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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(4S)-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C31H31ClN4O2S
2-[(4S)-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4S)-4-(3-fluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C30H29FN4O3S
2-[(4S)-4-(3-fluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4R)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C30H38N4O4S
2-[(4R)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4S)-1-(2-chlorophenyl)-4-(2,4-difluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C29H25ClF2N4O2S
2-[(4S)-1-(2-chlorophenyl)-4-(2,4-difluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4S)-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C30H28F2N4O2S
2-[(4S)-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4R)-1-(2-chlorophenyl)-4-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C30H29ClN4O2S
2-[(4R)-1-(2-chlorophenyl)-4-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4R)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C30H28F2N4O3S
2-[(4R)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4S)-1-(2-chlorophenyl)-4-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C30H29ClN4O2S
2-[(4S)-1-(2-chlorophenyl)-4-(2-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4R)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C31H31ClN4O4S
2-[(4R)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4S)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C29H26ClFN4O2S
2-[(4S)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4R)-3-(4-chlorophenyl)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C32H33ClN4O5S
2-[(4R)-3-(4-chlorophenyl)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C31H30N4O4S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4S)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C31H31ClN4O4S
2-[(4S)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4R)-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C31H31ClN4O2S
2-[(4R)-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4S)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C30H38N4O4S
2-[(4S)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4R)-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C30H28F2N4O2S
2-[(4R)-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4S)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C27H24ClFN4O2S2
2-[(4S)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4S)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C30H29ClN4O2S
2-[(4S)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— (4S)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C33H34N4O6S
(4S)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[[5-(4-fluorophenyl)tetrazol-2-yl]methyl]-6-methyl-5-[(2S)-2-methylbutyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C20H21FN6OS
2-[[5-(4-fluorophenyl)tetrazol-2-yl]methyl]-6-methyl-5-[(2S)-2-methylbutyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— N-[(Z)-1-(3-fluoro-4-methoxyphenyl)ethylideneamino]-2-morpholin-4-yl-1,3-thiazole-4-carboxamide —— C17H19FN4O3S
N-[(Z)-1-(3-fluoro-4-methoxyphenyl)ethylideneamino]-2-morpholin-4-yl-1,3-thiazole-4-carboxamide
—— 2-(4-chlorophenoxy)-N-[(1S)-1-[5-[(4-fluorophenyl)methylsulfanyl]-4-(4-nitrophenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]acetamide —— C31H25ClFN5O4S
2-(4-chlorophenoxy)-N-[(1S)-1-[5-[(4-fluorophenyl)methylsulfanyl]-4-(4-nitrophenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]acetamide
—— N-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]-5-(2,4-dimethoxyphenyl)-2-ethylpyrazole-3-carboxamide —— C21H27N3O3
N-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]-5-(2,4-dimethoxyphenyl)-2-ethylpyrazole-3-carboxamide
—— 3-(2-ethoxyphenyl)-N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]propanamide —— C24H28N4O2
3-(2-ethoxyphenyl)-N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]propanamide
—— 2-[4-[(Z)-[3-(4-ethoxyphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]iminomethyl]-2-methoxyphenoxy]acetonitrile —— C20H19N5O3S
2-[4-[(Z)-[3-(4-ethoxyphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]iminomethyl]-2-methoxyphenoxy]acetonitrile
—— 2-[(5S,7S)-3-bromo-1-adamantyl]-N-[3-(tetrazol-1-yl)phenyl]acetamide —— C19H22BrN5O
2-[(5S,7S)-3-bromo-1-adamantyl]-N-[3-(tetrazol-1-yl)phenyl]acetamide
—— 2-[[4-amino-5-(2,4-dichlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2S,3S)-2,3-dimethylcyclohexyl]acetamide —— C18H23Cl2N5OS
2-[[4-amino-5-(2,4-dichlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2S,3S)-2,3-dimethylcyclohexyl]acetamide
—— 6,7-dimethoxy-2-[[5-(4-propan-2-ylphenyl)tetrazol-2-yl]methyl]-3H-quinazolin-4-one —— C21H22N6O3
6,7-dimethoxy-2-[[5-(4-propan-2-ylphenyl)tetrazol-2-yl]methyl]-3H-quinazolin-4-one
—— 2-(4-chlorophenoxy)-N-[(1R)-1-[5-[(4-fluorophenyl)methylsulfanyl]-4-(4-nitrophenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]acetamide —— C31H25ClFN5O4S
2-(4-chlorophenoxy)-N-[(1R)-1-[5-[(4-fluorophenyl)methylsulfanyl]-4-(4-nitrophenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]acetamide
—— 3-(3-bromophenyl)-4-[(Z)-(2-chlorophenyl)methylideneamino]-1H-1,2,4-triazole-5-thione —— C15H10BrClN4S
3-(3-bromophenyl)-4-[(Z)-(2-chlorophenyl)methylideneamino]-1H-1,2,4-triazole-5-thione
—— 2-[(5R,7R)-3-bromo-1-adamantyl]-N-[3-(tetrazol-1-yl)phenyl]acetamide —— C19H22BrN5O
2-[(5R,7R)-3-bromo-1-adamantyl]-N-[3-(tetrazol-1-yl)phenyl]acetamide
—— (2R)-N-[(E)-(4-bromophenyl)methylideneamino]-2-[[5-[(naphthalen-1-ylamino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C29H25BrN6OS
(2R)-N-[(E)-(4-bromophenyl)methylideneamino]-2-[[5-[(naphthalen-1-ylamino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 3-(3-bromophenyl)-4-[(Z)-(4-nitrophenyl)methylideneamino]-1H-1,2,4-triazole-5-thione —— C15H10BrN5O2S
3-(3-bromophenyl)-4-[(Z)-(4-nitrophenyl)methylideneamino]-1H-1,2,4-triazole-5-thione
—— 2-[[5-(2-chlorophenyl)tetrazol-2-yl]methyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H15ClN6OS
2-[[5-(2-chlorophenyl)tetrazol-2-yl]methyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 3-(4-ethoxyphenyl)-4-[(Z)-(3-hydroxy-4-methoxyphenyl)methylideneamino]-1H-1,2,4-triazole-5-thione —— C18H18N4O3S
3-(4-ethoxyphenyl)-4-[(Z)-(3-hydroxy-4-methoxyphenyl)methylideneamino]-1H-1,2,4-triazole-5-thione
—— 4-[(2,5-dimethylpyrrol-3-ylidene)methylamino]-3-(4-methylphenyl)-1H-1,2,4-triazole-5-thione —— C16H17N5S
4-[(2,5-dimethylpyrrol-3-ylidene)methylamino]-3-(4-methylphenyl)-1H-1,2,4-triazole-5-thione
—— N-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]-5-(2,4-dimethoxyphenyl)-2-ethylpyrazole-3-carboxamide —— C21H27N3O3
N-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]-5-(2,4-dimethoxyphenyl)-2-ethylpyrazole-3-carboxamide
—— N-[2-[[4-(4-chlorophenyl)-1-(4-methylphenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]thiophene-2-carboxamide —— C28H27ClN4O3S
N-[2-[[4-(4-chlorophenyl)-1-(4-methylphenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]thiophene-2-carboxamide
—— 2-[[5-(2-methylphenyl)tetrazol-2-yl]methyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H18N6OS
2-[[5-(2-methylphenyl)tetrazol-2-yl]methyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— N-[(1R)-1-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[5-(3,4-dimethoxyphenyl)tetrazol-2-yl]acetamide —— C20H27N5O3
N-[(1R)-1-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[5-(3,4-dimethoxyphenyl)tetrazol-2-yl]acetamide
—— 4-[(Z)-[3-(3-bromophenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]iminomethyl]benzoate —— C16H10BrN4O2S-
4-[(Z)-[3-(3-bromophenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]iminomethyl]benzoate
—— 6,7-dimethoxy-2-[[5-(2-methylphenyl)tetrazol-2-yl]methyl]-3H-quinazolin-4-one —— C19H18N6O3
6,7-dimethoxy-2-[[5-(2-methylphenyl)tetrazol-2-yl]methyl]-3H-quinazolin-4-one
—— 2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C29H35ClN4O2S
2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— (1-propyltetrazol-5-yl)methyl (5S,7R)-3-chloroadamantane-1-carboxylate —— C16H23ClN4O2
(1-propyltetrazol-5-yl)methyl (5S,7R)-3-chloroadamantane-1-carboxylate
—— 2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C29H35ClN4O2S
2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 3-(3-bromophenyl)-4-[(Z)-(4-methylsulfanylphenyl)methylideneamino]-1H-1,2,4-triazole-5-thione —— C16H13BrN4S2
3-(3-bromophenyl)-4-[(Z)-(4-methylsulfanylphenyl)methylideneamino]-1H-1,2,4-triazole-5-thione
—— 3-(4-ethoxyphenyl)-4-[(Z)-(4-methylsulfanylphenyl)methylideneamino]-1H-1,2,4-triazole-5-thione —— C18H18N4OS2
3-(4-ethoxyphenyl)-4-[(Z)-(4-methylsulfanylphenyl)methylideneamino]-1H-1,2,4-triazole-5-thione
—— 2-[[5-(4-bromophenyl)tetrazol-2-yl]methyl]-3H-quinazolin-4-one —— C16H11BrN6O
2-[[5-(4-bromophenyl)tetrazol-2-yl]methyl]-3H-quinazolin-4-one
—— 1-[(Z)-(1,3-diphenylpyrazol-4-yl)methylideneamino]-4,6-dimethyl-2-oxopyridine-3-carbonitrile —— C24H19N5O
1-[(Z)-(1,3-diphenylpyrazol-4-yl)methylideneamino]-4,6-dimethyl-2-oxopyridine-3-carbonitrile
—— N-[2-[[4-(4-chlorophenyl)-1-(4-methylphenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]thiophene-2-carboxamide —— C28H27ClN4O3S
N-[2-[[4-(4-chlorophenyl)-1-(4-methylphenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]thiophene-2-carboxamide