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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(1S)-2-methyl-1-thiophen-2-ylpropyl]propanamide —— C19H20ClN3O2S
3-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(1S)-2-methyl-1-thiophen-2-ylpropyl]propanamide
—— [(1R,2S,5R)-5-methyl-2-propan-2-ylcyclohexyl] 2-[[4-(2,2-dimethoxyethyl)-5-[3-(dimethylsulfamoyl)phenyl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C26H40N4O6S2
[(1R,2S,5R)-5-methyl-2-propan-2-ylcyclohexyl] 2-[[4-(2,2-dimethoxyethyl)-5-[3-(dimethylsulfamoyl)phenyl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— [(1R,2S,5S)-5-methyl-2-propan-2-ylcyclohexyl] 2-[[4-(2,2-dimethoxyethyl)-5-[3-(dimethylsulfamoyl)phenyl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C26H40N4O6S2
[(1R,2S,5S)-5-methyl-2-propan-2-ylcyclohexyl] 2-[[4-(2,2-dimethoxyethyl)-5-[3-(dimethylsulfamoyl)phenyl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— 2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[2-(4-fluorophenyl)ethyl]acetamide —— C20H22FN5O2S
2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[2-(4-fluorophenyl)ethyl]acetamide
—— (1S,2S,3S,4S)-3-[[(1S)-1-(1-ethyl-3-methylpyrazol-4-yl)ethyl]carbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C17H23N3O3
(1S,2S,3S,4S)-3-[[(1S)-1-(1-ethyl-3-methylpyrazol-4-yl)ethyl]carbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— (1S,2S,3S,4R)-3-[(1,3,5-trimethylpyrazol-4-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C16H21N3O3
(1S,2S,3S,4R)-3-[(1,3,5-trimethylpyrazol-4-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— (2R)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-methyl-2-[1-(2-methylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C16H21N5O3S2
(2R)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-methyl-2-[1-(2-methylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— (1S,2S,3S,4S)-3-[(1,5-dimethylpyrazol-4-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C15H19N3O3
(1S,2S,3S,4S)-3-[(1,5-dimethylpyrazol-4-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— (2R)-N-(2-chlorophenyl)-2-[1-(2-methylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C17H16ClN5OS
(2R)-N-(2-chlorophenyl)-2-[1-(2-methylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— (3-Cyano-4-imino-2-oxopentyl) 2-phenyl-1,3-thiazole-4-carboxylate —— C16H13N3O3S
(3-Cyano-4-imino-2-oxopentyl) 2-phenyl-1,3-thiazole-4-carboxylate
—— (E)-3-(2-ethyl-1-benzofuran-3-yl)-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]prop-2-enamide —— C24H24N4O2
(E)-3-(2-ethyl-1-benzofuran-3-yl)-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]prop-2-enamide
—— (1S,2S,3S,4S)-3-[[(1R)-1-(1-ethyl-3-methylpyrazol-4-yl)ethyl]carbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C17H23N3O3
(1S,2S,3S,4S)-3-[[(1R)-1-(1-ethyl-3-methylpyrazol-4-yl)ethyl]carbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— (1S,2S,3R,4R)-3-(3-pyrazol-1-ylpropylcarbamoyl)bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C15H19N3O3
(1S,2S,3R,4R)-3-(3-pyrazol-1-ylpropylcarbamoyl)bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-3-phenyl-1H-pyrazole-5-carboxamide —— C19H26N4O
N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-3-phenyl-1H-pyrazole-5-carboxamide
—— Methyl 2-[(5-phenyl-1,3-oxazol-2-yl)methoxy]benzoate —— C18H15NO4
Methyl 2-[(5-phenyl-1,3-oxazol-2-yl)methoxy]benzoate
—— 2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide —— C32H33ClN4O3S
2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide
—— (4S)-3-(4-chlorophenyl)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C33H33ClN4O5S
(4S)-3-(4-chlorophenyl)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3,5-dimethyl-1-[(4-methylphenyl)methyl]pyrazole-4-carboxamide —— C22H26N4O2
N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3,5-dimethyl-1-[(4-methylphenyl)methyl]pyrazole-4-carboxamide
—— [(1S)-2-(3-chloro-4-methylanilino)-2-oxo-1-phenylethyl] 1-(4-chlorophenyl)-3-methylthieno[2,3-c]pyrazole-5-carboxylate —— C28H21Cl2N3O3S
[(1S)-2-(3-chloro-4-methylanilino)-2-oxo-1-phenylethyl] 1-(4-chlorophenyl)-3-methylthieno[2,3-c]pyrazole-5-carboxylate
—— (4R)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H28N4O3S2
(4R)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C30H38N4O4S
2-[(4R)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— 2-[[4-(2,4-dimethylphenyl)-5-(naphthalen-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(3S)-1,1-dioxothiolan-3-yl]-N-methylacetamide —— C28H30N4O3S2
2-[[4-(2,4-dimethylphenyl)-5-(naphthalen-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(3S)-1,1-dioxothiolan-3-yl]-N-methylacetamide
—— (1S,2S,3S,4S)-3-(3-pyrazol-1-ylpropylcarbamoyl)bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C15H19N3O3
(1S,2S,3S,4S)-3-(3-pyrazol-1-ylpropylcarbamoyl)bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— 2-[[5-(3-morpholin-4-ylsulfonylphenyl)-4-[(1R)-1-phenylethyl]-1,2,4-triazol-3-yl]sulfanyl]-1-pyrrolidin-1-ylethanone —— C26H31N5O4S2
2-[[5-(3-morpholin-4-ylsulfonylphenyl)-4-[(1R)-1-phenylethyl]-1,2,4-triazol-3-yl]sulfanyl]-1-pyrrolidin-1-ylethanone
—— 6-[(5-Cyclopropyl-1-phenyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3,5-triazine-2,4-diamine —— C15H16N8S
6-[(5-Cyclopropyl-1-phenyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3,5-triazine-2,4-diamine
—— (1S,2S,3S,4R)-3-[(1,5-dimethylpyrazol-4-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C15H19N3O3
(1S,2S,3S,4R)-3-[(1,5-dimethylpyrazol-4-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-1-phenylpyrazole-4-carboxamide —— C18H18N4O2
N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-1-phenylpyrazole-4-carboxamide
—— N-benzyl-2-[[4-(2,4-dimethylphenyl)-5-(naphthalen-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(3S)-1,1-dioxothiolan-3-yl]acetamide —— C34H34N4O3S2
N-benzyl-2-[[4-(2,4-dimethylphenyl)-5-(naphthalen-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(3S)-1,1-dioxothiolan-3-yl]acetamide
—— (Z)-N-[3-(tetrazol-1-yl)phenyl]-3-thiophen-2-ylprop-2-enamide —— C14H11N5OS
(Z)-N-[3-(tetrazol-1-yl)phenyl]-3-thiophen-2-ylprop-2-enamide
—— 2-[(4S)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C30H38N4O4S
2-[(4S)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— N-[(1R)-1-(1,3-benzothiazol-2-yl)ethyl]-N-methyl-3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide —— C22H22N4O2S
N-[(1R)-1-(1,3-benzothiazol-2-yl)ethyl]-N-methyl-3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
—— N-ethyl-2-[[5-(3-morpholin-4-ylsulfonylphenyl)-4-[(1R)-1-phenylethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-phenylacetamide —— C30H33N5O4S2
N-ethyl-2-[[5-(3-morpholin-4-ylsulfonylphenyl)-4-[(1R)-1-phenylethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-phenylacetamide
—— 2-[2-[(3S)-3-methyl-2,5-dioxopyrrolidin-1-yl]-1,3-thiazol-4-yl]acetic acid —— C10H10N2O4S
2-[2-[(3S)-3-methyl-2,5-dioxopyrrolidin-1-yl]-1,3-thiazol-4-yl]acetic acid
—— 4-(2-amino-2-oxoethoxy)-3-methoxy-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]benzamide —— C21H23N5O4
4-(2-amino-2-oxoethoxy)-3-methoxy-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]benzamide
—— N-methyl-3-(3-methyl-4-oxoquinazolin-2-yl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]propanamide —— C23H24N6O2
N-methyl-3-(3-methyl-4-oxoquinazolin-2-yl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]propanamide
—— N-[[4-(diethylsulfamoyl)phenyl]methyl]-3-phenyl-1H-pyrazole-5-carboxamide —— C21H24N4O3S
N-[[4-(diethylsulfamoyl)phenyl]methyl]-3-phenyl-1H-pyrazole-5-carboxamide
—— (1S,2S,3S,4R)-3-[(1-methylpyrazol-4-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C14H17N3O3
(1S,2S,3S,4R)-3-[(1-methylpyrazol-4-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— N-ethyl-2-[[5-(3-morpholin-4-ylsulfonylphenyl)-4-[(1S)-1-phenylethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-phenylacetamide —— C30H33N5O4S2
N-ethyl-2-[[5-(3-morpholin-4-ylsulfonylphenyl)-4-[(1S)-1-phenylethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-phenylacetamide
—— (4R)-3-(4-chlorophenyl)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C33H33ClN4O5S
(4R)-3-(4-chlorophenyl)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 1-benzyl-5-chloro-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-methylpyrazole-4-carboxamide —— C20H21ClN4O2
1-benzyl-5-chloro-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-methylpyrazole-4-carboxamide
—— 3-methyl-N'-[3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]propanoyl]-1-benzofuran-2-carbohydrazide —— C22H20N4O4
3-methyl-N'-[3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]propanoyl]-1-benzofuran-2-carbohydrazide
—— ethyl (3R)-1-[2-[6-[1-(2-ethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C29H33N5O4S
ethyl (3R)-1-[2-[6-[1-(2-ethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate
—— diethyl-[[4-[[(3-phenyl-1H-pyrazole-5-carbonyl)amino]methyl]phenyl]methyl]azanium —— C22H27N4O+
diethyl-[[4-[[(3-phenyl-1H-pyrazole-5-carbonyl)amino]methyl]phenyl]methyl]azanium
—— N-methyl-3-(3-methyl-4-oxoquinazolin-2-yl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]propanamide —— C23H24N6O2
N-methyl-3-(3-methyl-4-oxoquinazolin-2-yl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]propanamide
—— N-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl]-2-methyl-4-phenyl-1,3-thiazole-5-carboxamide —— C21H19ClN2O3S
N-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl]-2-methyl-4-phenyl-1,3-thiazole-5-carboxamide
—— (2S)-1-[[5-(4-fluorophenoxy)-1-methyl-3-phenylpyrazol-4-yl]methyl-(furan-2-ylmethyl)amino]-3-(furan-2-ylmethoxy)propan-2-ol —— C30H30FN3O5
(2S)-1-[[5-(4-fluorophenoxy)-1-methyl-3-phenylpyrazol-4-yl]methyl-(furan-2-ylmethyl)amino]-3-(furan-2-ylmethoxy)propan-2-ol
—— (2R)-N-[(2R)-2-phenylbutyl]-2-(1-phenyltetrazol-5-yl)sulfanylpropanamide —— C20H23N5OS
(2R)-N-[(2R)-2-phenylbutyl]-2-(1-phenyltetrazol-5-yl)sulfanylpropanamide
—— (1S,2S,3R,4S)-3-[(1,5-dimethylpyrazol-4-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C15H19N3O3
(1S,2S,3R,4S)-3-[(1,5-dimethylpyrazol-4-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylacetamide —— C22H26N4O2S
N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylacetamide
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C31H26ClN5O2S2
2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide