中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
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2-[(4R)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[2-(dimethylamino)ethyl]acetamide |
—— |
C32H34ClN5O4S |
|
—— |
2-[(4S)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C32H33ClN4O5S |
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—— |
2-[(4S)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide |
—— |
C31H31ClN4O5S |
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2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide |
—— |
C28H27ClN4O4S2 |
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(4S)-3-(4-chlorophenyl)-4-(2,5-dimethoxyphenyl)-1-(4-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C33H33ClN4O4S |
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(4S)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C32H31ClN4O5S |
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—— |
2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C30H25ClN4O4S2 |
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—— |
2-[(4R)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide |
—— |
C31H29ClN4O4S |
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—— |
2-[(4S)-3-(4-chlorophenyl)-4-(2,5-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide |
—— |
C32H31ClN4O4S |
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—— |
N-[(2R)-butan-2-yl]-2-[(4S)-3-(4-chlorophenyl)-4-(2,5-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C33H35ClN4O4S |
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—— |
2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide |
—— |
C28H25ClN4O3S2 |
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—— |
(4R)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C32H31ClN4O5S |
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—— |
2-[(4S)-4-(4-fluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide |
—— |
C31H31FN4O3S |
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—— |
2-[(4S)-3-(4-chlorophenyl)-4-(2,5-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide |
—— |
C32H33ClN4O5S |
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—— |
(4S)-3-(4-chlorophenyl)-4-(2,5-dimethoxyphenyl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C33H33ClN4O5S |
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—— |
2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide |
—— |
C31H26ClN5O3S2 |
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—— |
2-[(4R)-3-(4-chlorophenyl)-4-(2,5-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide |
—— |
C32H31ClN4O4S |
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—— |
1-(3-fluorophenyl)-4-methyl-5-(4-nitro-2-pyrrolidin-1-ylsulfonylphenoxy)-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide |
—— |
C26H28FN5O7S |
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—— |
2-[(4S)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide |
—— |
C31H29ClN4O4S |
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—— |
2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide |
—— |
C31H26ClN5O3S2 |
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—— |
2-[(4S)-3-(4-chlorophenyl)-4-(2,5-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide |
—— |
C32H33ClN4O4S |
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—— |
2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C30H25ClN4O4S2 |
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—— |
N-[(2R)-butan-2-yl]-1-(3-fluorophenyl)-4-methyl-5-[4-nitro-2-(propan-2-ylsulfamoyl)phenoxy]pyrazole-3-carboxamide |
—— |
C24H28FN5O6S |
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—— |
5-[[(2R)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-ium-1-yl]methyl]-3-(4-chlorophenyl)-1,2,4-oxadiazole |
—— |
C20H18ClN4OS+ |
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—— |
N-[(2S)-butan-2-yl]-1-(3-fluorophenyl)-4-methyl-5-[4-nitro-2-(propan-2-ylsulfamoyl)phenoxy]pyrazole-3-carboxamide |
—— |
C24H28FN5O6S |
|
—— |
4-methyl-5-[4-[[(2S)-2-methylbutanoyl]amino]-2-morpholin-4-ylsulfonylphenoxy]-1-phenylpyrazole-3-carboxylic acid |
—— |
C26H30N4O7S |
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—— |
(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C29H33ClN4O4S |
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—— |
1-(3-fluorophenyl)-4-methyl-5-(4-nitro-2-pyrrolidin-1-ylsulfonylphenoxy)-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide |
—— |
C26H28FN5O7S |
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—— |
2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide |
—— |
C28H33ClN4O3S |
|
—— |
N-cyclopropyl-1-(3-fluorophenyl)-4-methyl-5-(4-nitro-2-pyrrolidin-1-ylsulfonylphenoxy)pyrazole-3-carboxamide |
—— |
C24H24FN5O6S |
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—— |
N-[(2S)-butan-2-yl]-2-[(4S)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C29H29ClN4O2S2 |
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—— |
2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide |
—— |
C28H31ClN4O3S |
|
—— |
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-fluorophenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C32H38FN5O3S |
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—— |
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-(pyridin-3-ylmethyl)pyrazole-3-carboxamide |
—— |
C27H27FN6O6S |
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—— |
4-methyl-1-(4-methylphenyl)-5-[4-[[(3R)-oxolane-3-carbonyl]amino]-2-(2-pyridin-2-ylethylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid |
—— |
C30H31N5O7S |
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—— |
2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C30H30F2N4O3S |
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—— |
2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C30H35ClN4O4S |
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—— |
N-(4-pyrrolidin-1-ylphenyl)-2-[5-[3-(trifluoromethyl)phenyl]tetrazol-2-yl]acetamide |
—— |
C20H19F3N6O |
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—— |
4-methyl-5-[4-[[(2R)-2-methylbutanoyl]amino]-2-morpholin-4-ylsulfonylphenoxy]-1-phenylpyrazole-3-carboxylic acid |
—— |
C26H30N4O7S |
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—— |
N-[(2R)-butan-2-yl]-2-[(4R)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C29H29ClN4O2S2 |
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—— |
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-(cyclopropanecarbonylamino)phenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxylic acid |
—— |
C25H27FN4O6S |
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5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-4-methyl-N-propylpyrazole-3-carboxamide |
—— |
C24H28FN5O6S |
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—— |
1-(3-chlorophenyl)-5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide |
—— |
C25H26ClN5O7S |
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—— |
2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide |
—— |
C28H31ClN4O3S |
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—— |
2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C30H35ClN4O4S |
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—— |
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-N-cyclopropyl-1-(4-fluorophenyl)-4-methylpyrazole-3-carboxamide |
—— |
C24H26FN5O6S |
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—— |
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-N,4-dimethyl-N-propylpyrazole-3-carboxamide |
—— |
C25H30FN5O6S |
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—— |
(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C29H33ClN4O3S |
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—— |
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-(cyclopropanecarbonylamino)phenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxylic acid |
—— |
C25H27FN4O6S |
|
—— |
2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C30H34F2N4O3S |
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