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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-2-chloro-1-[4-[1-(4-fluorophenyl)-3-methyl-6-[(4-methylphenyl)methyl]pyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-1-yl]-2-phenylethanone —— C33H32ClFN6O
(2R)-2-chloro-1-[4-[1-(4-fluorophenyl)-3-methyl-6-[(4-methylphenyl)methyl]pyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-1-yl]-2-phenylethanone
—— (2R)-2-[[5-(4-tert-butylphenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-N,N-dimethylpropanamide —— C18H26N4OS
(2R)-2-[[5-(4-tert-butylphenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-N,N-dimethylpropanamide
—— (2R)-2-[[5-(4-tert-butylphenyl)-4-(2-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(3,5-dimethylphenyl)-2-phenylacetamide —— C34H33ClN4OS
(2R)-2-[[5-(4-tert-butylphenyl)-4-(2-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(3,5-dimethylphenyl)-2-phenylacetamide
—— [(1S)-2-oxo-1-phenyl-2-piperidin-1-ylethyl] 4-(tetrazol-1-yl)benzoate —— C21H21N5O3
[(1S)-2-oxo-1-phenyl-2-piperidin-1-ylethyl] 4-(tetrazol-1-yl)benzoate
—— [2-(6-Amino-1-methyl-2,4-dioxopyrimidin-5-yl)-2-oxoethyl] 1-benzyl-3,5-dimethylpyrazole-4-carboxylate —— C20H21N5O5
[2-(6-Amino-1-methyl-2,4-dioxopyrimidin-5-yl)-2-oxoethyl] 1-benzyl-3,5-dimethylpyrazole-4-carboxylate
—— (2R)-N-(4-acetamidophenyl)-2-[[4-cyclohexyl-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C28H35N5O5S
(2R)-N-(4-acetamidophenyl)-2-[[4-cyclohexyl-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 2-[[5-(4-methoxyphenyl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-pentylacetamide —— C22H26N4O2S
2-[[5-(4-methoxyphenyl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-pentylacetamide
—— (2R)-2-[[4-benzyl-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,3-dihydro-1,4-benzodioxin-6-yl)propanamide —— C30H31N5O6S2
(2R)-2-[[4-benzyl-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,3-dihydro-1,4-benzodioxin-6-yl)propanamide
—— (2-phenyl-1,3-thiazol-4-yl)methyl (1S,5S)-9-oxobicyclo[3.3.1]nonane-3-carboxylate —— C20H21NO3S
(2-phenyl-1,3-thiazol-4-yl)methyl (1S,5S)-9-oxobicyclo[3.3.1]nonane-3-carboxylate
—— [2-[benzyl-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]-2-oxoethyl] (1S,5S)-9-oxobicyclo[3.3.1]nonane-3-carboxylate —— C28H27ClN2O4S
[2-[benzyl-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]-2-oxoethyl] (1S,5S)-9-oxobicyclo[3.3.1]nonane-3-carboxylate
—— N-[4-[[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]phenyl]acetamide —— C17H14ClN3O2S
N-[4-[[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]phenyl]acetamide
—— [3-(4-Ethylphenyl)-1,2,4-oxadiazol-5-yl]methyl quinoxaline-6-carboxylate —— C20H16N4O3
[3-(4-Ethylphenyl)-1,2,4-oxadiazol-5-yl]methyl quinoxaline-6-carboxylate
—— 2-[(1S)-1-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-5-(4-methylphenyl)-1,3,4-oxadiazole —— C22H23N5O2S
2-[(1S)-1-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-5-(4-methylphenyl)-1,3,4-oxadiazole
—— (2S)-N-(4-acetamidophenyl)-2-[[4-cyclohexyl-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C28H35N5O5S
(2S)-N-(4-acetamidophenyl)-2-[[4-cyclohexyl-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl 4-(tetrazol-1-yl)benzoate —— C18H15ClN4O4
(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl 4-(tetrazol-1-yl)benzoate
—— (1-propyltetrazol-5-yl)methyl 2-[(5S,7R)-3-bromo-1-adamantyl]acetate —— C17H25BrN4O2
(1-propyltetrazol-5-yl)methyl 2-[(5S,7R)-3-bromo-1-adamantyl]acetate
—— (2S)-2-[[4-benzyl-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,3-dihydro-1,4-benzodioxin-6-yl)propanamide —— C30H31N5O6S2
(2S)-2-[[4-benzyl-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,3-dihydro-1,4-benzodioxin-6-yl)propanamide
—— (2-phenyl-1,3-thiazol-4-yl)methyl (1R,5R)-9-oxobicyclo[3.3.1]nonane-3-carboxylate —— C20H21NO3S
(2-phenyl-1,3-thiazol-4-yl)methyl (1R,5R)-9-oxobicyclo[3.3.1]nonane-3-carboxylate
—— (2R)-2-[1-(4-chlorophenyl)imidazol-2-yl]sulfanyl-N-(3-fluorophenyl)propanamide —— C18H15ClFN3OS
(2R)-2-[1-(4-chlorophenyl)imidazol-2-yl]sulfanyl-N-(3-fluorophenyl)propanamide
—— [2-oxo-2-[(4-phenyl-1,3-thiazol-2-yl)-prop-2-enylamino]ethyl] (1R,5R)-9-oxobicyclo[3.3.1]nonane-3-carboxylate —— C24H26N2O4S
[2-oxo-2-[(4-phenyl-1,3-thiazol-2-yl)-prop-2-enylamino]ethyl] (1R,5R)-9-oxobicyclo[3.3.1]nonane-3-carboxylate
—— [2-(4-chlorophenyl)-1,3-thiazol-4-yl]methyl (1S,5S)-9-oxobicyclo[3.3.1]nonane-3-carboxylate —— C20H20ClNO3S
[2-(4-chlorophenyl)-1,3-thiazol-4-yl]methyl (1S,5S)-9-oxobicyclo[3.3.1]nonane-3-carboxylate
—— 2-[(1R)-1-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-5-(4-methylphenyl)-1,3,4-oxadiazole —— C22H23N5O2S
2-[(1R)-1-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-5-(4-methylphenyl)-1,3,4-oxadiazole
—— [2-[benzyl-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]-2-oxoethyl] (1R,5R)-9-oxobicyclo[3.3.1]nonane-3-carboxylate —— C28H27ClN2O4S
[2-[benzyl-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]-2-oxoethyl] (1R,5R)-9-oxobicyclo[3.3.1]nonane-3-carboxylate
—— 6-[[5-(4-Methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3,5-triazine-2,4-diamine —— C16H18N8OS
6-[[5-(4-Methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3,5-triazine-2,4-diamine
—— 2-[[5-(4-methoxyphenyl)-4-(2-methylpropyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2S)-5-methylhexan-2-yl]acetamide —— C22H34N4O2S
2-[[5-(4-methoxyphenyl)-4-(2-methylpropyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2S)-5-methylhexan-2-yl]acetamide
—— [2-oxo-2-[(4-phenyl-1,3-thiazol-2-yl)-prop-2-enylamino]ethyl] (1S,5S)-9-oxobicyclo[3.3.1]nonane-3-carboxylate —— C24H26N2O4S
[2-oxo-2-[(4-phenyl-1,3-thiazol-2-yl)-prop-2-enylamino]ethyl] (1S,5S)-9-oxobicyclo[3.3.1]nonane-3-carboxylate
—— (2S)-2-[(3aS,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]-N-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]propanamide —— C23H26N4O3
(2S)-2-[(3aS,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]-N-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]propanamide
—— (2S)-2-[1-(4-chlorophenyl)imidazol-2-yl]sulfanyl-N-(2-methylpropyl)propanamide —— C16H20ClN3OS
(2S)-2-[1-(4-chlorophenyl)imidazol-2-yl]sulfanyl-N-(2-methylpropyl)propanamide
—— (2R)-2-[[5-(3-chlorophenyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(2,5-dimethylphenyl)propanamide —— C21H23ClN4OS
(2R)-2-[[5-(3-chlorophenyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(2,5-dimethylphenyl)propanamide
—— (2S)-2-[1-(4-chlorophenyl)imidazol-2-yl]sulfanyl-N-(2-ethoxyphenyl)propanamide —— C20H20ClN3O2S
(2S)-2-[1-(4-chlorophenyl)imidazol-2-yl]sulfanyl-N-(2-ethoxyphenyl)propanamide
—— (2S)-N-(1,3-benzodioxol-5-yl)-2-[[4-[(4-fluorophenyl)methyl]-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C29H28FN5O6S2
(2S)-N-(1,3-benzodioxol-5-yl)-2-[[4-[(4-fluorophenyl)methyl]-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 2-[5-(2-chlorophenyl)-1,2,4-triazol-1-yl]-N-methyl-N-[(2-methylphenyl)methyl]acetamide —— C19H19ClN4O
2-[5-(2-chlorophenyl)-1,2,4-triazol-1-yl]-N-methyl-N-[(2-methylphenyl)methyl]acetamide
—— (2R)-2-[1-(4-chlorophenyl)imidazol-2-yl]sulfanyl-N-[(4-fluorophenyl)methyl]propanamide —— C19H17ClFN3OS
(2R)-2-[1-(4-chlorophenyl)imidazol-2-yl]sulfanyl-N-[(4-fluorophenyl)methyl]propanamide
—— 4-chloro-N-[[3-ethyl-5-(4-fluorophenoxy)-1-phenylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide —— C30H29ClFN3O3
4-chloro-N-[[3-ethyl-5-(4-fluorophenoxy)-1-phenylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide
—— (2R)-2-[1-(4-chlorophenyl)imidazol-2-yl]sulfanyl-N-[(4-methylphenyl)methyl]propanamide —— C20H20ClN3OS
(2R)-2-[1-(4-chlorophenyl)imidazol-2-yl]sulfanyl-N-[(4-methylphenyl)methyl]propanamide
—— (2S)-2-[1-(4-chlorophenyl)imidazol-2-yl]sulfanyl-N-[(3R)-1,1-dioxothiolan-3-yl]-N-methylpropanamide —— C17H20ClN3O3S2
(2S)-2-[1-(4-chlorophenyl)imidazol-2-yl]sulfanyl-N-[(3R)-1,1-dioxothiolan-3-yl]-N-methylpropanamide
—— (2R)-1-[4-[6-benzyl-1-(4-fluorophenyl)-3-methylpyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-1-yl]-2-chloro-2-phenylethanone —— C32H30ClFN6O
(2R)-1-[4-[6-benzyl-1-(4-fluorophenyl)-3-methylpyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-1-yl]-2-chloro-2-phenylethanone
—— (2S)-2-[(3aS,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]-N-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]propanamide —— C23H26N4O3
(2S)-2-[(3aS,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]-N-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]propanamide
—— 2-[(4S)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C30H29FN4O3S2
2-[(4S)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-[(4S)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C30H25ClN4O3S2
2-[(4S)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— (2S)-1-[4-[6-benzyl-1-(4-fluorophenyl)-3-methylpyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-1-yl]-2-chloro-2-phenylethanone —— C32H30ClFN6O
(2S)-1-[4-[6-benzyl-1-(4-fluorophenyl)-3-methylpyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-1-yl]-2-chloro-2-phenylethanone
—— (2R)-2-[[5-(4-chlorophenyl)-4-(3-methoxypropyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[4-chloro-3-(trifluoromethyl)phenyl]propanamide —— C22H21Cl2F3N4O2S
(2R)-2-[[5-(4-chlorophenyl)-4-(3-methoxypropyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[4-chloro-3-(trifluoromethyl)phenyl]propanamide
—— (2S)-2-[[5-(4-chlorophenyl)-4-(3-methoxypropyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[4-chloro-3-(trifluoromethyl)phenyl]propanamide —— C22H21Cl2F3N4O2S
(2S)-2-[[5-(4-chlorophenyl)-4-(3-methoxypropyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[4-chloro-3-(trifluoromethyl)phenyl]propanamide
—— 4-butoxy-N-[(1S)-1-[5-[(3-methylphenyl)methylsulfanyl]-4-(4-nitrophenyl)-1,2,4-triazol-3-yl]ethyl]benzamide —— C29H31N5O4S
4-butoxy-N-[(1S)-1-[5-[(3-methylphenyl)methylsulfanyl]-4-(4-nitrophenyl)-1,2,4-triazol-3-yl]ethyl]benzamide
—— ethyl 2-[[2-[[5-(4-chlorophenyl)-4-[(2S)-2-methylhexyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]-4-(2-methylpropyl)thiophene-3-carboxylate —— C28H37ClN4O3S2
ethyl 2-[[2-[[5-(4-chlorophenyl)-4-[(2S)-2-methylhexyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]-4-(2-methylpropyl)thiophene-3-carboxylate
—— 2-[5-(2-chlorophenyl)-1,2,4-triazol-1-yl]-N-[(R)-cyclopropyl(phenyl)methyl]acetamide —— C20H19ClN4O
2-[5-(2-chlorophenyl)-1,2,4-triazol-1-yl]-N-[(R)-cyclopropyl(phenyl)methyl]acetamide
—— (2R)-2-[[5-(4-tert-butylphenyl)-4-cyclopentyl-1,2,4-triazol-3-yl]sulfanyl]-N-(3,5-dichlorophenyl)-2-phenylacetamide —— C31H32Cl2N4OS
(2R)-2-[[5-(4-tert-butylphenyl)-4-cyclopentyl-1,2,4-triazol-3-yl]sulfanyl]-N-(3,5-dichlorophenyl)-2-phenylacetamide
—— 4-butoxy-N-[(1R)-1-[5-[(3-methylphenyl)methylsulfanyl]-4-(4-nitrophenyl)-1,2,4-triazol-3-yl]ethyl]benzamide —— C29H31N5O4S
4-butoxy-N-[(1R)-1-[5-[(3-methylphenyl)methylsulfanyl]-4-(4-nitrophenyl)-1,2,4-triazol-3-yl]ethyl]benzamide
—— N-[[3-benzyl-2-[(2-fluorophenyl)methylsulfonyl]imidazol-4-yl]methyl]-3,3-dimethyl-N-[[(2R)-oxolan-2-yl]methyl]butanamide —— C29H36FN3O4S
N-[[3-benzyl-2-[(2-fluorophenyl)methylsulfonyl]imidazol-4-yl]methyl]-3,3-dimethyl-N-[[(2R)-oxolan-2-yl]methyl]butanamide
—— 2-[[4-benzyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[2-[(5E)-2,4-dioxo-5-(pyridin-3-ylmethylidene)-1,3-thiazolidin-3-yl]ethyl]acetamide —— C28H23FN6O3S2
2-[[4-benzyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[2-[(5E)-2,4-dioxo-5-(pyridin-3-ylmethylidene)-1,3-thiazolidin-3-yl]ethyl]acetamide