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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[[4-benzyl-5-(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]acetamide —— C26H29ClN4OS
2-[[4-benzyl-5-(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]acetamide
—— N-butyl-2,2-dichloro-N-[2-[(2R)-2-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]acetamide —— C21H25Cl3N4O3
N-butyl-2,2-dichloro-N-[2-[(2R)-2-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]acetamide
—— 2-[(4S)-1-(2,3-dimethylphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C32H34N4O2S
2-[(4S)-1-(2,3-dimethylphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-[(2-methoxyacetyl)amino]phenoxy]-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxylic acid —— C25H30N4O8S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-[(2-methoxyacetyl)amino]phenoxy]-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxylic acid
—— N-butyl-2,2-dichloro-N-[2-[(2S)-2-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]acetamide —— C21H25Cl3N4O3
N-butyl-2,2-dichloro-N-[2-[(2S)-2-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]acetamide
—— 2-[[4-benzyl-5-(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]acetamide —— C26H29ClN4OS
2-[[4-benzyl-5-(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C31H30ClN5O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 2-[(4S)-3-tert-butyl-1-(2-chlorophenyl)-4-(3,4-dimethoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C32H34ClN5O4S
2-[(4S)-3-tert-butyl-1-(2-chlorophenyl)-4-(3,4-dimethoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— 2,3-dichloro-N-[4-(tetrazol-1-yl)phenyl]benzenesulfonamide —— C13H9Cl2N5O2S
2,3-dichloro-N-[4-(tetrazol-1-yl)phenyl]benzenesulfonamide
—— [3-(3-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl 2-anilino-4-oxofuran-3-carboxylate —— C20H14ClN3O5
[3-(3-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl 2-anilino-4-oxofuran-3-carboxylate
—— [3-(4-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl 2-anilino-4-oxofuran-3-carboxylate —— C20H14ClN3O5
[3-(4-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl 2-anilino-4-oxofuran-3-carboxylate
—— 2,3,5,6-tetramethyl-N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]benzenesulfonamide —— C23H28N4O2S
2,3,5,6-tetramethyl-N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]benzenesulfonamide
—— 3-(4-fluorophenyl)-4-[(Z)-[4-[2-hydroxyethyl(methyl)amino]phenyl]methylideneamino]-1H-1,2,4-triazole-5-thione —— C18H18FN5OS
3-(4-fluorophenyl)-4-[(Z)-[4-[2-hydroxyethyl(methyl)amino]phenyl]methylideneamino]-1H-1,2,4-triazole-5-thione
—— 4-methyl-N-[4-(tetrazol-1-yl)phenyl]benzenesulfonamide 878929-12-5 C14H13N5O2S
4-methyl-N-[4-(tetrazol-1-yl)phenyl]benzenesulfonamide
—— 3-chloro-4-fluoro-N-[4-(tetrazol-1-yl)phenyl]benzenesulfonamide —— C13H9ClFN5O2S
3-chloro-4-fluoro-N-[4-(tetrazol-1-yl)phenyl]benzenesulfonamide
—— 4-bromo-3-methyl-N-[4-(tetrazol-1-yl)phenyl]benzenesulfonamide —— C14H12BrN5O2S
4-bromo-3-methyl-N-[4-(tetrazol-1-yl)phenyl]benzenesulfonamide
—— (2S)-1-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl-(2-methoxyethyl)amino]-3-phenylmethoxypropan-2-ol —— C30H33F2N3O4
(2S)-1-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl-(2-methoxyethyl)amino]-3-phenylmethoxypropan-2-ol
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H30FN5O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— (4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methylphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C32H37N5O5S
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methylphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 1-(5-Bromothiophen-2-yl)-2-[5-(2-methylphenyl)tetrazol-2-yl]ethanone —— C14H11BrN4OS
1-(5-Bromothiophen-2-yl)-2-[5-(2-methylphenyl)tetrazol-2-yl]ethanone
—— (2S)-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[[4-(furan-2-ylmethyl)-5-[(4-methoxyphenoxy)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C29H30N6O5S
(2S)-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[[4-(furan-2-ylmethyl)-5-[(4-methoxyphenoxy)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 2-[[5-(2-chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(2-methoxyphenyl)methyl]-N-methylacetamide —— C20H21ClN4O2S
2-[[5-(2-chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(2-methoxyphenyl)methyl]-N-methylacetamide
—— 3-methylsulfanyl-5-(4-nitrophenyl)-4-[(Z)-2-pyrrolidin-1-ylprop-1-enyl]-1,2,4-triazole —— C16H19N5O2S
3-methylsulfanyl-5-(4-nitrophenyl)-4-[(Z)-2-pyrrolidin-1-ylprop-1-enyl]-1,2,4-triazole
—— N-[(1R)-1-[5-[(4-fluorophenyl)methylsulfanyl]-4-(4-nitrophenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]-4-pentylbenzamide —— C35H34FN5O3S
N-[(1R)-1-[5-[(4-fluorophenyl)methylsulfanyl]-4-(4-nitrophenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]-4-pentylbenzamide
—— N-[(1S)-1-[5-[(4-fluorophenyl)methylsulfanyl]-4-(4-nitrophenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]-4-pentylbenzamide —— C35H34FN5O3S
N-[(1S)-1-[5-[(4-fluorophenyl)methylsulfanyl]-4-(4-nitrophenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]-4-pentylbenzamide
—— N-[(5-chlorothiophen-2-yl)methyl]-2-[5-(2-methylphenyl)tetrazol-2-yl]-N-prop-2-enylacetamide —— C18H18ClN5OS
N-[(5-chlorothiophen-2-yl)methyl]-2-[5-(2-methylphenyl)tetrazol-2-yl]-N-prop-2-enylacetamide
—— 2-(2,5-Dimethylfuran-3-yl)-5-[(4-ethyl-5-phenyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3,4-oxadiazole —— C19H19N5O2S
2-(2,5-Dimethylfuran-3-yl)-5-[(4-ethyl-5-phenyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3,4-oxadiazole
—— 2-[(4S)-4-(3-methylphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-phenylacetamide —— C34H30N4O2S
2-[(4S)-4-(3-methylphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-phenylacetamide
—— 2-[(4R)-3-tert-butyl-4-(2-chlorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C32H32ClFN4O2S
2-[(4R)-3-tert-butyl-4-(2-chlorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— (2R)-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[[4-(furan-2-ylmethyl)-5-[(4-methoxyphenoxy)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C29H30N6O5S
(2R)-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[[4-(furan-2-ylmethyl)-5-[(4-methoxyphenoxy)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C34H29N5O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4R)-3-tert-butyl-1-(4-fluorophenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C32H32F2N4O2S
2-[(4R)-3-tert-butyl-1-(4-fluorophenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— (4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C34H34N4O5S
(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (2S)-1-[[3-ethyl-5-(2-fluorophenoxy)-1-phenylpyrazol-4-yl]methyl-[[(2S)-oxolan-2-yl]methyl]amino]-3-phenoxypropan-2-ol —— C32H36FN3O4
(2S)-1-[[3-ethyl-5-(2-fluorophenoxy)-1-phenylpyrazol-4-yl]methyl-[[(2S)-oxolan-2-yl]methyl]amino]-3-phenoxypropan-2-ol
—— 2-[(4S)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H26ClN5O2S2
2-[(4S)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4S)-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C29H26F2N4O2S
2-[(4S)-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— (2R)-1-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl-(2-methoxyethyl)amino]-3-phenylmethoxypropan-2-ol —— C30H33F2N3O4
(2R)-1-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl-(2-methoxyethyl)amino]-3-phenylmethoxypropan-2-ol
—— 2-[(4R)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C31H26ClN5O2S2
2-[(4R)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 2-[(4S)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C30H29ClN4O3S2
2-[(4S)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-[(4S)-1-(2,3-dimethylphenyl)-4-(3-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C35H30F2N4O2S
2-[(4S)-1-(2,3-dimethylphenyl)-4-(3-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 2-[(4R)-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C34H31N5O4S
2-[(4R)-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4S)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H26FN5O2S2
2-[(4S)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— (1S,2R)-1-chloro-2-fluoro-N-[3-[5-(2-fluorophenyl)-3-[2-(4-methoxyphenyl)ethoxy]-1,2,4-triazol-1-yl]phenyl]cyclopropane-1-carboxamide —— C27H23ClF2N4O3
(1S,2R)-1-chloro-2-fluoro-N-[3-[5-(2-fluorophenyl)-3-[2-(4-methoxyphenyl)ethoxy]-1,2,4-triazol-1-yl]phenyl]cyclopropane-1-carboxamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C34H29N5O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 2-[(4S)-3-tert-butyl-4-(3-methylphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C33H35FN4O2S
2-[(4S)-3-tert-butyl-4-(3-methylphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C31H30ClN5O4S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— (4R)-4-(3-chlorophenyl)-1-(4-methylphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H31ClN4O2S2
(4R)-4-(3-chlorophenyl)-1-(4-methylphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— N-[(4-fluorophenyl)methyl]-2-[(4S)-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C35H31FN4O4S
N-[(4-fluorophenyl)methyl]-2-[(4S)-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— N-[(4-fluorophenyl)methyl]-2-[(4S)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C35H31FN4O3S
N-[(4-fluorophenyl)methyl]-2-[(4S)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— 2-[(4R)-3-tert-butyl-4-(3-methylphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C33H35FN4O2S
2-[(4R)-3-tert-butyl-4-(3-methylphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide