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中文名称 英文名称 CAS号 化学式 结构式图片
—— [(2S)-1-(cycloheptylamino)-1-oxopropan-2-yl] 4-pyrazol-1-ylbenzoate —— C20H25N3O3
[(2S)-1-(cycloheptylamino)-1-oxopropan-2-yl] 4-pyrazol-1-ylbenzoate
—— (2R)-2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-ethylpropanamide —— C14H19N5OS
(2R)-2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-ethylpropanamide
—— (2S)-2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-ethylpropanamide —— C14H19N5OS
(2S)-2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-ethylpropanamide
—— 2-[[3-(3-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-5-(furan-2-yl)-1,3,4-oxadiazole —— C15H9ClN4O3S
2-[[3-(3-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-5-(furan-2-yl)-1,3,4-oxadiazole
—— [(2S)-1-oxo-1-(2-propan-2-ylanilino)propan-2-yl] 4-pyrazol-1-ylbenzoate —— C22H23N3O3
[(2S)-1-oxo-1-(2-propan-2-ylanilino)propan-2-yl] 4-pyrazol-1-ylbenzoate
—— 2-[(4S)-3-tert-butyl-4-(2-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C28H32F2N4O3S
2-[(4S)-3-tert-butyl-4-(2-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— (4S)-4-(2,5-dimethoxyphenyl)-1-methyl-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H34N4O4S
(4S)-4-(2,5-dimethoxyphenyl)-1-methyl-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(3-chlorophenyl)-1-(2-methylphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H36ClN5O3S
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(3-chlorophenyl)-1-(2-methylphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— [(2S)-1-[benzyl(tert-butyl)amino]-1-oxopropan-2-yl] 4-pyrazol-1-ylbenzoate —— C24H27N3O3
[(2S)-1-[benzyl(tert-butyl)amino]-1-oxopropan-2-yl] 4-pyrazol-1-ylbenzoate
—— [(2R)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] 2-[(1R)-2-(benzenesulfonyl)-3,4-dihydro-1H-isoquinolin-1-yl]acetate —— C31H32N4O6S
[(2R)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] 2-[(1R)-2-(benzenesulfonyl)-3,4-dihydro-1H-isoquinolin-1-yl]acetate
—— (4Z,5R)-5-(4-fluorophenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(3-morpholin-4-ylpropyl)pyrrolidine-2,3-dione —— C28H29FN4O4
(4Z,5R)-5-(4-fluorophenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(3-morpholin-4-ylpropyl)pyrrolidine-2,3-dione
—— [2-(1-methyl-2-oxo-3H-indol-5-yl)-2-oxoethyl] 4-pyrazol-1-ylbenzoate —— C21H17N3O4
[2-(1-methyl-2-oxo-3H-indol-5-yl)-2-oxoethyl] 4-pyrazol-1-ylbenzoate
—— 3-[[3-(4-Ethylphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-5-(4-methoxyphenyl)-1,2,4-triazol-4-amine —— C20H20N6O2S
3-[[3-(4-Ethylphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-5-(4-methoxyphenyl)-1,2,4-triazol-4-amine
—— [3-(4-Ethylphenyl)-1,2,4-oxadiazol-5-yl]methyl 3-(3,5-dimethyl-1,2-oxazol-4-yl)propanoate —— C19H21N3O4
[3-(4-Ethylphenyl)-1,2,4-oxadiazol-5-yl]methyl 3-(3,5-dimethyl-1,2-oxazol-4-yl)propanoate
—— 3-[[3-(2-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-5-(4-methylphenyl)-1,2,4-triazol-4-amine —— C18H15ClN6OS
3-[[3-(2-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-5-(4-methylphenyl)-1,2,4-triazol-4-amine
—— (2R)-1-[[5-(4-fluorophenoxy)-1-methyl-3-phenylpyrazol-4-yl]methyl-(furan-2-ylmethyl)amino]-3-(furan-2-ylmethoxy)propan-2-ol —— C30H30FN3O5
(2R)-1-[[5-(4-fluorophenoxy)-1-methyl-3-phenylpyrazol-4-yl]methyl-(furan-2-ylmethyl)amino]-3-(furan-2-ylmethoxy)propan-2-ol
—— [2-oxo-2-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethyl] 1-(4-fluorophenyl)-3-methylthieno[2,3-c]pyrazole-5-carboxylate —— C25H28FN3O3S
[2-oxo-2-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethyl] 1-(4-fluorophenyl)-3-methylthieno[2,3-c]pyrazole-5-carboxylate
