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中文名称 英文名称 CAS号 化学式 结构式图片
—— (4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C28H34N4O3S2
(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-chlorophenyl)-4-methyl-N-propylpyrazole-3-carboxamide —— C24H28ClN5O6S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-chlorophenyl)-4-methyl-N-propylpyrazole-3-carboxamide
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-fluorophenyl)-N-(2-methoxyethyl)-4-methylpyrazole-3-carboxamide —— C24H28FN5O7S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-fluorophenyl)-N-(2-methoxyethyl)-4-methylpyrazole-3-carboxamide
—— 5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]-1-phenylpyrazole-3-carboxamide —— C26H31N5O7S
5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]-1-phenylpyrazole-3-carboxamide
—— 2-[(4R)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C31H31ClN4O3S
2-[(4R)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-methoxyphenyl)-N,4-dimethyl-N-propylpyrazole-3-carboxamide —— C26H33N5O7S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-methoxyphenyl)-N,4-dimethyl-N-propylpyrazole-3-carboxamide
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]-1-phenylpyrazole-3-carboxamide —— C26H31N5O7S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]-1-phenylpyrazole-3-carboxamide
—— 1-[(4-phenyl-1,2,4-triazol-3-yl)methyl]-3-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]urea —— C20H27N5O
1-[(4-phenyl-1,2,4-triazol-3-yl)methyl]-3-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]urea
—— 1-[(4-phenyl-1,2,4-triazol-3-yl)methyl]-3-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]urea —— C20H27N5O
1-[(4-phenyl-1,2,4-triazol-3-yl)methyl]-3-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]urea
—— (4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(3-chlorophenyl)-1-(4-fluorophenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C30H33ClFN5O3S
(4R)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-4-(3-chlorophenyl)-1-(4-fluorophenyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— N-[(2R)-butan-2-yl]-5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxamide —— C25H30FN5O6S
N-[(2R)-butan-2-yl]-5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxamide
—— (4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C28H34N4O3S2
(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-N-cyclopropyl-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxamide —— C25H29N5O7S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-N-cyclopropyl-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxamide
—— 1-(2,5-dimethylphenyl)-N-(2-methoxyethyl)-4-methyl-5-[2-(2-methylpropylsulfamoyl)-4-nitrophenoxy]pyrazole-3-carboxamide —— C26H33N5O7S
1-(2,5-dimethylphenyl)-N-(2-methoxyethyl)-4-methyl-5-[2-(2-methylpropylsulfamoyl)-4-nitrophenoxy]pyrazole-3-carboxamide
—— N-[(2S)-butan-2-yl]-1-(3-chlorophenyl)-4-methyl-5-[2-(2-methylpropylsulfamoyl)-4-nitrophenoxy]pyrazole-3-carboxamide —— C25H30ClN5O6S
N-[(2S)-butan-2-yl]-1-(3-chlorophenyl)-4-methyl-5-[2-(2-methylpropylsulfamoyl)-4-nitrophenoxy]pyrazole-3-carboxamide
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-chlorophenyl)-N-(furan-2-ylmethyl)-4-methylpyrazole-3-carboxamide —— C26H26ClN5O7S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-chlorophenyl)-N-(furan-2-ylmethyl)-4-methylpyrazole-3-carboxamide
—— (4S)-1-tert-butyl-4-(2,4-difluorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C28H30F2N4O3S
(4S)-1-tert-butyl-4-(2,4-difluorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-chlorophenyl)-4-methyl-N-propylpyrazole-3-carboxamide —— C24H28ClN5O6S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-chlorophenyl)-4-methyl-N-propylpyrazole-3-carboxamide
—— 2-[(4S)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide —— C31H30F2N4O3S
2-[(4S)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methylpropyl)acetamide
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-chlorophenyl)-N-(furan-2-ylmethyl)-4-methylpyrazole-3-carboxamide —— C26H26ClN5O7S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-chlorophenyl)-N-(furan-2-ylmethyl)-4-methylpyrazole-3-carboxamide
—— (4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-1-(2,4-dimethylphenyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C30H37N5O3S2
(4S)-8-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-tert-butyl-1-(2,4-dimethylphenyl)-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— N-[(2R)-butan-2-yl]-2-[2-(4-methoxyphenyl)-4-methyl-5-(pyrrolidine-1-carbonyl)pyrazol-3-yl]oxy-5-nitrobenzenesulfonamide —— C26H31N5O7S
N-[(2R)-butan-2-yl]-2-[2-(4-methoxyphenyl)-4-methyl-5-(pyrrolidine-1-carbonyl)pyrazol-3-yl]oxy-5-nitrobenzenesulfonamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C31H30N4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-fluorophenyl)-4-methyl-N-propylpyrazole-3-carboxamide —— C24H28FN5O6S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-fluorophenyl)-4-methyl-N-propylpyrazole-3-carboxamide
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-fluorophenyl)-4-methyl-N-propylpyrazole-3-carboxamide —— C24H28FN5O6S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-fluorophenyl)-4-methyl-N-propylpyrazole-3-carboxamide
—— N-[(2S)-butan-2-yl]-2-[2-(4-methoxyphenyl)-4-methyl-5-(pyrrolidine-1-carbonyl)pyrazol-3-yl]oxy-5-nitrobenzenesulfonamide —— C26H31N5O7S
N-[(2S)-butan-2-yl]-2-[2-(4-methoxyphenyl)-4-methyl-5-(pyrrolidine-1-carbonyl)pyrazol-3-yl]oxy-5-nitrobenzenesulfonamide
—— 2-[(4S)-3-tert-butyl-1-(3-fluorophenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C31H32FN5O2S
2-[(4S)-3-tert-butyl-1-(3-fluorophenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— 2-[(4S)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C31H31ClN4O3S
2-[(4S)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— 1-(2,3-dimethylphenyl)-N-(2-methoxyethyl)-4-methyl-5-[2-(2-methylpropylsulfamoyl)-4-nitrophenoxy]pyrazole-3-carboxamide —— C26H33N5O7S
1-(2,3-dimethylphenyl)-N-(2-methoxyethyl)-4-methyl-5-[2-(2-methylpropylsulfamoyl)-4-nitrophenoxy]pyrazole-3-carboxamide
—— N-[(2S)-butan-2-yl]-5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxamide —— C25H30FN5O6S
N-[(2S)-butan-2-yl]-5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxamide
—— N-[(2S)-butan-2-yl]-5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxamide —— C25H30FN5O6S
N-[(2S)-butan-2-yl]-5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxamide
—— 2-[(4R)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C32H31ClN4O3S
2-[(4R)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— N-[(2R)-butan-2-yl]-1-(3-chlorophenyl)-4-methyl-5-[2-(2-methylpropylsulfamoyl)-4-nitrophenoxy]pyrazole-3-carboxamide —— C25H30ClN5O6S
N-[(2R)-butan-2-yl]-1-(3-chlorophenyl)-4-methyl-5-[2-(2-methylpropylsulfamoyl)-4-nitrophenoxy]pyrazole-3-carboxamide
—— 2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C28H36N4O3S2
2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-N-cyclopropyl-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxamide —— C25H29N5O7S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-N-cyclopropyl-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxamide
—— 5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]-1-phenylpyrazole-3-carboxamide —— C26H31N5O7S
5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]-1-phenylpyrazole-3-carboxamide
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-N-(furan-2-ylmethyl)-4-methyl-1-phenylpyrazole-3-carboxamide —— C26H27N5O7S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-N-(furan-2-ylmethyl)-4-methyl-1-phenylpyrazole-3-carboxamide
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-N-(furan-2-ylmethyl)-4-methylpyrazole-3-carboxamide —— C26H26FN5O7S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(4-fluorophenyl)-N-(furan-2-ylmethyl)-4-methylpyrazole-3-carboxamide
—— N'-ethyl-N'-phenyl-N-(1-phenyltetrazol-5-yl)propane-1,3-diamine —— C18H22N6
N'-ethyl-N'-phenyl-N-(1-phenyltetrazol-5-yl)propane-1,3-diamine
—— (Z)-3-(2-methyl-1,3-thiazol-4-yl)-N-(2-pyridin-2-ylethyl)prop-2-enamide —— C14H15N3OS
(Z)-3-(2-methyl-1,3-thiazol-4-yl)-N-(2-pyridin-2-ylethyl)prop-2-enamide
—— (4S)-1-(4-methoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H32N4O3S2
(4S)-1-(4-methoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C32H31ClN4O3S
2-[(4R)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-fluorophenyl)-N-(furan-2-ylmethyl)-4-methylpyrazole-3-carboxamide —— C26H26FN5O7S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-(3-fluorophenyl)-N-(furan-2-ylmethyl)-4-methylpyrazole-3-carboxamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C31H30N4O5S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]-1-phenylpyrazole-3-carboxamide —— C26H31N5O7S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]-1-phenylpyrazole-3-carboxamide
—— 2-[(4R)-4-(2-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C31H31ClN4O4S
2-[(4R)-4-(2-chlorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— 2-[(4R)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C32H27ClN4O3S
2-[(4R)-4-(3-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— (E)-1-[4-(5,6-dihydro-4H-1,3-thiazin-2-ylamino)phenyl]-3-(1-phenylpyrazol-4-yl)prop-2-en-1-one —— C22H20N4OS
(E)-1-[4-(5,6-dihydro-4H-1,3-thiazin-2-ylamino)phenyl]-3-(1-phenylpyrazol-4-yl)prop-2-en-1-one
—— 2-[(4S)-4-(2-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C33H28ClN5O2S
2-[(4S)-4-(2-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— 2-[(4R)-4-(2-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C33H28ClN5O2S
2-[(4R)-4-(2-chlorophenyl)-1-(4-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide