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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(4R)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C30H23ClFN5O2S2
2-[(4R)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— [2-[[(2S)-butan-2-yl]-[(3S)-1,1-dioxothiolan-3-yl]amino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate —— C19H24N4O5S
[2-[[(2S)-butan-2-yl]-[(3S)-1,1-dioxothiolan-3-yl]amino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate
—— 5-methoxy-3-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-1-benzofuran-2-carboxamide —— C21H20N4O3
5-methoxy-3-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-1-benzofuran-2-carboxamide
—— 2-[(4R)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H25F2N5O2S2
2-[(4R)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— [2-[[(1S)-1-(4-ethylphenyl)ethyl]amino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate —— C21H22N4O3
[2-[[(1S)-1-(4-ethylphenyl)ethyl]amino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate
—— N'-[2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]-3-phenyl-1H-pyrazole-5-carbohydrazide —— C19H22N4O2
N'-[2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]-3-phenyl-1H-pyrazole-5-carbohydrazide
—— N-[(1S)-1-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[5-(3,4-dimethoxyphenyl)tetrazol-2-yl]acetamide —— C20H27N5O3
N-[(1S)-1-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[5-(3,4-dimethoxyphenyl)tetrazol-2-yl]acetamide
—— N-[(1S)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[5-(3,4-dimethoxyphenyl)tetrazol-2-yl]acetamide —— C20H27N5O3
N-[(1S)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[5-(3,4-dimethoxyphenyl)tetrazol-2-yl]acetamide
—— [(2S)-1-[2-[(2R)-butan-2-yl]anilino]-1-oxopropan-2-yl] 4-(1,2,4-triazol-1-yl)benzoate —— C22H24N4O3
[(2S)-1-[2-[(2R)-butan-2-yl]anilino]-1-oxopropan-2-yl] 4-(1,2,4-triazol-1-yl)benzoate
—— (2R)-N-[(E)-(3-bromophenyl)methylideneamino]-2-[[5-[(naphthalen-1-ylamino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C29H25BrN6OS
(2R)-N-[(E)-(3-bromophenyl)methylideneamino]-2-[[5-[(naphthalen-1-ylamino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— [(1S)-2-(4-methylanilino)-2-oxo-1-phenylethyl] 4-(1,2,4-triazol-1-yl)benzoate —— C24H20N4O3
[(1S)-2-(4-methylanilino)-2-oxo-1-phenylethyl] 4-(1,2,4-triazol-1-yl)benzoate
—— 2-[(4R)-4-(2-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H26ClN5O2S2
2-[(4R)-4-(2-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— [2-[Di(propan-2-yl)amino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate —— C17H22N4O3
[2-[Di(propan-2-yl)amino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate
—— 2-[(4S)-3-tert-butyl-1-(3-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C28H33ClFN5O2S
2-[(4S)-3-tert-butyl-1-(3-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— [2-[[(3S)-1,1-dioxothiolan-3-yl]-(2-methylpropyl)amino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate —— C19H24N4O5S
[2-[[(3S)-1,1-dioxothiolan-3-yl]-(2-methylpropyl)amino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate
—— 2-[(4R)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C30H23ClFN5O2S2
2-[(4R)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4R)-3-tert-butyl-1-(3-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C28H33ClFN5O2S
2-[(4R)-3-tert-butyl-1-(3-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— (2-Oxo-2-piperidin-1-ylethyl) 4-(1,2,4-triazol-1-yl)benzoate —— C16H18N4O3
(2-Oxo-2-piperidin-1-ylethyl) 4-(1,2,4-triazol-1-yl)benzoate
—— (3S)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-2,3-dihydro-1,4-benzodioxine-3-carboxamide —— C19H18N4O3
(3S)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-2,3-dihydro-1,4-benzodioxine-3-carboxamide
—— 2-[(4S)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H25F2N5O2S2
2-[(4S)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4R)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H26FN5O2S2
2-[(4R)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— [(2R)-1-(cyclohexylamino)-1-oxopropan-2-yl] 4-(1,2,4-triazol-1-yl)benzoate —— C18H22N4O3
[(2R)-1-(cyclohexylamino)-1-oxopropan-2-yl] 4-(1,2,4-triazol-1-yl)benzoate
—— [2-(5-Chloro-2-nitroanilino)-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate —— C17H12ClN5O5
[2-(5-Chloro-2-nitroanilino)-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate
—— (3R)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-2,3-dihydro-1,4-benzodioxine-3-carboxamide —— C19H18N4O3
(3R)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-2,3-dihydro-1,4-benzodioxine-3-carboxamide
—— N-[4-(4-ethylphenyl)-1,3-thiazol-2-yl]-3-methyl-5-propan-2-yl-1,2-oxazole-4-carboxamide —— C19H21N3O2S
N-[4-(4-ethylphenyl)-1,3-thiazol-2-yl]-3-methyl-5-propan-2-yl-1,2-oxazole-4-carboxamide
—— (2S)-N-[(E)-(5-bromo-2-methoxyphenyl)methylideneamino]-2-[[5-[(4-methylanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C27H27BrN6O2S
(2S)-N-[(E)-(5-bromo-2-methoxyphenyl)methylideneamino]-2-[[5-[(4-methylanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 2-[(4S)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C30H23ClFN5O2S2
2-[(4S)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— 2-[(4S)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H26FN5O2S2
2-[(4S)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— (2R)-2-[[5-[(4-chloroanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(E)-naphthalen-1-ylmethylideneamino]propanamide —— C29H25ClN6OS
(2R)-2-[[5-[(4-chloroanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(E)-naphthalen-1-ylmethylideneamino]propanamide
—— N-[(1R)-1-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-4-nitrobenzamide —— C18H16N4O5
N-[(1R)-1-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-4-nitrobenzamide
—— 4-N-[(E)-1,3-benzodioxol-5-ylmethylideneamino]-5-N-[(Z)-1,3-benzodioxol-5-ylmethylideneamino]-1-(4-nitrophenyl)triazole-4,5-dicarboxamide —— C26H18N8O8
4-N-[(E)-1,3-benzodioxol-5-ylmethylideneamino]-5-N-[(Z)-1,3-benzodioxol-5-ylmethylideneamino]-1-(4-nitrophenyl)triazole-4,5-dicarboxamide
—— 2-[(4R)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C31H25F2N5O2S2
2-[(4R)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— N-[(1S)-1-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]-2-(4-methoxyphenyl)acetamide —— C19H18ClN3O3
N-[(1S)-1-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]-2-(4-methoxyphenyl)acetamide
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-chlorophenyl)-4-methyl-N-(pyridin-3-ylmethyl)pyrazole-3-carboxamide —— C27H27ClN6O6S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-chlorophenyl)-4-methyl-N-(pyridin-3-ylmethyl)pyrazole-3-carboxamide
—— 2-[(4S)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C30H23ClFN5O2S2
2-[(4S)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— (5R,7R)-3-chloro-N-(3-imidazol-1-ylphenyl)adamantane-1-carboxamide —— C20H22ClN3O
(5R,7R)-3-chloro-N-(3-imidazol-1-ylphenyl)adamantane-1-carboxamide
—— (2S)-2-[[5-[(4-chloroanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(E)-naphthalen-1-ylmethylideneamino]propanamide —— C29H25ClN6OS
(2S)-2-[[5-[(4-chloroanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(E)-naphthalen-1-ylmethylideneamino]propanamide
—— 2-[(4S)-4-(4-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H26FN5O2S2
2-[(4S)-4-(4-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 4-N-[(Z)-1,3-benzodioxol-5-ylmethylideneamino]-5-N-[(E)-1,3-benzodioxol-5-ylmethylideneamino]-1-(4-nitrophenyl)triazole-4,5-dicarboxamide —— C26H18N8O8
4-N-[(Z)-1,3-benzodioxol-5-ylmethylideneamino]-5-N-[(E)-1,3-benzodioxol-5-ylmethylideneamino]-1-(4-nitrophenyl)triazole-4,5-dicarboxamide
—— 2-[(4R)-4-(4-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H26FN5O2S2
2-[(4R)-4-(4-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-chlorophenyl)-4-methyl-N-(pyridin-3-ylmethyl)pyrazole-3-carboxamide —— C27H27ClN6O6S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-chlorophenyl)-4-methyl-N-(pyridin-3-ylmethyl)pyrazole-3-carboxamide
—— 4-N-[(E)-(4-ethoxyphenyl)methylideneamino]-5-N-[(Z)-(4-ethoxyphenyl)methylideneamino]-1-(4-nitrophenyl)triazole-4,5-dicarboxamide —— C28H26N8O6
4-N-[(E)-(4-ethoxyphenyl)methylideneamino]-5-N-[(Z)-(4-ethoxyphenyl)methylideneamino]-1-(4-nitrophenyl)triazole-4,5-dicarboxamide
—— N-[(1S)-1-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-4-nitrobenzamide —— C18H16N4O5
N-[(1S)-1-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-4-nitrobenzamide
—— 2-[(4S)-4-(2-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H26ClN5O2S2
2-[(4S)-4-(2-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— N-[(Z)-1-(1,3-benzothiazol-2-yl)ethylideneamino]-2-(5-phenyltetrazol-2-yl)acetamide —— C18H15N7OS
N-[(Z)-1-(1,3-benzothiazol-2-yl)ethylideneamino]-2-(5-phenyltetrazol-2-yl)acetamide
—— 2-(2-morpholin-4-yl-1,3-thiazol-4-yl)-N-[(Z)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethylideneamino]acetamide —— C19H21N7O2S
2-(2-morpholin-4-yl-1,3-thiazol-4-yl)-N-[(Z)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethylideneamino]acetamide
—— [2-oxo-2-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]amino]ethyl] 4-(1,2,4-triazol-1-yl)benzoate —— C21H20N4O3
[2-oxo-2-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]amino]ethyl] 4-(1,2,4-triazol-1-yl)benzoate
—— [(2R)-1-(2,3-dihydroindol-1-yl)-1-oxopropan-2-yl] 4-(1,2,4-triazol-1-yl)benzoate —— C20H18N4O3
[(2R)-1-(2,3-dihydroindol-1-yl)-1-oxopropan-2-yl] 4-(1,2,4-triazol-1-yl)benzoate
—— [2-(2,5-Difluoroanilino)-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate —— C17H12F2N4O3
[2-(2,5-Difluoroanilino)-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate
—— N-(1,3-benzothiazol-2-yl)-4-methoxy-1-phenylpyrazole-3-carboxamide —— C18H14N4O2S
N-(1,3-benzothiazol-2-yl)-4-methoxy-1-phenylpyrazole-3-carboxamide