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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(1R)-1-(3-nitrophenyl)ethyl]propanamide —— C20H19FN4O4
3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(1R)-1-(3-nitrophenyl)ethyl]propanamide
—— N-(4-bromophenyl)-3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide —— C17H13BrFN3O2
N-(4-bromophenyl)-3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide
—— 3-Amino-2-[2-[[4-(3,4-dimethylphenyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]but-2-enenitrile —— C22H21N5OS
3-Amino-2-[2-[[4-(3,4-dimethylphenyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]but-2-enenitrile
—— 4-[5-[(5-Fluoro-2-methoxyphenyl)methylsulfanyl]-4-(3-fluorophenyl)-1,2,4-triazol-3-yl]morpholine —— C20H20F2N4O2S
4-[5-[(5-Fluoro-2-methoxyphenyl)methylsulfanyl]-4-(3-fluorophenyl)-1,2,4-triazol-3-yl]morpholine
—— N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazole-4-carboxamide —— C18H15N3O3
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazole-4-carboxamide
—— N-(3-bromophenyl)-3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide —— C17H13BrFN3O2
N-(3-bromophenyl)-3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide
—— 4-[4-(3-Fluorophenyl)-5-[2-(3-methylphenoxy)ethylsulfanyl]-1,2,4-triazol-3-yl]morpholine —— C21H23FN4O2S
4-[4-(3-Fluorophenyl)-5-[2-(3-methylphenoxy)ethylsulfanyl]-1,2,4-triazol-3-yl]morpholine
—— [4-[(4-Methoxyphenyl)methyl]piperazin-1-yl]-(4-pyrazol-1-ylphenyl)methanone —— C22H24N4O2
[4-[(4-Methoxyphenyl)methyl]piperazin-1-yl]-(4-pyrazol-1-ylphenyl)methanone
—— ethyl (E)-2-cyano-3-[[4-(5-methylfuran-2-yl)-1,3-thiazol-2-yl]amino]prop-2-enoate —— C14H13N3O3S
ethyl (E)-2-cyano-3-[[4-(5-methylfuran-2-yl)-1,3-thiazol-2-yl]amino]prop-2-enoate
—— 2-[[4-(3-fluorophenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]-N-(3-methoxypropyl)acetamide —— C18H24FN5O3S
2-[[4-(3-fluorophenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]-N-(3-methoxypropyl)acetamide
—— 4-[4-(3-fluorophenyl)-5-[[(2R)-oxolan-2-yl]methylsulfanyl]-1,2,4-triazol-3-yl]morpholine —— C17H21FN4O2S
4-[4-(3-fluorophenyl)-5-[[(2R)-oxolan-2-yl]methylsulfanyl]-1,2,4-triazol-3-yl]morpholine
—— 4-[4-(3-fluorophenyl)-5-[[(2R)-oxan-2-yl]methylsulfanyl]-1,2,4-triazol-3-yl]morpholine —— C18H23FN4O2S
4-[4-(3-fluorophenyl)-5-[[(2R)-oxan-2-yl]methylsulfanyl]-1,2,4-triazol-3-yl]morpholine
—— 2-[[[4-(4-Methylphenyl)-1,3-thiazol-2-yl]amino]methylidene]propanedinitrile —— C14H10N4S
2-[[[4-(4-Methylphenyl)-1,3-thiazol-2-yl]amino]methylidene]propanedinitrile
—— ethyl (E)-3-[[4-(2-chlorophenyl)-1,3-thiazol-2-yl]amino]-2-cyanoprop-2-enoate —— C15H12ClN3O2S
ethyl (E)-3-[[4-(2-chlorophenyl)-1,3-thiazol-2-yl]amino]-2-cyanoprop-2-enoate
—— (2R)-2-[[4-(3-fluorophenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C15H18FN5O2S
(2R)-2-[[4-(3-fluorophenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 2-[[4-(3-fluorophenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]-N-propylacetamide —— C17H22FN5O2S
2-[[4-(3-fluorophenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]-N-propylacetamide
—— (2S)-3-[[4-(3-fluorophenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]-2-methylpropanenitrile —— C16H18FN5OS
(2S)-3-[[4-(3-fluorophenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]-2-methylpropanenitrile
—— Ethyl 5-(2,2-dicyanoethenylamino)-1-(3,5-dimethylphenyl)pyrazole-4-carboxylate —— C18H17N5O2
Ethyl 5-(2,2-dicyanoethenylamino)-1-(3,5-dimethylphenyl)pyrazole-4-carboxylate
—— 4-[[4-(3-Fluorophenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]butanenitrile —— C16H18FN5OS
