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中文名称 英文名称 CAS号 化学式 结构式图片
—— (4S)-1-tert-butyl-4-(2,5-dimethoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C32H40N4O4S
(4S)-1-tert-butyl-4-(2,5-dimethoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-1-(4-fluorophenyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C28H32FN5O3S2
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-1-(4-fluorophenyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4Z,5R)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-(4-methoxyphenyl)pyrrolidine-2,3-dione —— C26H28N4O4
(4Z,5R)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-(4-methoxyphenyl)pyrrolidine-2,3-dione
—— 2-[5-(4-Fluorophenyl)tetrazol-2-yl]-1-(1-methylsulfonyl-2,3-dihydroindol-5-yl)ethanone —— C18H16FN5O3S
2-[5-(4-Fluorophenyl)tetrazol-2-yl]-1-(1-methylsulfonyl-2,3-dihydroindol-5-yl)ethanone
—— 5-(4-Chlorophenyl)-2-[[5-(furan-2-yl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-oxazole —— C17H13ClN4O2S
5-(4-Chlorophenyl)-2-[[5-(furan-2-yl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-oxazole
—— [3-(2-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 4-methylsulfonylbenzoate —— C18H16N2O6S
[3-(2-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 4-methylsulfonylbenzoate
—— (2S)-2-[[5-(4-chlorophenyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-ethylpropanamide —— C15H19ClN4OS
(2S)-2-[[5-(4-chlorophenyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-ethylpropanamide
—— [3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl (E)-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enoate —— C19H20N4O4
[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl (E)-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enoate
—— [3-(2,4-Dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 4,5,6,7-tetrahydro-1-benzothiophene-2-carboxylate —— C20H20N2O5S
[3-(2,4-Dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 4,5,6,7-tetrahydro-1-benzothiophene-2-carboxylate
—— [3-(2-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 4-(1,3-dithiolan-2-yl)benzoate —— C20H18N2O4S2
[3-(2-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 4-(1,3-dithiolan-2-yl)benzoate
—— 3-(4-Fluorophenyl)-5-[(2,5,6-trimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylmethyl]-1,2,4-oxadiazole —— C18H15FN4OS2
3-(4-Fluorophenyl)-5-[(2,5,6-trimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylmethyl]-1,2,4-oxadiazole
—— [3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl (E)-3-(2-chloroimidazo[1,2-a]pyridin-3-yl)prop-2-enoate —— C20H15ClN4O4
[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl (E)-3-(2-chloroimidazo[1,2-a]pyridin-3-yl)prop-2-enoate
—— 2-[[5-(4-chlorophenyl)-4-(2-propan-2-ylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R)-1-(3,4-dichlorophenyl)ethyl]acetamide —— C27H25Cl3N4OS
2-[[5-(4-chlorophenyl)-4-(2-propan-2-ylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R)-1-(3,4-dichlorophenyl)ethyl]acetamide
—— [2-Oxo-2-(thiophene-2-carbonylamino)ethyl] 5-methyl-2-phenyl-1,3-oxazole-4-carboxylate —— C18H14N2O5S
[2-Oxo-2-(thiophene-2-carbonylamino)ethyl] 5-methyl-2-phenyl-1,3-oxazole-4-carboxylate
—— [3-(2-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 5-methyl-2-phenyl-1,3-oxazole-4-carboxylate —— C21H17N3O5
[3-(2-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 5-methyl-2-phenyl-1,3-oxazole-4-carboxylate
—— (4S)-4-methyl-5-[2-[3-(tetrazol-1-yl)phenoxy]acetyl]-3,4-dihydro-1H-1,5-benzodiazepin-2-one —— C19H18N6O3
(4S)-4-methyl-5-[2-[3-(tetrazol-1-yl)phenoxy]acetyl]-3,4-dihydro-1H-1,5-benzodiazepin-2-one
—— [2-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methylamino]-2-oxoethyl] 5-methyl-2-phenyl-1,3-oxazole-4-carboxylate —— C22H20N2O6
[2-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methylamino]-2-oxoethyl] 5-methyl-2-phenyl-1,3-oxazole-4-carboxylate
—— (4S)-4-(2,5-dimethoxyphenyl)-1-(2,4-dimethylphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C36H40N4O4S
(4S)-4-(2,5-dimethoxyphenyl)-1-(2,4-dimethylphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 6-amino-5-[(2S)-2-[[5-(4-chlorophenyl)-4-(2-propan-2-ylphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]-1,3-dimethylpyrimidine-2,4-dione —— C26H27ClN6O3S
6-amino-5-[(2S)-2-[[5-(4-chlorophenyl)-4-(2-propan-2-ylphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]-1,3-dimethylpyrimidine-2,4-dione
—— (4S)-4-(2,5-dimethoxyphenyl)-1-(2,4-dimethylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C34H36N4O5S
(4S)-4-(2,5-dimethoxyphenyl)-1-(2,4-dimethylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C33H37N5O3S
2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— (4R)-4-(2,5-dimethoxyphenyl)-1-(2,4-dimethylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C34H36N4O5S
(4R)-4-(2,5-dimethoxyphenyl)-1-(2,4-dimethylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[[5-(4-chlorophenyl)-4-(2-propan-2-ylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-(3,4-dichlorophenyl)ethyl]acetamide —— C27H25Cl3N4OS
2-[[5-(4-chlorophenyl)-4-(2-propan-2-ylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-(3,4-dichlorophenyl)ethyl]acetamide
—— 2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C32H36N4O4S
2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 1-(4-fluorophenyl)-4-methyl-5-[4-[[(2S)-2-methylbutanoyl]amino]-2-(2-methylpropylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid —— C26H31FN4O6S
1-(4-fluorophenyl)-4-methyl-5-[4-[[(2S)-2-methylbutanoyl]amino]-2-(2-methylpropylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C30H29ClN4O5S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— (4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H32F2N4O3S
(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[[4-(3-chloro-4-methylphenyl)-5-(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(3R)-1,1-dioxothiolan-3-yl]-N-ethylacetamide —— C23H24Cl2N4O3S2
2-[[4-(3-chloro-4-methylphenyl)-5-(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(3R)-1,1-dioxothiolan-3-yl]-N-ethylacetamide
—— 2-[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]-5-[(5-phenyl-1,3-oxazol-2-yl)methylsulfanyl]-1,3,4-oxadiazole —— C20H15N3O4S
2-[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]-5-[(5-phenyl-1,3-oxazol-2-yl)methylsulfanyl]-1,3,4-oxadiazole
—— 2-[[4-(3-chloro-4-fluorophenyl)-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[2,5-dimethyl-1-[[(2R)-oxolan-2-yl]methyl]pyrrol-3-yl]ethanone —— C28H28ClFN4O3S
2-[[4-(3-chloro-4-fluorophenyl)-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[2,5-dimethyl-1-[[(2R)-oxolan-2-yl]methyl]pyrrol-3-yl]ethanone
—— (4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-1-(2-methylphenyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H35N5O3S2
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-1-(2-methylphenyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— [(1S,2R,5S)-5-methyl-2-propan-2-ylcyclohexyl] 2-[[4-(3-chloro-4-methylphenyl)-5-(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetate —— C27H31Cl2N3O2S
[(1S,2R,5S)-5-methyl-2-propan-2-ylcyclohexyl] 2-[[4-(3-chloro-4-methylphenyl)-5-(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetate
—— 2-[[4-(3-chloro-4-methylphenyl)-5-(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(3S)-1,1-dioxothiolan-3-yl]-N-ethylacetamide —— C23H24Cl2N4O3S2
2-[[4-(3-chloro-4-methylphenyl)-5-(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(3S)-1,1-dioxothiolan-3-yl]-N-ethylacetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C30H29ClN4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— (2S)-N-ethyl-2-[[4-(2-methoxyethyl)-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C17H24N4O2S
(2S)-N-ethyl-2-[[4-(2-methoxyethyl)-5-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (1R,2S,3S,4R)-3-(1H-pyrazol-4-ylmethylcarbamoyl)bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C13H15N3O3
(1R,2S,3S,4R)-3-(1H-pyrazol-4-ylmethylcarbamoyl)bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— [3-(2,4-Dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 4-(difluoromethoxy)benzoate —— C19H16F2N2O6
[3-(2,4-Dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 4-(difluoromethoxy)benzoate
—— [3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl (3S)-2,3-dihydro-1,4-benzodioxine-3-carboxylate —— C18H13ClN2O5
[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl (3S)-2,3-dihydro-1,4-benzodioxine-3-carboxylate
—— [(1S)-2-(dimethylamino)-2-oxo-1-phenylethyl] 2-(2,4-dimethylphenyl)-5-methyltriazole-4-carboxylate —— C22H24N4O3
[(1S)-2-(dimethylamino)-2-oxo-1-phenylethyl] 2-(2,4-dimethylphenyl)-5-methyltriazole-4-carboxylate
—— (2S)-N-ethyl-2-[[5-(4-methoxyphenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C19H26N4O3S
(2S)-N-ethyl-2-[[5-(4-methoxyphenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 2-[(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C33H37N5O3S
2-[(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— (1-Propyltetrazol-5-yl)methyl 2-(4-methylphenyl)-1,3-thiazole-4-carboxylate —— C16H17N5O2S
(1-Propyltetrazol-5-yl)methyl 2-(4-methylphenyl)-1,3-thiazole-4-carboxylate
—— [3-(2,4-Dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 1-benzofuran-2-carboxylate —— C20H16N2O6
[3-(2,4-Dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 1-benzofuran-2-carboxylate
—— N-[(1R)-1-phenylethyl]-2-[[4-phenyl-5-(3-pyrrolidin-1-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C28H29N5O3S2
N-[(1R)-1-phenylethyl]-2-[[4-phenyl-5-(3-pyrrolidin-1-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— 3-(3-chlorophenyl)-5-[[5-[(2-methylphenoxy)methyl]-1H-1,2,4-triazol-3-yl]sulfanylmethyl]-1,2,4-oxadiazole —— C19H16ClN5O2S
3-(3-chlorophenyl)-5-[[5-[(2-methylphenoxy)methyl]-1H-1,2,4-triazol-3-yl]sulfanylmethyl]-1,2,4-oxadiazole
—— 5-[[5-(4-Chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-3-(4-ethylphenyl)-1,2,4-oxadiazole —— C20H18ClN5OS
5-[[5-(4-Chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-3-(4-ethylphenyl)-1,2,4-oxadiazole
—— [(1R)-2-(cyclopropylamino)-2-oxo-1-phenylethyl] 2-(2,4-dimethylphenyl)-5-methyltriazole-4-carboxylate —— C23H24N4O3
[(1R)-2-(cyclopropylamino)-2-oxo-1-phenylethyl] 2-(2,4-dimethylphenyl)-5-methyltriazole-4-carboxylate
—— [3-(2-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl 4-(difluoromethoxy)benzoate —— C17H11ClF2N2O4
[3-(2-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl 4-(difluoromethoxy)benzoate
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C33H34N4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— (1R,2S,3R,4R)-3-(1H-pyrazol-4-ylmethylcarbamoyl)bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C13H15N3O3
(1R,2S,3R,4R)-3-(1H-pyrazol-4-ylmethylcarbamoyl)bicyclo[2.2.1]hept-5-ene-2-carboxylic acid