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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]-2-(thiophen-2-ylmethylsulfanyl)acetamide —— C20H22N4OS2
N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]-2-(thiophen-2-ylmethylsulfanyl)acetamide
—— [2-[Methyl(thiophen-2-ylmethyl)amino]-2-oxoethyl] 3,5-dimethyl-1-phenylpyrazole-4-carboxylate —— C20H21N3O3S
[2-[Methyl(thiophen-2-ylmethyl)amino]-2-oxoethyl] 3,5-dimethyl-1-phenylpyrazole-4-carboxylate
—— [2-[Furan-2-ylmethyl(methyl)amino]-2-oxoethyl] 3,5-dimethyl-1-phenylpyrazole-4-carboxylate —— C20H21N3O4
[2-[Furan-2-ylmethyl(methyl)amino]-2-oxoethyl] 3,5-dimethyl-1-phenylpyrazole-4-carboxylate
—— N-[4-[[(17S)-15-methyl-13-phenyl-17-(3,4,5-trimethoxyphenyl)-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-yl]amino]phenyl]acetamide —— C36H33N7O4
N-[4-[[(17S)-15-methyl-13-phenyl-17-(3,4,5-trimethoxyphenyl)-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-yl]amino]phenyl]acetamide
—— [2-(2-fluoro-4-methylanilino)-2-oxoethyl] (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate —— C23H22FN3O3
[2-(2-fluoro-4-methylanilino)-2-oxoethyl] (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate
—— N-[[4-(morpholine-4-carbonyl)cyclohexyl]methyl]pyrazolo[1,5-b]pyridazine-3-carboxamide —— C19H25N5O3
N-[[4-(morpholine-4-carbonyl)cyclohexyl]methyl]pyrazolo[1,5-b]pyridazine-3-carboxamide
—— N-[[4-(2-methylpropylcarbamoyl)cyclohexyl]methyl]pyrazolo[1,5-b]pyridazine-3-carboxamide —— C19H27N5O2
N-[[4-(2-methylpropylcarbamoyl)cyclohexyl]methyl]pyrazolo[1,5-b]pyridazine-3-carboxamide
—— [2-(2,6-Difluoroanilino)-2-oxoethyl] 3,5-dimethyl-1-phenylpyrazole-4-carboxylate —— C20H17F2N3O3
[2-(2,6-Difluoroanilino)-2-oxoethyl] 3,5-dimethyl-1-phenylpyrazole-4-carboxylate
—— 2-(5-methyl-4H-imidazol-2-yl)ethanamine —— C6H11N3
2-(5-methyl-4H-imidazol-2-yl)ethanamine
—— [2-[[(1R)-1-cyano-1-cyclopropylethyl]amino]-2-oxoethyl] (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate —— C22H24N4O3
[2-[[(1R)-1-cyano-1-cyclopropylethyl]amino]-2-oxoethyl] (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate
—— [2-(2-Acetylhydrazinyl)-2-oxoethyl] 1-benzyl-5-chloro-3-methylpyrazole-4-carboxylate —— C16H17ClN4O4
[2-(2-Acetylhydrazinyl)-2-oxoethyl] 1-benzyl-5-chloro-3-methylpyrazole-4-carboxylate
—— N-[[4-(cyclohexylcarbamoyl)cyclohexyl]methyl]-2-phenylpyrazolo[1,5-b]pyridazine-3-carboxamide —— C27H33N5O2
N-[[4-(cyclohexylcarbamoyl)cyclohexyl]methyl]-2-phenylpyrazolo[1,5-b]pyridazine-3-carboxamide
—— [(2S)-1-oxo-1-piperidin-1-ylpropan-2-yl] 3,5-dimethyl-1-phenylpyrazole-4-carboxylate —— C20H25N3O3
[(2S)-1-oxo-1-piperidin-1-ylpropan-2-yl] 3,5-dimethyl-1-phenylpyrazole-4-carboxylate
—— N-[[4-(furan-2-ylmethylcarbamoyl)cyclohexyl]methyl]-2-phenylpyrazolo[1,5-b]pyridazine-3-carboxamide —— C26H27N5O3
N-[[4-(furan-2-ylmethylcarbamoyl)cyclohexyl]methyl]-2-phenylpyrazolo[1,5-b]pyridazine-3-carboxamide
—— (17S)-N-(4-bromophenyl)-17-[4-(dimethylamino)phenyl]-15-methyl-13-(2-methylphenyl)-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C34H30BrN7
(17S)-N-(4-bromophenyl)-17-[4-(dimethylamino)phenyl]-15-methyl-13-(2-methylphenyl)-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— (17R)-N-(4-bromophenyl)-17-[4-(dimethylamino)phenyl]-15-methyl-13-(2-methylphenyl)-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C34H30BrN7
