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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(2S)-butan-2-yl]-2-[(4R)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C29H29ClN4O2S2
N-[(2S)-butan-2-yl]-2-[(4R)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-propylpyrazole-3-carboxamide —— C24H28FN5O6S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-propylpyrazole-3-carboxamide
—— 4-methyl-1-(4-methylphenyl)-5-(2-morpholin-4-ylsulfonyl-4-nitrophenoxy)-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C27H31N5O8S
4-methyl-1-(4-methylphenyl)-5-(2-morpholin-4-ylsulfonyl-4-nitrophenoxy)-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 4-methyl-5-(3-methyl-4-nitrophenoxy)-1-(4-methylphenyl)-N-[[3-(trifluoromethyl)phenyl]methyl]pyrazole-3-carboxamide —— C27H23F3N4O4
4-methyl-5-(3-methyl-4-nitrophenoxy)-1-(4-methylphenyl)-N-[[3-(trifluoromethyl)phenyl]methyl]pyrazole-3-carboxamide
—— 2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide —— C28H33ClN4O3S
2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide
—— 2-[(4R)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide —— C28H27ClN4O2S2
2-[(4R)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide
—— 2-[(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C30H34F2N4O3S
2-[(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-[(4S)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C32H36N4O5S
2-[(4S)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C30H34F2N4O3S
2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— N-(furan-2-ylmethyl)-4-methyl-5-[4-nitro-2-(propan-2-ylsulfamoyl)phenoxy]-1-phenylpyrazole-3-carboxamide —— C25H25N5O7S
N-(furan-2-ylmethyl)-4-methyl-5-[4-nitro-2-(propan-2-ylsulfamoyl)phenoxy]-1-phenylpyrazole-3-carboxamide
—— 2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C30H35ClN4O4S
2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— (4S)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(3-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H38N4O4S
(4S)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(3-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C30H34F2N4O3S
2-[(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 4-methyl-1-(4-methylphenyl)-5-[4-[[(3S)-oxolane-3-carbonyl]amino]-2-(2-pyridin-2-ylethylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid —— C30H31N5O7S
4-methyl-1-(4-methylphenyl)-5-[4-[[(3S)-oxolane-3-carbonyl]amino]-2-(2-pyridin-2-ylethylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid
—— N-[(2S)-butan-2-yl]-2-[2-(4-fluorophenyl)-4-methyl-5-(morpholine-4-carbonyl)pyrazol-3-yl]oxy-5-nitrobenzenesulfonamide —— C25H28FN5O7S
N-[(2S)-butan-2-yl]-2-[2-(4-fluorophenyl)-4-methyl-5-(morpholine-4-carbonyl)pyrazol-3-yl]oxy-5-nitrobenzenesulfonamide
—— (4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-fluorophenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C32H38FN5O3S
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-fluorophenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C26H30FN5O7S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— N-[(2R)-butan-2-yl]-1-(3-chlorophenyl)-5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-4-methylpyrazole-3-carboxamide —— C24H26ClN5O6S
N-[(2R)-butan-2-yl]-1-(3-chlorophenyl)-5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-4-methylpyrazole-3-carboxamide
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-N,4-dimethyl-N-propylpyrazole-3-carboxamide —— C25H30FN5O6S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-N,4-dimethyl-N-propylpyrazole-3-carboxamide
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C26H30FN5O7S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 2-[(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C30H30F2N4O3S
2-[(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 4-methyl-1-(4-methylphenyl)-5-(2-morpholin-4-ylsulfonyl-4-nitrophenoxy)-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C27H31N5O8S
4-methyl-1-(4-methylphenyl)-5-(2-morpholin-4-ylsulfonyl-4-nitrophenoxy)-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-N-cyclopropyl-1-(4-fluorophenyl)-4-methylpyrazole-3-carboxamide —— C24H26FN5O6S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-N-cyclopropyl-1-(4-fluorophenyl)-4-methylpyrazole-3-carboxamide
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-(pyridin-3-ylmethyl)pyrazole-3-carboxamide —— C27H27FN6O6S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-(pyridin-3-ylmethyl)pyrazole-3-carboxamide
—— (4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H33ClN4O3S
(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— N-[(2S)-butan-2-yl]-1-(3-chlorophenyl)-5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-4-methylpyrazole-3-carboxamide —— C24H26ClN5O6S
N-[(2S)-butan-2-yl]-1-(3-chlorophenyl)-5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-4-methylpyrazole-3-carboxamide
—— N-[(2S)-butan-2-yl]-5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxamide —— C25H30FN5O6S
N-[(2S)-butan-2-yl]-5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxamide
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C26H30FN5O7S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— N-[(2R)-butan-2-yl]-5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxamide —— C25H30FN5O6S
N-[(2R)-butan-2-yl]-5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxamide
—— 1-(3-chlorophenyl)-5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-4-methyl-N-propan-2-ylpyrazole-3-carboxamide —— C23H24ClN5O6S
1-(3-chlorophenyl)-5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-4-methyl-N-propan-2-ylpyrazole-3-carboxamide
—— 5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-1-(3-fluorophenyl)-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C26H30FN5O7S
5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-1-(3-fluorophenyl)-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C26H30FN5O7S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-(2-methylpropanoylamino)phenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxylic acid —— C25H29FN4O6S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-(2-methylpropanoylamino)phenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxylic acid
—— (4R)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(3-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H38N4O4S
(4R)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(3-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-(3-methylbutanoylamino)phenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxylic acid —— C26H31FN4O6S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-(3-methylbutanoylamino)phenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxylic acid
—— 5-[[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]sulfonyl]-2-chloro-4-methyl-1,3-thiazole —— C10H13ClN2O2S2
5-[[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]sulfonyl]-2-chloro-4-methyl-1,3-thiazole
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-(3-methylbutanoylamino)phenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxylic acid —— C26H31FN4O6S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-(3-methylbutanoylamino)phenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxylic acid
—— 1-(3-chlorophenyl)-5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C25H26ClN5O7S
1-(3-chlorophenyl)-5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 2-[(4S)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide —— C28H27ClN4O2S2
2-[(4S)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide
—— N-[1-(4-fluorophenyl)-4-phenylimidazol-2-yl]-2-[(4-methoxyphenyl)sulfonyl-[[(2R)-oxolan-2-yl]methyl]amino]acetamide —— C29H29FN4O5S
N-[1-(4-fluorophenyl)-4-phenylimidazol-2-yl]-2-[(4-methoxyphenyl)sulfonyl-[[(2R)-oxolan-2-yl]methyl]amino]acetamide
—— (4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(3-fluorophenyl)-1-(4-fluorophenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C30H33F2N5O3S
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(3-fluorophenyl)-1-(4-fluorophenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(3-fluorophenyl)-1-(4-fluorophenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C30H33F2N5O3S
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(3-fluorophenyl)-1-(4-fluorophenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (Z)-N-ethyl-N-(2-methylprop-2-enyl)-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C13H18N2OS
(Z)-N-ethyl-N-(2-methylprop-2-enyl)-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— 2-[(4S)-1,4-bis(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C33H34N4O3S
2-[(4S)-1,4-bis(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-[(4R)-4-(3-fluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide —— C31H31FN4O3S
2-[(4R)-4-(3-fluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide
—— 2-[(4S)-4-(3,4-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C33H29FN4O5S
2-[(4S)-4-(3,4-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 2-[(4R)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C33H37N5O5S
2-[(4R)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 2-[(4S)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C29H32F2N4O3S
2-[(4S)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2-chlorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C31H29ClN4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2-chlorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— 2-[(4S)-4-(3,4-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C33H33FN4O5S
2-[(4S)-4-(3,4-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide