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中文名称 英文名称 CAS号 化学式 结构式图片
—— [(2S)-4-cyano-4-(1,3-dihydrobenzimidazol-2-ylidene)-3-oxobutan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate —— C22H18N6O3
[(2S)-4-cyano-4-(1,3-dihydrobenzimidazol-2-ylidene)-3-oxobutan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate
—— (2-methyl-5-phenylpyrazol-3-yl)-[(5R)-5-(morpholin-4-ylmethyl)-1,4-thiazepan-4-yl]methanone —— C21H28N4O2S
(2-methyl-5-phenylpyrazol-3-yl)-[(5R)-5-(morpholin-4-ylmethyl)-1,4-thiazepan-4-yl]methanone
—— 2,4-dibromo-6-[[[1-[(E)-(2,4-dichlorophenyl)methylideneamino]-4-phenylimidazol-2-yl]amino]methylidene]cyclohexa-2,4-dien-1-one —— C23H14Br2Cl2N4O
2,4-dibromo-6-[[[1-[(E)-(2,4-dichlorophenyl)methylideneamino]-4-phenylimidazol-2-yl]amino]methylidene]cyclohexa-2,4-dien-1-one
—— N-[2-[[1-(3,4-dimethoxyphenyl)-4-phenylimidazol-2-yl]amino]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]furan-2-carboxamide —— C29H30N4O6
N-[2-[[1-(3,4-dimethoxyphenyl)-4-phenylimidazol-2-yl]amino]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]furan-2-carboxamide
—— [(2R)-1-(2-methylpropylamino)-1-oxopropan-2-yl] 1-benzyl-3-phenylpyrazole-4-carboxylate —— C24H27N3O3
[(2R)-1-(2-methylpropylamino)-1-oxopropan-2-yl] 1-benzyl-3-phenylpyrazole-4-carboxylate
—— 5-[2-[5-(4-fluorophenyl)tetrazol-2-yl]acetyl]-1-methyl-3H-indol-2-one —— C18H14FN5O2
5-[2-[5-(4-fluorophenyl)tetrazol-2-yl]acetyl]-1-methyl-3H-indol-2-one
—— N-[2-[[4-(4-chlorophenyl)-1-(3,4-dimethoxyphenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]furan-2-carboxamide —— C29H29ClN4O6
N-[2-[[4-(4-chlorophenyl)-1-(3,4-dimethoxyphenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]furan-2-carboxamide
—— N-[2-(dimethylamino)ethyl]-2-[(4S)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C31H32FN5O3S
N-[2-(dimethylamino)ethyl]-2-[(4S)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— (4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(2,5-dimethoxyphenyl)-1-methyl-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H33N5O5S
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(2,5-dimethoxyphenyl)-1-methyl-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— N-[2-(dimethylamino)ethyl]-2-[(4R)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C31H32FN5O3S
N-[2-(dimethylamino)ethyl]-2-[(4R)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H30ClN5O4S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— N-[2-[[1-(3,4-dimethoxyphenyl)-4-phenylimidazol-2-yl]amino]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]furan-2-carboxamide —— C29H30N4O6
N-[2-[[1-(3,4-dimethoxyphenyl)-4-phenylimidazol-2-yl]amino]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]furan-2-carboxamide
—— [(2R)-1-[(4-fluorophenyl)methylamino]-1-oxopropan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate —— C20H19FN4O3
[(2R)-1-[(4-fluorophenyl)methylamino]-1-oxopropan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate
—— 2-[(4R)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C33H28FN5O3S
2-[(4R)-1-(4-fluorophenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— (4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(2,5-dimethoxyphenyl)-1-methyl-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H33N5O5S
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(2,5-dimethoxyphenyl)-1-methyl-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— [(2R)-1-(methoxycarbonylamino)-1-oxopropan-2-yl] 2-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]acetate —— C16H15ClN2O5S
[(2R)-1-(methoxycarbonylamino)-1-oxopropan-2-yl] 2-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]acetate
—— 3-ethyl-1-[[2-[(4-fluorophenyl)methylsulfonyl]-3-[[(2R)-oxolan-2-yl]methyl]imidazol-4-yl]methyl]-1-(2-morpholin-4-ylethyl)urea —— C25H36FN5O5S
3-ethyl-1-[[2-[(4-fluorophenyl)methylsulfonyl]-3-[[(2R)-oxolan-2-yl]methyl]imidazol-4-yl]methyl]-1-(2-morpholin-4-ylethyl)urea
—— [4-[1-(4-fluorophenyl)-3-methyl-6-[(2R)-pentan-2-yl]pyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-1-yl]-[(1R,2R)-2-phenylcyclopropyl]methanone —— C32H37FN6O
[4-[1-(4-fluorophenyl)-3-methyl-6-[(2R)-pentan-2-yl]pyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-1-yl]-[(1R,2R)-2-phenylcyclopropyl]methanone
—— [4-[1-(4-fluorophenyl)-3-methyl-6-[(2S)-pentan-2-yl]pyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-1-yl]-[(1R,2R)-2-phenylcyclopropyl]methanone —— C32H37FN6O
[4-[1-(4-fluorophenyl)-3-methyl-6-[(2S)-pentan-2-yl]pyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-1-yl]-[(1R,2R)-2-phenylcyclopropyl]methanone
—— [(2S)-1-(methoxycarbonylamino)-1-oxopropan-2-yl] 2-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]acetate —— C16H15ClN2O5S
[(2S)-1-(methoxycarbonylamino)-1-oxopropan-2-yl] 2-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]acetate
—— (2S)-2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methylpropyl)propanamide —— C18H23FN4OS
(2S)-2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methylpropyl)propanamide
—— 3-cyclopropyl-1-[[2-[(4-fluorophenyl)methylsulfonyl]-3-[[(2S)-oxolan-2-yl]methyl]imidazol-4-yl]methyl]-1-(2-morpholin-4-ylethyl)thiourea —— C26H36FN5O4S2
3-cyclopropyl-1-[[2-[(4-fluorophenyl)methylsulfonyl]-3-[[(2S)-oxolan-2-yl]methyl]imidazol-4-yl]methyl]-1-(2-morpholin-4-ylethyl)thiourea
—— (2S)-2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(4-fluorophenyl)methyl]propanamide —— C19H20FN5OS
(2S)-2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(4-fluorophenyl)methyl]propanamide
—— [(2S)-1-(3-chloro-4-fluoroanilino)-1-oxopropan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate —— C19H16ClFN4O3
[(2S)-1-(3-chloro-4-fluoroanilino)-1-oxopropan-2-yl] 5-methyl-2-phenyltriazole-4-carboxylate
—— (2R)-2-[[4-amino-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,3-dihydro-1H-inden-5-yl)propanamide —— C21H23N5O2S
(2R)-2-[[4-amino-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,3-dihydro-1H-inden-5-yl)propanamide
—— (2R)-2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(thiophen-2-ylmethyl)propanamide —— C19H19FN4OS2
(2R)-2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(thiophen-2-ylmethyl)propanamide
—— (Z)-N-[(2R)-1-methoxypropan-2-yl]-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide —— C13H21N3O2
(Z)-N-[(2R)-1-methoxypropan-2-yl]-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide
—— (2S)-2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,5-dimethylphenyl)propanamide —— C22H23FN4OS
(2S)-2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,5-dimethylphenyl)propanamide
—— (2S)-N-cycloheptyl-2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C21H27FN4OS
(2S)-N-cycloheptyl-2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (Z)-N-[(2S)-1-methoxypropan-2-yl]-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide —— C13H21N3O2
(Z)-N-[(2S)-1-methoxypropan-2-yl]-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide
—— N-[1-(3-ethoxyphenyl)-4-phenylimidazol-2-yl]-2-[(4-methoxyphenyl)sulfonyl-[[(2R)-oxolan-2-yl]methyl]amino]acetamide —— C31H34N4O6S
N-[1-(3-ethoxyphenyl)-4-phenylimidazol-2-yl]-2-[(4-methoxyphenyl)sulfonyl-[[(2R)-oxolan-2-yl]methyl]amino]acetamide
—— (2R)-2-[[4-amino-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(4-fluorophenyl)methyl]propanamide —— C19H20FN5O2S
(2R)-2-[[4-amino-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(4-fluorophenyl)methyl]propanamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H30ClN5O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-ethyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C22H30N4OS
N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-ethyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— (2R)-2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(3-fluoro-4-methylphenyl)propanamide —— C19H20FN5OS
(2R)-2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(3-fluoro-4-methylphenyl)propanamide
—— 3-(4-methoxyphenyl)-5-[(1R)-1-(3-nitrophenyl)ethyl]sulfanyl-1,2,4-triazol-4-amine —— C17H17N5O3S
3-(4-methoxyphenyl)-5-[(1R)-1-(3-nitrophenyl)ethyl]sulfanyl-1,2,4-triazol-4-amine
—— N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-ethyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C22H30N4OS
N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-ethyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— (2R)-2-[[4-amino-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-chloropyridin-3-yl)propanamide —— C17H17ClN6O2S
(2R)-2-[[4-amino-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-chloropyridin-3-yl)propanamide
—— (2S)-2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methylpropyl)propanamide —— C16H23N5OS
(2S)-2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methylpropyl)propanamide
—— 2-[tert-butylcarbamoyl-[[(2R)-oxolan-2-yl]methyl]amino]-N-[4-(4-chlorophenyl)-1-(3-methoxyphenyl)imidazol-2-yl]acetamide —— C28H34ClN5O4
2-[tert-butylcarbamoyl-[[(2R)-oxolan-2-yl]methyl]amino]-N-[4-(4-chlorophenyl)-1-(3-methoxyphenyl)imidazol-2-yl]acetamide
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-N-(2-methoxyethyl)-4-methyl-1-phenylpyrazole-3-carboxamide —— C24H29N5O7S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-N-(2-methoxyethyl)-4-methyl-1-phenylpyrazole-3-carboxamide
—— 3-cyclopropyl-1-[[2-[(4-fluorophenyl)methylsulfonyl]-3-[[(2R)-oxolan-2-yl]methyl]imidazol-4-yl]methyl]-1-(2-morpholin-4-ylethyl)thiourea —— C26H36FN5O4S2
3-cyclopropyl-1-[[2-[(4-fluorophenyl)methylsulfonyl]-3-[[(2R)-oxolan-2-yl]methyl]imidazol-4-yl]methyl]-1-(2-morpholin-4-ylethyl)thiourea
—— N-[1-(3-ethoxyphenyl)-4-phenylimidazol-2-yl]-2-[(4-methoxyphenyl)sulfonyl-[[(2S)-oxolan-2-yl]methyl]amino]acetamide —— C31H34N4O6S
N-[1-(3-ethoxyphenyl)-4-phenylimidazol-2-yl]-2-[(4-methoxyphenyl)sulfonyl-[[(2S)-oxolan-2-yl]methyl]amino]acetamide
—— (2R)-2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2-chlorophenyl)methyl]propanamide —— C19H20ClN5OS
(2R)-2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2-chlorophenyl)methyl]propanamide
—— 3-ethyl-1-[[2-[(4-fluorophenyl)methylsulfonyl]-3-[[(2S)-oxolan-2-yl]methyl]imidazol-4-yl]methyl]-1-(2-morpholin-4-ylethyl)urea —— C25H36FN5O5S
3-ethyl-1-[[2-[(4-fluorophenyl)methylsulfonyl]-3-[[(2S)-oxolan-2-yl]methyl]imidazol-4-yl]methyl]-1-(2-morpholin-4-ylethyl)urea
—— N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-ethyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C22H30N4OS
N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-ethyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— (2S)-2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-propan-2-ylphenyl)propanamide —— C21H25N5OS
(2S)-2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-propan-2-ylphenyl)propanamide
—— (2R)-2-[[4-amino-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(3-fluorophenyl)propanamide —— C18H18FN5O2S
(2R)-2-[[4-amino-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(3-fluorophenyl)propanamide
—— (2R)-2-[[4-amino-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(4-ethoxyphenyl)propanamide —— C20H23N5O3S
(2R)-2-[[4-amino-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(4-ethoxyphenyl)propanamide
—— (Z)-N-(3-methylbutyl)-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide —— C14H23N3O
(Z)-N-(3-methylbutyl)-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide