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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-[2-[2-[(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-2-oxoethyl]tetrazol-5-yl]benzamide —— C19H24N6O2
4-[2-[2-[(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-2-oxoethyl]tetrazol-5-yl]benzamide
—— 4-ethyl-5-(4-methoxyphenyl)-2-[[(2R)-2-thiophen-2-ylpyrrolidin-1-yl]methyl]-1,2,4-triazole-3-thione —— C20H24N4OS2
4-ethyl-5-(4-methoxyphenyl)-2-[[(2R)-2-thiophen-2-ylpyrrolidin-1-yl]methyl]-1,2,4-triazole-3-thione
—— 4-[2-[2-(Dibutylamino)-2-oxoethyl]tetrazol-5-yl]benzamide —— C18H26N6O2
4-[2-[2-(Dibutylamino)-2-oxoethyl]tetrazol-5-yl]benzamide
—— 4-[2-[2-[[(1R)-1-cyclopropylethyl]-(2,2,2-trifluoroethyl)amino]-2-oxoethyl]tetrazol-5-yl]benzamide —— C17H19F3N6O2
4-[2-[2-[[(1R)-1-cyclopropylethyl]-(2,2,2-trifluoroethyl)amino]-2-oxoethyl]tetrazol-5-yl]benzamide
—— (4Z,5R)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-(4-methylphenyl)-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione —— C28H30N4O4
(4Z,5R)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-(4-methylphenyl)-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione
—— 4-[2-[2-[[(1S)-1-(4-chlorophenyl)ethyl]amino]-2-oxoethyl]tetrazol-5-yl]benzamide —— C18H17ClN6O2
4-[2-[2-[[(1S)-1-(4-chlorophenyl)ethyl]amino]-2-oxoethyl]tetrazol-5-yl]benzamide
—— N-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]-2-ethyl-5-(2-methoxyphenyl)pyrazole-3-carboxamide —— C20H25N3O2
N-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]-2-ethyl-5-(2-methoxyphenyl)pyrazole-3-carboxamide
—— 5-methyl-4-(3-methylphenyl)-2-[[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]methyl]-1,2,4-triazole-3-thione —— C19H22N4S2
5-methyl-4-(3-methylphenyl)-2-[[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]methyl]-1,2,4-triazole-3-thione
—— 5-methyl-4-phenyl-2-[[(2R)-2-thiophen-2-ylpyrrolidin-1-ium-1-yl]methyl]-1,2,4-triazole-3-thione —— C18H21N4S2+
5-methyl-4-phenyl-2-[[(2R)-2-thiophen-2-ylpyrrolidin-1-ium-1-yl]methyl]-1,2,4-triazole-3-thione
—— 4-[2-[2-Oxo-2-(3-phenylsulfanylpropylamino)ethyl]tetrazol-5-yl]benzamide —— C19H20N6O2S
4-[2-[2-Oxo-2-(3-phenylsulfanylpropylamino)ethyl]tetrazol-5-yl]benzamide
—— 5-phenyl-4-prop-2-enyl-2-[[(2S)-2-thiophen-2-ylpyrrolidin-1-ium-1-yl]methyl]-1,2,4-triazole-3-thione —— C20H23N4S2+
5-phenyl-4-prop-2-enyl-2-[[(2S)-2-thiophen-2-ylpyrrolidin-1-ium-1-yl]methyl]-1,2,4-triazole-3-thione
—— 4-[2-[2-(5-Ethylthiophen-2-yl)-2-oxoethyl]tetrazol-5-yl]benzamide —— C16H15N5O2S
4-[2-[2-(5-Ethylthiophen-2-yl)-2-oxoethyl]tetrazol-5-yl]benzamide
—— 4-[2-[2-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-2-oxoethyl]tetrazol-5-yl]benzamide —— C19H24N6O2
4-[2-[2-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-2-oxoethyl]tetrazol-5-yl]benzamide
—— 5-(4-chlorophenyl)-4-methyl-2-[[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]methyl]-1,2,4-triazole-3-thione —— C18H19ClN4S2
5-(4-chlorophenyl)-4-methyl-2-[[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]methyl]-1,2,4-triazole-3-thione
—— 4-[2-[2-[2-(Difluoromethoxy)anilino]-2-oxoethyl]tetrazol-5-yl]benzamide —— C17H14F2N6O3
4-[2-[2-[2-(Difluoromethoxy)anilino]-2-oxoethyl]tetrazol-5-yl]benzamide
—— Methyl 2-[[5-(4-carbamoylphenyl)tetrazol-2-yl]methyl]-4-methylquinoline-3-carboxylate —— C21H18N6O3
Methyl 2-[[5-(4-carbamoylphenyl)tetrazol-2-yl]methyl]-4-methylquinoline-3-carboxylate
—— 1-(2,5-dimethylphenyl)-4-[[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]methyl]tetrazole-5-thione —— C18H21N5S2
1-(2,5-dimethylphenyl)-4-[[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]methyl]tetrazole-5-thione
—— 5-(4-methoxyphenyl)-4-prop-2-enyl-2-[[(2R)-2-thiophen-2-ylpyrrolidin-1-ium-1-yl]methyl]-1,2,4-triazole-3-thione —— C21H25N4OS2+
5-(4-methoxyphenyl)-4-prop-2-enyl-2-[[(2R)-2-thiophen-2-ylpyrrolidin-1-ium-1-yl]methyl]-1,2,4-triazole-3-thione
—— 4-ethyl-5-phenyl-2-[[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]methyl]-1,2,4-triazole-3-thione —— C19H22N4S2
4-ethyl-5-phenyl-2-[[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]methyl]-1,2,4-triazole-3-thione
—— 4-[2-[2-(5-Chloro-2-fluoroanilino)-2-oxoethyl]tetrazol-5-yl]benzamide —— C16H12ClFN6O2
4-[2-[2-(5-Chloro-2-fluoroanilino)-2-oxoethyl]tetrazol-5-yl]benzamide
—— 4-[2-[2-(2,4-Dichlorophenoxy)ethyl]tetrazol-5-yl]benzamide —— C16H13Cl2N5O2
4-[2-[2-(2,4-Dichlorophenoxy)ethyl]tetrazol-5-yl]benzamide
—— 4-[2-[2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-oxoethyl]tetrazol-5-yl]benzamide —— C19H17N5O4
4-[2-[2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-oxoethyl]tetrazol-5-yl]benzamide
—— (4Z,5S)-5-(3-chlorophenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione —— C27H27ClN4O4
(4Z,5S)-5-(3-chlorophenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione
—— (4Z,5R)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-(4-methylphenyl)pyrrolidine-2,3-dione —— C26H28N4O3
(4Z,5R)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-(4-methylphenyl)pyrrolidine-2,3-dione
—— 4-[2-[2-[1-(2-Methoxyethyl)-2,5-dimethylpyrrol-3-yl]-2-oxoethyl]tetrazol-5-yl]benzamide —— C19H22N6O3
4-[2-[2-[1-(2-Methoxyethyl)-2,5-dimethylpyrrol-3-yl]-2-oxoethyl]tetrazol-5-yl]benzamide
—— 4-[2-[(4-Methylsulfanylphenyl)methyl]tetrazol-5-yl]benzamide —— C16H15N5OS
4-[2-[(4-Methylsulfanylphenyl)methyl]tetrazol-5-yl]benzamide
—— 2-[(4-Hydroxypiperidin-1-ium-1-yl)methyl]-4-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-thione —— C18H21N4OS2+
2-[(4-Hydroxypiperidin-1-ium-1-yl)methyl]-4-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-thione
—— 4-[2-[2-[[(1R,2S)-2-methylcyclohexyl]amino]-2-oxoethyl]tetrazol-5-yl]benzamide —— C17H22N6O2
4-[2-[2-[[(1R,2S)-2-methylcyclohexyl]amino]-2-oxoethyl]tetrazol-5-yl]benzamide
—— (4S)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H28F2N4O4S
(4S)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[[(3S)-3-(1,3-benzothiazol-2-yl)piperidin-1-yl]methyl]-4-phenyl-1,2,4-triazole-3-thione —— C21H21N5S2
2-[[(3S)-3-(1,3-benzothiazol-2-yl)piperidin-1-yl]methyl]-4-phenyl-1,2,4-triazole-3-thione
—— [3-(4-Ethylphenyl)-1,2,4-oxadiazol-5-yl]methyl 3,5-difluorobenzoate —— C18H14F2N2O3
[3-(4-Ethylphenyl)-1,2,4-oxadiazol-5-yl]methyl 3,5-difluorobenzoate
—— 4-[2-[2-(Dimethylamino)-2-oxoethyl]tetrazol-5-yl]benzamide —— C12H14N6O2
4-[2-[2-(Dimethylamino)-2-oxoethyl]tetrazol-5-yl]benzamide
—— 4-[2-[2-[Cyclohexyl(ethyl)amino]-2-oxoethyl]tetrazol-5-yl]benzamide —— C18H24N6O2
4-[2-[2-[Cyclohexyl(ethyl)amino]-2-oxoethyl]tetrazol-5-yl]benzamide
—— Methyl 5-[[5-(4-carbamoylphenyl)tetrazol-2-yl]methyl]-2-methylfuran-3-carboxylate —— C16H15N5O4
