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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(4R)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C30H28F2N4O3S2
2-[(4R)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-(4-chlorophenoxy)-N-[2-[(2S)-2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]-N-(2-methoxyethyl)acetamide —— C26H28Cl2N4O5
2-(4-chlorophenoxy)-N-[2-[(2S)-2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]-N-(2-methoxyethyl)acetamide
—— 2-[(4S)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C28H26F2N4O3S2
2-[(4S)-4-(2,4-difluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— (4S)-4-(2-fluorophenyl)-1-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H27FN4O3S2
(4S)-4-(2-fluorophenyl)-1-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[[4-amino-5-(2,4-dichlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C20H25Cl2N5OS
2-[[4-amino-5-(2,4-dichlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— (4R)-1-(3-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H28N4O3S2
(4R)-1-(3-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C32H30N4O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— N-[(4-fluorophenyl)methyl]-2-[(4R)-4-(4-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C32H26F2N4O2S2
N-[(4-fluorophenyl)methyl]-2-[(4R)-4-(4-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— N-[(4-fluorophenyl)methyl]-2-[(4S)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C32H26F2N4O2S2
N-[(4-fluorophenyl)methyl]-2-[(4S)-4-(2-fluorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— (E)-N-[(1R)-1-cyclopropylethyl]-3-[3-(2-methoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enamide —— C24H25N3O2
(E)-N-[(1R)-1-cyclopropylethyl]-3-[3-(2-methoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enamide
—— 2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C27H24Cl2N4O3S2
2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— N-[(2R)-butan-2-yl]-1-(4-methoxyphenyl)-4-methyl-5-[2-(2-methylpropylsulfamoyl)-4-nitrophenoxy]pyrazole-3-carboxamide —— C26H33N5O7S
N-[(2R)-butan-2-yl]-1-(4-methoxyphenyl)-4-methyl-5-[2-(2-methylpropylsulfamoyl)-4-nitrophenoxy]pyrazole-3-carboxamide
—— 1-[(1R)-1-[5-benzylsulfanyl-4-(4-methylphenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]-3-(4-cyanophenyl)urea —— C32H28N6OS
1-[(1R)-1-[5-benzylsulfanyl-4-(4-methylphenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]-3-(4-cyanophenyl)urea
—— ethyl 4-[[(1S)-1-[5-benzylsulfanyl-4-(4-methylphenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]carbamoylamino]benzoate —— C34H33N5O3S
ethyl 4-[[(1S)-1-[5-benzylsulfanyl-4-(4-methylphenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]carbamoylamino]benzoate
—— (4S)-3-tert-butyl-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C27H32N4O4S2
(4S)-3-tert-butyl-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— [5-(2-chlorophenyl)-2-(3-chlorophenyl)pyrazol-3-yl]-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C26H27Cl2N3O
[5-(2-chlorophenyl)-2-(3-chlorophenyl)pyrazol-3-yl]-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— ethyl 4-[[(1S)-1-[4-(4-methylphenyl)-5-[(3-methylphenyl)methylsulfanyl]-1,2,4-triazol-3-yl]-2-phenylethyl]carbamoylamino]benzoate —— C35H35N5O3S
ethyl 4-[[(1S)-1-[4-(4-methylphenyl)-5-[(3-methylphenyl)methylsulfanyl]-1,2,4-triazol-3-yl]-2-phenylethyl]carbamoylamino]benzoate
—— 1-[(1S)-1-[5-benzylsulfanyl-4-(4-methylphenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]-3-(3-chloro-4-methylphenyl)urea —— C32H30ClN5OS
1-[(1S)-1-[5-benzylsulfanyl-4-(4-methylphenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]-3-(3-chloro-4-methylphenyl)urea
—— 2-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C23H30N4OS
2-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— (4S)-1-(3-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H28N4O3S2
(4S)-1-(3-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— N-cyclopropyl-2-[(4R)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C29H28N4O2S2
N-cyclopropyl-2-[(4R)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— 2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C30H37FN4O3S
2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— N-[[5-(4-chlorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-4-methoxy-N-[[(2S)-oxolan-2-yl]methyl]benzamide —— C30H30ClN3O4
N-[[5-(4-chlorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-4-methoxy-N-[[(2S)-oxolan-2-yl]methyl]benzamide
—— 2-methyl-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]-4-phenyl-1,3-thiazole-5-carboxamide —— C20H27N3OS
2-methyl-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]-4-phenyl-1,3-thiazole-5-carboxamide
—— 1-[(1R)-1-[5-benzylsulfanyl-4-(4-methylphenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]-3-(3,4-dichlorophenyl)urea —— C31H27Cl2N5OS
1-[(1R)-1-[5-benzylsulfanyl-4-(4-methylphenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]-3-(3,4-dichlorophenyl)urea
—— ethyl (3S)-1-[2-[7-methyl-6-[5-methyl-1-(4-methylphenyl)pyrazol-3-yl]-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C28H31N5O4S
