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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-(4-Fluorophenyl)-5-[(1-methyltetrazol-5-yl)sulfanylmethyl]-1,2,4-oxadiazole —— C11H9FN6OS
3-(4-Fluorophenyl)-5-[(1-methyltetrazol-5-yl)sulfanylmethyl]-1,2,4-oxadiazole
—— 3-[(E)-2-(1-benzyl-3-phenylpyrazol-4-yl)ethenyl]-1H-quinoxalin-2-one —— C26H20N4O
3-[(E)-2-(1-benzyl-3-phenylpyrazol-4-yl)ethenyl]-1H-quinoxalin-2-one
—— N-(2-methyl-6-propan-2-ylphenyl)-2-[(4-pyrazol-1-ylphenyl)methylsulfanyl]acetamide —— C22H25N3OS
N-(2-methyl-6-propan-2-ylphenyl)-2-[(4-pyrazol-1-ylphenyl)methylsulfanyl]acetamide
—— N-phenyl-2-[(4-pyrazol-1-ylphenyl)methylsulfanyl]acetamide —— C18H17N3OS
N-phenyl-2-[(4-pyrazol-1-ylphenyl)methylsulfanyl]acetamide
—— 3-[(E)-2-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]ethenyl]-1H-quinoxalin-2-one —— C21H17FN4O
3-[(E)-2-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]ethenyl]-1H-quinoxalin-2-one
—— 2-[(5S)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-5-[(5-phenyl-1,3-oxazol-2-yl)methylsulfanyl]-1,3,4-oxadiazole —— C21H19N3O2S2
2-[(5S)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-5-[(5-phenyl-1,3-oxazol-2-yl)methylsulfanyl]-1,3,4-oxadiazole
—— 3-[(E)-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)ethenyl]-1H-quinoxalin-2-one —— C21H18N4O
3-[(E)-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)ethenyl]-1H-quinoxalin-2-one
—— [3-(4-Fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl 2,3-dimethylbenzoate —— C18H15FN2O3
[3-(4-Fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl 2,3-dimethylbenzoate
—— (4Z,5R)-5-(3-chlorophenyl)-1-[3-(dimethylamino)propyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]pyrrolidine-2,3-dione —— C26H27ClN4O3
(4Z,5R)-5-(3-chlorophenyl)-1-[3-(dimethylamino)propyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]pyrrolidine-2,3-dione
—— Methyl 4-[(5-phenyl-1,3-oxazol-2-yl)methoxy]benzoate —— C18H15NO4
Methyl 4-[(5-phenyl-1,3-oxazol-2-yl)methoxy]benzoate
—— 3-[(E)-2-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)ethenyl]-1H-quinoxalin-2-one —— C20H15ClN4O
3-[(E)-2-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)ethenyl]-1H-quinoxalin-2-one
—— 2-[(4S)-3-tert-butyl-1-(2-chlorophenyl)-4-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C27H30ClFN4O3S
2-[(4S)-3-tert-butyl-1-(2-chlorophenyl)-4-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— 5-[2-(2-methoxyethylsulfamoyl)-4-nitrophenoxy]-1-(4-methoxyphenyl)-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C26H31N5O9S
5-[2-(2-methoxyethylsulfamoyl)-4-nitrophenoxy]-1-(4-methoxyphenyl)-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 5,6-dimethyl-2-[(1R)-1-(1-methyl-5-phenylimidazol-2-yl)sulfanylethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C20H20N4OS2
5,6-dimethyl-2-[(1R)-1-(1-methyl-5-phenylimidazol-2-yl)sulfanylethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— 5-(4-methoxyphenyl)-3-[[1-[[(2S)-oxolan-2-yl]methyl]-5-pyrrolidin-1-ylsulfonylbenzimidazol-2-yl]sulfanylmethyl]-1,2,4-oxadiazole —— C26H29N5O5S2
5-(4-methoxyphenyl)-3-[[1-[[(2S)-oxolan-2-yl]methyl]-5-pyrrolidin-1-ylsulfonylbenzimidazol-2-yl]sulfanylmethyl]-1,2,4-oxadiazole
—— 4-methyl-5-[4-nitro-2-(propylsulfamoyl)phenoxy]-N-[[(2R)-oxolan-2-yl]methyl]-1-phenylpyrazole-3-carboxamide —— C25H29N5O7S
4-methyl-5-[4-nitro-2-(propylsulfamoyl)phenoxy]-N-[[(2R)-oxolan-2-yl]methyl]-1-phenylpyrazole-3-carboxamide
—— 2-[(4R)-3-tert-butyl-1-(2-chlorophenyl)-4-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C28H32ClFN4O3S
2-[(4R)-3-tert-butyl-1-(2-chlorophenyl)-4-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— (4Z,5R)-4-[hydroxy(phenyl)methylidene]-1-(3-imidazol-1-ylpropyl)-5-thiophen-2-ylpyrrolidine-2,3-dione —— C21H19N3O3S
(4Z,5R)-4-[hydroxy(phenyl)methylidene]-1-(3-imidazol-1-ylpropyl)-5-thiophen-2-ylpyrrolidine-2,3-dione
—— 4-methyl-5-[4-nitro-2-(propylsulfamoyl)phenoxy]-N-[[(2S)-oxolan-2-yl]methyl]-1-phenylpyrazole-3-carboxamide —— C25H29N5O7S
4-methyl-5-[4-nitro-2-(propylsulfamoyl)phenoxy]-N-[[(2S)-oxolan-2-yl]methyl]-1-phenylpyrazole-3-carboxamide
—— 2-[(4S)-3-tert-butyl-1-(2-chlorophenyl)-4-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C28H32ClFN4O3S
2-[(4S)-3-tert-butyl-1-(2-chlorophenyl)-4-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— 5-[2-(2-methoxyethylsulfamoyl)-4-nitrophenoxy]-4-methyl-1-(4-methylphenyl)-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C26H31N5O8S
5-[2-(2-methoxyethylsulfamoyl)-4-nitrophenoxy]-4-methyl-1-(4-methylphenyl)-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 1-(3-fluorophenyl)-4-methyl-5-[4-nitro-2-(propylsulfamoyl)phenoxy]-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C25H28FN5O7S
1-(3-fluorophenyl)-4-methyl-5-[4-nitro-2-(propylsulfamoyl)phenoxy]-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 5-[2-(2-methoxyethylsulfamoyl)-4-nitrophenoxy]-4-methyl-1-(4-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C26H31N5O8S
5-[2-(2-methoxyethylsulfamoyl)-4-nitrophenoxy]-4-methyl-1-(4-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 2-[(4R)-3-tert-butyl-1-(2-chlorophenyl)-4-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C27H30ClFN4O3S
2-[(4R)-3-tert-butyl-1-(2-chlorophenyl)-4-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— 1-(4-methoxyphenyl)-4-methyl-5-[4-nitro-2-(propylsulfamoyl)phenoxy]-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C26H31N5O8S
1-(4-methoxyphenyl)-4-methyl-5-[4-nitro-2-(propylsulfamoyl)phenoxy]-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 5-(4-methoxyphenyl)-3-[[1-[[(2R)-oxolan-2-yl]methyl]-5-pyrrolidin-1-ylsulfonylbenzimidazol-2-yl]sulfanylmethyl]-1,2,4-oxadiazole —— C26H29N5O5S2
5-(4-methoxyphenyl)-3-[[1-[[(2R)-oxolan-2-yl]methyl]-5-pyrrolidin-1-ylsulfonylbenzimidazol-2-yl]sulfanylmethyl]-1,2,4-oxadiazole
—— (4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H27ClN4O2S2
(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H27ClN4O4S2
(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-chloro-N-[[1-(4-chlorophenyl)-3-methyl-5-phenoxypyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide —— C29H27Cl2N3O3
2-chloro-N-[[1-(4-chlorophenyl)-3-methyl-5-phenoxypyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide
—— 2-[(4S)-3-(4-chlorophenyl)-4-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C32H31ClN4O5S
2-[(4S)-3-(4-chlorophenyl)-4-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— 2-chloro-N-[[1-(4-chlorophenyl)-3-methyl-5-phenoxypyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide —— C29H27Cl2N3O3
2-chloro-N-[[1-(4-chlorophenyl)-3-methyl-5-phenoxypyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide
—— (4S)-3-(4-chlorophenyl)-4-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C33H33ClN4O5S
(4S)-3-(4-chlorophenyl)-4-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-3-(4-chlorophenyl)-4-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C32H31ClN4O5S
2-[(4R)-3-(4-chlorophenyl)-4-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— (4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H27ClN4O2S2
(4R)-3-(4-chlorophenyl)-1-(4-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H27ClN4O4S2
(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— [3-(4-Fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl 3-fluorobenzoate —— C16H10F2N2O3
[3-(4-Fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl 3-fluorobenzoate
—— 4-pyrazol-1-yl-N-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]benzamide —— C20H25N3O
4-pyrazol-1-yl-N-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]benzamide
—— (2R)-2-[[5-(4-chlorophenyl)-4-(2-ethoxyethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-ethoxyphenyl)-2-phenylacetamide —— C28H29ClN4O3S
(2R)-2-[[5-(4-chlorophenyl)-4-(2-ethoxyethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-ethoxyphenyl)-2-phenylacetamide
—— [3-(2-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 2-(2,4-dichlorophenyl)acetate —— C18H14Cl2N2O4
[3-(2-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 2-(2,4-dichlorophenyl)acetate
—— 2-[(4S)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C31H30F2N4O4S
2-[(4S)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— 5,6-dimethyl-2-[(1S)-1-(1-methyl-5-phenylimidazol-2-yl)sulfanylethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C20H20N4OS2
5,6-dimethyl-2-[(1S)-1-(1-methyl-5-phenylimidazol-2-yl)sulfanylethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— [3-(4-Fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl thiophene-2-carboxylate —— C14H9FN2O3S
[3-(4-Fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl thiophene-2-carboxylate
—— N-[2-(3-fluorophenyl)ethyl]-3-[1-(3-methoxyphenyl)-3,5-dimethylpyrazol-4-yl]propanamide —— C23H26FN3O2
N-[2-(3-fluorophenyl)ethyl]-3-[1-(3-methoxyphenyl)-3,5-dimethylpyrazol-4-yl]propanamide
—— (2R)-2-[[4-amino-5-(2-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,4-difluorophenyl)propanamide —— C17H14ClF2N5OS
(2R)-2-[[4-amino-5-(2-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,4-difluorophenyl)propanamide
—— 4-pyrazol-1-yl-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]benzamide —— C20H25N3O
4-pyrazol-1-yl-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]benzamide
—— (4Z,5S)-1-[3-(dimethylamino)propyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-phenylpyrrolidine-2,3-dione —— C26H28N4O3
(4Z,5S)-1-[3-(dimethylamino)propyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-phenylpyrrolidine-2,3-dione
—— ethyl 2-[(2R,3Z)-2-(furan-2-yl)-3-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C24H22N2O7S
ethyl 2-[(2R,3Z)-2-(furan-2-yl)-3-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— (4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(3,4-dimethoxyphenyl)-1-methyl-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H33N5O5S
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(3,4-dimethoxyphenyl)-1-methyl-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (2R)-2-[(3-oxo-4-phenyl-4,5,7,9-tetrazatricyclo[7.5.0.02,6]tetradeca-1,5,7-trien-8-yl)sulfanyl]-N-[3-(trifluoromethyl)phenyl]propanamide —— C26H24F3N5O2S
(2R)-2-[(3-oxo-4-phenyl-4,5,7,9-tetrazatricyclo[7.5.0.02,6]tetradeca-1,5,7-trien-8-yl)sulfanyl]-N-[3-(trifluoromethyl)phenyl]propanamide
—— ethyl 2-[(2S,3Z)-2-(furan-2-yl)-3-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C24H22N2O7S
ethyl 2-[(2S,3Z)-2-(furan-2-yl)-3-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate