin-4-ylethylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-chlorophenyl)-N-(2-methoxyethyl)-4-methylpyrazole-3-carboxamide —— C24H28ClN5O7S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-chlorophenyl)-N-(2-methoxyethyl)-4-methylpyrazole-3-carboxamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C32H32N4O5S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— 5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-1-(3-chlorophenyl)-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C26H30ClN5O7S
5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-1-(3-chlorophenyl)-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-1-(3-chlorophenyl)-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C26H30ClN5O7S
5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-1-(3-chlorophenyl)-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C33H32N4O5S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— (4R)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C32H30N4O5S
(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[tert-butylcarbamoyl-[[(2R)-oxolan-2-yl]methyl]amino]-N-[4-(4-chlorophenyl)-1-(3,4-dimethylphenyl)imidazol-2-yl]acetamide —— C29H36ClN5O3
2-[tert-butylcarbamoyl-[[(2R)-oxolan-2-yl]methyl]amino]-N-[4-(4-chlorophenyl)-1-(3,4-dimethylphenyl)imidazol-2-yl]acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C33H32N4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— (4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C32H30N4O4S
(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (2S)-N-(5-chloro-2-methylphenyl)-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propanamide —— C19H19ClN4OS
(2S)-N-(5-chloro-2-methylphenyl)-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propanamide