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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(4R)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C27H22Cl2N4O2S2
2-[(4R)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— 2-[(4R)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C33H36N4O5S2
2-[(4R)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-[(4R)-4-(4-fluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C34H28F2N4O3S
2-[(4R)-4-(4-fluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 2-[(4R)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C29H26Cl2N4O3S2
2-[(4R)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— (2R)-N-(4-acetamidophenyl)-2-[[5-(4-tert-butylphenyl)-4-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C31H35N5O3S
(2R)-N-(4-acetamidophenyl)-2-[[5-(4-tert-butylphenyl)-4-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 2-[(4R)-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C36H33FN4O3S
2-[(4R)-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 5-Cyclopropyl-2-[(4-methylpiperidin-1-yl)methyl]-4-phenyl-1,2,4-triazole-3-thione —— C18H24N4S
5-Cyclopropyl-2-[(4-methylpiperidin-1-yl)methyl]-4-phenyl-1,2,4-triazole-3-thione
—— 2-[(4R)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide —— C28H26F2N4O2S2
2-[(4R)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C32H30ClFN4O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 2-[(4S)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide —— C33H36N4O5S
2-[(4S)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide
—— 4-[4-(2-Ethylphenyl)-5-[(2-methoxyphenyl)methylsulfanyl]-1,2,4-triazol-3-yl]morpholine —— C22H26N4O2S
4-[4-(2-Ethylphenyl)-5-[(2-methoxyphenyl)methylsulfanyl]-1,2,4-triazol-3-yl]morpholine
—— N-cyclopropyl-2-[[4-(2-ethylphenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C19H25N5O2S
N-cyclopropyl-2-[[4-(2-ethylphenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— N-(2,6-dimethylphenyl)-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]acetamide —— C23H27N5OS
N-(2,6-dimethylphenyl)-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]acetamide
—— 2-[(4-Phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]-1-(1,2,5-trimethylpyrrol-3-yl)ethanone —— C22H27N5OS
2-[(4-Phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]-1-(1,2,5-trimethylpyrrol-3-yl)ethanone
—— 3-(3-Chlorophenyl)-5-[[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]-1,2,4-oxadiazole —— C18H15ClN6OS
3-(3-Chlorophenyl)-5-[[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]-1,2,4-oxadiazole
—— N-[3-(4-cyclopentyl-5-methylsulfanyl-1,2,4-triazol-3-yl)propyl]-4-(5-methylpyrazol-1-yl)benzamide —— C22H28N6OS
N-[3-(4-cyclopentyl-5-methylsulfanyl-1,2,4-triazol-3-yl)propyl]-4-(5-methylpyrazol-1-yl)benzamide
—— [2-(2-Methoxyethylamino)-2-oxoethyl] 2-(3-chlorophenyl)-4-methyl-1,3-thiazole-5-carboxylate —— C16H17ClN2O4S
[2-(2-Methoxyethylamino)-2-oxoethyl] 2-(3-chlorophenyl)-4-methyl-1,3-thiazole-5-carboxylate
—— (2S)-N-(furan-2-ylmethyl)-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]propanamide —— C21H25N5O2S
(2S)-N-(furan-2-ylmethyl)-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]propanamide
—— [2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl] 2-(3-chlorophenyl)-4-methyl-1,3-thiazole-5-carboxylate —— C18H19ClN2O4S
[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl] 2-(3-chlorophenyl)-4-methyl-1,3-thiazole-5-carboxylate
—— [(1S)-2-oxocyclohexyl] 2-(3-chlorophenyl)-4-methyl-1,3-thiazole-5-carboxylate —— C17H16ClNO3S
[(1S)-2-oxocyclohexyl] 2-(3-chlorophenyl)-4-methyl-1,3-thiazole-5-carboxylate
—— 2-(3-chlorophenyl)-5-[(1S)-1-(1-ethyl-5-phenylimidazol-2-yl)sulfanylethyl]-1,3,4-oxadiazole —— C21H19ClN4OS
2-(3-chlorophenyl)-5-[(1S)-1-(1-ethyl-5-phenylimidazol-2-yl)sulfanylethyl]-1,3,4-oxadiazole
—— N-[(2S)-3-methylbutan-2-yl]-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]acetamide —— C20H29N5OS
N-[(2S)-3-methylbutan-2-yl]-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]acetamide
—— 2-(1-ethyl-5-phenylimidazol-2-yl)sulfanyl-N-[4-(2-oxopyrrolidin-1-yl)phenyl]acetamide —— C23H24N4O2S
2-(1-ethyl-5-phenylimidazol-2-yl)sulfanyl-N-[4-(2-oxopyrrolidin-1-yl)phenyl]acetamide
—— 2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]-N-propylacetamide —— C18H25N5OS
2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]-N-propylacetamide
—— [3-(2-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 2-(4-methylphenyl)acetate —— C19H18N2O4
[3-(2-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 2-(4-methylphenyl)acetate
—— [(2R)-1-(ethylamino)-1-oxopropan-2-yl] 2-[2-(4-methylphenyl)-1,3-thiazol-4-yl]acetate —— C17H20N2O3S
[(2R)-1-(ethylamino)-1-oxopropan-2-yl] 2-[2-(4-methylphenyl)-1,3-thiazol-4-yl]acetate
—— (2R)-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]-1-pyrrolidin-1-ylpropan-1-one —— C20H27N5OS
(2R)-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]-1-pyrrolidin-1-ylpropan-1-one
—— 3-methyl-1-phenyl-N-(3-pyrrolidin-1-ylpropyl)thieno[2,3-c]pyrazole-5-carboxamide —— C20H24N4OS
3-methyl-1-phenyl-N-(3-pyrrolidin-1-ylpropyl)thieno[2,3-c]pyrazole-5-carboxamide
—— [4-[(4-Methoxyphenyl)methyl]piperazin-1-yl]-[4-(5-methylpyrazol-1-yl)phenyl]methanone —— C23H26N4O2
[4-[(4-Methoxyphenyl)methyl]piperazin-1-yl]-[4-(5-methylpyrazol-1-yl)phenyl]methanone
—— (2R)-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]propanamide —— C16H21N5OS
(2R)-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]propanamide
—— [2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl] 2-(3-chlorophenyl)-4-methyl-1,3-thiazole-5-carboxylate —— C18H19ClN2O4S
[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl] 2-(3-chlorophenyl)-4-methyl-1,3-thiazole-5-carboxylate
—— N-cyclohexyl-3-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]propanamide —— C18H24N4OS
N-cyclohexyl-3-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]propanamide
—— N-(1-cyanocyclohexyl)-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]acetamide —— C22H28N6OS
N-(1-cyanocyclohexyl)-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]acetamide
—— 2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanylmethyl]-3H-quinazolin-4-one —— C22H22N6OS
2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanylmethyl]-3H-quinazolin-4-one
—— (2R)-N-methyl-N-phenyl-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]propanamide —— C23H27N5OS
(2R)-N-methyl-N-phenyl-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]propanamide
—— N-[(1R)-1-cyano-1-cyclopropylethyl]-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]acetamide —— C21H26N6OS
N-[(1R)-1-cyano-1-cyclopropylethyl]-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]acetamide
—— 1-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]ethanone —— C21H29N5O2S
1-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]ethanone
—— N-[3-(4-cyclopentyl-5-methylsulfanyl-1,2,4-triazol-3-yl)propyl]-4-pyrazol-1-ylbenzamide —— C21H26N6OS
N-[3-(4-cyclopentyl-5-methylsulfanyl-1,2,4-triazol-3-yl)propyl]-4-pyrazol-1-ylbenzamide
—— N-(4-methoxyphenyl)-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]acetamide —— C22H25N5O2S
N-(4-methoxyphenyl)-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]acetamide
—— (2S)-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-ethylpropanamide —— C14H19N5OS
(2S)-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-ethylpropanamide
—— 4-[[4-(2-Ethylphenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]butanenitrile —— C18H23N5OS
4-[[4-(2-Ethylphenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanyl]butanenitrile
—— (2R)-N-ethyl-2-(1-ethyl-5-phenylimidazol-2-yl)sulfanylpropanamide —— C16H21N3OS
(2R)-N-ethyl-2-(1-ethyl-5-phenylimidazol-2-yl)sulfanylpropanamide
—— N-[(1R,2R)-2-methylcyclohexyl]-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]acetamide —— C22H31N5OS
N-[(1R,2R)-2-methylcyclohexyl]-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]acetamide
—— N-[(2R)-3-methylbutan-2-yl]-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]acetamide —— C20H29N5OS
N-[(2R)-3-methylbutan-2-yl]-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]acetamide
—— (2R)-1-(4-ethylpiperazin-1-yl)-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]propan-1-one —— C22H32N6OS
(2R)-1-(4-ethylpiperazin-1-yl)-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]propan-1-one
—— 1-[(3R)-3-methylpiperidin-1-yl]-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]ethanone —— C21H29N5OS
1-[(3R)-3-methylpiperidin-1-yl]-2-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanyl]ethanone
—— 3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-methyl-N-[(1S)-1-(3-nitrophenyl)ethyl]propanamide —— C23H26N4O3
3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-methyl-N-[(1S)-1-(3-nitrophenyl)ethyl]propanamide
—— (E)-N-(2,4-dimethylphenyl)-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C20H19N3O
(E)-N-(2,4-dimethylphenyl)-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— 2-[[4-(3-Fluorophenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-benzoxazole —— C20H18FN5O2S
2-[[4-(3-Fluorophenyl)-5-morpholin-4-yl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-benzoxazole
—— N-(1,3-benzodioxol-5-yl)-3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide —— C18H14FN3O4
N-(1,3-benzodioxol-5-yl)-3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide