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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5E)-2-[(Z)-2-(3,4-dimethoxyphenyl)ethenyl]-5-[[3-(3-fluoro-4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylidene]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one —— C31H24FN5O4S
(5E)-2-[(Z)-2-(3,4-dimethoxyphenyl)ethenyl]-5-[[3-(3-fluoro-4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylidene]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one
—— (5Z)-3-benzyl-5-[(2,5-diphenyl-1,2,4-triazol-3-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C25H18N4OS2
(5Z)-3-benzyl-5-[(2,5-diphenyl-1,2,4-triazol-3-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetamide —— C20H27N5OS
N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetamide
—— [(2S)-1-(3-methoxyanilino)-1-oxopropan-2-yl] 4-methoxy-1-phenylpyrazole-3-carboxylate —— C21H21N3O5
[(2S)-1-(3-methoxyanilino)-1-oxopropan-2-yl] 4-methoxy-1-phenylpyrazole-3-carboxylate
—— (2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C21H27ClN4OS
(2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (1R,2S,3R,4R)-3-[[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C20H20FN3O3
(1R,2S,3R,4R)-3-[[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— (2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C21H27ClN4OS
(2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetamide —— C20H27N5OS
N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetamide
—— (Z)-2-cyano-N-(3,4-dimethylphenyl)-3-(8-methyl-2-phenylimidazo[1,2-a]pyridin-3-yl)prop-2-enamide —— C26H22N4O
(Z)-2-cyano-N-(3,4-dimethylphenyl)-3-(8-methyl-2-phenylimidazo[1,2-a]pyridin-3-yl)prop-2-enamide
—— 1-(5-Ethylthiophen-2-yl)-2-[1-(3-fluorophenyl)tetrazol-5-yl]sulfanylethanone —— C15H13FN4OS2
1-(5-Ethylthiophen-2-yl)-2-[1-(3-fluorophenyl)tetrazol-5-yl]sulfanylethanone
—— (5Z)-3-methyl-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C20H16N4OS2
(5Z)-3-methyl-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— methyl (Z)-3-[5-(4-chlorophenyl)-2-phenyl-1,2,4-triazol-3-yl]-2-cyanoprop-2-enoate —— C19H13ClN4O2
methyl (Z)-3-[5-(4-chlorophenyl)-2-phenyl-1,2,4-triazol-3-yl]-2-cyanoprop-2-enoate
—— (2S)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C21H29N5OS
(2S)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— (2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C21H29N5OS
(2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— (2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)sulfanylpropanamide —— C23H27N5OS
(2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)sulfanylpropanamide
—— 2-(4-chlorophenoxy)-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-methylpropanamide —— C21H22ClN3O3
2-(4-chlorophenoxy)-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-methylpropanamide
—— (2R)-2-[[4-amino-5-(2-bromophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]propanamide —— C20H26BrN5OS
(2R)-2-[[4-amino-5-(2-bromophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]propanamide
—— (1R,2S,3R,4R)-3-[(3-fluoro-4-imidazol-1-ylphenyl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C19H18FN3O3
(1R,2S,3R,4R)-3-[(3-fluoro-4-imidazol-1-ylphenyl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— (2R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C20H25FN4OS
(2R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (Z)-2-cyano-3-[3-[3-(diethylsulfamoyl)phenyl]-1-phenylpyrazol-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide —— C28H31N5O4S
(Z)-2-cyano-3-[3-[3-(diethylsulfamoyl)phenyl]-1-phenylpyrazol-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide
—— 3-[(3aS,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)propanamide —— C22H24N4O4
3-[(3aS,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)propanamide
—— methyl (Z)-2-cyano-3-[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]prop-2-enoate —— C20H16N4O2
methyl (Z)-2-cyano-3-[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]prop-2-enoate
—— (2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C21H29N5OS
(2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C19H23FN4OS
N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— (5Z)-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-3-propan-2-yl-2-sulfanylidene-1,3-thiazolidin-4-one —— C22H20N4OS2
(5Z)-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-3-propan-2-yl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-3-(2-methoxyethyl)-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C22H20N4O2S2
(5Z)-3-(2-methoxyethyl)-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (4E)-4-[(2,4-dichlorophenyl)methylidene]-5-oxo-1-phenylpyrazole-3-carboxylic acid —— C17H10Cl2N2O3
(4E)-4-[(2,4-dichlorophenyl)methylidene]-5-oxo-1-phenylpyrazole-3-carboxylic acid
—— (2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-phenyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C25H35N5OS
(2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-phenyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C25H33FN4O2S
(2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetamide —— C20H27N5OS
N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetamide
—— (2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C25H33FN4O2S
(2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-fluorophenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (5Z)-5-[[5-(4-chlorophenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-3-methyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C19H13ClN4OS2
(5Z)-5-[[5-(4-chlorophenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-3-methyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (2R)-2-[[4-amino-5-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]propanamide —— C21H29N5O2S
(2R)-2-[[4-amino-5-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]propanamide
—— (2R)-2-[[4-amino-5-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]propanamide —— C21H29N5O2S
(2R)-2-[[4-amino-5-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]propanamide
—— (5Z)-3-[(2R)-butan-2-yl]-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C23H22N4OS2
(5Z)-3-[(2R)-butan-2-yl]-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetamide —— C20H27N5OS
N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetamide
—— (2S)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C21H29N5OS
(2S)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— (2R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)sulfanylpropanamide —— C23H27N5OS
(2R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)sulfanylpropanamide
—— (2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)sulfanylpropanamide —— C23H27N5OS
(2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)sulfanylpropanamide
—— (2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)sulfanylpropanamide —— C23H27N5OS
(2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)sulfanylpropanamide
—— 2-[(5S,7S)-3-bromo-1-adamantyl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)acetamide —— C17H23BrN2OS
2-[(5S,7S)-3-bromo-1-adamantyl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)acetamide
—— N-[[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]methyl]-2-[4-(tetrazol-1-yl)phenyl]acetamide —— C17H21N5O
N-[[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]methyl]-2-[4-(tetrazol-1-yl)phenyl]acetamide
—— (2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C23H29FN4OS
(2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— N-[[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]methyl]-2-[4-(tetrazol-1-yl)phenyl]acetamide —— C17H21N5O
N-[[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]methyl]-2-[4-(tetrazol-1-yl)phenyl]acetamide
—— (2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[(4-ethyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propanamide —— C22H30N4OS
(2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[(4-ethyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propanamide
—— 2-[(5R,7R)-3-bromo-1-adamantyl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)acetamide —— C17H23BrN2OS
2-[(5R,7R)-3-bromo-1-adamantyl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)acetamide
—— 5-[[1-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-4,5-dimethylimidazol-2-yl]sulfonylmethyl]-3-(4-methoxyphenyl)-1,2,4-oxadiazole —— C24H30N4O4S
5-[[1-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-4,5-dimethylimidazol-2-yl]sulfonylmethyl]-3-(4-methoxyphenyl)-1,2,4-oxadiazole
—— 5-[[1-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-4,5-dimethylimidazol-2-yl]sulfonylmethyl]-3-(4-methoxyphenyl)-1,2,4-oxadiazole —— C24H30N4O4S
5-[[1-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-4,5-dimethylimidazol-2-yl]sulfonylmethyl]-3-(4-methoxyphenyl)-1,2,4-oxadiazole
—— (2R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C23H29FN4OS
(2R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 5-[[1-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-4,5-dimethylimidazol-2-yl]sulfonylmethyl]-3-(4-methoxyphenyl)-1,2,4-oxadiazole —— C24H30N4O4S
5-[[1-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-4,5-dimethylimidazol-2-yl]sulfonylmethyl]-3-(4-methoxyphenyl)-1,2,4-oxadiazole