(17R)-N-(4-bromophenyl)-17-[4-(dimethylamino)phenyl]-15-methyl-13-(2-methylphenyl)-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— N-[[4-(benzylcarbamoyl)cyclohexyl]methyl]pyrazolo[1,5-b]pyridazine-3-carboxamide —— C22H25N5O2
N-[[4-(benzylcarbamoyl)cyclohexyl]methyl]pyrazolo[1,5-b]pyridazine-3-carboxamide
—— 2-phenyl-N-[[4-(pyrrolidine-1-carbonyl)cyclohexyl]methyl]pyrazolo[1,5-b]pyridazine-3-carboxamide —— C25H29N5O2
2-phenyl-N-[[4-(pyrrolidine-1-carbonyl)cyclohexyl]methyl]pyrazolo[1,5-b]pyridazine-3-carboxamide
—— N-[[4-[(4-fluorophenyl)carbamoyl]cyclohexyl]methyl]-2-phenylpyrazolo[1,5-b]pyridazine-3-carboxamide —— C27H26FN5O2
N-[[4-[(4-fluorophenyl)carbamoyl]cyclohexyl]methyl]-2-phenylpyrazolo[1,5-b]pyridazine-3-carboxamide
—— N-[[4-(2,3-dihydroindole-1-carbonyl)cyclohexyl]methyl]-2-phenylpyrazolo[1,5-b]pyridazine-3-carboxamide —— C29H29N5O2
N-[[4-(2,3-dihydroindole-1-carbonyl)cyclohexyl]methyl]-2-phenylpyrazolo[1,5-b]pyridazine-3-carboxamide
—— 2-(2,4-dimethylphenyl)-5-methyl-N-pentan-3-yltriazole-4-carboxamide —— C17H24N4O
2-(2,4-dimethylphenyl)-5-methyl-N-pentan-3-yltriazole-4-carboxamide
—— 2-phenyl-N-[[4-(propan-2-ylcarbamoyl)cyclohexyl]methyl]pyrazolo[1,5-b]pyridazine-3-carboxamide —— C24H29N5O2
2-phenyl-N-[[4-(propan-2-ylcarbamoyl)cyclohexyl]methyl]pyrazolo[1,5-b]pyridazine-3-carboxamide
—— (17S)-N-(4-bromophenyl)-15-methyl-17-(3-nitrophenyl)-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C31H22BrN7O2
(17S)-N-(4-bromophenyl)-15-methyl-17-(3-nitrophenyl)-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— methyl 4-[(17S)-15-methyl-13-phenyl-9-[3-(trifluoromethyl)anilino]-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-17-yl]benzoate —— C34H25F3N6O2
methyl 4-[(17S)-15-methyl-13-phenyl-9-[3-(trifluoromethyl)anilino]-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-17-yl]benzoate
—— [2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl] (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate —— C21H25N3O4
[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl] (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate
—— 7-oxo-2-phenyl-N-[[4-(piperidine-1-carbonyl)cyclohexyl]methyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H31N5O3
7-oxo-2-phenyl-N-[[4-(piperidine-1-carbonyl)cyclohexyl]methyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— N-[[4-(pyrrolidine-1-carbonyl)cyclohexyl]methyl]pyrazolo[1,5-b]pyridazine-3-carboxamide —— C19H25N5O2
N-[[4-(pyrrolidine-1-carbonyl)cyclohexyl]methyl]pyrazolo[1,5-b]pyridazine-3-carboxamide
—— [(2R)-1-oxo-1-(prop-2-enylamino)propan-2-yl] 3-(3-methylphenyl)-1-phenylpyrazole-4-carboxylate —— C23H23N3O3
[(2R)-1-oxo-1-(prop-2-enylamino)propan-2-yl] 3-(3-methylphenyl)-1-phenylpyrazole-4-carboxylate
—— [(2S)-1-oxo-1-piperidin-1-ylpropan-2-yl] (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate —— C22H27N3O3
[(2S)-1-oxo-1-piperidin-1-ylpropan-2-yl] (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate
—— [2-[2-(cyclohexen-1-yl)ethylamino]-2-oxoethyl] (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate —— C24H29N3O3
[2-[2-(cyclohexen-1-yl)ethylamino]-2-oxoethyl] (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate
—— N-[[4-[(3,4-difluorophenyl)carbamoyl]cyclohexyl]methyl]-2-phenylpyrazolo[1,5-b]pyridazine-3-carboxamide —— C27H25F2N5O2
N-[[4-[(3,4-difluorophenyl)carbamoyl]cyclohexyl]methyl]-2-phenylpyrazolo[1,5-b]pyridazine-3-carboxamide
—— 7-oxo-2-phenyl-N-[[4-(propan-2-ylcarbamoyl)cyclohexyl]methyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C24H29N5O3
7-oxo-2-phenyl-N-[[4-(propan-2-ylcarbamoyl)cyclohexyl]methyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 2-(2-methylphenyl)-N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]acetamide —— C22H24N4O
2-(2-methylphenyl)-N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]acetamide
—— (5-methyl-4H-imidazol-2-yl)methanamine —— C5H9N3
(5-methyl-4H-imidazol-2-yl)methanamine
—— methyl 4-[(17R)-15-methyl-13-phenyl-9-[3-(trifluoromethyl)anilino]-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-17-yl]benzoate —— C34H25F3N6O2
methyl 4-[(17R)-15-methyl-13-phenyl-9-[3-(trifluoromethyl)anilino]-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-17-yl]benzoate
—— [2-oxo-2-[[(1S)-1-thiophen-2-ylethyl]amino]ethyl] (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate —— C22H23N3O3S
[2-oxo-2-[[(1S)-1-thiophen-2-ylethyl]amino]ethyl] (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate
—— [2-[(3-fluorophenyl)methyl-methylamino]-2-oxoethyl] (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate —— C24H24FN3O3
[2-[(3-fluorophenyl)methyl-methylamino]-2-oxoethyl] (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate
—— 7-oxo-2-phenyl-N-[[4-(pyrrolidine-1-carbonyl)cyclohexyl]methyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H29N5O3
7-oxo-2-phenyl-N-[[4-(pyrrolidine-1-carbonyl)cyclohexyl]methyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 6-bromo-4H-benzimidazol-2-amine —— C7H6BrN3
6-bromo-4H-benzimidazol-2-amine
—— (17R)-N-(1,3-benzodioxol-5-yl)-17-(3,4-dichlorophenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C32H22Cl2N6O2
(17R)-N-(1,3-benzodioxol-5-yl)-17-(3,4-dichlorophenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— 2-bromo-5-methyl-4H-imidazole —— C4H5BrN2
2-bromo-5-methyl-4H-imidazole
—— (3aS)-5-propan-2-yl-3aH-benzimidazol-2-amine —— C10H13N3
(3aS)-5-propan-2-yl-3aH-benzimidazol-2-amine
—— (3aR)-5-propan-2-yl-3aH-benzimidazol-2-amine —— C10H13N3
(3aR)-5-propan-2-yl-3aH-benzimidazol-2-amine
—— [2-(3-Chloro-4-methoxyanilino)-2-oxoethyl] 3,5-dimethyl-1-phenylpyrazole-4-carboxylate —— C21H20ClN3O4
[2-(3-Chloro-4-methoxyanilino)-2-oxoethyl] 3,5-dimethyl-1-phenylpyrazole-4-carboxylate
—— (17S)-N-(1,3-benzodioxol-5-yl)-17-(3,4-dichlorophenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine —— C32H22Cl2N6O2
(17S)-N-(1,3-benzodioxol-5-yl)-17-(3,4-dichlorophenyl)-15-methyl-13-phenyl-1,8,11,13,14-pentazatetracyclo[8.7.0.02,7.012,16]heptadeca-2,4,6,8,10,12(16),14-heptaen-9-amine
—— (4R)-4-(chloromethyl)-5-methyl-4H-imidazole —— C5H7ClN2
(4R)-4-(chloromethyl)-5-methyl-4H-imidazole
—— (2R)-N-(1-cyanocyclohexyl)-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]propanamide —— C18H21N5OS
(2R)-N-(1-cyanocyclohexyl)-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]propanamide
—— 6-fluoro-4H-benzimidazol-2-amine —— C7H6FN3
6-fluoro-4H-benzimidazol-2-amine
—— N-cyclopropyl-2-(2,5-dimethylphenyl)-5-(3,4-dimethylphenyl)pyrazole-3-carboxamide —— C23H25N3O
N-cyclopropyl-2-(2,5-dimethylphenyl)-5-(3,4-dimethylphenyl)pyrazole-3-carboxamide
—— ethyl 2-[2-[[2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]acetyl]amino]-1,3-thiazol-4-yl]acetate —— C17H17N5O3S2
ethyl 2-[2-[[2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]acetyl]amino]-1,3-thiazol-4-yl]acetate