Methyl 5-[[5-(4-carbamoylphenyl)tetrazol-2-yl]methyl]-2-methylfuran-3-carboxylate
—— 2-[(4S)-1-tert-butyl-4-(2,5-dimethoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C31H34N4O5S
2-[(4S)-1-tert-butyl-4-(2,5-dimethoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 4-[2-[2-(2-Bromoanilino)-2-oxoethyl]tetrazol-5-yl]benzamide —— C16H13BrN6O2
4-[2-[2-(2-Bromoanilino)-2-oxoethyl]tetrazol-5-yl]benzamide
—— (4Z,5S)-5-(4-bromophenyl)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]pyrrolidine-2,3-dione —— C25H25BrN4O3
(4Z,5S)-5-(4-bromophenyl)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]pyrrolidine-2,3-dione
—— 4-[2-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl]tetrazol-5-yl]benzamide —— C17H22N6O2
4-[2-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl]tetrazol-5-yl]benzamide
—— 5-(4-Chlorophenyl)-2-[(4-hydroxypiperidin-1-yl)methyl]-4-(3-methylphenyl)-1,2,4-triazole-3-thione —— C21H23ClN4OS
5-(4-Chlorophenyl)-2-[(4-hydroxypiperidin-1-yl)methyl]-4-(3-methylphenyl)-1,2,4-triazole-3-thione
—— 2-[(4-Hydroxypiperidin-1-yl)methyl]-5-(4-methylphenyl)-4-(2-propan-2-ylphenyl)-1,2,4-triazole-3-thione —— C24H30N4OS
2-[(4-Hydroxypiperidin-1-yl)methyl]-5-(4-methylphenyl)-4-(2-propan-2-ylphenyl)-1,2,4-triazole-3-thione
—— 2-[(4-Hydroxypiperidin-1-ium-1-yl)methyl]-5-[(2-methylphenoxy)methyl]-4-phenyl-1,2,4-triazole-3-thione —— C22H27N4O2S+
2-[(4-Hydroxypiperidin-1-ium-1-yl)methyl]-5-[(2-methylphenoxy)methyl]-4-phenyl-1,2,4-triazole-3-thione
—— 4-[2-[2-(2,4-Difluoroanilino)-2-oxoethyl]tetrazol-5-yl]benzamide —— C16H12F2N6O2
4-[2-[2-(2,4-Difluoroanilino)-2-oxoethyl]tetrazol-5-yl]benzamide
—— 5-(4-Chlorophenyl)-2-[(4-hydroxypiperidin-1-ium-1-yl)methyl]-4-phenyl-1,2,4-triazole-3-thione —— C20H22ClN4OS+
5-(4-Chlorophenyl)-2-[(4-hydroxypiperidin-1-ium-1-yl)methyl]-4-phenyl-1,2,4-triazole-3-thione
—— 2-[[(3S)-3-(1,3-benzothiazol-2-yl)piperidin-1-yl]methyl]-4-(2-methylphenyl)-1,2,4-triazole-3-thione —— C22H23N5S2
2-[[(3S)-3-(1,3-benzothiazol-2-yl)piperidin-1-yl]methyl]-4-(2-methylphenyl)-1,2,4-triazole-3-thione
—— methyl 2-[(4Z,5S)-4-[hydroxy-(4-propoxyphenyl)methylidene]-2,3-dioxo-5-thiophen-2-ylpyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C24H22N2O6S2
methyl 2-[(4Z,5S)-4-[hydroxy-(4-propoxyphenyl)methylidene]-2,3-dioxo-5-thiophen-2-ylpyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— 4-[2-[2-(2,6-Dichloroanilino)-2-oxoethyl]tetrazol-5-yl]benzamide —— C16H12Cl2N6O2
4-[2-[2-(2,6-Dichloroanilino)-2-oxoethyl]tetrazol-5-yl]benzamide
—— [5-(2-bromophenyl)-3-sulfanylidene-1H-1,2,4-triazol-2-yl]methyl-[(4-fluorophenyl)methyl]-methylazanium —— C17H17BrFN4S+
[5-(2-bromophenyl)-3-sulfanylidene-1H-1,2,4-triazol-2-yl]methyl-[(4-fluorophenyl)methyl]-methylazanium
—— 4-[2-[2-(2-Chloro-4-methylanilino)-2-oxoethyl]tetrazol-5-yl]benzamide —— C17H15ClN6O2
4-[2-[2-(2-Chloro-4-methylanilino)-2-oxoethyl]tetrazol-5-yl]benzamide
—— 4-[2-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]tetrazol-5-yl]benzamide —— C17H22N6O2
4-[2-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]tetrazol-5-yl]benzamide
—— [3-(2,4-Dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 3-(4-methoxyphenyl)propanoate —— C21H22N2O6
[3-(2,4-Dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 3-(4-methoxyphenyl)propanoate