4-[[4-(3-Fluorophenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]butanenitrile
—— ethyl (E)-2-cyano-3-[[4-(4-methylphenyl)-1,3-thiazol-2-yl]amino]prop-2-enoate —— C16H15N3O2S
ethyl (E)-2-cyano-3-[[4-(4-methylphenyl)-1,3-thiazol-2-yl]amino]prop-2-enoate
—— N-ethyl-2-[[4-(3-fluorophenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methylprop-2-enyl)acetamide —— C20H26FN5O2S
N-ethyl-2-[[4-(3-fluorophenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methylprop-2-enyl)acetamide
—— 2-[[5-(4-tert-butylphenyl)-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(3R)-1,1-dioxothiolan-3-yl]-N-ethylacetamide —— C27H34N4O4S2
2-[[5-(4-tert-butylphenyl)-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(3R)-1,1-dioxothiolan-3-yl]-N-ethylacetamide
—— 4-[5-Benzylsulfanyl-4-(3-fluorophenyl)-1,2,4-triazol-3-yl]morpholine —— C19H19FN4OS
4-[5-Benzylsulfanyl-4-(3-fluorophenyl)-1,2,4-triazol-3-yl]morpholine
—— 2-[[(5-Benzyl-1,3-thiazol-2-yl)amino]methylidene]propanedinitrile —— C14H10N4S
2-[[(5-Benzyl-1,3-thiazol-2-yl)amino]methylidene]propanedinitrile
—— (7R)-2-[(1S)-1-[[4,5-bis(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C27H23Cl2N5OS2
(7R)-2-[(1S)-1-[[4,5-bis(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 2-[[[4-(2,5-Dimethyl-1-propylpyrrol-3-yl)-1,3-thiazol-2-yl]amino]methylidene]propanedinitrile —— C16H17N5S
2-[[[4-(2,5-Dimethyl-1-propylpyrrol-3-yl)-1,3-thiazol-2-yl]amino]methylidene]propanedinitrile
—— N-[5-(3,4-dimethoxyphenyl)-1H-1,2,4-triazol-3-yl]-4-fluorobenzamide —— C17H15FN4O3
N-[5-(3,4-dimethoxyphenyl)-1H-1,2,4-triazol-3-yl]-4-fluorobenzamide
—— (Z)-3-amino-2-[2-[[5-(4-tert-butylphenyl)-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]but-2-enenitrile —— C23H25N5O2S
(Z)-3-amino-2-[2-[[5-(4-tert-butylphenyl)-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]but-2-enenitrile
—— ethyl (E)-2-cyano-3-[(4-pyridin-3-yl-1,3-thiazol-2-yl)amino]prop-2-enoate —— C14H12N4O2S
ethyl (E)-2-cyano-3-[(4-pyridin-3-yl-1,3-thiazol-2-yl)amino]prop-2-enoate
—— (2S)-N-(4-acetamidophenyl)-2-[[5-(4-tert-butylphenyl)-4-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C31H35N5O3S
(2S)-N-(4-acetamidophenyl)-2-[[5-(4-tert-butylphenyl)-4-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— [(2S)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] (Z)-3-[5-chloro-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]prop-2-enoate —— C25H28ClN5O6S
[(2S)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] (Z)-3-[5-chloro-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]prop-2-enoate
—— N-[2-[6-(2,5-dimethoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]ethyl]-4-methoxy-N-[[(2S)-oxolan-2-yl]methyl]benzenesulfonamide —— C27H31N3O6S2
N-[2-[6-(2,5-dimethoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]ethyl]-4-methoxy-N-[[(2S)-oxolan-2-yl]methyl]benzenesulfonamide
—— 1-(4-nitrophenyl)-4-N-[(Z)-pyridin-4-ylmethylideneamino]-5-N-[(E)-pyridin-4-ylmethylideneamino]triazole-4,5-dicarboxamide —— C22H16N10O4
1-(4-nitrophenyl)-4-N-[(Z)-pyridin-4-ylmethylideneamino]-5-N-[(E)-pyridin-4-ylmethylideneamino]triazole-4,5-dicarboxamide
—— (4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(4-fluorophenyl)-1-(4-methoxyphenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C33H32FN5O4S
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(4-fluorophenyl)-1-(4-methoxyphenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 3-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[[2-[(dimethylamino)methyl]phenyl]methyl]propanamide —— C21H23ClN4O2
3-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[[2-[(dimethylamino)methyl]phenyl]methyl]propanamide
—— (5S,7S)-3-chloro-N-[2-(1,2,4-triazol-1-yl)-5-(trifluoromethyl)phenyl]adamantane-1-carboxamide —— C20H20ClF3N4O
(5S,7S)-3-chloro-N-[2-(1,2,4-triazol-1-yl)-5-(trifluoromethyl)phenyl]adamantane-1-carboxamide
—— (E)-N-benzyl-4-[[5-(4-tert-butylphenyl)-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-cyano-3-hydroxybut-2-enamide —— C31H31N5O3S
(E)-N-benzyl-4-[[5-(4-tert-butylphenyl)-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-cyano-3-hydroxybut-2-enamide
—— (2R)-2-[4-(5-acetyl-4-methyl-1,3-thiazol-2-yl)phenoxy]-N-benzyl-N-methylpropanamide —— C23H24N2O3S
(2R)-2-[4-(5-acetyl-4-methyl-1,3-thiazol-2-yl)phenoxy]-N-benzyl-N-methylpropanamide
—— 2-[[5-(4-tert-butylphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-1-[(3R)-5-(4-chlorophenyl)-3-(furan-2-yl)-3,4-dihydropyrazol-2-yl]ethanone —— C30H30ClN5O2S
2-[[5-(4-tert-butylphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-1-[(3R)-5-(4-chlorophenyl)-3-(furan-2-yl)-3,4-dihydropyrazol-2-yl]ethanone
—— 2-[(4-bromophenyl)sulfonyl-butylamino]-N-[2-(4-chlorophenyl)-5-phenylpyrazol-3-yl]acetamide —— C27H26BrClN4O3S
2-[(4-bromophenyl)sulfonyl-butylamino]-N-[2-(4-chlorophenyl)-5-phenylpyrazol-3-yl]acetamide
—— 2-[4-(5-acetyl-4-methyl-1,3-thiazol-2-yl)phenoxy]-N-(3-phenylpropyl)acetamide —— C23H24N2O3S
2-[4-(5-acetyl-4-methyl-1,3-thiazol-2-yl)phenoxy]-N-(3-phenylpropyl)acetamide
—— 2-[[5-(4-tert-butylphenyl)-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(3S)-1,1-dioxothiolan-3-yl]-N-ethylacetamide —— C27H34N4O4S2
2-[[5-(4-tert-butylphenyl)-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(3S)-1,1-dioxothiolan-3-yl]-N-ethylacetamide
—— N-[2-[6-(2,5-dimethoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]ethyl]-4-methoxy-N-[[(2R)-oxolan-2-yl]methyl]benzenesulfonamide —— C27H31N3O6S2
N-[2-[6-(2,5-dimethoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]ethyl]-4-methoxy-N-[[(2R)-oxolan-2-yl]methyl]benzenesulfonamide
—— 1-[2-[4-[[(1S)-2,2-dichlorocyclopropyl]methoxy]phenyl]-4-methyl-1,3-thiazol-5-yl]ethanone —— C16H15Cl2NO2S
1-[2-[4-[[(1S)-2,2-dichlorocyclopropyl]methoxy]phenyl]-4-methyl-1,3-thiazol-5-yl]ethanone
—— (E)-N-benzyl-4-[[4-(4-chlorophenyl)-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-cyano-3-hydroxybut-2-enamide —— C27H22ClN5O3S
(E)-N-benzyl-4-[[4-(4-chlorophenyl)-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-cyano-3-hydroxybut-2-enamide
—— 2-[4-(5-acetyl-4-methyl-1,3-thiazol-2-yl)phenoxy]-N-[(2S)-3-methylbutan-2-yl]acetamide —— C19H24N2O3S
2-[4-(5-acetyl-4-methyl-1,3-thiazol-2-yl)phenoxy]-N-[(2S)-3-methylbutan-2-yl]acetamide
—— 2-[(4S)-4-(4-fluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C34H28F2N4O3S
2-[(4S)-4-(4-fluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— N-[[2-[(dimethylamino)methyl]phenyl]methyl]-3-[1-(3-methoxyphenyl)-3,5-dimethylpyrazol-4-yl]propanamide —— C25H32N4O2
N-[[2-[(dimethylamino)methyl]phenyl]methyl]-3-[1-(3-methoxyphenyl)-3,5-dimethylpyrazol-4-yl]propanamide
—— 2-[4-(5-acetyl-4-methyl-1,3-thiazol-2-yl)phenoxy]-N-benzylacetamide —— C21H20N2O3S
2-[4-(5-acetyl-4-methyl-1,3-thiazol-2-yl)phenoxy]-N-benzylacetamide
—— [(2S)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] (Z)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]prop-2-enoate —— C25H28ClN5O6S
[(2S)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] (Z)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]prop-2-enoate