ethyl (3S)-1-[2-[7-methyl-6-[5-methyl-1-(4-methylphenyl)pyrazol-3-yl]-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate
—— (4R)-3-tert-butyl-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C27H32N4O4S2
(4R)-3-tert-butyl-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— N-[(1R)-1-[5-benzylsulfanyl-4-(4-nitrophenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]-3,5-dichlorobenzamide —— C30H23Cl2N5O3S
N-[(1R)-1-[5-benzylsulfanyl-4-(4-nitrophenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]-3,5-dichlorobenzamide
—— N-[3-[(2R)-2-methylpiperidin-1-ium-1-yl]propyl]-2-thiophen-3-yl-1,3-thiazole-4-carboxamide —— C17H24N3OS2+
N-[3-[(2R)-2-methylpiperidin-1-ium-1-yl]propyl]-2-thiophen-3-yl-1,3-thiazole-4-carboxamide
—— 1-[(1S)-1-[5-benzylsulfanyl-4-(4-methylphenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]-3-(3-cyanophenyl)urea —— C32H28N6OS
1-[(1S)-1-[5-benzylsulfanyl-4-(4-methylphenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]-3-(3-cyanophenyl)urea
—— ethyl 1-[3-[[(1S,5S)-9-oxobicyclo[3.3.1]nonane-3-carbonyl]amino]phenyl]pyrazole-3-carboxylate —— C22H25N3O4
ethyl 1-[3-[[(1S,5S)-9-oxobicyclo[3.3.1]nonane-3-carbonyl]amino]phenyl]pyrazole-3-carboxylate
—— ethyl (3R)-1-[2-[7-methyl-6-[5-methyl-1-(4-methylphenyl)pyrazol-3-yl]-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C28H31N5O4S
ethyl (3R)-1-[2-[7-methyl-6-[5-methyl-1-(4-methylphenyl)pyrazol-3-yl]-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate
—— 1-[(1R)-1-[5-benzylsulfanyl-4-(4-methylphenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]-3-(3-cyanophenyl)urea —— C32H28N6OS
1-[(1R)-1-[5-benzylsulfanyl-4-(4-methylphenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]-3-(3-cyanophenyl)urea
—— ethyl 1-[3-[[(1R,5R)-9-oxobicyclo[3.3.1]nonane-3-carbonyl]amino]phenyl]pyrazole-3-carboxylate —— C22H25N3O4
ethyl 1-[3-[[(1R,5R)-9-oxobicyclo[3.3.1]nonane-3-carbonyl]amino]phenyl]pyrazole-3-carboxylate
—— N-[2-(2-fluorophenyl)ethyl]-2-thiophen-3-yl-1,3-thiazole-4-carboxamide —— C16H13FN2OS2
N-[2-(2-fluorophenyl)ethyl]-2-thiophen-3-yl-1,3-thiazole-4-carboxamide
—— 2-[[5-(2-bromophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C20H25BrN4OS
2-[[5-(2-bromophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— N-[(1S)-1-[5-benzylsulfanyl-4-(4-nitrophenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]-3,4-dichlorobenzamide —— C30H23Cl2N5O3S
N-[(1S)-1-[5-benzylsulfanyl-4-(4-nitrophenyl)-1,2,4-triazol-3-yl]-2-phenylethyl]-3,4-dichlorobenzamide
—— 2-[[5-(2-bromophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C20H25BrN4OS
2-[[5-(2-bromophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— 2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]-N-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C20H26N4OS
2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]-N-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— N-[4-[[(1S)-1-[4-(4-methylphenyl)-5-[(2-methylphenyl)methylsulfanyl]-1,2,4-triazol-3-yl]ethyl]sulfamoyl]phenyl]acetamide —— C27H29N5O3S2
N-[4-[[(1S)-1-[4-(4-methylphenyl)-5-[(2-methylphenyl)methylsulfanyl]-1,2,4-triazol-3-yl]ethyl]sulfamoyl]phenyl]acetamide
—— 2-(4-chlorophenoxy)-N-[2-[(2R)-2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]-N-(2-methoxyethyl)acetamide —— C26H28Cl2N4O5
2-(4-chlorophenoxy)-N-[2-[(2R)-2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]-N-(2-methoxyethyl)acetamide
—— N-[[5-(4-chlorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-4-methoxy-N-[[(2R)-oxolan-2-yl]methyl]benzamide —— C30H30ClN3O4
N-[[5-(4-chlorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-4-methoxy-N-[[(2R)-oxolan-2-yl]methyl]benzamide
—— 2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C20H26N4OS
2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— [5-(2-chlorophenyl)-2-(3-chlorophenyl)pyrazol-3-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C26H27Cl2N3O
[5-(2-chlorophenyl)-2-(3-chlorophenyl)pyrazol-3-yl]-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— 2-methyl-N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-4-phenyl-1,3-thiazole-5-carboxamide —— C20H27N3OS
2-methyl-N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-4-phenyl-1,3-thiazole-5-carboxamide
—— [4-[(3-Fluoro-4-methoxyphenyl)methyl]piperazin-4-ium-1-yl]-(2-thiophen-3-yl-1,3-thiazol-4-yl)methanone —— C20H21FN3O2S2+
[4-[(3-Fluoro-4-methoxyphenyl)methyl]piperazin-4-ium-1-yl]-(2-thiophen-3-yl-1,3-thiazol-4-yl)methanone
—— 2-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanyl]-N-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C23H30N4OS
2-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanyl]-N-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— 2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C22H31N5O2S
2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— (4R)-4-(2-chlorophenyl)-1-(4-fluorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C30H26ClFN4O3S
(4R)-4-(2-chlorophenyl)-1-(4-fluorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4S)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide —— C29H30N4O3S2
2-[(4S)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide