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中文名称 英文名称 CAS号 化学式 结构式图片
—— (4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(4-fluorophenyl)-1-(4-methoxyphenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C33H32FN5O4S
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(4-fluorophenyl)-1-(4-methoxyphenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— methyl (2R)-2-[[5-(3-morpholin-4-ylsulfonylphenyl)-4-[3-(trifluoromethyl)phenyl]-1,2,4-triazol-3-yl]sulfanyl]propanoate —— C23H23F3N4O5S2
methyl (2R)-2-[[5-(3-morpholin-4-ylsulfonylphenyl)-4-[3-(trifluoromethyl)phenyl]-1,2,4-triazol-3-yl]sulfanyl]propanoate
—— 2-[4-(5-acetyl-4-methyl-1,3-thiazol-2-yl)phenoxy]-N-pentan-3-ylacetamide —— C19H24N2O3S
2-[4-(5-acetyl-4-methyl-1,3-thiazol-2-yl)phenoxy]-N-pentan-3-ylacetamide
—— 2-[(4R)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide —— C33H36N4O5S
2-[(4R)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide
—— 2-[[5-[3-(diethylsulfamoyl)phenyl]-4-(2-phenylethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S,2R)-2-methylcyclohexyl]acetamide —— C29H39N5O3S2
2-[[5-[3-(diethylsulfamoyl)phenyl]-4-(2-phenylethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S,2R)-2-methylcyclohexyl]acetamide
—— methyl (2S)-2-[[5-(3-morpholin-4-ylsulfonylphenyl)-4-[3-(trifluoromethyl)phenyl]-1,2,4-triazol-3-yl]sulfanyl]propanoate —— C23H23F3N4O5S2
methyl (2S)-2-[[5-(3-morpholin-4-ylsulfonylphenyl)-4-[3-(trifluoromethyl)phenyl]-1,2,4-triazol-3-yl]sulfanyl]propanoate
—— (2S)-2-[[5-(furan-2-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-2-phenyl-N-[3-(trifluoromethyl)phenyl]acetamide —— C27H19F3N4O2S
(2S)-2-[[5-(furan-2-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-2-phenyl-N-[3-(trifluoromethyl)phenyl]acetamide
—— 2-[[5-[3-(diethylsulfamoyl)phenyl]-4-(2-phenylethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S,2S)-2-methylcyclohexyl]acetamide —— C29H39N5O3S2
2-[[5-[3-(diethylsulfamoyl)phenyl]-4-(2-phenylethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S,2S)-2-methylcyclohexyl]acetamide
—— [4-(tetrazol-1-yl)phenyl] 2-(2,3-dihydro-1H-inden-5-yloxy)acetate —— C18H16N4O3
[4-(tetrazol-1-yl)phenyl] 2-(2,3-dihydro-1H-inden-5-yloxy)acetate
—— N-[[2-[(dimethylamino)methyl]phenyl]methyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)propanamide —— C24H30N4O
N-[[2-[(dimethylamino)methyl]phenyl]methyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)propanamide
—— (2R)-2-[[5-(furan-2-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-2-phenyl-N-[3-(trifluoromethyl)phenyl]acetamide —— C27H19F3N4O2S
(2R)-2-[[5-(furan-2-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-2-phenyl-N-[3-(trifluoromethyl)phenyl]acetamide
—— 2-Methyl-4-[[1-(3-methylphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-thiazole —— C13H13N5S2
2-Methyl-4-[[1-(3-methylphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-thiazole
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C34H30N4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— (2R)-2-[[5-(2-methylfuran-3-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-2-phenyl-N-[3-(trifluoromethyl)phenyl]acetamide —— C28H21F3N4O2S
(2R)-2-[[5-(2-methylfuran-3-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-2-phenyl-N-[3-(trifluoromethyl)phenyl]acetamide
—— (2R)-2-[[5-[(4-chloroanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(E)-(4-chlorophenyl)methylideneamino]propanamide —— C25H22Cl2N6OS
(2R)-2-[[5-[(4-chloroanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(E)-(4-chlorophenyl)methylideneamino]propanamide
—— (2S)-2-[[5-[3-(diethylsulfamoyl)phenyl]-4-(2-phenylethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[3-(trifluoromethyl)phenyl]propanamide —— C30H32F3N5O3S2
(2S)-2-[[5-[3-(diethylsulfamoyl)phenyl]-4-(2-phenylethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[3-(trifluoromethyl)phenyl]propanamide
—— (2R)-2-[[4-cyclohexyl-5-(3,4-dimethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,5-dimethylphenyl)-2-phenylacetamide —— C32H36N4O3S
(2R)-2-[[4-cyclohexyl-5-(3,4-dimethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,5-dimethylphenyl)-2-phenylacetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C35H31N5O4S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C34H30N4O5S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— (2S)-2-[[5-(2-methylfuran-3-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-2-phenyl-N-[3-(trifluoromethyl)phenyl]acetamide —— C28H21F3N4O2S
(2S)-2-[[5-(2-methylfuran-3-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-2-phenyl-N-[3-(trifluoromethyl)phenyl]acetamide
—— 1-[(3S)-5-(4-chlorophenyl)-3-(furan-2-yl)-3,4-dihydropyrazol-2-yl]-2-[[5-(2-methylfuran-3-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]ethanone —— C28H22ClN5O3S
1-[(3S)-5-(4-chlorophenyl)-3-(furan-2-yl)-3,4-dihydropyrazol-2-yl]-2-[[5-(2-methylfuran-3-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]ethanone
—— 2-[(4,5-diphenyl-1H-imidazol-2-yl)sulfanyl]-1-[(3R)-3-(furan-2-yl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]ethanone —— C31H26N4O3S
2-[(4,5-diphenyl-1H-imidazol-2-yl)sulfanyl]-1-[(3R)-3-(furan-2-yl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]ethanone
—— 1-[(3R)-5-(4-chlorophenyl)-3-(furan-2-yl)-3,4-dihydropyrazol-2-yl]-2-[[5-(2-methylfuran-3-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]ethanone —— C28H22ClN5O3S
1-[(3R)-5-(4-chlorophenyl)-3-(furan-2-yl)-3,4-dihydropyrazol-2-yl]-2-[[5-(2-methylfuran-3-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]ethanone
—— 2-[[5-(3-nitrophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(E)-[(Z)-3-phenylprop-2-enylidene]amino]acetamide —— C22H20N6O3S
2-[[5-(3-nitrophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(E)-[(Z)-3-phenylprop-2-enylidene]amino]acetamide
—— 2-[[5-[3-(diethylsulfamoyl)phenyl]-4-(2-phenylethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2S)-2-methylcyclohexyl]acetamide —— C29H39N5O3S2
2-[[5-[3-(diethylsulfamoyl)phenyl]-4-(2-phenylethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2S)-2-methylcyclohexyl]acetamide
—— 2-[[5-[3-(diethylsulfamoyl)phenyl]-4-(2-phenylethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R)-2-methylcyclohexyl]acetamide —— C29H39N5O3S2
2-[[5-[3-(diethylsulfamoyl)phenyl]-4-(2-phenylethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R)-2-methylcyclohexyl]acetamide
—— 1-[(3R)-3-(4-methoxyphenyl)-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]ethanone —— C31H27N5O3S
1-[(3R)-3-(4-methoxyphenyl)-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]ethanone
—— (2R)-2-[[5-[3-(diethylsulfamoyl)phenyl]-4-(2-phenylethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[3-(trifluoromethyl)phenyl]propanamide —— C30H32F3N5O3S2
(2R)-2-[[5-[3-(diethylsulfamoyl)phenyl]-4-(2-phenylethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[3-(trifluoromethyl)phenyl]propanamide
—— N-[(Z)-1-(4-aminophenyl)ethylideneamino]-2-[5-[3-(trifluoromethyl)phenyl]tetrazol-2-yl]acetamide —— C18H16F3N7O
N-[(Z)-1-(4-aminophenyl)ethylideneamino]-2-[5-[3-(trifluoromethyl)phenyl]tetrazol-2-yl]acetamide
—— 2-[[5-(3-nitrophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(Z)-[(Z)-3-phenylprop-2-enylidene]amino]acetamide —— C22H20N6O3S
2-[[5-(3-nitrophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(Z)-[(Z)-3-phenylprop-2-enylidene]amino]acetamide
—— 2-[(4,5-diphenyl-1H-imidazol-2-yl)sulfanyl]-1-[(3S)-3-(furan-2-yl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]ethanone —— C31H26N4O3S
2-[(4,5-diphenyl-1H-imidazol-2-yl)sulfanyl]-1-[(3S)-3-(furan-2-yl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]ethanone
—— 1-[(3-bromophenyl)methyl]-4-N-[(Z)-pyridin-4-ylmethylideneamino]-5-N-[(E)-pyridin-4-ylmethylideneamino]imidazole-4,5-dicarboxamide —— C24H19BrN8O2
1-[(3-bromophenyl)methyl]-4-N-[(Z)-pyridin-4-ylmethylideneamino]-5-N-[(E)-pyridin-4-ylmethylideneamino]imidazole-4,5-dicarboxamide
—— (2S)-2-[[5-[(4-chloroanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(E)-(4-chlorophenyl)methylideneamino]propanamide —— C25H22Cl2N6OS
(2S)-2-[[5-[(4-chloroanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(E)-(4-chlorophenyl)methylideneamino]propanamide
—— (2S)-2-[[4-cyclohexyl-5-(3,4-dimethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,5-dimethylphenyl)-2-phenylacetamide —— C32H36N4O3S
(2S)-2-[[4-cyclohexyl-5-(3,4-dimethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,5-dimethylphenyl)-2-phenylacetamide
—— N-[(4-fluorophenyl)methyl]-2-[(4R)-4-(3-methylphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C35H31FN4O2S
N-[(4-fluorophenyl)methyl]-2-[(4R)-4-(3-methylphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— 2-[[4-cyclopentyl-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2S)-4-phenylbutan-2-yl]acetamide —— C29H37N5O4S2
2-[[4-cyclopentyl-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2S)-4-phenylbutan-2-yl]acetamide
—— N-[(4-fluorophenyl)methyl]-2-[(4S)-4-(3-methylphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C35H31FN4O2S
N-[(4-fluorophenyl)methyl]-2-[(4S)-4-(3-methylphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— [(1R,2R,5R)-5-methyl-2-propan-2-ylcyclohexyl] 2-[[4-cyclopentyl-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetate —— C29H42N4O5S2
[(1R,2R,5R)-5-methyl-2-propan-2-ylcyclohexyl] 2-[[4-cyclopentyl-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetate
—— N-butyl-N-[2-[(2R)-2-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]nonanamide —— C28H41ClN4O3
N-butyl-N-[2-[(2R)-2-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]nonanamide
—— ethyl (4S)-6-[[4-cyclopentyl-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C26H34N6O6S2
ethyl (4S)-6-[[4-cyclopentyl-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 2-[(4S)-4-(2,5-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C34H32N4O5S
2-[(4S)-4-(2,5-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 2-[(4S)-1-(2,4-dimethylphenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C35H30F2N4O2S
2-[(4S)-1-(2,4-dimethylphenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C35H31N5O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— (4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-(2-chlorophenyl)-4-(2-fluorophenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C32H29ClFN5O3S
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-(2-chlorophenyl)-4-(2-fluorophenyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[[4-cyclopentyl-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide —— C29H35N5O4S2
2-[[4-cyclopentyl-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide
—— N-[6-(dimethylamino)pyridin-3-yl]-4-ethoxy-1-phenylpyrazole-3-carboxamide —— C19H21N5O2
N-[6-(dimethylamino)pyridin-3-yl]-4-ethoxy-1-phenylpyrazole-3-carboxamide
—— 2-[[4-cyclopentyl-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2R)-4-phenylbutan-2-yl]acetamide —— C29H37N5O4S2
2-[[4-cyclopentyl-5-(3-morpholin-4-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2R)-4-phenylbutan-2-yl]acetamide
—— N-(3-chloro-4-fluorophenyl)-2-[5-(2-methylphenyl)tetrazol-2-yl]acetamide —— C16H13ClFN5O
N-(3-chloro-4-fluorophenyl)-2-[5-(2-methylphenyl)tetrazol-2-yl]acetamide
—— 2-[(4R)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C33H29FN4O2S2
2-[(4R)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 1-[(3S)-3-(4-methoxyphenyl)-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]ethanone —— C31H27N5O3S
1-[(3S)-3-(4-methoxyphenyl)-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]ethanone