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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(4R)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C33H33ClN4O4S
2-[(4R)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-[(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C28H25ClN4O2S2
2-[(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— (2R)-1-(2,6-dimethylphenoxy)-3-[[5-(4-fluorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]propan-2-ol —— C22H24FN3O2S
(2R)-1-(2,6-dimethylphenoxy)-3-[[5-(4-fluorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]propan-2-ol
—— 2-[(4S)-3-(4-chlorophenyl)-4-(2-methylphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C33H33ClN4O3S
2-[(4S)-3-(4-chlorophenyl)-4-(2-methylphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— (4R)-4-(2-chlorophenyl)-1-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H27ClN4O3S2
(4R)-4-(2-chlorophenyl)-1-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4S)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C31H31ClN4O4S
2-[(4S)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— [(5S)-3,5-bis(difluoromethyl)-5-hydroxy-4H-pyrazol-1-yl]-[(5S,7S)-3-(tetrazol-2-yl)-1-adamantyl]methanone —— C17H20F4N6O2
[(5S)-3,5-bis(difluoromethyl)-5-hydroxy-4H-pyrazol-1-yl]-[(5S,7S)-3-(tetrazol-2-yl)-1-adamantyl]methanone
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C28H27ClN4O2S2
2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4R)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C24H18Cl2N4O2S2
2-[(4R)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— (2S)-1-[[5-(4-methoxyphenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-3-[[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]oxy]propan-2-ol —— C23H27N3O3S
(2S)-1-[[5-(4-methoxyphenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-3-[[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]oxy]propan-2-ol
—— (E)-2-(5-morpholin-4-yl-4-phenyl-1,2,4-triazol-3-yl)-3-(2,4,5-trimethylphenyl)prop-2-enenitrile —— C24H25N5O
(E)-2-(5-morpholin-4-yl-4-phenyl-1,2,4-triazol-3-yl)-3-(2,4,5-trimethylphenyl)prop-2-enenitrile
—— 2-[(4S)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C33H33ClN4O4S
2-[(4S)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— N-[(2R)-butan-2-yl]-2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C29H29ClN4O2S2
N-[(2R)-butan-2-yl]-2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— 2-[(4R)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide —— C32H33ClN4O3S
2-[(4R)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide
—— (4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H27ClN4O2S2
(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4R)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C28H24ClFN4O3S2
(4R)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4S)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C32H31ClN4O4S
(4S)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-3-(4-chlorophenyl)-4-(2-methylphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C33H29ClN4O3S
2-[(4R)-3-(4-chlorophenyl)-4-(2-methylphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— (E)-2-cyano-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C19H17N5O2S
(E)-2-cyano-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— (4S)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C28H24ClFN4O3S2
(4S)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 3-[[5-(4-methoxyphenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methyl-4-oxopentan-2-yl)propanamide —— C19H26N4O3S
3-[[5-(4-methoxyphenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methyl-4-oxopentan-2-yl)propanamide
—— (2S)-1-[(2-fluorophenyl)methoxy]-3-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanyl]propan-2-ol —— C21H22FN3O2S
(2S)-1-[(2-fluorophenyl)methoxy]-3-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanyl]propan-2-ol
—— 2-[(4S)-4-(2-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C32H26ClFN4O2S2
2-[(4S)-4-(2-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C28H25ClN4O2S2
2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— (3R,4S)-4-[(4-ethyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]-1,1-dioxothiolan-3-ol —— C14H17N3O3S2
(3R,4S)-4-[(4-ethyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]-1,1-dioxothiolan-3-ol
—— 2-[(4R)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C28H26Cl2N4O3S2
2-[(4R)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— 2-[(4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C32H30ClFN4O3S
2-[(4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C24H18Cl2N4O2S2
2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— 2-[(4R)-3-(4-chlorophenyl)-4-(2-methylphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C31H29ClN4O2S
2-[(4R)-3-(4-chlorophenyl)-4-(2-methylphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— 2-[(4S)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide —— C32H33ClN4O3S
2-[(4S)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide
—— (4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H28ClFN4O3S
(4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide —— C29H29ClN4O2S2
2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide
—— N-[[5-(2,4-difluorophenoxy)-3-ethyl-1-(4-methoxyphenyl)pyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]thiophene-2-carboxamide —— C29H29F2N3O4S
N-[[5-(2,4-difluorophenoxy)-3-ethyl-1-(4-methoxyphenyl)pyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]thiophene-2-carboxamide
—— (4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H28ClFN4O2S
(4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (2R)-2-[[5-(4-methoxyphenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]pentanedinitrile —— C16H17N5OS
(2R)-2-[[5-(4-methoxyphenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]pentanedinitrile
—— (3S,4R)-4-[[5-(4-fluorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-1,1-dioxothiolan-3-ol —— C15H16FN3O3S2
(3S,4R)-4-[[5-(4-fluorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-1,1-dioxothiolan-3-ol
—— N-[[5-(2,4-difluorophenoxy)-3-ethyl-1-(4-methoxyphenyl)pyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide —— C31H31F2N3O4
N-[[5-(2,4-difluorophenoxy)-3-ethyl-1-(4-methoxyphenyl)pyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide
—— (2R)-1-[(4-ethyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]-3-(2-fluorophenoxy)propan-2-ol —— C19H20FN3O2S
(2R)-1-[(4-ethyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]-3-(2-fluorophenoxy)propan-2-ol
—— 3-tert-butyl-1-[[5-(2,4-difluorophenoxy)-3-ethyl-1-(4-methoxyphenyl)pyrazol-4-yl]methyl]-1-[[(2R)-oxolan-2-yl]methyl]urea —— C29H36F2N4O4
3-tert-butyl-1-[[5-(2,4-difluorophenoxy)-3-ethyl-1-(4-methoxyphenyl)pyrazol-4-yl]methyl]-1-[[(2R)-oxolan-2-yl]methyl]urea
—— 2-[(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C30H25ClN4O3S2
2-[(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 2-fluoro-N-[[5-(3-fluorophenoxy)-1-phenyl-3-propan-2-ylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide —— C31H31F2N3O3
2-fluoro-N-[[5-(3-fluorophenoxy)-1-phenyl-3-propan-2-ylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide
—— (2S)-1-[[5-(4-fluorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-3-(3-methylphenoxy)propan-2-ol —— C21H22FN3O2S
(2S)-1-[[5-(4-fluorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-3-(3-methylphenoxy)propan-2-ol
—— (2S)-1-[(4-ethyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]-3-naphthalen-1-yloxypropan-2-ol —— C23H23N3O2S
(2S)-1-[(4-ethyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]-3-naphthalen-1-yloxypropan-2-ol
—— 2-[(4R)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C33H33ClN4O4S
2-[(4R)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— N-(2-methyl-4-oxopentan-2-yl)-3-[1-(4-propan-2-ylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C19H27N5O2S
N-(2-methyl-4-oxopentan-2-yl)-3-[1-(4-propan-2-ylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— (4S)-4-(2-chlorophenyl)-1-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H27ClN4O3S2
(4S)-4-(2-chlorophenyl)-1-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H28ClFN4O2S
(4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— N-[[5-(2,4-difluorophenoxy)-3-ethyl-1-(4-methoxyphenyl)pyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]furan-2-carboxamide —— C29H29F2N3O5
N-[[5-(2,4-difluorophenoxy)-3-ethyl-1-(4-methoxyphenyl)pyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]furan-2-carboxamide
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide —— C28H27ClN4O2S2
2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide
—— 2-[(4R)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C32H33ClN4O4S
2-[(4R)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide