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中文名称 英文名称 CAS号 化学式 结构式图片
—— (1R,2S,4R)-N-[[2-(2-methylimidazol-1-yl)phenyl]methyl]bicyclo[2.2.1]heptane-2-carboxamide —— C19H23N3O
(1R,2S,4R)-N-[[2-(2-methylimidazol-1-yl)phenyl]methyl]bicyclo[2.2.1]heptane-2-carboxamide
—— (2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(4-fluorophenyl)-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C26H36FN5OS
(2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(4-fluorophenyl)-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (Z)-2-[[5-(4-chlorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-3-(5-nitrofuran-2-yl)prop-2-enoate —— C15H8ClN4O5S-
(Z)-2-[[5-(4-chlorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-3-(5-nitrofuran-2-yl)prop-2-enoate
—— (E)-2-[[5-(4-chlorophenyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-3-(5-methylfuran-2-yl)prop-2-enoate —— C18H15ClN3O3S-
(E)-2-[[5-(4-chlorophenyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-3-(5-methylfuran-2-yl)prop-2-enoate
—— (E)-2-[[5-(4-chlorophenyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-3-thiophen-2-ylprop-2-enoate —— C17H13ClN3O2S2-
(E)-2-[[5-(4-chlorophenyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-3-thiophen-2-ylprop-2-enoate
—— 2-[(5S,7S)-3-bromo-1-adamantyl]-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide —— C17H23BrN2O2
2-[(5S,7S)-3-bromo-1-adamantyl]-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
—— N-[[(5S,7S)-3-chloro-1-adamantyl]methyl]-2-(methoxymethyl)-1,3-thiazole-4-carboxamide —— C17H23ClN2O2S
N-[[(5S,7S)-3-chloro-1-adamantyl]methyl]-2-(methoxymethyl)-1,3-thiazole-4-carboxamide
—— (2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C20H25FN4OS
(2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C19H23FN4OS
N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— (2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-phenyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C26H37N5OS
(2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-phenyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 4-[5-[(E)-[6-oxo-2-(3,4,5-trimethoxyphenyl)-[1,3]thiazolo[3,2-b][1,2,4]triazol-5-ylidene]methyl]furan-2-yl]benzenesulfonamide —— C24H20N4O7S2
4-[5-[(E)-[6-oxo-2-(3,4,5-trimethoxyphenyl)-[1,3]thiazolo[3,2-b][1,2,4]triazol-5-ylidene]methyl]furan-2-yl]benzenesulfonamide
—— [2-(1-Benzofuran-2-yl)-2-oxoethyl] 4-methoxy-1-phenylpyrazole-3-carboxylate —— C21H16N2O5
[2-(1-Benzofuran-2-yl)-2-oxoethyl] 4-methoxy-1-phenylpyrazole-3-carboxylate
—— (2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(4-fluorophenyl)-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C26H36FN5OS
(2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(4-fluorophenyl)-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(4-fluorophenyl)-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C26H36FN5OS
(2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(4-fluorophenyl)-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C20H25FN4OS
(2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (5E)-5-[[3-(3-bromo-4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylidene]-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-1,3-thiazol-4-one —— C26H25BrN4O3S
(5E)-5-[[3-(3-bromo-4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylidene]-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-1,3-thiazol-4-one
—— (2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-phenyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C25H35N5OS
(2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-phenyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (4-Oxo-1,2,3-benzotriazin-3-yl)methyl 4-methoxy-1-phenylpyrazole-3-carboxylate —— C19H15N5O4
(4-Oxo-1,2,3-benzotriazin-3-yl)methyl 4-methoxy-1-phenylpyrazole-3-carboxylate
—— N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C19H23FN4OS
N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— (5E)-2-[(E)-2-(3,4-dimethoxyphenyl)ethenyl]-5-[[3-(3-fluoro-4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylidene]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one —— C31H24FN5O4S
(5E)-2-[(E)-2-(3,4-dimethoxyphenyl)ethenyl]-5-[[3-(3-fluoro-4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylidene]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one
—— (5E)-3-benzyl-5-[(3-methyl-1-phenyl-5-phenylsulfanylpyrazol-4-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C27H21N3OS3
(5E)-3-benzyl-5-[(3-methyl-1-phenyl-5-phenylsulfanylpyrazol-4-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-phenyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C26H37N5OS
(2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-phenyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— [2-[2-(4-Methoxyphenyl)ethylamino]-2-oxoethyl] 4-methoxy-1-phenylpyrazole-3-carboxylate —— C22H23N3O5
[2-[2-(4-Methoxyphenyl)ethylamino]-2-oxoethyl] 4-methoxy-1-phenylpyrazole-3-carboxylate
—— 1,4-dimethyl-5-phenyl-N-propylpyrazole-3-carboxamide —— C15H19N3O
1,4-dimethyl-5-phenyl-N-propylpyrazole-3-carboxamide
—— ethyl 2-[2-[(Z)-2-oxohex-4-enyl]-1,3-thiazol-4-yl]acetate —— C13H17NO3S
ethyl 2-[2-[(Z)-2-oxohex-4-enyl]-1,3-thiazol-4-yl]acetate
—— (5E)-5-[[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]methylidene]-2-[(E)-2-(3,4-dimethoxyphenyl)ethenyl]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one —— C32H25N5O5S
(5E)-5-[[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]methylidene]-2-[(E)-2-(3,4-dimethoxyphenyl)ethenyl]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one
—— (2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-phenyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C26H37N5OS
(2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-phenyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-phenyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C25H35N5OS
(2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-phenyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— [(2R)-1-(3-methylanilino)-1-oxopropan-2-yl] 4-methoxy-1-phenylpyrazole-3-carboxylate —— C21H21N3O4
[(2R)-1-(3-methylanilino)-1-oxopropan-2-yl] 4-methoxy-1-phenylpyrazole-3-carboxylate
—— [(2R)-1-(1-adamantylamino)-1-oxopropan-2-yl] 4-methoxy-1-phenylpyrazole-3-carboxylate —— C24H29N3O4
[(2R)-1-(1-adamantylamino)-1-oxopropan-2-yl] 4-methoxy-1-phenylpyrazole-3-carboxylate
—— [2-(2-Methyl-6-propan-2-ylanilino)-2-oxoethyl] 4-methoxy-1-phenylpyrazole-3-carboxylate —— C23H25N3O4
[2-(2-Methyl-6-propan-2-ylanilino)-2-oxoethyl] 4-methoxy-1-phenylpyrazole-3-carboxylate
—— [2-(2-Methoxy-5-methylanilino)-2-oxoethyl] 4-methoxy-1-phenylpyrazole-3-carboxylate —— C21H21N3O5
[2-(2-Methoxy-5-methylanilino)-2-oxoethyl] 4-methoxy-1-phenylpyrazole-3-carboxylate
—— (2R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-phenyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C25H35N5OS
(2R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-phenyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— N-[[(5R,7R)-3-chloro-1-adamantyl]methyl]-2-(methoxymethyl)-1,3-thiazole-4-carboxamide —— C17H23ClN2O2S
N-[[(5R,7R)-3-chloro-1-adamantyl]methyl]-2-(methoxymethyl)-1,3-thiazole-4-carboxamide
—— (2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C20H25FN4OS
(2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (5Z)-2-[(Z)-2-(3,4-dimethoxyphenyl)ethenyl]-5-[[3-(3-fluoro-4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylidene]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one —— C31H24FN5O4S
(5Z)-2-[(Z)-2-(3,4-dimethoxyphenyl)ethenyl]-5-[[3-(3-fluoro-4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylidene]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one
—— [2-[(2-Methoxybenzoyl)amino]-2-oxoethyl] 4-methoxy-1-phenylpyrazole-3-carboxylate —— C21H19N3O6
[2-[(2-Methoxybenzoyl)amino]-2-oxoethyl] 4-methoxy-1-phenylpyrazole-3-carboxylate
—— (5Z)-5-[[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]methylidene]-2-[(Z)-2-(3,4-dimethoxyphenyl)ethenyl]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one —— C32H25N5O5S
(5Z)-5-[[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]methylidene]-2-[(Z)-2-(3,4-dimethoxyphenyl)ethenyl]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one
—— ethyl (Z)-3-[7-methyl-2-(4-methylphenyl)imidazo[1,2-a]pyridin-3-yl]prop-2-enoate —— C20H20N2O2
ethyl (Z)-3-[7-methyl-2-(4-methylphenyl)imidazo[1,2-a]pyridin-3-yl]prop-2-enoate
—— N-[(4-methoxyphenyl)methyl]-N,1,4-trimethyl-5-phenylpyrazole-3-carboxamide —— C21H23N3O2
N-[(4-methoxyphenyl)methyl]-N,1,4-trimethyl-5-phenylpyrazole-3-carboxamide
—— (5Z)-3-[(2S)-butan-2-yl]-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C23H22N4OS2
(5Z)-3-[(2S)-butan-2-yl]-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (2R)-2-[[4-amino-5-(2-bromophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]propanamide —— C20H26BrN5OS
(2R)-2-[[4-amino-5-(2-bromophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]propanamide
—— (5Z)-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-3-[[(2R)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C24H22N4O2S2
(5Z)-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-3-[[(2R)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (1R,2S,3S,4R)-3-[(3-fluoro-4-imidazol-1-ylphenyl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C19H18FN3O3
(1R,2S,3S,4R)-3-[(3-fluoro-4-imidazol-1-ylphenyl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— (2R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C25H33FN4O2S
(2R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C19H23FN4OS
N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— (5Z)-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-3-[[(2S)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C24H22N4O2S2
(5Z)-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-3-[[(2S)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-3-octyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C27H30N4OS2
(5Z)-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-3-octyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-3-heptyl-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C26H28N4OS2
(5Z)-3-heptyl-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (Z)-2-cyano-3-[3-[3-(diethylsulfamoyl)phenyl]-1-phenylpyrazol-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide —— C28H31N5O4S
(Z)-2-cyano-3-[3-[3-(diethylsulfamoyl)phenyl]-1-phenylpyrazol-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide