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中文名称 英文名称 CAS号 化学式 结构式图片
—— (4R)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H38N4O6S
(4R)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 5-[[3-(3-bromophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-N-methyl-1,3,4-thiadiazol-2-amine —— C12H10BrN5OS2
5-[[3-(3-bromophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-N-methyl-1,3,4-thiadiazol-2-amine
—— (4S)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H38N4O6S
(4S)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-(4-Tert-butylphenyl)-5-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propylsulfanyl]-1,3,4-oxadiazole —— C23H24N4O2S
2-(4-Tert-butylphenyl)-5-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propylsulfanyl]-1,3,4-oxadiazole
—— [5-(Furan-2-yl)-1,2-oxazol-3-yl]methyl 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate —— C18H11ClN2O4S
[5-(Furan-2-yl)-1,2-oxazol-3-yl]methyl 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate
—— 2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C30H29ClN4O4S2
2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C30H29ClN4O4S2
2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— (4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(2-chlorophenyl)-1-(2-methylphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H36ClN5O3S
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(2-chlorophenyl)-1-(2-methylphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-(cyclopropanecarbonylamino)phenoxy]-1-(4-chlorophenyl)-4-methylpyrazole-3-carboxylic acid —— C25H27ClN4O6S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-(cyclopropanecarbonylamino)phenoxy]-1-(4-chlorophenyl)-4-methylpyrazole-3-carboxylic acid
—— 1-(3-chlorophenyl)-4-methyl-5-[4-nitro-2-(propylsulfamoyl)phenoxy]-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C25H28ClN5O7S
1-(3-chlorophenyl)-4-methyl-5-[4-nitro-2-(propylsulfamoyl)phenoxy]-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 1-(4-methoxyphenyl)-4-methyl-5-(2-morpholin-4-ylsulfonyl-4-nitrophenoxy)-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C27H31N5O9S
1-(4-methoxyphenyl)-4-methyl-5-(2-morpholin-4-ylsulfonyl-4-nitrophenoxy)-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— (5-Phenyl-1,2-oxazol-3-yl)methyl 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate —— C20H13ClN2O3S
(5-Phenyl-1,2-oxazol-3-yl)methyl 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate
—— 2-[[3-(3,4-Dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-5,6-dimethyl-3-oxopyridazine-4-carbonitrile —— C18H17N5O4
2-[[3-(3,4-Dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-5,6-dimethyl-3-oxopyridazine-4-carbonitrile
—— 2-(morpholin-4-yl)-N'-(2-phenylethenesulfonyl)-1,3-thiazole-4-carbohydrazide —— C16H18N4O4S2
2-(morpholin-4-yl)-N'-(2-phenylethenesulfonyl)-1,3-thiazole-4-carbohydrazide
—— N-[(2S)-butan-2-yl]-1-(4-fluorophenyl)-4-methyl-5-[2-(2-methylpropylsulfamoyl)-4-nitrophenoxy]pyrazole-3-carboxamide —— C25H30FN5O6S
N-[(2S)-butan-2-yl]-1-(4-fluorophenyl)-4-methyl-5-[2-(2-methylpropylsulfamoyl)-4-nitrophenoxy]pyrazole-3-carboxamide
—— 5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-1-(2,5-dimethylphenyl)-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C27H31N5O7S
5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-1-(2,5-dimethylphenyl)-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-(3,3-dimethylbutanoylamino)phenoxy]-1-(4-fluorophenyl)-4-methylpyrazole-3-carboxylic acid —— C27H33FN4O6S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-(3,3-dimethylbutanoylamino)phenoxy]-1-(4-fluorophenyl)-4-methylpyrazole-3-carboxylic acid
—— N-[(2R)-butan-2-yl]-1-(4-fluorophenyl)-4-methyl-5-[2-(2-methylpropylsulfamoyl)-4-nitrophenoxy]pyrazole-3-carboxamide —— C25H30FN5O6S
N-[(2R)-butan-2-yl]-1-(4-fluorophenyl)-4-methyl-5-[2-(2-methylpropylsulfamoyl)-4-nitrophenoxy]pyrazole-3-carboxamide
—— (4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H31ClN4O2S2
(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-1-(2,3-dimethylphenyl)-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C27H31N5O7S
5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-1-(2,3-dimethylphenyl)-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 2-[(4S)-4-(2-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-phenylacetamide —— C33H27ClN4O2S
2-[(4S)-4-(2-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-phenylacetamide
—— N-(1,3-benzodioxol-5-ylmethyl)-4-[[5-(2-chlorophenyl)-4-[(2R)-1-methoxypropan-2-yl]-1,2,4-triazol-3-yl]sulfanylmethyl]benzamide —— C28H27ClN4O4S
N-(1,3-benzodioxol-5-ylmethyl)-4-[[5-(2-chlorophenyl)-4-[(2R)-1-methoxypropan-2-yl]-1,2,4-triazol-3-yl]sulfanylmethyl]benzamide
—— (4S)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C33H33FN4O3S
(4S)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 1-(3-fluoro-4-methylphenyl)-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]thiourea —— C18H18FN5S
1-(3-fluoro-4-methylphenyl)-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]thiourea
—— 1-[(4-fluorophenyl)methyl]-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]thiourea —— C18H18FN5S
1-[(4-fluorophenyl)methyl]-3-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]thiourea
—— 1-(4-methoxyphenyl)-4-methyl-5-(2-morpholin-4-ylsulfonyl-4-nitrophenoxy)-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C27H31N5O9S
1-(4-methoxyphenyl)-4-methyl-5-(2-morpholin-4-ylsulfonyl-4-nitrophenoxy)-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-(cyclopropanecarbonylamino)phenoxy]-1-(4-chlorophenyl)-4-methylpyrazole-3-carboxylic acid —— C25H27ClN4O6S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-(cyclopropanecarbonylamino)phenoxy]-1-(4-chlorophenyl)-4-methylpyrazole-3-carboxylic acid
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C30H29ClN4O4S2
2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C33H28N4O5S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 3-(3-fluoro-4-methylphenyl)-1-methyl-1-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]thiourea —— C19H20FN5S
3-(3-fluoro-4-methylphenyl)-1-methyl-1-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]thiourea
—— N-cyclopropyl-2-[2-(2,3-dimethylphenyl)-4-methyl-5-(pyrrolidine-1-carbonyl)pyrazol-3-yl]oxy-5-nitrobenzenesulfonamide —— C26H29N5O6S
N-cyclopropyl-2-[2-(2,3-dimethylphenyl)-4-methyl-5-(pyrrolidine-1-carbonyl)pyrazol-3-yl]oxy-5-nitrobenzenesulfonamide
—— (Z)-1-[(1R)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-en-1-one —— C15H17N3OS
(Z)-1-[(1R)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-en-1-one
—— (1R,2R)-1-chloro-N-[3-[5-(3,4-dichlorophenyl)-3-[2-(4-methoxyphenyl)ethoxy]-1,2,4-triazol-1-yl]phenyl]-2-fluorocyclopropane-1-carboxamide —— C27H22Cl3FN4O3
(1R,2R)-1-chloro-N-[3-[5-(3,4-dichlorophenyl)-3-[2-(4-methoxyphenyl)ethoxy]-1,2,4-triazol-1-yl]phenyl]-2-fluorocyclopropane-1-carboxamide
—— (Z)-1-[(1S)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-en-1-one —— C15H17N3OS
(Z)-1-[(1S)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-en-1-one
—— 2-[(4R)-4-(2-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-phenylacetamide —— C33H27ClN4O2S
2-[(4R)-4-(2-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-phenylacetamide
—— 3-[(2R)-2-ethylhexyl]-1-methyl-1-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]thiourea —— C20H31N5S
3-[(2R)-2-ethylhexyl]-1-methyl-1-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]thiourea
—— (Z)-N-methyl-3-(5-methylfuran-2-yl)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]prop-2-enamide —— C14H16N2O3
(Z)-N-methyl-3-(5-methylfuran-2-yl)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]prop-2-enamide
—— (4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(2-chlorophenyl)-1-(2-methylphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H36ClN5O3S
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(2-chlorophenyl)-1-(2-methylphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (7S)-3-[[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H20N4O3S
(7S)-3-[[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H31ClN4O2S2
(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 1-(4-fluorophenyl)-4-methyl-5-[2-(2-methylpropylsulfamoyl)-4-nitrophenoxy]-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C26H30FN5O7S
1-(4-fluorophenyl)-4-methyl-5-[2-(2-methylpropylsulfamoyl)-4-nitrophenoxy]-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— (1S,2S)-1-chloro-N-[3-[5-(3,4-dichlorophenyl)-3-[2-(4-methoxyphenyl)ethoxy]-1,2,4-triazol-1-yl]phenyl]-2-fluorocyclopropane-1-carboxamide —— C27H22Cl3FN4O3
(1S,2S)-1-chloro-N-[3-[5-(3,4-dichlorophenyl)-3-[2-(4-methoxyphenyl)ethoxy]-1,2,4-triazol-1-yl]phenyl]-2-fluorocyclopropane-1-carboxamide
—— 1-(3-chlorophenyl)-4-methyl-5-[4-nitro-2-(propylsulfamoyl)phenoxy]-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C25H28ClN5O7S
1-(3-chlorophenyl)-4-methyl-5-[4-nitro-2-(propylsulfamoyl)phenoxy]-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C33H28N4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— N-(1,3-benzodioxol-5-ylmethyl)-4-[[5-(2-chlorophenyl)-4-[(2S)-1-methoxypropan-2-yl]-1,2,4-triazol-3-yl]sulfanylmethyl]benzamide —— C28H27ClN4O4S
N-(1,3-benzodioxol-5-ylmethyl)-4-[[5-(2-chlorophenyl)-4-[(2S)-1-methoxypropan-2-yl]-1,2,4-triazol-3-yl]sulfanylmethyl]benzamide
—— (4R)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C33H33FN4O3S
(4R)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (1S,2R)-1-chloro-N-[3-[5-(3,4-dichlorophenyl)-3-[2-(4-methoxyphenyl)ethoxy]-1,2,4-triazol-1-yl]phenyl]-2-fluorocyclopropane-1-carboxamide —— C27H22Cl3FN4O3
(1S,2R)-1-chloro-N-[3-[5-(3,4-dichlorophenyl)-3-[2-(4-methoxyphenyl)ethoxy]-1,2,4-triazol-1-yl]phenyl]-2-fluorocyclopropane-1-carboxamide
—— [4-[[6-(1-benzothiophen-2-yl)-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1S,3S)-3-methoxycyclohexyl]methanone —— C34H35ClN4O2S
[4-[[6-(1-benzothiophen-2-yl)-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1S,3S)-3-methoxycyclohexyl]methanone
—— [4-[[6-(1-benzothiophen-2-yl)-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1R,3S)-3-methoxycyclohexyl]methanone —— C34H35ClN4O2S
[4-[[6-(1-benzothiophen-2-yl)-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1R,3S)-3-methoxycyclohexyl]methanone
—— (1R,2S)-1-chloro-N-[3-[5-(3,4-dichlorophenyl)-3-[2-(4-methoxyphenyl)ethoxy]-1,2,4-triazol-1-yl]phenyl]-2-fluorocyclopropane-1-carboxamide —— C27H22Cl3FN4O3
(1R,2S)-1-chloro-N-[3-[5-(3,4-dichlorophenyl)-3-[2-(4-methoxyphenyl)ethoxy]-1,2,4-triazol-1-yl]phenyl]-2-fluorocyclopropane-1-carboxamide