中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
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2-[(4R)-4-(2,4-difluorophenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide |
—— |
C29H25F3N4O3S |
|
—— |
(4R)-3-tert-butyl-1-(2-chlorophenyl)-4-(3,4-dimethoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C30H35ClN4O5S |
|
—— |
2-[(4R)-4-(2,5-dimethoxyphenyl)-1-methyl-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide |
—— |
C30H29FN4O4S |
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—— |
2-[[4-amino-5-(2-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide |
—— |
C20H26ClN5OS |
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—— |
(5S)-3-[2-(dimethylamino)ethyl]-5-(3,5-dimethyl-1-phenylpyrazol-4-yl)-2-sulfanylideneimidazolidin-4-one |
—— |
C18H23N5OS |
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—— |
(5S)-5-(3,5-dimethyl-1-phenylpyrazol-4-yl)-3-[(2R)-1-methoxypropan-2-yl]-2-sulfanylideneimidazolidin-4-one |
—— |
C18H22N4O2S |
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—— |
(4S)-4-(4-fluorophenyl)-1-(2-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C29H27FN4O2S2 |
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—— |
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-methoxyphenyl)-4-methyl-N-propylpyrazole-3-carboxamide |
—— |
C25H31N5O7S |
|
—— |
2-[(4S)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C30H29FN4O3S2 |
|
—— |
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide |
—— |
C29H32N4O4S |
|
—— |
(4R)-4-(4-fluorophenyl)-1-(2-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C29H27FN4O2S2 |
|
—— |
N-cyclopropyl-2-[(4S)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C29H28N4O2S2 |
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—— |
2-[(4R)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide |
—— |
C29H29ClN4O2S2 |
|
—— |
(4R)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C29H26F2N4O3S2 |
|
—— |
N-cyclopropyl-2-[(4R)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C28H26N4O3S2 |
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—— |
2-[(4S)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C30H29FN4O3S2 |
|
—— |
N-cyclopropyl-2-[(4R)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C29H28N4O2S2 |
|
—— |
N-cyclopropyl-2-[(4R)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C28H25FN4O2S2 |
|
—— |
2-[(4R)-1-(2-chlorophenyl)-7-oxo-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide |
—— |
C27H23ClN4O2S2 |
|
—— |
2-[(4S)-3-tert-butyl-1-(3-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C29H28ClFN4O3S |
|
—— |
(4R)-4-(2-fluorophenyl)-1-(2-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C29H27FN4O2S2 |
|
—— |
2-[(4R)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C30H29FN4O3S2 |
|
—— |
N-[(2S)-butan-2-yl]-1-(4-methoxyphenyl)-4-methyl-5-[2-(2-methylpropylsulfamoyl)-4-nitrophenoxy]pyrazole-3-carboxamide |
—— |
C26H33N5O7S |
|
—— |
2-[(4R)-3-tert-butyl-1-(3-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C29H28ClFN4O3S |
|
—— |
2-[(4R)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C30H29FN4O3S2 |
|
—— |
N-[(2S)-butan-2-yl]-2-[(4S)-4-(4-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C29H29FN4O2S2 |
|
—— |
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-methoxyphenyl)-4-methyl-N-propylpyrazole-3-carboxamide |
—— |
C25H31N5O7S |
|
—— |
(4R)-4-(4-fluorophenyl)-1-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C29H27FN4O3S2 |
|
—— |
2-[(4R)-4-(3,4-dimethoxyphenyl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-phenylacetamide |
—— |
C35H32N4O4S |
|
—— |
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide |
—— |
C32H30N4O4S |
|
—— |
2-[(4S)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide |
—— |
C28H27FN4O3S2 |
|
—— |
N-[(2S)-butan-2-yl]-2-[(4R)-4-(4-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C29H29FN4O2S2 |
|
—— |
2-[(4S)-4-(2,4-difluorophenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide |
—— |
C29H25F3N4O3S |
|
—— |
2-[(4R)-4-(4-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide |
—— |
C29H29FN4O2S2 |
|
—— |
2-[(4S)-4-(4-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide |
—— |
C28H27FN4O3S2 |
|
—— |
2-[(4R)-4-(2,5-dimethoxyphenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C32H34N4O5S2 |
|
—— |
(4S)-4-(4-fluorophenyl)-1-(2-methylphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H31FN4O2S2 |
|
—— |
2-[(4S)-4-(2,5-dimethoxyphenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide |
—— |
C30H32N4O5S2 |
|
—— |
2-[(4R)-4-(2,5-dimethoxyphenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C32H34N4O5S2 |
|
—— |
N-cyclopropyl-2-[(4R)-4-(4-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C28H25FN4O2S2 |
|
—— |
2-[(4S)-4-(4-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide |
—— |
C29H29FN4O2S2 |
|
—— |
2-[(4R)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide |
—— |
C27H24Cl2N4O3S2 |
|
—— |
2-[(5R,7R)-3-bromo-1-adamantyl]-N-[[5-(2-methyl-1,3-thiazol-4-yl)furan-2-yl]methyl]acetamide |
—— |
C21H25BrN2O2S |
|
—— |
N-[(1R)-1-[5-benzylsulfanyl-4-(4-nitrophenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]-3,4-dichlorobenzamide |
—— |
C30H23Cl2N5O3S |
|
—— |
2-[(4S)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C30H28F2N4O3S2 |
|
—— |
2-[(4R)-4-(2,5-dimethoxyphenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide |
—— |
C30H32N4O5S2 |
|
—— |
(4S)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C29H26F2N4O3S2 |
|
—— |
N-[(2R)-butan-2-yl]-2-[(4R)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C29H29FN4O2S2 |
|
—— |
2-[(4S)-4-(4-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C30H29FN4O3S2 |
|
—— |
2-[(4S)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide |
—— |
C29H29ClN4O2S2 |
|