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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2,4,6-trimethyl-N-[[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-N-prop-2-enylbenzenesulfonamide —— C22H25N3O3S
2,4,6-trimethyl-N-[[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-N-prop-2-enylbenzenesulfonamide
—— 3-(4-Chlorophenyl)-5-[[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-6-methyl-2-sulfanylidene-[1,3]thiazolo[4,5-d]pyrimidin-7-one —— C21H13ClFN5O2S3
3-(4-Chlorophenyl)-5-[[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-6-methyl-2-sulfanylidene-[1,3]thiazolo[4,5-d]pyrimidin-7-one
—— 3-(3-Methoxyphenyl)-5-(4-propoxyphenyl)-1,2,4-oxadiazole —— C18H18N2O3
3-(3-Methoxyphenyl)-5-(4-propoxyphenyl)-1,2,4-oxadiazole
—— 2,4,6-trimethyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-prop-2-enylbenzenesulfonamide —— C21H23N3O3S
2,4,6-trimethyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-prop-2-enylbenzenesulfonamide
—— 4-methyl-3-[1-[(3R)-oxan-3-yl]tetrazol-5-yl]aniline —— C13H17N5O
4-methyl-3-[1-[(3R)-oxan-3-yl]tetrazol-5-yl]aniline
—— N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C20H26N4O2S
N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— 3-(4-Chlorophenyl)-6-methyl-2-sulfanylidene-5-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methylsulfanyl]-[1,3]thiazolo[4,5-d]pyrimidin-7-one —— C22H13ClF3N5O2S3
3-(4-Chlorophenyl)-6-methyl-2-sulfanylidene-5-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methylsulfanyl]-[1,3]thiazolo[4,5-d]pyrimidin-7-one
—— 2-chloro-5-[1-[(3R)-oxan-3-yl]tetrazol-5-yl]aniline —— C12H14ClN5O
2-chloro-5-[1-[(3R)-oxan-3-yl]tetrazol-5-yl]aniline
—— 5-[[3-(4-Tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-6-methyl-3-(4-methylphenyl)-2-sulfanylidene-[1,3]thiazolo[4,5-d]pyrimidin-7-one —— C26H25N5O2S3
5-[[3-(4-Tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-6-methyl-3-(4-methylphenyl)-2-sulfanylidene-[1,3]thiazolo[4,5-d]pyrimidin-7-one
—— 3-(4-chlorophenyl)-5-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-2-sulfanylidene-6H-[1,3]thiazolo[4,5-d]pyrimidin-7-one —— C21H14ClN5O2S4
3-(4-chlorophenyl)-5-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-2-sulfanylidene-6H-[1,3]thiazolo[4,5-d]pyrimidin-7-one
—— N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(3-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C19H23ClN4OS
N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(3-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— 4-[1-[(3S)-oxan-3-yl]tetrazol-5-yl]aniline —— C12H15N5O
4-[1-[(3S)-oxan-3-yl]tetrazol-5-yl]aniline
—— (2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(3-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C20H25ClN4OS
(2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(3-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (3R)-3-(chloromethyl)-1-(1,2-dimethylimidazol-4-yl)sulfonylpiperidine —— C11H18ClN3O2S
(3R)-3-(chloromethyl)-1-(1,2-dimethylimidazol-4-yl)sulfonylpiperidine
—— 3-(3-Methoxyphenyl)-5-(3-phenylmethoxyphenyl)-1,2,4-oxadiazole —— C22H18N2O3
3-(3-Methoxyphenyl)-5-(3-phenylmethoxyphenyl)-1,2,4-oxadiazole
—— (2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(3-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C20H25ClN4OS
(2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(3-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C20H26N4O2S
N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— (2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(3-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C20H25ClN4OS
(2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(3-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— N-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2,4,6-trimethylbenzenesulfonamide —— C19H21N3O4S
N-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2,4,6-trimethylbenzenesulfonamide
—— 3-(benzyloxy)-N-{[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide —— C24H21N3O3
3-(benzyloxy)-N-{[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
—— N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(3-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C19H23ClN4OS
N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(3-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— (2R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(3-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C20H25ClN4OS
(2R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(3-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (3S)-3-(chloromethyl)-1-(1,2-dimethylimidazol-4-yl)sulfonylpiperidine —— C11H18ClN3O2S
(3S)-3-(chloromethyl)-1-(1,2-dimethylimidazol-4-yl)sulfonylpiperidine
—— 6-(2,3-Dimethylphenyl)-4-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-pyrrolidin-1-yl-[1,3]thiazolo[4,5-d]pyrimidine-5,7-dione —— C27H26N6O3S2
6-(2,3-Dimethylphenyl)-4-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-pyrrolidin-1-yl-[1,3]thiazolo[4,5-d]pyrimidine-5,7-dione
—— 1-[6-[[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-cyclopropylpiperidine-4-carboxamide —— C27H31N7O3S
1-[6-[[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-cyclopropylpiperidine-4-carboxamide
—— (3S)-1-[6-[[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-cyclopropylpiperidine-3-carboxamide —— C27H31N7O3S
(3S)-1-[6-[[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-cyclopropylpiperidine-3-carboxamide
—— 2-[4-(Piperidine-1-carbonyl)piperidin-1-yl]-6-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,3]thiazolo[4,5-d]pyrimidin-7-one —— C26H26F3N7O3S
2-[4-(Piperidine-1-carbonyl)piperidin-1-yl]-6-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,3]thiazolo[4,5-d]pyrimidin-7-one
—— N-cyclopropyl-1-[6-[[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]piperidine-4-carboxamide —— C25H27N7O5S
N-cyclopropyl-1-[6-[[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]piperidine-4-carboxamide
—— N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C20H26N4O2S
N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— (2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C21H28N4O2S
(2R)-N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 7-Methyl-5-[4-(trifluoromethyl)phenyl]-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-c]pyrimidin-3-one —— C23H14F6N6O2
7-Methyl-5-[4-(trifluoromethyl)phenyl]-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-c]pyrimidin-3-one
—— N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C20H26N4O2S
N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— 4-[[3-(4-Tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-6-(2,3-dimethylphenyl)-2-pyrrolidin-1-yl-[1,3]thiazolo[4,5-d]pyrimidine-5,7-dione —— C30H32N6O3S
4-[[3-(4-Tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-6-(2,3-dimethylphenyl)-2-pyrrolidin-1-yl-[1,3]thiazolo[4,5-d]pyrimidine-5,7-dione
—— (3S)-N-cyclopropyl-1-[7-oxo-6-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]piperidine-3-carboxamide —— C24H22F3N7O3S
(3S)-N-cyclopropyl-1-[7-oxo-6-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]piperidine-3-carboxamide
—— 6-[[3-(2,3-Dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]-[1,3]thiazolo[4,5-d]pyrimidin-7-one —— C27H31N7O5S
6-[[3-(2,3-Dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]-[1,3]thiazolo[4,5-d]pyrimidin-7-one
—— (3R)-N-cyclopropyl-1-[7-oxo-6-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]piperidine-3-carboxamide —— C24H22F3N7O3S
(3R)-N-cyclopropyl-1-[7-oxo-6-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]piperidine-3-carboxamide
—— (2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C21H28N4O2S
(2R)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 6-(2,3-Dimethylphenyl)-2-pyrrolidin-1-yl-4-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,3]thiazolo[4,5-d]pyrimidine-5,7-dione —— C27H23F3N6O3S
6-(2,3-Dimethylphenyl)-2-pyrrolidin-1-yl-4-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,3]thiazolo[4,5-d]pyrimidine-5,7-dione
—— N-cyclopropyl-1-[7-oxo-6-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]piperidine-4-carboxamide —— C24H22F3N7O3S
N-cyclopropyl-1-[7-oxo-6-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]piperidine-4-carboxamide
—— (2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C21H28N4O2S
(2R)-N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 4-[[3-(2,3-Dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-6-(2,3-dimethylphenyl)-2-pyrrolidin-1-yl-[1,3]thiazolo[4,5-d]pyrimidine-5,7-dione —— C28H28N6O5S
4-[[3-(2,3-Dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-6-(2,3-dimethylphenyl)-2-pyrrolidin-1-yl-[1,3]thiazolo[4,5-d]pyrimidine-5,7-dione
—— (3R)-N-cyclopropyl-1-[6-[[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]piperidine-3-carboxamide —— C25H27N7O5S
(3R)-N-cyclopropyl-1-[6-[[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]piperidine-3-carboxamide
—— (3R)-1-[6-[[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-cyclopropylpiperidine-3-carboxamide —— C27H31N7O3S
(3R)-1-[6-[[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]-N-cyclopropylpiperidine-3-carboxamide
—— (2R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C21H28N4O2S
(2R)-N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (3S)-N-cyclopropyl-1-[6-[[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]piperidine-3-carboxamide —— C25H27N7O5S
(3S)-N-cyclopropyl-1-[6-[[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-7-oxo-[1,3]thiazolo[4,5-d]pyrimidin-2-yl]piperidine-3-carboxamide
—— N-[(2R)-2-chloropropyl]-1-ethyl-N,2-dimethylimidazole-4-sulfonamide —— C10H18ClN3O2S
N-[(2R)-2-chloropropyl]-1-ethyl-N,2-dimethylimidazole-4-sulfonamide
—— N-[(2S)-2-chloropropyl]-1-ethyl-N,2-dimethylimidazole-4-sulfonamide —— C10H18ClN3O2S
N-[(2S)-2-chloropropyl]-1-ethyl-N,2-dimethylimidazole-4-sulfonamide
—— Ethyl 1-[2-[[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxo-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl]piperidine-4-carboxylate —— C28H29N7O6
Ethyl 1-[2-[[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxo-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl]piperidine-4-carboxylate
—— 8-[(4-Chlorophenyl)methylsulfanyl]-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one —— C22H14ClF3N6O2S
8-[(4-Chlorophenyl)methylsulfanyl]-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrazin-3-one
—— Ethyl 1-[2-[[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxo-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl]piperidine-4-carboxylate —— C30H33N7O4
Ethyl 1-[2-[[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxo-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl]piperidine-4-carboxylate