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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5Z)-5-[[1-benzyl-3-(2-methoxyphenyl)pyrazol-4-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C21H17N3O2S2
(5Z)-5-[[1-benzyl-3-(2-methoxyphenyl)pyrazol-4-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— N-[(Z)-1-(4-fluorophenyl)ethylideneamino]-4-phenyl-1,3-thiazol-2-amine —— C17H14FN3S
N-[(Z)-1-(4-fluorophenyl)ethylideneamino]-4-phenyl-1,3-thiazol-2-amine
—— (E)-3-[1-benzyl-3-(3,4-dimethylphenyl)pyrazol-4-yl]-2-cyano-N-prop-2-enylprop-2-enamide —— C25H24N4O
(E)-3-[1-benzyl-3-(3,4-dimethylphenyl)pyrazol-4-yl]-2-cyano-N-prop-2-enylprop-2-enamide
—— 2-methoxyethyl (E)-3-[4-chloro-2-(3-chloro-4-methylanilino)-1,3-thiazol-5-yl]-2-cyanoprop-2-enoate —— C17H15Cl2N3O3S
2-methoxyethyl (E)-3-[4-chloro-2-(3-chloro-4-methylanilino)-1,3-thiazol-5-yl]-2-cyanoprop-2-enoate
—— N-[(Z)-1-(2,5-difluorophenyl)ethylideneamino]-4-phenyl-1,3-thiazol-2-amine —— C17H13F2N3S
N-[(Z)-1-(2,5-difluorophenyl)ethylideneamino]-4-phenyl-1,3-thiazol-2-amine
—— 2-[[1-Benzyl-3-(4-ethylphenyl)pyrazol-4-yl]methylidene]propanedinitrile —— C22H18N4
2-[[1-Benzyl-3-(4-ethylphenyl)pyrazol-4-yl]methylidene]propanedinitrile
—— N-[(Z)-[(3S)-3-methylpentan-2-ylidene]amino]-4-phenyl-1,3-thiazol-2-amine —— C15H19N3S
N-[(Z)-[(3S)-3-methylpentan-2-ylidene]amino]-4-phenyl-1,3-thiazol-2-amine
—— 1-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3-[(2R)-2-ethylhexyl]thiourea —— C20H30N4OS
1-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3-[(2R)-2-ethylhexyl]thiourea
—— 2-[(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C33H34F2N4O2S
2-[(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 1,4-dimethyl-5-[(Z)-[methyl(phenyl)hydrazinylidene]methyl]-2-phenylpyrazol-3-one —— C19H20N4O
1,4-dimethyl-5-[(Z)-[methyl(phenyl)hydrazinylidene]methyl]-2-phenylpyrazol-3-one
—— 1-(1,5-Dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3-(3-fluoro-4-methylphenyl)thiourea —— C19H19FN4OS
1-(1,5-Dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3-(3-fluoro-4-methylphenyl)thiourea
—— 1-(4-phenyl-1,3-thiazol-2-yl)-2-(1-pyrrol-2-ylideneethyl)hydrazine —— C15H14N4S
1-(4-phenyl-1,3-thiazol-2-yl)-2-(1-pyrrol-2-ylideneethyl)hydrazine
—— 1-(4-fluorophenyl)-4-methyl-5-[4-[[(2R)-2-methylbutanoyl]amino]-2-morpholin-4-ylsulfonylphenoxy]pyrazole-3-carboxylic acid —— C26H29FN4O7S
1-(4-fluorophenyl)-4-methyl-5-[4-[[(2R)-2-methylbutanoyl]amino]-2-morpholin-4-ylsulfonylphenoxy]pyrazole-3-carboxylic acid
—— N-[(Z)-[2,5-dimethyl-1-[[(2R)-oxolan-2-yl]methyl]pyrrol-3-yl]methylideneamino]-4-phenyl-1,3-thiazol-2-amine —— C21H24N4OS
N-[(Z)-[2,5-dimethyl-1-[[(2R)-oxolan-2-yl]methyl]pyrrol-3-yl]methylideneamino]-4-phenyl-1,3-thiazol-2-amine
—— N-[(E)-[(1S,5R)-6-bicyclo[3.2.0]hept-2-enylidene]amino]-4-phenyl-1,3-thiazol-2-amine —— C16H15N3S
N-[(E)-[(1S,5R)-6-bicyclo[3.2.0]hept-2-enylidene]amino]-4-phenyl-1,3-thiazol-2-amine
—— 3-fluoro-N-[[5-(2-fluorophenoxy)-1-phenyl-3-propan-2-ylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide —— C31H31F2N3O3
3-fluoro-N-[[5-(2-fluorophenoxy)-1-phenyl-3-propan-2-ylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide
—— N-(pentan-3-ylideneamino)-4-phenyl-1,3-thiazol-2-amine —— C14H17N3S
N-(pentan-3-ylideneamino)-4-phenyl-1,3-thiazol-2-amine
—— N-[(Z)-pentan-2-ylideneamino]-4-phenyl-1,3-thiazol-2-amine —— C14H17N3S
N-[(Z)-pentan-2-ylideneamino]-4-phenyl-1,3-thiazol-2-amine
—— N-[(Z)-(3-methylthiophen-2-yl)methylideneamino]-4-phenyl-1,3-thiazol-2-amine —— C15H13N3S2
N-[(Z)-(3-methylthiophen-2-yl)methylideneamino]-4-phenyl-1,3-thiazol-2-amine
—— 3-fluoro-N-[[5-(2-fluorophenoxy)-1-phenyl-3-propan-2-ylpyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide —— C31H31F2N3O3
3-fluoro-N-[[5-(2-fluorophenoxy)-1-phenyl-3-propan-2-ylpyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide
—— 2-[(4R)-3-tert-butyl-4-(2-methylphenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C32H35N5O2S
2-[(4R)-3-tert-butyl-4-(2-methylphenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— (Z)-N-methyl-N-[(2-methylphenyl)methyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C16H18N2OS
(Z)-N-methyl-N-[(2-methylphenyl)methyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— 3-(2-methylphenyl)-4-[(Z)-(5-phenylthiophen-2-yl)methylideneamino]-1H-1,2,4-triazole-5-thione —— C20H16N4S2
3-(2-methylphenyl)-4-[(Z)-(5-phenylthiophen-2-yl)methylideneamino]-1H-1,2,4-triazole-5-thione
—— 2-[(4R)-1-(2,3-dimethylphenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C32H33FN4O3S
2-[(4R)-1-(2,3-dimethylphenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— 4-[(Z)-[1-benzyl-3-(4-methylphenyl)pyrazol-4-yl]methylideneamino]-1H-1,2,4-triazole-5-thione —— C20H18N6S
4-[(Z)-[1-benzyl-3-(4-methylphenyl)pyrazol-4-yl]methylideneamino]-1H-1,2,4-triazole-5-thione
—— 3-(4-methylphenyl)-4-[(Z)-(5-phenylthiophen-2-yl)methylideneamino]-1H-1,2,4-triazole-5-thione —— C20H16N4S2
3-(4-methylphenyl)-4-[(Z)-(5-phenylthiophen-2-yl)methylideneamino]-1H-1,2,4-triazole-5-thione
—— 2-[[5-[(1-Methylpyrrol-2-yl)methyl]-4-[3-(trifluoromethyl)phenyl]-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C17H16F3N5OS
2-[[5-[(1-Methylpyrrol-2-yl)methyl]-4-[3-(trifluoromethyl)phenyl]-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— 7-[(2,4-Dichlorophenyl)methylsulfanyl]-3-(4-fluorophenyl)triazolo[4,5-d]pyrimidine —— C17H10Cl2FN5S
7-[(2,4-Dichlorophenyl)methylsulfanyl]-3-(4-fluorophenyl)triazolo[4,5-d]pyrimidine
—— 2-[(4S)-3-tert-butyl-4-(2-methylphenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C32H35N5O2S
2-[(4S)-3-tert-butyl-4-(2-methylphenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 3-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-4-(2-phenylethyl)-1H-1,2,4-triazol-5-one —— C20H19N5O2S
3-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-4-(2-phenylethyl)-1H-1,2,4-triazol-5-one
—— N-(5-ethyl-1,3,4-thiadiazol-2-yl)-1-(4-fluorophenyl)-3-(4-methylphenyl)pyrazole-4-carboxamide —— C21H18FN5OS
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-1-(4-fluorophenyl)-3-(4-methylphenyl)pyrazole-4-carboxamide
—— 4-methyl-5-[4-[[(2S)-2-methylbutanoyl]amino]-2-(2-morpholin-4-ylethylsulfamoyl)phenoxy]-1-phenylpyrazole-3-carboxylic acid —— C28H35N5O7S
4-methyl-5-[4-[[(2S)-2-methylbutanoyl]amino]-2-(2-morpholin-4-ylethylsulfamoyl)phenoxy]-1-phenylpyrazole-3-carboxylic acid
—— (4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-tert-butyl-4-(2,5-dimethoxyphenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C32H39N5O5S
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-tert-butyl-4-(2,5-dimethoxyphenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-(2,3-dimethylphenyl)-4-(4-fluorophenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C34H34FN5O3S
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-(2,3-dimethylphenyl)-4-(4-fluorophenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C33H28N4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— (4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-tert-butyl-4-(2,5-dimethoxyphenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C32H39N5O5S
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-tert-butyl-4-(2,5-dimethoxyphenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-(2,3-dimethylphenyl)-4-(4-fluorophenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C34H34FN5O3S
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-(2,3-dimethylphenyl)-4-(4-fluorophenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C28H25ClN4O3S2
2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C34H29N5O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 1-(3-fluorophenyl)-4-methyl-5-[4-[[(2S)-2-methylbutanoyl]amino]-2-(2-morpholin-4-ylethylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid —— C28H34FN5O7S
1-(3-fluorophenyl)-4-methyl-5-[4-[[(2S)-2-methylbutanoyl]amino]-2-(2-morpholin-4-ylethylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid
—— 2-[(4R)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C34H28F2N4O3S
2-[(4R)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C29H29ClN4O4S2
2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C33H28N4O5S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 2-[(4S)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C34H28F2N4O3S
2-[(4S)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 1-(3-fluorophenyl)-4-methyl-5-[4-[[(2S)-2-methylbutanoyl]amino]-2-(3-morpholin-4-ylpropylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid —— C29H36FN5O7S
1-(3-fluorophenyl)-4-methyl-5-[4-[[(2S)-2-methylbutanoyl]amino]-2-(3-morpholin-4-ylpropylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid
—— 1-(3-fluorophenyl)-4-methyl-5-[4-[[(2R)-2-methylbutanoyl]amino]-2-(2-morpholin-4-ylethylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid —— C28H34FN5O7S
1-(3-fluorophenyl)-4-methyl-5-[4-[[(2R)-2-methylbutanoyl]amino]-2-(2-morpholin-4-ylethylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid
—— 2-[(4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C33H27ClFN5O2S
2-[(4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 5-amino-3-[(E)-1-cyano-2-[3,5-dichloro-2-[(2,4-dichlorophenyl)methoxy]phenyl]ethenyl]-1-phenylpyrazole-4-carbonitrile —— C26H15Cl4N5O
5-amino-3-[(E)-1-cyano-2-[3,5-dichloro-2-[(2,4-dichlorophenyl)methoxy]phenyl]ethenyl]-1-phenylpyrazole-4-carbonitrile
—— 2-[(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C29H30ClN5O2S2
2-[(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C34H29N5O4S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide