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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C29H29ClN4O4S2
2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H26ClN5O2S2
2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— N-[(2R)-butan-2-yl]-1-(3-fluorophenyl)-5-[2-(2-methoxyethylsulfamoyl)-4-nitrophenoxy]-4-methylpyrazole-3-carboxamide —— C24H28FN5O7S
N-[(2R)-butan-2-yl]-1-(3-fluorophenyl)-5-[2-(2-methoxyethylsulfamoyl)-4-nitrophenoxy]-4-methylpyrazole-3-carboxamide
—— 4-methyl-5-[4-[[(2R)-2-methylbutanoyl]amino]-2-(2-morpholin-4-ylethylsulfamoyl)phenoxy]-1-phenylpyrazole-3-carboxylic acid —— C28H35N5O7S
4-methyl-5-[4-[[(2R)-2-methylbutanoyl]amino]-2-(2-morpholin-4-ylethylsulfamoyl)phenoxy]-1-phenylpyrazole-3-carboxylic acid
—— (2R)-N-[(1R)-1-(4-fluorophenyl)ethyl]-2-[1-[[(2R)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylpropanamide —— C25H28FN3O2S
(2R)-N-[(1R)-1-(4-fluorophenyl)ethyl]-2-[1-[[(2R)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylpropanamide
—— 2-[(4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C31H31ClFN5O2S
2-[(4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— (2S)-N-[(1R)-1-(4-fluorophenyl)ethyl]-2-[1-[[(2R)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylpropanamide —— C25H28FN3O2S
(2S)-N-[(1R)-1-(4-fluorophenyl)ethyl]-2-[1-[[(2R)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylpropanamide
—— 2-[(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H26ClN5O2S2
2-[(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C29H30ClN5O2S2
2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 1-(3-fluorophenyl)-5-[2-(2-methoxyethylsulfamoyl)-4-nitrophenoxy]-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C25H28FN5O8S
1-(3-fluorophenyl)-5-[2-(2-methoxyethylsulfamoyl)-4-nitrophenoxy]-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 2-[(4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C31H31ClFN5O2S
2-[(4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 2-[(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C33H37N5O2S
2-[(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 4-[(Z)-[1-benzyl-3-(4-methylphenyl)pyrazol-4-yl]methylideneamino]-3-ethyl-1H-1,2,4-triazole-5-thione —— C22H22N6S
4-[(Z)-[1-benzyl-3-(4-methylphenyl)pyrazol-4-yl]methylideneamino]-3-ethyl-1H-1,2,4-triazole-5-thione
—— 1-(3-chlorophenyl)-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-3-methylthieno[2,3-c]pyrazole-5-carboxamide —— C17H14ClN5OS2
1-(3-chlorophenyl)-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-3-methylthieno[2,3-c]pyrazole-5-carboxamide
—— 2-[(4R)-3-(4-chlorophenyl)-4-(2-methylphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C34H30ClN5O2S
2-[(4R)-3-(4-chlorophenyl)-4-(2-methylphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— N-[(2S)-butan-2-yl]-1-(3-fluorophenyl)-5-[2-(2-methoxyethylsulfamoyl)-4-nitrophenoxy]-4-methylpyrazole-3-carboxamide —— C24H28FN5O7S
N-[(2S)-butan-2-yl]-1-(3-fluorophenyl)-5-[2-(2-methoxyethylsulfamoyl)-4-nitrophenoxy]-4-methylpyrazole-3-carboxamide
—— 2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C33H37N5O2S
2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 2-[(4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C33H27ClFN5O2S
2-[(4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 5-amino-3-[(E)-2-[5-bromo-2-[(2,4-dichlorophenyl)methoxy]phenyl]-1-cyanoethenyl]-1-phenylpyrazole-4-carbonitrile —— C26H16BrCl2N5O
5-amino-3-[(E)-2-[5-bromo-2-[(2,4-dichlorophenyl)methoxy]phenyl]-1-cyanoethenyl]-1-phenylpyrazole-4-carbonitrile
—— 2-[(4R)-3-(4-chlorophenyl)-4-(2-methylphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C32H34ClN5O2S
2-[(4R)-3-(4-chlorophenyl)-4-(2-methylphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[[5-[(4-methoxyphenoxy)methyl]-4-methyl-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C18H21N5O3S2
N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[[5-[(4-methoxyphenoxy)methyl]-4-methyl-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— (Z)-2-[[5-(5-chloro-2-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-3-(5-methylfuran-2-yl)prop-2-enoic acid —— C17H14ClN3O4S
(Z)-2-[[5-(5-chloro-2-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-3-(5-methylfuran-2-yl)prop-2-enoic acid
—— (1-propyltetrazol-5-yl)methyl (5S,7S)-3-chloroadamantane-1-carboxylate —— C16H23ClN4O2
(1-propyltetrazol-5-yl)methyl (5S,7S)-3-chloroadamantane-1-carboxylate
—— (1S,5S)-N-[4-(1,3-benzoxazol-2-yl)phenyl]-9-oxobicyclo[3.3.1]nonane-3-carboxamide —— C23H22N2O3
(1S,5S)-N-[4-(1,3-benzoxazol-2-yl)phenyl]-9-oxobicyclo[3.3.1]nonane-3-carboxamide
—— 1-(3,4-dihydro-2H-quinolin-1-yl)-2-[[4-ethyl-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethanone —— C22H24N4OS
1-(3,4-dihydro-2H-quinolin-1-yl)-2-[[4-ethyl-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethanone
—— 2-[(4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C33H27ClFN5O2S
2-[(4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 5-[4-(3,3-dimethylbutanoylamino)-2-(4-methylpiperazin-1-yl)sulfonylphenoxy]-4-methyl-1-phenylpyrazole-3-carboxylic acid —— C28H35N5O6S
5-[4-(3,3-dimethylbutanoylamino)-2-(4-methylpiperazin-1-yl)sulfonylphenoxy]-4-methyl-1-phenylpyrazole-3-carboxylic acid
—— 2-[(4S)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C32H34ClN5O3S
2-[(4S)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— (E)-2-[[5-(3,5-dimethoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-3-(5-methylfuran-2-yl)prop-2-enoate —— C18H16N3O5S-
(E)-2-[[5-(3,5-dimethoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-3-(5-methylfuran-2-yl)prop-2-enoate
—— (Z)-N,N-diethyl-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C11H16N2OS
(Z)-N,N-diethyl-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— 5-(2,4-dichlorophenyl)-3-[2-(4-methoxyphenoxy)ethylsulfanyl]-1H-1,2,4-triazole —— C17H15Cl2N3O2S
5-(2,4-dichlorophenyl)-3-[2-(4-methoxyphenoxy)ethylsulfanyl]-1H-1,2,4-triazole
—— (1-propyltetrazol-5-yl)methyl (5R,7R)-3-chloroadamantane-1-carboxylate —— C16H23ClN4O2
(1-propyltetrazol-5-yl)methyl (5R,7R)-3-chloroadamantane-1-carboxylate
—— (Z)-3-[2-(difluoromethylsulfonylamino)-1,3-thiazol-5-yl]prop-2-enoic acid —— C7H6F2N2O4S2
(Z)-3-[2-(difluoromethylsulfonylamino)-1,3-thiazol-5-yl]prop-2-enoic acid
—— N-[[4-(3-fluorophenyl)-5-propylsulfanyl-1,2,4-triazol-3-yl]methyl]adamantane-1-carboxamide —— C23H29FN4OS
N-[[4-(3-fluorophenyl)-5-propylsulfanyl-1,2,4-triazol-3-yl]methyl]adamantane-1-carboxamide
—— 2-[[3-(2,6-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-4-propan-2-yl-1H-pyrimidin-6-one —— C18H20N4O4S
2-[[3-(2,6-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-4-propan-2-yl-1H-pyrimidin-6-one
—— (3R)-5-[2-[[4-(2-methoxyphenyl)-5-piperidin-1-yl-1,2,4-triazol-3-yl]sulfanyl]acetyl]-3-methyl-1,3-dihydroindol-2-one —— C25H27N5O3S
(3R)-5-[2-[[4-(2-methoxyphenyl)-5-piperidin-1-yl-1,2,4-triazol-3-yl]sulfanyl]acetyl]-3-methyl-1,3-dihydroindol-2-one
—— (Z)-3-[2-(butylsulfonylamino)-1,3-thiazol-5-yl]prop-2-enoic acid —— C10H14N2O4S2
(Z)-3-[2-(butylsulfonylamino)-1,3-thiazol-5-yl]prop-2-enoic acid
—— N-[[4-(4-fluorophenyl)-5-propylsulfanyl-1,2,4-triazol-3-yl]methyl]adamantane-1-carboxamide —— C23H29FN4OS
N-[[4-(4-fluorophenyl)-5-propylsulfanyl-1,2,4-triazol-3-yl]methyl]adamantane-1-carboxamide
—— N-[[5-[(2R)-butan-2-yl]sulfanyl-4-(3-fluorophenyl)-1,2,4-triazol-3-yl]methyl]-4-methoxybenzamide —— C21H23FN4O2S
N-[[5-[(2R)-butan-2-yl]sulfanyl-4-(3-fluorophenyl)-1,2,4-triazol-3-yl]methyl]-4-methoxybenzamide
—— (Z)-3-phenyl-N-[2-(1-phenyltetrazol-5-yl)sulfanylethyl]prop-2-en-1-amine —— C18H19N5S
(Z)-3-phenyl-N-[2-(1-phenyltetrazol-5-yl)sulfanylethyl]prop-2-en-1-amine
—— 2-[(4-butyl-5-oxo-1H-1,2,4-triazol-3-yl)sulfanyl]-N-[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]acetamide —— C20H26N6O2S
2-[(4-butyl-5-oxo-1H-1,2,4-triazol-3-yl)sulfanyl]-N-[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]acetamide
—— (1R,5R)-N-[4-(1,3-benzoxazol-2-yl)phenyl]-9-oxobicyclo[3.3.1]nonane-3-carboxamide —— C23H22N2O3
(1R,5R)-N-[4-(1,3-benzoxazol-2-yl)phenyl]-9-oxobicyclo[3.3.1]nonane-3-carboxamide
—— N-benzyl-2-{[5-(2-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetamide —— C18H18N4OS
N-benzyl-2-{[5-(2-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetamide
—— 2-[(4S)-3-(4-chlorophenyl)-4-(2-methylphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C32H34ClN5O2S
2-[(4S)-3-(4-chlorophenyl)-4-(2-methylphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 2-[(4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C33H27ClFN5O2S
2-[(4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— (Z)-3-[2-(propylsulfonylamino)-1,3-thiazol-5-yl]prop-2-enoic acid —— C9H12N2O4S2
(Z)-3-[2-(propylsulfonylamino)-1,3-thiazol-5-yl]prop-2-enoic acid
—— N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-{[4-ethyl-5-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetamide —— C18H21N5O2S2
N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-{[4-ethyl-5-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetamide
—— N-(1-adamantyl)-2-[[4-ethyl-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C23H30N4OS
N-(1-adamantyl)-2-[[4-ethyl-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— 1-(3,4-dihydro-2H-quinolin-1-yl)-2-[[4-methyl-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethanone —— C21H22N4OS
1-(3,4-dihydro-2H-quinolin-1-yl)-2-[[4-methyl-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethanone
—— 3-(4-methoxyphenyl)-5-[(2-phenoxyethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazole —— C20H21N3O2S
3-(4-methoxyphenyl)-5-[(2-phenoxyethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazole