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中文名称 英文名称 CAS号 化学式 结构式图片
—— Ethyl 1-[2-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxo-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl]piperidine-4-carboxylate —— C27H27N7O4S
Ethyl 1-[2-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxo-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl]piperidine-4-carboxylate
—— Ethyl 1-[1-oxo-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl]piperidine-4-carboxylate —— C27H24F3N7O4
Ethyl 1-[1-oxo-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl]piperidine-4-carboxylate
—— 4-[3-[2-(3-Hydroxypyridin-1-ium-1-yl)acetyl]-2,5-dimethylpyrrol-1-yl]-1,5-dimethyl-2-phenylpyrazol-3-one —— C24H25N4O3+
4-[3-[2-(3-Hydroxypyridin-1-ium-1-yl)acetyl]-2,5-dimethylpyrrol-1-yl]-1,5-dimethyl-2-phenylpyrazol-3-one
—— N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]propanamide —— C21H28N4OS
N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]propanamide
—— (3R)-1-[7-oxo-6-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-propylpiperidine-3-carboxamide —— C24H24F3N7O3S
(3R)-1-[7-oxo-6-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-propylpiperidine-3-carboxamide
—— N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]propanamide —— C21H28N4OS
N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]propanamide
—— (2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propanamide —— C21H28N4OS
(2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propanamide
—— (2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propanamide —— C21H28N4OS
(2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propanamide
—— N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]acetamide —— C20H26N4OS
N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]acetamide
—— Cyclopropyl-[[3-(4-ethylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[(4-methoxyphenyl)methyl]azanium —— C22H26N3O2+
Cyclopropyl-[[3-(4-ethylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[(4-methoxyphenyl)methyl]azanium
—— N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]propanamide —— C21H28N4OS
N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]propanamide
—— (3S)-1-[7-oxo-6-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-propylpiperidine-3-carboxamide —— C24H24F3N7O3S
(3S)-1-[7-oxo-6-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-propylpiperidine-3-carboxamide
—— N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]acetamide —— C20H26N4OS
N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]acetamide
—— 1-[6-[[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-propan-2-ylpiperidine-4-carboxamide —— C27H33N7O3S
1-[6-[[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-propan-2-ylpiperidine-4-carboxamide
—— N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]acetamide —— C20H26N4OS
N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]acetamide
—— (3S)-1-[6-[[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-propylpiperidine-3-carboxamide —— C25H29N7O5S
(3S)-1-[6-[[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-propylpiperidine-3-carboxamide
—— 1-[6-[[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-propan-2-ylpiperidine-4-carboxamide —— C25H29N7O5S
1-[6-[[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-propan-2-ylpiperidine-4-carboxamide
—— (3S)-1-[6-[[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-propylpiperidine-3-carboxamide —— C27H33N7O3S
(3S)-1-[6-[[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-propylpiperidine-3-carboxamide
—— (3R)-1-[6-[[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-propylpiperidine-3-carboxamide —— C25H29N7O5S
(3R)-1-[6-[[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-propylpiperidine-3-carboxamide
—— (2R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propanamide —— C21H28N4OS
(2R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propanamide
—— 1-[7-oxo-6-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-propan-2-ylpiperidine-4-carboxamide —— C24H24F3N7O3S
1-[7-oxo-6-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-propan-2-ylpiperidine-4-carboxamide
—— N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]propanamide —— C21H28N4OS
N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]propanamide
—— (2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propanamide —— C21H28N4OS
(2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propanamide
—— 6-(4-Methylphenyl)-3-propyl-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methylsulfanyl]thieno[3,2-d]pyrimidin-4-one —— C26H21F3N4O2S2
6-(4-Methylphenyl)-3-propyl-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methylsulfanyl]thieno[3,2-d]pyrimidin-4-one
—— 6-[(4-Chlorophenyl)methylsulfanyl]-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-b]pyridazin-3-one —— C22H14ClF3N6O2S
6-[(4-Chlorophenyl)methylsulfanyl]-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-b]pyridazin-3-one
—— 2-[[3-(4-Tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-6-(4-methylphenyl)-3-propylthieno[3,2-d]pyrimidin-4-one —— C29H30N4O2S2
2-[[3-(4-Tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-6-(4-methylphenyl)-3-propylthieno[3,2-d]pyrimidin-4-one
—— (2R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(furan-2-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C24H28N4O2S
(2R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(furan-2-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— Methyl 2-[2,4-dioxo-1-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]quinazolin-3-yl]benzoate —— C26H17F3N4O5
Methyl 2-[2,4-dioxo-1-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]quinazolin-3-yl]benzoate
—— (2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(furan-2-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C24H28N4O2S
(2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(furan-2-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(furan-2-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C24H28N4O2S
(2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(furan-2-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— [(3R)-3-(chloromethyl)pyrrolidin-1-yl]-(1,3,5-trimethylpyrazol-4-yl)methanone —— C12H18ClN3O
[(3R)-3-(chloromethyl)pyrrolidin-1-yl]-(1,3,5-trimethylpyrazol-4-yl)methanone
—— 1-[(4-Methyl-2-morpholin-4-yl-1,3-thiazole-5-carbonyl)amino]-3-propylthiourea —— C13H21N5O2S2
1-[(4-Methyl-2-morpholin-4-yl-1,3-thiazole-5-carbonyl)amino]-3-propylthiourea
—— 1-(2-Methoxyethyl)-3-[(2-morpholin-4-yl-1,3-thiazole-4-carbonyl)amino]thiourea —— C12H19N5O3S2
1-(2-Methoxyethyl)-3-[(2-morpholin-4-yl-1,3-thiazole-4-carbonyl)amino]thiourea
—— [(3S)-3-(chloromethyl)pyrrolidin-1-yl]-(1,3,5-trimethylpyrazol-4-yl)methanone —— C12H18ClN3O
[(3S)-3-(chloromethyl)pyrrolidin-1-yl]-(1,3,5-trimethylpyrazol-4-yl)methanone
—— 1-[(1S,2R)-2-methylcyclohexyl]-3-[(4-methyl-2-morpholin-4-yl-1,3-thiazole-5-carbonyl)amino]thiourea —— C17H27N5O2S2
1-[(1S,2R)-2-methylcyclohexyl]-3-[(4-methyl-2-morpholin-4-yl-1,3-thiazole-5-carbonyl)amino]thiourea
—— 1-[(4-methyl-2-morpholin-4-yl-1,3-thiazole-5-carbonyl)amino]-3-[[(2S)-oxolan-2-yl]methyl]thiourea —— C15H23N5O3S2
1-[(4-methyl-2-morpholin-4-yl-1,3-thiazole-5-carbonyl)amino]-3-[[(2S)-oxolan-2-yl]methyl]thiourea
—— 1-[(4-Methoxyphenyl)methyl]-3-[(4-methyl-2-morpholin-4-yl-1,3-thiazole-5-carbonyl)amino]thiourea —— C18H23N5O3S2
1-[(4-Methoxyphenyl)methyl]-3-[(4-methyl-2-morpholin-4-yl-1,3-thiazole-5-carbonyl)amino]thiourea
—— 1-(Furan-2-ylmethyl)-3-[(4-methyl-2-morpholin-4-yl-1,3-thiazole-5-carbonyl)amino]thiourea —— C15H19N5O3S2
1-(Furan-2-ylmethyl)-3-[(4-methyl-2-morpholin-4-yl-1,3-thiazole-5-carbonyl)amino]thiourea
—— 1-Methyl-3-[(2-morpholin-4-yl-1,3-thiazole-4-carbonyl)amino]thiourea —— C10H15N5O2S2
1-Methyl-3-[(2-morpholin-4-yl-1,3-thiazole-4-carbonyl)amino]thiourea
—— 1-Cyclopropyl-3-[(4-methyl-2-morpholin-4-yl-1,3-thiazole-5-carbonyl)amino]thiourea —— C13H19N5O2S2
1-Cyclopropyl-3-[(4-methyl-2-morpholin-4-yl-1,3-thiazole-5-carbonyl)amino]thiourea
—— 1-[(1R,2S)-2-methylcyclohexyl]-3-[(4-methyl-2-morpholin-4-yl-1,3-thiazole-5-carbonyl)amino]thiourea —— C17H27N5O2S2
1-[(1R,2S)-2-methylcyclohexyl]-3-[(4-methyl-2-morpholin-4-yl-1,3-thiazole-5-carbonyl)amino]thiourea
—— [3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl-[(R)-(4-ethylphenyl)-thiophen-2-ylmethyl]azanium —— C22H21ClN3OS+
[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl-[(R)-(4-ethylphenyl)-thiophen-2-ylmethyl]azanium
—— 4-[(3R)-3-(chloromethyl)pyrrolidin-1-yl]sulfonyl-1-ethyl-2-methylimidazole —— C11H18ClN3O2S
4-[(3R)-3-(chloromethyl)pyrrolidin-1-yl]sulfonyl-1-ethyl-2-methylimidazole
—— 2-[5-[3-(Trifluoromethyl)phenyl]tetrazol-2-yl]acetonitrile —— C10H6F3N5
2-[5-[3-(Trifluoromethyl)phenyl]tetrazol-2-yl]acetonitrile
—— (1R)-1-(4-ethyl-5-methyl-1,3-thiazol-2-yl)-N-propan-2-ylheptan-1-amine —— C16H30N2S
(1R)-1-(4-ethyl-5-methyl-1,3-thiazol-2-yl)-N-propan-2-ylheptan-1-amine
—— N-cycloheptyl-2-[5-(thiophen-2-yl)-2H-tetrazol-2-yl]acetamide —— C14H19N5OS
N-cycloheptyl-2-[5-(thiophen-2-yl)-2H-tetrazol-2-yl]acetamide
—— 2-[(4-amino-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]acetamide —— C19H25N5OS
2-[(4-amino-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]acetamide
—— 4-[(3S)-3-(chloromethyl)pyrrolidin-1-yl]sulfonyl-1-ethyl-2-methylimidazole —— C11H18ClN3O2S
4-[(3S)-3-(chloromethyl)pyrrolidin-1-yl]sulfonyl-1-ethyl-2-methylimidazole
—— 2-[(4-amino-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]acetamide —— C19H25N5OS
2-[(4-amino-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]acetamide
—— 2-[(4-amino-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]acetamide —— C19H25N5OS
2-[(4-amino-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]acetamide