—— [(2R)-1-(2,6-dimethylanilino)-1-oxopropan-2-yl] 4-pyrazol-1-ylbenzoate —— C21H21N3O3
[(2R)-1-(2,6-dimethylanilino)-1-oxopropan-2-yl] 4-pyrazol-1-ylbenzoate
—— 2-[(4R)-4-(2,5-dimethoxyphenyl)-1-methyl-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C29H29N5O4S
2-[(4R)-4-(2,5-dimethoxyphenyl)-1-methyl-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— [(2R)-1-(2-ethoxyanilino)-1-oxopropan-2-yl] 4-pyrazol-1-ylbenzoate —— C21H21N3O4
[(2R)-1-(2-ethoxyanilino)-1-oxopropan-2-yl] 4-pyrazol-1-ylbenzoate
—— [(2R)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] 2-[(3,4-difluorophenyl)sulfonylamino]benzoate —— C27H24F2N4O6S
[(2R)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] 2-[(3,4-difluorophenyl)sulfonylamino]benzoate
—— 2-[[3-(3-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-5-[(3-methylphenoxy)methyl]-1,3,4-oxadiazole —— C19H15ClN4O3S
2-[[3-(3-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-5-[(3-methylphenoxy)methyl]-1,3,4-oxadiazole
—— 4-Cyclopropyl-3-(2-fluorophenyl)-5-[3-(4-methoxyphenoxy)propylsulfanyl]-1,2,4-triazole —— C21H22FN3O2S
4-Cyclopropyl-3-(2-fluorophenyl)-5-[3-(4-methoxyphenoxy)propylsulfanyl]-1,2,4-triazole
—— 3-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methylsulfanyl]-5-(4-methoxyphenyl)-1,2,4-triazol-4-amine —— C19H19ClN4O3S
3-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methylsulfanyl]-5-(4-methoxyphenyl)-1,2,4-triazol-4-amine
—— 2-[(4S)-4-(2,4-difluorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C31H30F2N4O3S
2-[(4S)-4-(2,4-difluorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— [3-(3-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl 3-(3,5-dimethyl-1,2-oxazol-4-yl)propanoate —— C17H16ClN3O4
[3-(3-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl 3-(3,5-dimethyl-1,2-oxazol-4-yl)propanoate
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C28H31FN4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— (4Z,5R)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)-5-phenylpyrrolidine-2,3-dione —— C27H28N4O4
(4Z,5R)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)-5-phenylpyrrolidine-2,3-dione
—— (4S)-3-tert-butyl-1-(2-chlorophenyl)-4-(3-fluorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C28H30ClFN4O3S
(4S)-3-tert-butyl-1-(2-chlorophenyl)-4-(3-fluorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— ethyl (2S)-2-(4-methyl-1,3-thiazol-2-yl)-4-(4-nitroimidazol-1-yl)-3-oxobutanoate —— C13H14N4O5S
ethyl (2S)-2-(4-methyl-1,3-thiazol-2-yl)-4-(4-nitroimidazol-1-yl)-3-oxobutanoate
—— ethyl (2R)-2-(4-methyl-1,3-thiazol-2-yl)-4-(4-nitroimidazol-1-yl)-3-oxobutanoate —— C13H14N4O5S
ethyl (2R)-2-(4-methyl-1,3-thiazol-2-yl)-4-(4-nitroimidazol-1-yl)-3-oxobutanoate
—— [3-(3-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 2,3-dichlorobenzoate —— C17H12Cl2N2O4
[3-(3-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 2,3-dichlorobenzoate
—— (4Z,5S)-1-(4,5-dimethyl-1,3-thiazol-2-yl)-4-[(4-ethoxyphenyl)-hydroxymethylidene]-5-thiophen-2-ylpyrrolidine-2,3-dione —— C22H20N2O4S2
(4Z,5S)-1-(4,5-dimethyl-1,3-thiazol-2-yl)-4-[(4-ethoxyphenyl)-hydroxymethylidene]-5-thiophen-2-ylpyrrolidine-2,3-dione
—— [(1S)-2-(4-methyl-2-nitroanilino)-2-oxo-1-phenylethyl] (Z)-3-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C34H28N4O6
[(1S)-2-(4-methyl-2-nitroanilino)-2-oxo-1-phenylethyl] (Z)-3-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [3-(3-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 4-(diethylamino)benzoate —— C21H23N3O4
[3-(3-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 4-(diethylamino)benzoate
—— (4Z,5R)-1-(4,5-dimethyl-1,3-thiazol-2-yl)-4-[(4-ethoxyphenyl)-hydroxymethylidene]-5-thiophen-2-ylpyrrolidine-2,3-dione —— C22H20N2O4S2
(4Z,5R)-1-(4,5-dimethyl-1,3-thiazol-2-yl)-4-[(4-ethoxyphenyl)-hydroxymethylidene]-5-thiophen-2-ylpyrrolidine-2,3-dione
—— [2-[ethyl(naphthalen-1-yl)amino]-2-oxoethyl] (Z)-3-[3-(3,4-dimethoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C34H31N3O5
[2-[ethyl(naphthalen-1-yl)amino]-2-oxoethyl] (Z)-3-[3-(3,4-dimethoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [2-[4-nitro-2-(trifluoromethyl)anilino]-2-oxoethyl] (Z)-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enoate —— C25H17F3N4O5S
[2-[4-nitro-2-(trifluoromethyl)anilino]-2-oxoethyl] (Z)-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enoate
—— [(2R)-1-oxo-1-[(4-phenyl-1,3-thiazol-2-yl)amino]propan-2-yl] (Z)-3-[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C30H23FN4O3S
[(2R)-1-oxo-1-[(4-phenyl-1,3-thiazol-2-yl)amino]propan-2-yl] (Z)-3-[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 2,5-dichlorobenzoate —— C17H11Cl2NO3
(5-Phenyl-1,3-oxazol-2-yl)methyl 2,5-dichlorobenzoate
—— [(1S)-2-(2-methoxy-5-methylanilino)-2-oxo-1-phenylethyl] (Z)-3-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C35H31N3O5
[(1S)-2-(2-methoxy-5-methylanilino)-2-oxo-1-phenylethyl] (Z)-3-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [(1R)-2-(4-methyl-2-nitroanilino)-2-oxo-1-phenylethyl] (E)-3-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C34H28N4O6
[(1R)-2-(4-methyl-2-nitroanilino)-2-oxo-1-phenylethyl] (E)-3-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [2-[[(3S)-1,1-dioxothiolan-3-yl]-ethylamino]-2-oxoethyl] (Z)-3-[3-(1-benzofuran-2-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C28H27N3O6S
[2-[[(3S)-1,1-dioxothiolan-3-yl]-ethylamino]-2-oxoethyl] (Z)-3-[3-(1-benzofuran-2-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [2-[[(3R)-1,1-dioxothiolan-3-yl]-ethylamino]-2-oxoethyl] (Z)-3-[3-(1-benzofuran-2-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C28H27N3O6S
[2-[[(3R)-1,1-dioxothiolan-3-yl]-ethylamino]-2-oxoethyl] (Z)-3-[3-(1-benzofuran-2-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [(1S)-2-(4-chloro-3-nitroanilino)-2-oxo-1-phenylethyl] (Z)-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enoate —— C30H21ClN4O5S
[(1S)-2-(4-chloro-3-nitroanilino)-2-oxo-1-phenylethyl] (Z)-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enoate
—— [(1R)-2-(4-chloro-3-nitroanilino)-2-oxo-1-phenylethyl] (E)-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enoate —— C30H21ClN4O5S
[(1R)-2-(4-chloro-3-nitroanilino)-2-oxo-1-phenylethyl] (E)-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enoate
—— (3-Phenyl-1,2,4-oxadiazol-5-yl)methyl 5-bromopyridine-3-carboxylate —— C15H10BrN3O3
(3-Phenyl-1,2,4-oxadiazol-5-yl)methyl 5-bromopyridine-3-carboxylate
—— [2-(4-cyanoanilino)-2-oxoethyl] (Z)-3-[3-(4-bromophenyl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C27H19BrN4O3
[2-(4-cyanoanilino)-2-oxoethyl] (Z)-3-[3-(4-bromophenyl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [(1R)-2-(2-ethoxyanilino)-2-oxo-1-phenylethyl] (Z)-3-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C35H31N3O5
[(1R)-2-(2-ethoxyanilino)-2-oxo-1-phenylethyl] (Z)-3-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [(1R)-2-(4-methyl-2-nitroanilino)-2-oxo-1-phenylethyl] (Z)-3-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C34H28N4O6
[(1R)-2-(4-methyl-2-nitroanilino)-2-oxo-1-phenylethyl] (Z)-3-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoate