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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(4S)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C28H27FN4O3S2
2-[(4S)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— 3-(4-Methylphenyl)-5-[(5-phenyl-1,2-oxazol-3-yl)methylsulfanyl]-1,2,4-triazol-4-amine —— C19H17N5OS
3-(4-Methylphenyl)-5-[(5-phenyl-1,2-oxazol-3-yl)methylsulfanyl]-1,2,4-triazol-4-amine
—— [2-[[(1R)-1-(furan-2-yl)ethyl]amino]-2-oxoethyl] 4-pyrazol-1-ylbenzoate —— C18H17N3O4
[2-[[(1R)-1-(furan-2-yl)ethyl]amino]-2-oxoethyl] 4-pyrazol-1-ylbenzoate
—— (1R,9S,13E)-13-[(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylidene]-9-methyl-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraen-14-one —— C24H19ClN4O2S
(1R,9S,13E)-13-[(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylidene]-9-methyl-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraen-14-one
—— [2-(2,2-dimethyl-3-oxo-4H-quinoxalin-1-yl)-2-oxoethyl] 5-methyl-2-phenyltriazole-4-carboxylate —— C22H21N5O4
[2-(2,2-dimethyl-3-oxo-4H-quinoxalin-1-yl)-2-oxoethyl] 5-methyl-2-phenyltriazole-4-carboxylate
—— 2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2-methylphenyl)methyl]acetamide —— C19H21N5OS
2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2-methylphenyl)methyl]acetamide
—— [2-[[(1S)-1-(2,5-dimethoxyphenyl)ethyl]amino]-2-oxoethyl] 4-pyrazol-1-ylbenzoate —— C22H23N3O5
[2-[[(1S)-1-(2,5-dimethoxyphenyl)ethyl]amino]-2-oxoethyl] 4-pyrazol-1-ylbenzoate
—— [4-[[6-(1-benzothiophen-2-yl)-2-(4-methoxyphenyl)imidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1S,3R)-3-methoxycyclohexyl]methanone —— C35H38N4O3S
[4-[[6-(1-benzothiophen-2-yl)-2-(4-methoxyphenyl)imidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1S,3R)-3-methoxycyclohexyl]methanone
—— 3-[(1R)-1-[5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-yl]ethyl]sulfanyl-5-(4-methylphenyl)-1,2,4-triazol-4-amine —— C20H20N6O2S
3-[(1R)-1-[5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-yl]ethyl]sulfanyl-5-(4-methylphenyl)-1,2,4-triazol-4-amine
—— [2-[Di(propan-2-yl)amino]-2-oxoethyl] 5-methyl-2-phenyltriazole-4-carboxylate —— C18H24N4O3
[2-[Di(propan-2-yl)amino]-2-oxoethyl] 5-methyl-2-phenyltriazole-4-carboxylate
—— [4-[[6-(1-benzothiophen-2-yl)-2-(4-methoxyphenyl)imidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1R,3R)-3-methoxycyclohexyl]methanone —— C35H38N4O3S
[4-[[6-(1-benzothiophen-2-yl)-2-(4-methoxyphenyl)imidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1R,3R)-3-methoxycyclohexyl]methanone
—— 2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[2-(2-fluorophenyl)ethyl]acetamide —— C19H20FN5OS
2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[2-(2-fluorophenyl)ethyl]acetamide
—— [2-[2-[4-(Difluoromethoxy)phenyl]ethylamino]-2-oxoethyl] 4-pyrazol-1-ylbenzoate —— C21H19F2N3O4
[2-[2-[4-(Difluoromethoxy)phenyl]ethylamino]-2-oxoethyl] 4-pyrazol-1-ylbenzoate
—— [2-Oxo-2-(2-phenylethylamino)ethyl] 5-methyl-2-phenyltriazole-4-carboxylate —— C20H20N4O3
[2-Oxo-2-(2-phenylethylamino)ethyl] 5-methyl-2-phenyltriazole-4-carboxylate
—— 2-[5-(3-chlorophenyl)tetrazol-2-yl]-N-methyl-N-(thiophen-3-ylmethyl)acetamide —— C15H14ClN5OS
2-[5-(3-chlorophenyl)tetrazol-2-yl]-N-methyl-N-(thiophen-3-ylmethyl)acetamide
—— 2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2-fluorophenyl)methyl]-N-methylacetamide —— C19H20FN5OS
2-[[4-amino-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2-fluorophenyl)methyl]-N-methylacetamide
—— N-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]-5-(2-fluoro-4-methoxyphenyl)-2-methylpyrazole-3-carboxamide —— C19H22FN3O2
N-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]-5-(2-fluoro-4-methoxyphenyl)-2-methylpyrazole-3-carboxamide
—— (1-Propyltetrazol-5-yl)methyl 4-pyrazol-1-ylbenzoate —— C15H16N6O2
(1-Propyltetrazol-5-yl)methyl 4-pyrazol-1-ylbenzoate
—— [2-[[(2S)-2-ethylhexyl]amino]-2-oxoethyl] 4-pyrazol-1-ylbenzoate —— C20H27N3O3
[2-[[(2S)-2-ethylhexyl]amino]-2-oxoethyl] 4-pyrazol-1-ylbenzoate
—— [2-(2-Ethyl-6-methylanilino)-2-oxoethyl] 5-methyl-2-phenyltriazole-4-carboxylate —— C21H22N4O3
[2-(2-Ethyl-6-methylanilino)-2-oxoethyl] 5-methyl-2-phenyltriazole-4-carboxylate
—— N-[2-[[4-(4-methoxyphenyl)-1-(4-propan-2-ylphenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]thiophene-2-carboxamide —— C31H34N4O4S
N-[2-[[4-(4-methoxyphenyl)-1-(4-propan-2-ylphenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]thiophene-2-carboxamide
—— 2-[5-(3-chlorophenyl)tetrazol-2-yl]-N-[(4-ethylphenyl)methyl]-N-methylacetamide —— C19H20ClN5O
2-[5-(3-chlorophenyl)tetrazol-2-yl]-N-[(4-ethylphenyl)methyl]-N-methylacetamide
—— [2-[(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-2-oxoethyl] 4-pyrazol-1-ylbenzoate —— C21H25N3O3
[2-[(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-2-oxoethyl] 4-pyrazol-1-ylbenzoate
—— (3Z)-3-[(2R)-2-[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,3,5-tetrahydro-1,5-benzodiazepin-4-ylidene]-6-methylpyran-2,4-dione —— C25H22N4O4
(3Z)-3-[(2R)-2-[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,3,5-tetrahydro-1,5-benzodiazepin-4-ylidene]-6-methylpyran-2,4-dione
—— ethyl (4S)-4-ethyl-6-[(5-methyl-2-phenyltriazole-4-carbonyl)oxymethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H23N5O5
ethyl (4S)-4-ethyl-6-[(5-methyl-2-phenyltriazole-4-carbonyl)oxymethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— [2-[[(1R)-1-cyclopropylethyl]amino]-2-oxoethyl] 4-pyrazol-1-ylbenzoate —— C17H19N3O3
[2-[[(1R)-1-cyclopropylethyl]amino]-2-oxoethyl] 4-pyrazol-1-ylbenzoate
—— (E)-3-(5-ethylthiophen-2-yl)-2-(4-methyl-1,3-thiazol-2-yl)prop-2-enenitrile —— C13H12N2S2
(E)-3-(5-ethylthiophen-2-yl)-2-(4-methyl-1,3-thiazol-2-yl)prop-2-enenitrile
—— [2-(Azocan-1-yl)-2-oxoethyl] 4-pyrazol-1-ylbenzoate —— C19H23N3O3
[2-(Azocan-1-yl)-2-oxoethyl] 4-pyrazol-1-ylbenzoate
—— (E)-3-(5-benzylthiophen-2-yl)-2-(4-methyl-1,3-thiazol-2-yl)prop-2-enenitrile —— C18H14N2S2
(E)-3-(5-benzylthiophen-2-yl)-2-(4-methyl-1,3-thiazol-2-yl)prop-2-enenitrile
—— (3Z)-3-[(2S)-2-[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,3,5-tetrahydro-1,5-benzodiazepin-4-ylidene]-6-methylpyran-2,4-dione —— C25H22N4O4
(3Z)-3-[(2S)-2-[5-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,3,5-tetrahydro-1,5-benzodiazepin-4-ylidene]-6-methylpyran-2,4-dione
—— [4-[[6-(1-benzothiophen-2-yl)-2-(4-methoxyphenyl)imidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1R,3S)-3-methoxycyclohexyl]methanone —— C35H38N4O3S
[4-[[6-(1-benzothiophen-2-yl)-2-(4-methoxyphenyl)imidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1R,3S)-3-methoxycyclohexyl]methanone
—— 3-[[5-(3-Chlorophenyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanylmethyl]-5-phenyl-1,2-oxazole —— C20H17ClN4OS
3-[[5-(3-Chlorophenyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanylmethyl]-5-phenyl-1,2-oxazole
—— [4-[[6-(1-benzothiophen-2-yl)-2-(4-methoxyphenyl)imidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1S,3S)-3-methoxycyclohexyl]methanone —— C35H38N4O3S
[4-[[6-(1-benzothiophen-2-yl)-2-(4-methoxyphenyl)imidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1S,3S)-3-methoxycyclohexyl]methanone
—— 1-(2,3-dimethylphenyl)-4-methyl-5-[4-nitro-2-(propylsulfamoyl)phenoxy]-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C27H33N5O7S
1-(2,3-dimethylphenyl)-4-methyl-5-[4-nitro-2-(propylsulfamoyl)phenoxy]-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 2-methyl-6-[(4S)-3-methyl-5-oxo-1-phenyl-4H-pyrazole-4-carbonyl]pyridine-3-carbonitrile —— C18H14N4O2
2-methyl-6-[(4S)-3-methyl-5-oxo-1-phenyl-4H-pyrazole-4-carbonyl]pyridine-3-carbonitrile
—— 1-(2,3-dimethylphenyl)-4-methyl-5-[4-nitro-2-(propylsulfamoyl)phenoxy]-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C27H33N5O7S
1-(2,3-dimethylphenyl)-4-methyl-5-[4-nitro-2-(propylsulfamoyl)phenoxy]-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 2-methyl-6-[(4R)-3-methyl-5-oxo-1-phenyl-4H-pyrazole-4-carbonyl]pyridine-3-carbonitrile —— C18H14N4O2
2-methyl-6-[(4R)-3-methyl-5-oxo-1-phenyl-4H-pyrazole-4-carbonyl]pyridine-3-carbonitrile
—— 2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C28H27ClN4O3S2
2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4R)-1-(2-chlorophenyl)-4-(2,4-difluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C29H25ClF2N4O2S
2-[(4R)-1-(2-chlorophenyl)-4-(2,4-difluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4S)-4-(2,4-difluorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C31H30F2N4O2S
2-[(4S)-4-(2,4-difluorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4R)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C30H29ClN4O2S
2-[(4R)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C27H24Cl2N4O2S2
2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C29H35ClN4O2S
2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4S)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C30H28F2N4O3S
2-[(4S)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4S)-4-(3,4-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C32H34N4O4S
2-[(4S)-4-(3,4-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4R)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C28H28N4O3S2
2-[(4R)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C31H30N4O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— (4R)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C33H34N4O6S
(4R)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-4-(2,4-difluorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C31H30F2N4O2S
2-[(4R)-4-(2,4-difluorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4R)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C27H24ClFN4O2S2
2-[(4R)-1-(2-chlorophenyl)-4-(4-fluorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide