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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[[2-[[5-(3-chlorophenyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]-methylamino]-N-methylacetamide —— C16H20ClN5O2S
2-[[2-[[5-(3-chlorophenyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]-methylamino]-N-methylacetamide
—— 6-methyl-5-(4-methylphenyl)-2-[(5-phenyltetrazol-2-yl)methyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C22H18N6OS
6-methyl-5-(4-methylphenyl)-2-[(5-phenyltetrazol-2-yl)methyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— 3-[(Z)-[5-chloro-1-(2,5-dimethylphenyl)-3-methylpyrazol-4-yl]methylideneamino]-2-methylthieno[2,3-d]pyrimidin-4-one —— C20H18ClN5OS
3-[(Z)-[5-chloro-1-(2,5-dimethylphenyl)-3-methylpyrazol-4-yl]methylideneamino]-2-methylthieno[2,3-d]pyrimidin-4-one
—— N'-[(2,5-dimethylpyrrol-3-ylidene)methyl]-4-hydroxy-1-phenylpyrazole-3-carbohydrazide —— C17H17N5O2
N'-[(2,5-dimethylpyrrol-3-ylidene)methyl]-4-hydroxy-1-phenylpyrazole-3-carbohydrazide
—— 4-[(Z)-(3,4-difluorophenyl)methylideneamino]-3-(4-ethoxyphenyl)-1H-1,2,4-triazole-5-thione —— C17H14F2N4OS
4-[(Z)-(3,4-difluorophenyl)methylideneamino]-3-(4-ethoxyphenyl)-1H-1,2,4-triazole-5-thione
—— [2-(2-Benzoylhydrazinyl)-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate —— C18H15N5O4
[2-(2-Benzoylhydrazinyl)-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate
—— methyl 2,4-dimethyl-5-[(2S)-2-[4-(1,2,4-triazol-1-yl)benzoyl]oxypropanoyl]-1H-pyrrole-3-carboxylate —— C20H20N4O5
methyl 2,4-dimethyl-5-[(2S)-2-[4-(1,2,4-triazol-1-yl)benzoyl]oxypropanoyl]-1H-pyrrole-3-carboxylate
—— [2-(1,3-Benzodioxol-5-ylmethylamino)-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate —— C19H16N4O5
[2-(1,3-Benzodioxol-5-ylmethylamino)-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate
—— 2-(4-Chlorophenoxy)ethyl 4-(1,2,4-triazol-1-yl)benzoate —— C17H14ClN3O3
2-(4-Chlorophenoxy)ethyl 4-(1,2,4-triazol-1-yl)benzoate
—— [(2S)-1-[(5-chloropyridin-2-yl)amino]-1-oxopropan-2-yl] 4-(1,2,4-triazol-1-yl)benzoate —— C17H14ClN5O3
[(2S)-1-[(5-chloropyridin-2-yl)amino]-1-oxopropan-2-yl] 4-(1,2,4-triazol-1-yl)benzoate
—— [2-(5-Methylthiophen-2-yl)-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate —— C16H13N3O3S
[2-(5-Methylthiophen-2-yl)-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate
—— 2-[[5-(4-chlorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-1-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethanone —— C25H33ClN4O2S
2-[[5-(4-chlorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-1-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethanone
—— [3-(4-Propan-2-ylphenyl)-1,2,4-oxadiazol-5-yl]methyl 4-(1,2,4-triazol-1-yl)benzoate —— C21H19N5O3
[3-(4-Propan-2-ylphenyl)-1,2,4-oxadiazol-5-yl]methyl 4-(1,2,4-triazol-1-yl)benzoate
—— [(2R)-1-(2-cyanoanilino)-1-oxopropan-2-yl] 4-(1,2,4-triazol-1-yl)benzoate —— C19H15N5O3
[(2R)-1-(2-cyanoanilino)-1-oxopropan-2-yl] 4-(1,2,4-triazol-1-yl)benzoate
—— [2-[methyl-[(1S)-1-phenylethyl]amino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate —— C20H20N4O3
[2-[methyl-[(1S)-1-phenylethyl]amino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate
—— [5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-(1,2,4-triazol-1-yl)benzoate —— C18H12ClN5O3
[5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-(1,2,4-triazol-1-yl)benzoate
—— [(2R)-1-oxo-1-[[(2S)-2-phenylbutyl]amino]propan-2-yl] 4-(1,2,4-triazol-1-yl)benzoate —— C22H24N4O3
[(2R)-1-oxo-1-[[(2S)-2-phenylbutyl]amino]propan-2-yl] 4-(1,2,4-triazol-1-yl)benzoate
—— (2S)-2-[[5-[(naphthalen-1-ylamino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(E)-naphthalen-1-ylmethylideneamino]propanamide —— C33H28N6OS
(2S)-2-[[5-[(naphthalen-1-ylamino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(E)-naphthalen-1-ylmethylideneamino]propanamide
—— N-[(1R)-1-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]-2-(4-methoxyphenyl)acetamide —— C19H18ClN3O3
N-[(1R)-1-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]-2-(4-methoxyphenyl)acetamide
—— (2S)-N-[(E)-(4-bromophenyl)methylideneamino]-2-[[5-[(naphthalen-1-ylamino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C29H25BrN6OS
(2S)-N-[(E)-(4-bromophenyl)methylideneamino]-2-[[5-[(naphthalen-1-ylamino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— [2-[[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]amino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate —— C21H20N4O5
[2-[[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]amino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate
—— [(2S)-1-oxo-1-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]amino]propan-2-yl] 4-(1,2,4-triazol-1-yl)benzoate —— C22H22N4O3
[(2S)-1-oxo-1-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]amino]propan-2-yl] 4-(1,2,4-triazol-1-yl)benzoate
—— (2S)-N-[(E)-(3-bromophenyl)methylideneamino]-2-[[5-[(naphthalen-1-ylamino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C29H25BrN6OS
(2S)-N-[(E)-(3-bromophenyl)methylideneamino]-2-[[5-[(naphthalen-1-ylamino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— N-[(1R)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[5-(3,4-dimethoxyphenyl)tetrazol-2-yl]acetamide —— C20H27N5O3
N-[(1R)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[5-(3,4-dimethoxyphenyl)tetrazol-2-yl]acetamide
—— (2R)-N-[(E)-(4-methoxyphenyl)methylideneamino]-2-[[5-[(naphthalen-1-ylamino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C30H28N6O2S
(2R)-N-[(E)-(4-methoxyphenyl)methylideneamino]-2-[[5-[(naphthalen-1-ylamino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (2S)-2-[[5-[(4-chloro-2-methylanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(E)-(2-methoxyphenyl)methylideneamino]propanamide —— C27H27ClN6O2S
(2S)-2-[[5-[(4-chloro-2-methylanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(E)-(2-methoxyphenyl)methylideneamino]propanamide
—— 2-[[4-amino-5-(2,4-dichlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2S,3R)-2,3-dimethylcyclohexyl]acetamide —— C18H23Cl2N5OS
2-[[4-amino-5-(2,4-dichlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2S,3R)-2,3-dimethylcyclohexyl]acetamide
—— N-[(1R)-1-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl]pyridine-2-carboxamide —— C17H16N4O3
N-[(1R)-1-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl]pyridine-2-carboxamide
—— N-[(1S)-1-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]-3,5-dimethoxybenzamide —— C19H18ClN3O4
N-[(1S)-1-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]-3,5-dimethoxybenzamide
—— (2R)-2-[[5-[(4-chloro-2-methylanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(E)-(2-methoxyphenyl)methylideneamino]propanamide —— C27H27ClN6O2S
(2R)-2-[[5-[(4-chloro-2-methylanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(E)-(2-methoxyphenyl)methylideneamino]propanamide
—— N-[(1R)-1-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]-3,5-dimethoxybenzamide —— C19H18ClN3O4
N-[(1R)-1-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]-3,5-dimethoxybenzamide
—— 1-[(Z)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-4,6-dimethyl-2-oxopyridine-3-carbonitrile —— C19H16ClN5O
1-[(Z)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-4,6-dimethyl-2-oxopyridine-3-carbonitrile
—— (5S,7S)-3-chloro-N-(3-imidazol-1-ylphenyl)adamantane-1-carboxamide —— C20H22ClN3O
(5S,7S)-3-chloro-N-(3-imidazol-1-ylphenyl)adamantane-1-carboxamide
—— [2-[[(1R)-1-(2-chlorophenyl)ethyl]amino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate —— C19H17ClN4O3
[2-[[(1R)-1-(2-chlorophenyl)ethyl]amino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate
—— [(E)-3-phenylprop-2-enyl] 4-(1,2,4-triazol-1-yl)benzoate —— C18H15N3O2
[(E)-3-phenylprop-2-enyl] 4-(1,2,4-triazol-1-yl)benzoate
—— N'-[2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]-3-phenyl-1H-pyrazole-5-carbohydrazide —— C19H22N4O2
N'-[2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]-3-phenyl-1H-pyrazole-5-carbohydrazide
—— 2-[[4-amino-5-(2,4-dichlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]acetamide —— C18H23Cl2N5OS
2-[[4-amino-5-(2,4-dichlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]acetamide
—— 2-[[4-amino-5-(2,4-dichlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S,2S,3R)-2,3-dimethylcyclohexyl]acetamide —— C18H23Cl2N5OS
2-[[4-amino-5-(2,4-dichlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S,2S,3R)-2,3-dimethylcyclohexyl]acetamide
—— (2R)-N-[(E)-(5-bromo-2-methoxyphenyl)methylideneamino]-2-[[5-[(4-methylanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C27H27BrN6O2S
(2R)-N-[(E)-(5-bromo-2-methoxyphenyl)methylideneamino]-2-[[5-[(4-methylanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 2-[[5-(4-chlorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-1-[(1R,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethanone —— C25H33ClN4O2S
2-[[5-(4-chlorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-1-[(1R,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethanone
—— 2-[(4R)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C31H25F2N5O2S2
2-[(4R)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— (2R)-2-[[5-[(naphthalen-1-ylamino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(E)-naphthalen-1-ylmethylideneamino]propanamide —— C33H28N6OS
(2R)-2-[[5-[(naphthalen-1-ylamino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(E)-naphthalen-1-ylmethylideneamino]propanamide
—— 2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C30H23Cl2N5O2S2
2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— [2-[[(1R)-1-(3-chlorophenyl)ethyl]amino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate —— C19H17ClN4O3
[2-[[(1R)-1-(3-chlorophenyl)ethyl]amino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate
—— [2-[N-(cyanomethyl)anilino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate —— C19H15N5O3
[2-[N-(cyanomethyl)anilino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate
—— 2-[(4S)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C31H25F2N5O2S2
2-[(4S)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— [(2R)-1-oxo-1-[[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]amino]propan-2-yl] 4-(1,2,4-triazol-1-yl)benzoate —— C22H22N4O3
[(2R)-1-oxo-1-[[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]amino]propan-2-yl] 4-(1,2,4-triazol-1-yl)benzoate
—— [2-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methylamino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate —— C20H18N4O5
[2-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methylamino]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate
—— N-[(1S)-1-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl]pyridine-2-carboxamide —— C17H16N4O3
N-[(1S)-1-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl]pyridine-2-carboxamide
—— 2-[(4S)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C31H25F2N5O2S2
2-[(4S)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide