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中文名称 英文名称 CAS号 化学式 结构式图片
—— (4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C33H41N5O4S
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— ethyl (2S)-2-(4-methyl-1,3-thiazol-2-yl)-3-oxo-4-[1-(2-propan-2-ylphenyl)imidazol-2-yl]sulfanylbutanoate —— C22H25N3O3S2
ethyl (2S)-2-(4-methyl-1,3-thiazol-2-yl)-3-oxo-4-[1-(2-propan-2-ylphenyl)imidazol-2-yl]sulfanylbutanoate
—— ethyl (2R)-4-[1-(2,4-dimethylphenyl)imidazol-2-yl]sulfanyl-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate —— C21H23N3O3S2
ethyl (2R)-4-[1-(2,4-dimethylphenyl)imidazol-2-yl]sulfanyl-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate
—— [2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl] 2-thiophen-2-yl-1,3-thiazole-4-carboxylate —— C16H18N2O4S2
[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl] 2-thiophen-2-yl-1,3-thiazole-4-carboxylate
—— 2-[(6,7-Dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-ium-2-yl)methyl]-4-methyl-5-phenyl-1,2,4-triazole-3-thione —— C21H25N4O2S+
2-[(6,7-Dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-ium-2-yl)methyl]-4-methyl-5-phenyl-1,2,4-triazole-3-thione
—— 2-(Azocan-1-ium-1-ylmethyl)-5-(3-bromophenyl)-4-methyl-1,2,4-triazole-3-thione —— C17H24BrN4S+
2-(Azocan-1-ium-1-ylmethyl)-5-(3-bromophenyl)-4-methyl-1,2,4-triazole-3-thione
—— (2-Morpholin-4-yl-2-oxoethyl) 2-thiophen-2-yl-1,3-thiazole-4-carboxylate —— C14H14N2O4S2
(2-Morpholin-4-yl-2-oxoethyl) 2-thiophen-2-yl-1,3-thiazole-4-carboxylate
—— 2-[(4R)-3-tert-butyl-1-(2-chlorophenyl)-4-(3,4-dimethoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C31H33ClN4O5S
2-[(4R)-3-tert-butyl-1-(2-chlorophenyl)-4-(3,4-dimethoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— [2-[[(2S)-butan-2-yl]amino]-2-oxoethyl] 2-thiophen-2-yl-1,3-thiazole-4-carboxylate —— C14H16N2O3S2
[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl] 2-thiophen-2-yl-1,3-thiazole-4-carboxylate
—— (2S)-2-(5,7-dibromoquinolin-8-yl)oxy-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)propanamide —— C23H20Br2N4O3
(2S)-2-(5,7-dibromoquinolin-8-yl)oxy-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)propanamide
—— 2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C29H22Cl2N4O3S2
2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 5-Methyl-4-(2-methylphenyl)-2-[(4-methylpiperidin-1-ium-1-yl)methyl]-1,2,4-triazole-3-thione —— C17H25N4S+
5-Methyl-4-(2-methylphenyl)-2-[(4-methylpiperidin-1-ium-1-yl)methyl]-1,2,4-triazole-3-thione
—— Methyl 1-[[3-(4-methoxyphenyl)-4-(2-methylpropyl)-5-sulfanylidene-1,2,4-triazol-1-yl]methyl]piperidine-4-carboxylate —— C21H30N4O3S
Methyl 1-[[3-(4-methoxyphenyl)-4-(2-methylpropyl)-5-sulfanylidene-1,2,4-triazol-1-yl]methyl]piperidine-4-carboxylate
—— 4-(2-methoxyethyl)-5-(3-methylphenyl)-2-[(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)methyl]-1,2,4-triazole-3-thione —— C24H28N4OS
4-(2-methoxyethyl)-5-(3-methylphenyl)-2-[(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)methyl]-1,2,4-triazole-3-thione
—— 1-[3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanoyl]-N-phenylpiperidine-4-carboxamide —— C23H23FN4O3
1-[3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanoyl]-N-phenylpiperidine-4-carboxamide
—— 2-[(4S)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-phenylacetamide —— C31H25FN4O2S2
2-[(4S)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-phenylacetamide
—— (5R,7R)-3-chloro-N-[2-(1,2,4-triazol-1-yl)-5-(trifluoromethyl)phenyl]adamantane-1-carboxamide —— C20H20ClF3N4O
(5R,7R)-3-chloro-N-[2-(1,2,4-triazol-1-yl)-5-(trifluoromethyl)phenyl]adamantane-1-carboxamide
—— N-cyclopropyl-2-[(4S)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C31H32N4O4S2
N-cyclopropyl-2-[(4S)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— 2-[(4S)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C33H36N4O5S2
2-[(4S)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-[(4R)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C29H26Cl2N4O3S2
2-[(4R)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— (7S)-2-[(1S)-1-[[4,5-bis(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C27H23Cl2N5OS2
(7S)-2-[(1S)-1-[[4,5-bis(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1R)-1-[[4,5-bis(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C27H23Cl2N5OS2
(7R)-2-[(1R)-1-[[4,5-bis(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— methyl 1-[[5-(4-ethylphenyl)-3-sulfanylidene-1H-1,2,4-triazol-2-yl]methyl]piperidine-4-carboxylate —— C18H24N4O2S
methyl 1-[[5-(4-ethylphenyl)-3-sulfanylidene-1H-1,2,4-triazol-2-yl]methyl]piperidine-4-carboxylate
—— Methyl 1-[[3-(2,4-dimethylphenyl)-2-sulfanylideneimidazol-1-yl]methyl]piperidine-4-carboxylate —— C19H25N3O2S
Methyl 1-[[3-(2,4-dimethylphenyl)-2-sulfanylideneimidazol-1-yl]methyl]piperidine-4-carboxylate
—— 2-(Azocan-1-ium-1-ylmethyl)-4-(2,5-dimethylphenyl)-1,2,4-triazole-3-thione —— C18H27N4S+
2-(Azocan-1-ium-1-ylmethyl)-4-(2,5-dimethylphenyl)-1,2,4-triazole-3-thione
—— 2-(azocan-1-ium-1-ylmethyl)-5-thiophen-2-yl-1H-1,2,4-triazole-3-thione —— C14H21N4S2+
2-(azocan-1-ium-1-ylmethyl)-5-thiophen-2-yl-1H-1,2,4-triazole-3-thione
—— (2-Phenyl-1,3-thiazol-4-yl)methyl 2-thiophen-2-yl-1,3-thiazole-4-carboxylate —— C18H12N2O2S3
(2-Phenyl-1,3-thiazol-4-yl)methyl 2-thiophen-2-yl-1,3-thiazole-4-carboxylate
—— [2-[2-(4-Methoxyphenyl)ethylamino]-2-oxoethyl] 2-thiophen-2-yl-1,3-thiazole-4-carboxylate —— C19H18N2O4S2
[2-[2-(4-Methoxyphenyl)ethylamino]-2-oxoethyl] 2-thiophen-2-yl-1,3-thiazole-4-carboxylate
—— 2-[(4S)-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C36H33FN4O3S
2-[(4S)-1-(2,4-dimethylphenyl)-4-(2-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— (4R)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H28N4O3S2
(4R)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— [2-[(2-Methoxyphenyl)methylamino]-2-oxoethyl] 2-thiophen-2-yl-1,3-thiazole-4-carboxylate —— C18H16N2O4S2
[2-[(2-Methoxyphenyl)methylamino]-2-oxoethyl] 2-thiophen-2-yl-1,3-thiazole-4-carboxylate
—— 2-(Azocan-1-ylmethyl)-4-(2,4-dimethylphenyl)-1,2,4-triazole-3-thione —— C18H26N4S
2-(Azocan-1-ylmethyl)-4-(2,4-dimethylphenyl)-1,2,4-triazole-3-thione
—— (4R)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C28H24Cl2N4O3S2
(4R)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4S)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide —— C28H26F2N4O2S2
2-[(4S)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide
—— 2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C29H26Cl2N4O3S2
2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— (2R)-2-[[5-[4-(diethylamino)phenyl]-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-ethylpropanamide —— C19H29N5OS
(2R)-2-[[5-[4-(diethylamino)phenyl]-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-ethylpropanamide
—— (2-Morpholin-4-yl-2-oxoethyl) 2-(3-chlorophenyl)-4-methyl-1,3-thiazole-5-carboxylate —— C17H17ClN2O4S
(2-Morpholin-4-yl-2-oxoethyl) 2-(3-chlorophenyl)-4-methyl-1,3-thiazole-5-carboxylate
—— 2-[(4R)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C33H36N4O5S2
2-[(4R)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— [5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 2-thiophen-2-yl-1,3-thiazole-4-carboxylate —— C17H10ClN3O3S2
[5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 2-thiophen-2-yl-1,3-thiazole-4-carboxylate
—— 2-[(4S)-3-tert-butyl-1-(2-chlorophenyl)-4-(3,4-dimethoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C31H33ClN4O5S
2-[(4S)-3-tert-butyl-1-(2-chlorophenyl)-4-(3,4-dimethoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— (7S)-2-[(1R)-1-[[4,5-bis(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C27H23Cl2N5OS2
(7S)-2-[(1R)-1-[[4,5-bis(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C27H22Cl2N4O2S2
2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— 2-[(4S)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C33H36N4O5S2
2-[(4S)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-[(4R)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-phenylacetamide —— C31H25FN4O2S2
2-[(4R)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-phenylacetamide
—— (2R)-2-(5,7-dibromoquinolin-8-yl)oxy-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)propanamide —— C23H20Br2N4O3
(2R)-2-(5,7-dibromoquinolin-8-yl)oxy-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)propanamide
—— 2-[(4R)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C29H22Cl2N4O3S2
2-[(4R)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— (4S)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H28N4O3S2
(4S)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C28H24Cl2N4O3S2
(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 6-[[5-[4-(Diethylamino)phenyl]-4-ethyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3,5-triazine-2,4-diamine —— C18H25N9S
6-[[5-[4-(Diethylamino)phenyl]-4-ethyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3,5-triazine-2,4-diamine
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C32H30ClFN4O4S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide