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中文名称 英文名称 CAS号 化学式 结构式图片
—— Methyl-[(4-phenyl-5-sulfanylidenetetrazol-1-yl)methyl]-[(4-prop-2-enoxyphenyl)methyl]azanium —— C19H22N5OS+
Methyl-[(4-phenyl-5-sulfanylidenetetrazol-1-yl)methyl]-[(4-prop-2-enoxyphenyl)methyl]azanium
—— (4Z,5R)-5-(4-fluorophenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione —— C27H27FN4O4
(4Z,5R)-5-(4-fluorophenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione
—— 5-Cyclopropyl-2-[[methyl-[[4-(trifluoromethyl)phenyl]methyl]amino]methyl]-4-phenyl-1,2,4-triazole-3-thione —— C21H21F3N4S
5-Cyclopropyl-2-[[methyl-[[4-(trifluoromethyl)phenyl]methyl]amino]methyl]-4-phenyl-1,2,4-triazole-3-thione
—— [4-(4-Methoxyphenyl)-5-sulfanylidenetetrazol-1-yl]methyl-methyl-[(4-prop-2-enoxyphenyl)methyl]azanium —— C20H24N5O2S+
[4-(4-Methoxyphenyl)-5-sulfanylidenetetrazol-1-yl]methyl-methyl-[(4-prop-2-enoxyphenyl)methyl]azanium
—— 2-[[(2-Chloro-6-fluorophenyl)methyl-methylamino]methyl]-4-(3-methoxyphenyl)-1,2,4-triazole-3-thione —— C18H18ClFN4OS
2-[[(2-Chloro-6-fluorophenyl)methyl-methylamino]methyl]-4-(3-methoxyphenyl)-1,2,4-triazole-3-thione
—— (4Z,5S)-5-(4-fluorophenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione —— C27H27FN4O4
(4Z,5S)-5-(4-fluorophenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione
—— (2-Chloro-6-fluorophenyl)methyl-[[3-(4-methoxyphenyl)-4-methyl-5-sulfanylidene-1,2,4-triazol-1-yl]methyl]-methylazanium —— C19H21ClFN4OS+
(2-Chloro-6-fluorophenyl)methyl-[[3-(4-methoxyphenyl)-4-methyl-5-sulfanylidene-1,2,4-triazol-1-yl]methyl]-methylazanium
—— 5-(4-Fluorophenyl)-4-methyl-2-[[methyl-[(4-prop-2-enoxyphenyl)methyl]amino]methyl]-1,2,4-triazole-3-thione —— C21H23FN4OS
5-(4-Fluorophenyl)-4-methyl-2-[[methyl-[(4-prop-2-enoxyphenyl)methyl]amino]methyl]-1,2,4-triazole-3-thione
—— N-[3-(N-methylanilino)propyl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide —— C19H22N6OS
N-[3-(N-methylanilino)propyl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide
—— 1-[[Methyl-[(4-prop-2-enoxyphenyl)methyl]amino]methyl]-4-phenyltetrazole-5-thione —— C19H21N5OS
1-[[Methyl-[(4-prop-2-enoxyphenyl)methyl]amino]methyl]-4-phenyltetrazole-5-thione
—— (3S)-3-methyl-5-[2-(1-phenyltetrazol-5-yl)sulfanylacetyl]-1,3-dihydroindol-2-one —— C18H15N5O2S
(3S)-3-methyl-5-[2-(1-phenyltetrazol-5-yl)sulfanylacetyl]-1,3-dihydroindol-2-one
—— 2-[(4R)-3-tert-butyl-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C27H35N5O3S2
2-[(4R)-3-tert-butyl-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— (4Z,5S)-5-(2,3-dimethoxyphenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione —— C29H32N4O6
(4Z,5S)-5-(2,3-dimethoxyphenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione
—— N-[2-(2-fluorophenyl)ethyl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide —— C17H16FN5OS
N-[2-(2-fluorophenyl)ethyl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide
—— N-[2-(4-chlorophenoxy)ethyl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide —— C17H16ClN5O2S
N-[2-(4-chlorophenoxy)ethyl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide
—— (4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H27ClN4O3S2
(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (2S)-2-[[4-(2,4-difluorophenyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-methyl-2-nitrophenyl)-2-phenylacetamide —— C29H21F2N5O3S
(2S)-2-[[4-(2,4-difluorophenyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-methyl-2-nitrophenyl)-2-phenylacetamide
—— 1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(1-phenyltetrazol-5-yl)sulfanylethanone —— C18H16N4O3S
1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(1-phenyltetrazol-5-yl)sulfanylethanone
—— (4Z,5R)-5-(2,3-dimethoxyphenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione —— C29H32N4O6
(4Z,5R)-5-(2,3-dimethoxyphenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione
—— ethyl (4R)-6-[[4-(2,4-difluorophenyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanylmethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C28H23F2N5O3S
ethyl (4R)-6-[[4-(2,4-difluorophenyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanylmethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— [2-[[4-(Dimethylamino)phenyl]methyl-methylamino]-2-oxoethyl] 2-(3-methylbutylamino)-1,3-thiazole-4-carboxylate —— C21H30N4O3S
[2-[[4-(Dimethylamino)phenyl]methyl-methylamino]-2-oxoethyl] 2-(3-methylbutylamino)-1,3-thiazole-4-carboxylate
—— (2R)-2-[[4-(2,4-difluorophenyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-methyl-2-nitrophenyl)-2-phenylacetamide —— C29H21F2N5O3S
(2R)-2-[[4-(2,4-difluorophenyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-methyl-2-nitrophenyl)-2-phenylacetamide
—— [2-[[4-(Dimethylamino)phenyl]methylamino]-2-oxoethyl] 4-pyrazol-1-ylbenzoate —— C21H22N4O3
[2-[[4-(Dimethylamino)phenyl]methylamino]-2-oxoethyl] 4-pyrazol-1-ylbenzoate
—— N-cyclopropyl-N-[(4-methoxyphenyl)methyl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide —— C20H21N5O2S
N-cyclopropyl-N-[(4-methoxyphenyl)methyl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide
—— 6-chloro-2-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanylmethyl]-3H-quinazolin-4-one —— C20H16ClN5OS
6-chloro-2-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanylmethyl]-3H-quinazolin-4-one
—— (2S)-N-tert-butyl-2-[(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)sulfanyl]propanamide —— C18H21N5O2S
(2S)-N-tert-butyl-2-[(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)sulfanyl]propanamide
—— (2R)-2-[(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)sulfanyl]-N-propylpropanamide —— C17H19N5O2S
(2R)-2-[(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)sulfanyl]-N-propylpropanamide
—— 2-[[(2S)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-ium-1-yl]methyl]-4-(2-methylphenyl)-1,2,4-triazole-3-thione —— C21H22N5S2+
2-[[(2S)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-ium-1-yl]methyl]-4-(2-methylphenyl)-1,2,4-triazole-3-thione
—— ethyl (4S)-6-[[4-(2,4-difluorophenyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanylmethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C28H23F2N5O3S
ethyl (4S)-6-[[4-(2,4-difluorophenyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanylmethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-methyl-2-(1-phenyltetrazol-5-yl)sulfanylacetamide —— C19H19N5O3S
N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-methyl-2-(1-phenyltetrazol-5-yl)sulfanylacetamide
—— 4-chloro-N-[[3-ethyl-5-(3-fluorophenoxy)-1-phenylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide —— C30H29ClFN3O3
4-chloro-N-[[3-ethyl-5-(3-fluorophenoxy)-1-phenylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide
—— (4Z,5R)-5-(2,5-dimethoxyphenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione —— C29H32N4O6
(4Z,5R)-5-(2,5-dimethoxyphenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione
—— 4-chloro-N-[[3-ethyl-5-(3-fluorophenoxy)-1-phenylpyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide —— C30H29ClFN3O3
4-chloro-N-[[3-ethyl-5-(3-fluorophenoxy)-1-phenylpyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide
—— (2S)-N-(2-methoxyethyl)-2-[(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)sulfanyl]propanamide —— C17H19N5O3S
(2S)-N-(2-methoxyethyl)-2-[(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)sulfanyl]propanamide
—— N-[2-(2-methoxyphenyl)ethyl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide —— C18H19N5O2S
N-[2-(2-methoxyphenyl)ethyl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide
—— 2-[5-(3-fluorophenyl)tetrazol-2-yl]-N-[3-(N-methylanilino)propyl]acetamide —— C19H21FN6O
2-[5-(3-fluorophenyl)tetrazol-2-yl]-N-[3-(N-methylanilino)propyl]acetamide
—— 2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C33H29ClN4O4S
2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— [2-[2-(4-Nitroanilino)ethylamino]-2-oxoethyl] 4-pyrazol-1-ylbenzoate —— C20H19N5O5
[2-[2-(4-Nitroanilino)ethylamino]-2-oxoethyl] 4-pyrazol-1-ylbenzoate
—— (4Z,5S)-5-(2,5-dimethoxyphenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione —— C29H32N4O6
(4Z,5S)-5-(2,5-dimethoxyphenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C33H29ClN4O4S
2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 6-chloro-2-[[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]-3H-quinazolin-4-one —— C18H15ClN6OS
6-chloro-2-[[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]-3H-quinazolin-4-one
—— 2-[(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C29H30ClN5O2S2
2-[(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C28H27ClN4O3S2
2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— (4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H34ClN5O5S
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C32H39N5O5S
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4Z,5R)-1-[3-(dimethylamino)propyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dione —— C29H34N4O3
(4Z,5R)-1-[3-(dimethylamino)propyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-(4-propan-2-ylphenyl)pyrrolidine-2,3-dione
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide —— C29H30ClN5O2S2
2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H26ClN5O3S2
2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H26ClN5O2S2
2-[(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C32H30F2N4O4S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide