中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
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2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2-chlorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide |
—— |
C30H25ClN4O4S |
|
—— |
2-[(4S)-3-tert-butyl-4-(3-fluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide |
—— |
C32H32F2N4O2S |
|
—— |
N-[(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methyl]-1-(2,3-dimethoxyphenyl)-N-methylmethanamine |
—— |
C21H24ClN3O2 |
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—— |
2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide |
—— |
C29H35ClN4O3S |
|
—— |
N-[2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-methyl-4-(tetrazol-1-yl)benzamide |
—— |
C18H23N5O |
|
—— |
2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C29H32F2N4O3S |
|
—— |
2-[(4S)-1,4-bis(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide |
—— |
C34H31N5O2S |
|
—— |
(4S)-4-(1,3-benzodioxol-5-yl)-1-(2-chlorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H27ClN4O5S |
|
—— |
5-[[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]sulfonyl]-1H-pyrazole-4-carboxylic acid |
—— |
C10H13N3O4S |
|
—— |
2-[(4S)-1,4-bis(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C33H34N4O3S |
|
—— |
2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide |
—— |
C32H32F2N4O2S |
|
—— |
2-[(4S)-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide |
—— |
C32H34N4O3S |
|
—— |
2-[(4S)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide |
—— |
C33H37N5O5S |
|
—— |
N-[2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-methyl-4-(tetrazol-1-yl)benzamide |
—— |
C18H23N5O |
|
—— |
2-[(4R)-4-(2-methylphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C33H34N4O3S |
|
—— |
2-[(4R)-4-(3,4-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C34H32N4O5S |
|
—— |
2-[(4S)-4-(3,4-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C33H33FN4O5S |
|
—— |
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(2-chlorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide |
—— |
C31H29ClN4O5S |
|
—— |
(4R)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C34H36N4O3S |
|
—— |
2-[(4R)-4-(3,4-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C33H33FN4O5S |
|
—— |
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-1-(4-methylphenyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C29H35N5O3S2 |
|
—— |
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(2-fluorophenyl)-1-(4-methoxyphenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C31H36FN5O4S |
|
—— |
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-1-(4-methylphenyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C29H35N5O3S2 |
|
—— |
2-[(4R)-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide |
—— |
C32H34N4O3S |
|
—— |
2-[(4S)-4-(3,4-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C34H32N4O5S |
|
—— |
2-[(4S)-3-tert-butyl-1,4-bis(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C31H34N4O3S |
|
—— |
2-[(4R)-4-(3,4-dimethoxyphenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C33H33FN4O5S |
|
—— |
2-[(4S)-4-(2-methylphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C33H34N4O3S |
|
—— |
2-[(4R)-3-tert-butyl-1-(4-fluorophenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C30H35FN4O3S |
|
—— |
2-[[5-(4-bromophenyl)-4-(2-methylprop-2-enyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(E)-[(Z)-3-(2-methoxyphenyl)prop-2-enylidene]amino]acetamide |
—— |
C24H24BrN5O2S |
|
—— |
N-(furan-2-ylmethyl)-2-[(4S)-1-(4-methoxyphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide |
—— |
C33H30N4O4S |
|
—— |
2-[(4S)-4-(2-methylphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C33H34N4O3S |
|
—— |
[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl (1S,5S)-9-oxobicyclo[3.3.1]nonane-3-carboxylate |
—— |
C19H19FN2O4 |
|
—— |
1-(2-chlorophenyl)-N-(5-fluoropyridin-2-yl)-5-methyltriazole-4-carboxamide |
—— |
C15H11ClFN5O |
|
—— |
1-(3-fluorophenyl)-4-methyl-5-[4-[[(2S)-2-methylbutanoyl]amino]-2-morpholin-4-ylsulfonylphenoxy]pyrazole-3-carboxylic acid |
—— |
C26H29FN4O7S |
|
—— |
2-[(4R)-4-(3,4-dimethoxyphenyl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide |
—— |
C34H38N4O4S |
|
—— |
2-[(4R)-4-(3,4-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide |
—— |
C35H33N5O4S |
|
—— |
2-[(4S)-3-tert-butyl-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide |
—— |
C30H38N4O6S |
|
—— |
2-[(4R)-3-tert-butyl-1,4-bis(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide |
—— |
C31H34N4O3S |
|
—— |
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-(3-methylbutanoylamino)phenoxy]-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxylic acid |
—— |
C27H34N4O7S |
|
—— |
[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl (1R,5R)-9-oxobicyclo[3.3.1]nonane-3-carboxylate |
—— |
C19H19FN2O4 |
|
—— |
2-[(4R)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C33H34N4O4S |
|
—— |
2-[(4R)-4-(3,4-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C34H36N4O5S |
|
—— |
2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide |
—— |
C29H35ClN4O3S |
|
—— |
1-(3-fluorophenyl)-4-methyl-5-[4-[[(2R)-2-methylbutanoyl]amino]-2-(2-methylpropylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid |
—— |
C26H31FN4O6S |
|
—— |
2-[(4S)-4-(3-fluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide |
—— |
C31H31FN4O3S |
|
—— |
(4R)-4-(3,4-dimethoxyphenyl)-1-(4-fluorophenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one |
—— |
C32H31FN4O4S |
|
—— |
N-[1,4-bis(4-methylphenyl)imidazol-2-yl]-2-[(4-chlorophenyl)sulfonyl-[[(2S)-oxolan-2-yl]methyl]amino]acetamide |
—— |
C30H31ClN4O4S |
|
—— |
2-[(4S)-4-(3,4-dimethoxyphenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide |
—— |
C34H36N4O5S |
|
—— |
2-[(4S)-3-tert-butyl-1-(4-fluorophenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide |
—— |
C30H35FN4O3S |
|