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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-methyl-2-[5-(2-methylphenyl)tetrazol-2-yl]acetamide —— C20H21N5O3
N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-methyl-2-[5-(2-methylphenyl)tetrazol-2-yl]acetamide
—— 2-[5-(2-chlorophenyl)tetrazol-2-yl]-N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-ethylacetamide —— C20H20ClN5O3
2-[5-(2-chlorophenyl)tetrazol-2-yl]-N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-ethylacetamide
—— 2-[5-(2-chlorophenyl)tetrazol-2-yl]-N-cyclopropyl-N-[(4-methoxyphenyl)methyl]acetamide —— C20H20ClN5O2
2-[5-(2-chlorophenyl)tetrazol-2-yl]-N-cyclopropyl-N-[(4-methoxyphenyl)methyl]acetamide
—— N'-[(1S,2R,4S)-bicyclo[2.2.1]heptane-2-carbonyl]-3-phenyl-1H-pyrazole-5-carbohydrazide —— C18H20N4O2
N'-[(1S,2R,4S)-bicyclo[2.2.1]heptane-2-carbonyl]-3-phenyl-1H-pyrazole-5-carbohydrazide
—— N'-[(1S,2S,4R)-bicyclo[2.2.1]heptane-2-carbonyl]-3-phenyl-1H-pyrazole-5-carbohydrazide —— C18H20N4O2
N'-[(1S,2S,4R)-bicyclo[2.2.1]heptane-2-carbonyl]-3-phenyl-1H-pyrazole-5-carbohydrazide
—— N-[2-(4-chlorophenoxy)ethyl]-2-[5-(2-chlorophenyl)tetrazol-2-yl]-N-methylacetamide —— C18H17Cl2N5O2
N-[2-(4-chlorophenoxy)ethyl]-2-[5-(2-chlorophenyl)tetrazol-2-yl]-N-methylacetamide
—— 2-[5-(2-chlorophenyl)tetrazol-2-yl]-N-[(2S)-6-methylheptan-2-yl]acetamide —— C17H24ClN5O
2-[5-(2-chlorophenyl)tetrazol-2-yl]-N-[(2S)-6-methylheptan-2-yl]acetamide
—— N'-[(1S,2S,4S)-bicyclo[2.2.1]heptane-2-carbonyl]-3-phenyl-1H-pyrazole-5-carbohydrazide —— C18H20N4O2
N'-[(1S,2S,4S)-bicyclo[2.2.1]heptane-2-carbonyl]-3-phenyl-1H-pyrazole-5-carbohydrazide
—— N-[(1R)-1-(1-benzofuran-2-yl)ethyl]-2-[5-(2-methylphenyl)tetrazol-2-yl]acetamide —— C20H19N5O2
N-[(1R)-1-(1-benzofuran-2-yl)ethyl]-2-[5-(2-methylphenyl)tetrazol-2-yl]acetamide
—— N-[(2R)-5-(diethylamino)pentan-2-yl]-2-[6-[1-(4-fluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetamide —— C28H35FN6O2S
N-[(2R)-5-(diethylamino)pentan-2-yl]-2-[6-[1-(4-fluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetamide
—— 2-[5-(2-chlorophenyl)tetrazol-2-yl]-N-[(2-methylphenyl)methyl]acetamide —— C17H16ClN5O
2-[5-(2-chlorophenyl)tetrazol-2-yl]-N-[(2-methylphenyl)methyl]acetamide
—— 1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-[5-(2-methylphenyl)tetrazol-2-yl]ethanone —— C19H18N4O3
1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-[5-(2-methylphenyl)tetrazol-2-yl]ethanone
—— 1-[(4aS,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-2-[5-(2-chlorophenyl)tetrazol-2-yl]ethanone —— C18H22ClN5O
1-[(4aS,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-2-[5-(2-chlorophenyl)tetrazol-2-yl]ethanone
—— 2-[5-(2-chlorophenyl)tetrazol-2-yl]-N-cyclopropyl-N-[(2-fluorophenyl)methyl]acetamide —— C19H17ClFN5O
2-[5-(2-chlorophenyl)tetrazol-2-yl]-N-cyclopropyl-N-[(2-fluorophenyl)methyl]acetamide
—— N-[(2S)-5-(diethylamino)pentan-2-yl]-2-[6-[1-(4-fluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetamide —— C28H35FN6O2S
N-[(2S)-5-(diethylamino)pentan-2-yl]-2-[6-[1-(4-fluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetamide
—— (Z)-N-[4-(5-methyl-1,3-benzoxazol-2-yl)phenyl]-3-(3-nitrophenyl)prop-2-en-1-imine —— C23H17N3O3
(Z)-N-[4-(5-methyl-1,3-benzoxazol-2-yl)phenyl]-3-(3-nitrophenyl)prop-2-en-1-imine
—— N-ethyl-N-(4-fluorophenyl)-2-(5-phenyltetrazol-2-yl)acetamide —— C17H16FN5O
N-ethyl-N-(4-fluorophenyl)-2-(5-phenyltetrazol-2-yl)acetamide
—— N-[4-(propan-2-ylsulfamoyl)phenyl]-4-(2H-tetrazol-5-yl)benzenecarboximidate —— C17H17N6O3S-
N-[4-(propan-2-ylsulfamoyl)phenyl]-4-(2H-tetrazol-5-yl)benzenecarboximidate
—— (4E)-3-methyl-4-[(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)hydrazinylidene]-6,7-dihydro-5H-1-benzofuran-2-carboxylic acid —— C21H18N6O3
(4E)-3-methyl-4-[(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)hydrazinylidene]-6,7-dihydro-5H-1-benzofuran-2-carboxylic acid
—— 5-[(Z)-2-phenylethenyl]-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazole —— C17H11F3N2O
5-[(Z)-2-phenylethenyl]-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazole
—— [2-(2-Methylbutan-2-ylamino)-2-oxoethyl] 2-(3-chlorophenyl)-4-methyl-1,3-thiazole-5-carboxylate —— C18H21ClN2O3S
[2-(2-Methylbutan-2-ylamino)-2-oxoethyl] 2-(3-chlorophenyl)-4-methyl-1,3-thiazole-5-carboxylate
—— 5-[2-(5-Ethylthiophen-2-yl)-2-oxoethyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one —— C19H16N4O2S
5-[2-(5-Ethylthiophen-2-yl)-2-oxoethyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one
—— (Z)-3-(4-bromo-3-nitrophenyl)-N-[2-(4-methylphenyl)-1,3-benzoxazol-5-yl]prop-2-en-1-imine —— C23H16BrN3O3
(Z)-3-(4-bromo-3-nitrophenyl)-N-[2-(4-methylphenyl)-1,3-benzoxazol-5-yl]prop-2-en-1-imine
—— [2-[(2-Methylphenyl)methylamino]-2-oxoethyl] 2-(3-chlorophenyl)-4-methyl-1,3-thiazole-5-carboxylate —— C21H19ClN2O3S
[2-[(2-Methylphenyl)methylamino]-2-oxoethyl] 2-(3-chlorophenyl)-4-methyl-1,3-thiazole-5-carboxylate
—— 2-[(4S)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C30H39N5O3S
2-[(4S)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 2-[(4S)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C32H35N5O3S
2-[(4S)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— (Z)-N-[2-(cyclohexen-1-yl)ethyl]-3-(1-methylpyrazol-4-yl)prop-2-enamide —— C15H21N3O
(Z)-N-[2-(cyclohexen-1-yl)ethyl]-3-(1-methylpyrazol-4-yl)prop-2-enamide
—— 2-[(4R)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C30H39N5O3S
2-[(4R)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C32H33N5O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— (Z)-3-(1-methylpyrazol-4-yl)-N-[(1S)-1-thiophen-2-ylethyl]prop-2-enamide —— C13H15N3OS
(Z)-3-(1-methylpyrazol-4-yl)-N-[(1S)-1-thiophen-2-ylethyl]prop-2-enamide
—— (Z)-N-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]-N-methyl-3-(1-methylpyrazol-4-yl)prop-2-enamide —— C20H23N5O
(Z)-N-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]-N-methyl-3-(1-methylpyrazol-4-yl)prop-2-enamide
—— (Z)-N-(furan-2-ylmethyl)-N-methyl-3-(1-methylpyrazol-4-yl)prop-2-enamide —— C13H15N3O2
(Z)-N-(furan-2-ylmethyl)-N-methyl-3-(1-methylpyrazol-4-yl)prop-2-enamide
—— (3S)-3-(4-decoxyphenyl)-5-[(Z)-2-(4-decoxyphenyl)ethenyl]-2-phenyl-3,4-dihydropyrazole —— C43H60N2O2
(3S)-3-(4-decoxyphenyl)-5-[(Z)-2-(4-decoxyphenyl)ethenyl]-2-phenyl-3,4-dihydropyrazole
—— [2-[(2-Methylphenyl)methylamino]-2-oxoethyl] 2-[2-(2-chlorophenyl)-1,3-thiazol-4-yl]acetate —— C21H19ClN2O3S
[2-[(2-Methylphenyl)methylamino]-2-oxoethyl] 2-[2-(2-chlorophenyl)-1,3-thiazol-4-yl]acetate
—— 2-[(4S)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C29H36FN5O3S
2-[(4S)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— (Z)-3-(1-methylpyrazol-4-yl)-N-(2-thiophen-2-ylethyl)prop-2-enamide —— C13H15N3OS
(Z)-3-(1-methylpyrazol-4-yl)-N-(2-thiophen-2-ylethyl)prop-2-enamide
—— (Z)-3-(1-methylpyrazol-4-yl)-N-[(1R)-1-thiophen-2-ylethyl]prop-2-enamide —— C13H15N3OS
(Z)-3-(1-methylpyrazol-4-yl)-N-[(1R)-1-thiophen-2-ylethyl]prop-2-enamide
—— 2-[(4R)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C32H35N5O3S
2-[(4R)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— (Z)-3-(4-bromo-3-nitrophenyl)-N-[2-(2,5-dichlorophenyl)-1,3-benzoxazol-5-yl]prop-2-en-1-imine —— C22H12BrCl2N3O3
(Z)-3-(4-bromo-3-nitrophenyl)-N-[2-(2,5-dichlorophenyl)-1,3-benzoxazol-5-yl]prop-2-en-1-imine
—— 2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C29H36FN5O3S
2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C33H35N5O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— (4R)-3-tert-butyl-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C30H36N4O5S
(4R)-3-tert-butyl-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-3-tert-butyl-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C30H39N5O4S
2-[(4R)-3-tert-butyl-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 2-[(4R)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C33H35FN4O3S
2-[(4R)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 2-[(4S)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C33H35FN4O3S
2-[(4S)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— (Z)-3-(4-bromo-3-nitrophenyl)-N-[2-(4-tert-butylphenyl)-1,3-benzoxazol-5-yl]prop-2-en-1-imine —— C26H22BrN3O3
(Z)-3-(4-bromo-3-nitrophenyl)-N-[2-(4-tert-butylphenyl)-1,3-benzoxazol-5-yl]prop-2-en-1-imine
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C31H30FN5O4S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— N-[2-[[1-(3-chlorophenyl)-4-(4-chlorophenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]thiophene-2-carboxamide —— C27H24Cl2N4O3S
N-[2-[[1-(3-chlorophenyl)-4-(4-chlorophenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]thiophene-2-carboxamide
—— (4R)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C30H36N4O4S
(4R)-3-tert-butyl-1-(4-methoxyphenyl)-4-(3-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4S)-3-tert-butyl-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C30H33N5O2S2
2-[(4S)-3-tert-butyl-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide