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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-(2,4-Dimethylphenyl)-2-[[methyl-[(2-methylphenyl)methyl]amino]methyl]-1,2,4-triazole-3-thione —— C20H24N4S
4-(2,4-Dimethylphenyl)-2-[[methyl-[(2-methylphenyl)methyl]amino]methyl]-1,2,4-triazole-3-thione
—— 4-Methyl-2-[[methyl-[(4-propan-2-ylphenyl)methyl]amino]methyl]-5-phenyl-1,2,4-triazole-3-thione —— C21H26N4S
4-Methyl-2-[[methyl-[(4-propan-2-ylphenyl)methyl]amino]methyl]-5-phenyl-1,2,4-triazole-3-thione
—— (4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-(2,3-dimethylphenyl)-4-(3-fluorophenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C34H34FN5O3S
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-(2,3-dimethylphenyl)-4-(3-fluorophenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 5-(5-chloro-2-methoxyphenyl)-2-[[(3-fluorophenyl)methyl-methylamino]methyl]-1H-1,2,4-triazole-3-thione —— C18H18ClFN4OS
5-(5-chloro-2-methoxyphenyl)-2-[[(3-fluorophenyl)methyl-methylamino]methyl]-1H-1,2,4-triazole-3-thione
—— (4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H27ClN4O3S2
(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H26ClN5O3S2
2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C31H26ClN5O2S2
2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]-1-phenylpyrazole-3-carboxamide —— C25H27N5O7S
5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]-1-phenylpyrazole-3-carboxamide
—— (4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H27ClN4O3S2
(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 5-(4-Chlorophenyl)-4-ethyl-2-[[(3-fluorophenyl)methyl-methylamino]methyl]-1,2,4-triazole-3-thione —— C19H20ClFN4S
5-(4-Chlorophenyl)-4-ethyl-2-[[(3-fluorophenyl)methyl-methylamino]methyl]-1,2,4-triazole-3-thione
—— (3-Fluorophenyl)methyl-methyl-[[3-methyl-4-(2-methylphenyl)-5-sulfanylidene-1,2,4-triazol-1-yl]methyl]azanium —— C19H22FN4S+
(3-Fluorophenyl)methyl-methyl-[[3-methyl-4-(2-methylphenyl)-5-sulfanylidene-1,2,4-triazol-1-yl]methyl]azanium
—— Methyl-[[3-methyl-4-(2-methylphenyl)-5-sulfanylidene-1,2,4-triazol-1-yl]methyl]-[(2-methylphenyl)methyl]azanium —— C20H25N4S+
Methyl-[[3-methyl-4-(2-methylphenyl)-5-sulfanylidene-1,2,4-triazol-1-yl]methyl]-[(2-methylphenyl)methyl]azanium
—— (3-Fluorophenyl)methyl-methyl-[[4-(2-methylphenyl)-5-sulfanylidene-1,2,4-triazol-1-yl]methyl]azanium —— C18H20FN4S+
(3-Fluorophenyl)methyl-methyl-[[4-(2-methylphenyl)-5-sulfanylidene-1,2,4-triazol-1-yl]methyl]azanium
—— 2-[[(2R)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-ium-1-yl]methyl]-4-methyl-5-phenyl-1,2,4-triazole-3-thione —— C21H22N5S2+
2-[[(2R)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-ium-1-yl]methyl]-4-methyl-5-phenyl-1,2,4-triazole-3-thione
—— [5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 4-methylbenzoate —— C18H14ClNO3
[5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 4-methylbenzoate
—— (4Z,5S)-1-[3-(dimethylamino)propyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dione —— C29H34N4O3
(4Z,5S)-1-[3-(dimethylamino)propyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dione
—— 2-[[(2S)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-ium-1-yl]methyl]-4-methyl-5-phenyl-1,2,4-triazole-3-thione —— C21H22N5S2+
2-[[(2S)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-ium-1-yl]methyl]-4-methyl-5-phenyl-1,2,4-triazole-3-thione
—— (3-Fluorophenyl)methyl-[[4-(2-methoxyethyl)-3-(3-methylphenyl)-5-sulfanylidene-1,2,4-triazol-1-yl]methyl]-methylazanium —— C21H26FN4OS+
(3-Fluorophenyl)methyl-[[4-(2-methoxyethyl)-3-(3-methylphenyl)-5-sulfanylidene-1,2,4-triazol-1-yl]methyl]-methylazanium
—— (4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H34ClN5O5S
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-(2,3-dimethylphenyl)-4-(3-fluorophenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C34H34FN5O3S
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-(2,3-dimethylphenyl)-4-(3-fluorophenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C28H27ClN4O3S2
2-[(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— 2-[(4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C30H28ClFN4O3S
2-[(4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C32H30F2N4O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— (4Z,5S)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-(4-methoxyphenyl)pyrrolidine-2,3-dione —— C26H28N4O4
(4Z,5S)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-(4-methoxyphenyl)pyrrolidine-2,3-dione
—— (4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H27ClN4O3S2
(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H26ClN5O2S2
2-[(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4R)-3-(4-chlorophenyl)-4-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C32H33ClN4O5S
2-[(4R)-3-(4-chlorophenyl)-4-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— [3-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-5-sulfanylidene-1,2,4-triazol-1-yl]methyl-methyl-[(2-methylphenyl)methyl]azanium —— C23H28FN4OS+
[3-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-5-sulfanylidene-1,2,4-triazol-1-yl]methyl-methyl-[(2-methylphenyl)methyl]azanium
—— 5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]-1-phenylpyrazole-3-carboxamide —— C25H27N5O7S
5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]-1-phenylpyrazole-3-carboxamide
—— 2-[(4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C30H28ClFN4O3S
2-[(4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— 2-[(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C31H26ClN5O2S2
2-[(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H26ClN5O3S2
2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— (4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H27ClN4O4S2
(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 4-Methyl-2-[[methyl-[(2-methylphenyl)methyl]amino]methyl]-5-(2-methylphenyl)-1,2,4-triazole-3-thione —— C20H24N4S
4-Methyl-2-[[methyl-[(2-methylphenyl)methyl]amino]methyl]-5-(2-methylphenyl)-1,2,4-triazole-3-thione
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C29H30ClN5O3S2
2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— (3-Fluorophenyl)methyl-[[4-(4-methoxyphenyl)-5-sulfanylidenetetrazol-1-yl]methyl]-methylazanium —— C17H19FN5OS+
(3-Fluorophenyl)methyl-[[4-(4-methoxyphenyl)-5-sulfanylidenetetrazol-1-yl]methyl]-methylazanium
—— 2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C29H30ClN5O3S2
2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 5-(2-Chlorophenyl)-2-[[(3-fluorophenyl)methyl-methylamino]methyl]-4-methyl-1,2,4-triazole-3-thione —— C18H18ClFN4S
5-(2-Chlorophenyl)-2-[[(3-fluorophenyl)methyl-methylamino]methyl]-4-methyl-1,2,4-triazole-3-thione
—— 5-(2-Chlorophenyl)-4-methyl-2-[[methyl-[(2-methylphenyl)methyl]amino]methyl]-1,2,4-triazole-3-thione —— C19H21ClN4S
5-(2-Chlorophenyl)-4-methyl-2-[[methyl-[(2-methylphenyl)methyl]amino]methyl]-1,2,4-triazole-3-thione
—— Methyl-[[4-methyl-3-(2-methylphenyl)-5-sulfanylidene-1,2,4-triazol-1-yl]methyl]-[(2-methylphenyl)methyl]azanium —— C20H25N4S+
Methyl-[[4-methyl-3-(2-methylphenyl)-5-sulfanylidene-1,2,4-triazol-1-yl]methyl]-[(2-methylphenyl)methyl]azanium
—— [3-(4-Fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl 3-(ethoxymethyl)-1-benzofuran-2-carboxylate —— C21H17FN2O5
[3-(4-Fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl 3-(ethoxymethyl)-1-benzofuran-2-carboxylate
—— 2-[[(2R)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-ium-1-yl]methyl]-4-ethyl-5-phenyl-1,2,4-triazole-3-thione —— C22H24N5S2+
2-[[(2R)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-ium-1-yl]methyl]-4-ethyl-5-phenyl-1,2,4-triazole-3-thione
—— (4R)-1-tert-butyl-4-(2,5-dimethoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C32H40N4O4S
(4R)-1-tert-butyl-4-(2,5-dimethoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[5-(2-bromophenyl)tetrazol-2-yl]-N-[(2-methoxyphenyl)methyl]-N-methylacetamide —— C18H18BrN5O2
2-[5-(2-bromophenyl)tetrazol-2-yl]-N-[(2-methoxyphenyl)methyl]-N-methylacetamide
—— N-(2-chlorophenyl)-2-[[4-(2,5-dimethylphenyl)-5-sulfanylidenetetrazol-1-yl]methyl-methylamino]acetamide —— C19H21ClN6OS
N-(2-chlorophenyl)-2-[[4-(2,5-dimethylphenyl)-5-sulfanylidenetetrazol-1-yl]methyl-methylamino]acetamide
—— [3-(4-Methoxyphenyl)-4-methyl-5-sulfanylidene-1,2,4-triazol-1-yl]methyl-methyl-[(4-propan-2-ylphenyl)methyl]azanium —— C22H29N4OS+
[3-(4-Methoxyphenyl)-4-methyl-5-sulfanylidene-1,2,4-triazol-1-yl]methyl-methyl-[(4-propan-2-ylphenyl)methyl]azanium
—— 5-(4-Chlorophenyl)-2-[[(3-fluorophenyl)methyl-methylamino]methyl]-4-methyl-1,2,4-triazole-3-thione —— C18H18ClFN4S
5-(4-Chlorophenyl)-2-[[(3-fluorophenyl)methyl-methylamino]methyl]-4-methyl-1,2,4-triazole-3-thione
—— (4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-1-(4-fluorophenyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C28H32FN5O3S2
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-1-(4-fluorophenyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-1-(2-methylphenyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H35N5O3S2
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-1-(2-methylphenyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H32F2N4O3S
(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one