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中文名称 英文名称 CAS号 化学式 结构式图片
—— [3-(2-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 3-(4-chlorophenyl)sulfanylpropanoate —— C19H17ClN2O4S
[3-(2-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 3-(4-chlorophenyl)sulfanylpropanoate
—— [2-[(6-amino-1-butyl-2,4-dioxopyrimidin-5-yl)-pentylamino]-2-oxoethyl] (Z)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoate —— C28H34ClFN6O5
[2-[(6-amino-1-butyl-2,4-dioxopyrimidin-5-yl)-pentylamino]-2-oxoethyl] (Z)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoate
—— N-(2-(4-chlorophenyl)-5,5-dioxido-4,6-dihydro-2H-thieno[3,4-c]pyrazol-3-yl)-2-ethoxybenzamide —— C20H18ClN3O4S
N-(2-(4-chlorophenyl)-5,5-dioxido-4,6-dihydro-2H-thieno[3,4-c]pyrazol-3-yl)-2-ethoxybenzamide
—— 2-[(4S)-1-(2-chlorophenyl)-4-(2-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C30H28ClFN4O3S
2-[(4S)-1-(2-chlorophenyl)-4-(2-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— 2-(3,5-Dimethylphenyl)-5-[(3-phenyl-1,2,4-oxadiazol-5-yl)methylsulfanyl]-1,3,4-oxadiazole —— C19H16N4O2S
2-(3,5-Dimethylphenyl)-5-[(3-phenyl-1,2,4-oxadiazol-5-yl)methylsulfanyl]-1,3,4-oxadiazole
—— 2-[(4R)-1-(2-chlorophenyl)-4-(2-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C30H28ClFN4O3S
2-[(4R)-1-(2-chlorophenyl)-4-(2-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— 2-[(4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C30H26ClFN4O2S
2-[(4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— [2-(2-chloro-5-morpholin-4-ylsulfonylanilino)-2-oxoethyl] (Z)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]prop-2-enoate —— C26H26ClFN4O6S
[2-(2-chloro-5-morpholin-4-ylsulfonylanilino)-2-oxoethyl] (Z)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]prop-2-enoate
—— (4S)-2-(3-chlorophenyl)-4-[(R)-(2-chlorophenyl)-[2-(3-chlorophenyl)-5-methyl-3-oxo-1H-pyrazol-4-yl]methyl]-5-methyl-4H-pyrazol-3-one —— C27H21Cl3N4O2
(4S)-2-(3-chlorophenyl)-4-[(R)-(2-chlorophenyl)-[2-(3-chlorophenyl)-5-methyl-3-oxo-1H-pyrazol-4-yl]methyl]-5-methyl-4H-pyrazol-3-one
—— N-[4-chloro-3-(dimethylsulfamoyl)phenyl]-2-[[5-[(1S)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C22H26ClFN6O3S2
N-[4-chloro-3-(dimethylsulfamoyl)phenyl]-2-[[5-[(1S)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— (1-phenyltetrazol-5-yl)methyl (5R,7R)-3-chloroadamantane-1-carboxylate —— C19H21ClN4O2
(1-phenyltetrazol-5-yl)methyl (5R,7R)-3-chloroadamantane-1-carboxylate
—— 1-[(1R,4R)-7,7-dimethyl-2-oxo-1-bicyclo[2.2.1]heptanyl]-N-[2-(3,5-dimethylpyrazol-1-yl)phenyl]methanesulfonamide —— C21H27N3O3S
1-[(1R,4R)-7,7-dimethyl-2-oxo-1-bicyclo[2.2.1]heptanyl]-N-[2-(3,5-dimethylpyrazol-1-yl)phenyl]methanesulfonamide
—— (4S)-2-(3-chlorophenyl)-4-[(S)-(2-chlorophenyl)-[2-(3-chlorophenyl)-5-methyl-3-oxo-1H-pyrazol-4-yl]methyl]-5-methyl-4H-pyrazol-3-one —— C27H21Cl3N4O2
(4S)-2-(3-chlorophenyl)-4-[(S)-(2-chlorophenyl)-[2-(3-chlorophenyl)-5-methyl-3-oxo-1H-pyrazol-4-yl]methyl]-5-methyl-4H-pyrazol-3-one
—— (4R)-2-(3-chlorophenyl)-4-[(S)-(2-chlorophenyl)-[2-(3-chlorophenyl)-5-methyl-3-oxo-1H-pyrazol-4-yl]methyl]-5-methyl-4H-pyrazol-3-one —— C27H21Cl3N4O2
(4R)-2-(3-chlorophenyl)-4-[(S)-(2-chlorophenyl)-[2-(3-chlorophenyl)-5-methyl-3-oxo-1H-pyrazol-4-yl]methyl]-5-methyl-4H-pyrazol-3-one
—— (4R)-2-(3-chlorophenyl)-4-[(R)-(2-chlorophenyl)-[2-(3-chlorophenyl)-5-methyl-3-oxo-1H-pyrazol-4-yl]methyl]-5-methyl-4H-pyrazol-3-one —— C27H21Cl3N4O2
(4R)-2-(3-chlorophenyl)-4-[(R)-(2-chlorophenyl)-[2-(3-chlorophenyl)-5-methyl-3-oxo-1H-pyrazol-4-yl]methyl]-5-methyl-4H-pyrazol-3-one
—— 2-[[4-(4-fluorophenyl)-5-[(1R)-1-piperidin-1-ylethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[2-(4-sulfamoylphenyl)ethyl]acetamide —— C25H31FN6O3S2
2-[[4-(4-fluorophenyl)-5-[(1R)-1-piperidin-1-ylethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[2-(4-sulfamoylphenyl)ethyl]acetamide
—— N-[4-chloro-3-(dimethylsulfamoyl)phenyl]-2-[[5-[(1R)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C22H26ClFN6O3S2
N-[4-chloro-3-(dimethylsulfamoyl)phenyl]-2-[[5-[(1R)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— 2-[(4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C31H30ClFN4O3S
2-[(4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— 2-[[4-(4-chlorophenyl)-5-[(1R)-1-piperidin-1-ylethyl]-1,2,4-triazol-3-yl]sulfanyl]-1-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethanone —— C27H38ClN5OS
2-[[4-(4-chlorophenyl)-5-[(1R)-1-piperidin-1-ylethyl]-1,2,4-triazol-3-yl]sulfanyl]-1-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethanone
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C31H31ClN4O3S
2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— N-[(2S)-butan-2-yl]-2-[(4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C31H30ClFN4O2S
N-[(2S)-butan-2-yl]-2-[(4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— 1-[(1S,4S)-7,7-dimethyl-2-oxo-1-bicyclo[2.2.1]heptanyl]-N-[3-(4-ethyl-1,2,4-triazol-3-yl)phenyl]methanesulfonamide —— C20H26N4O3S
1-[(1S,4S)-7,7-dimethyl-2-oxo-1-bicyclo[2.2.1]heptanyl]-N-[3-(4-ethyl-1,2,4-triazol-3-yl)phenyl]methanesulfonamide
—— N-[(1S)-1-(1-adamantyl)ethyl]-1-benzyl-3,5-dimethylpyrazole-4-carboxamide —— C25H33N3O
N-[(1S)-1-(1-adamantyl)ethyl]-1-benzyl-3,5-dimethylpyrazole-4-carboxamide
—— 3-(2-methoxyphenyl)-5-(5H-[1,2,4]triazino[5,6-b]indol-3-ylsulfanylmethyl)-1,2,4-oxadiazole —— C19H14N6O2S
3-(2-methoxyphenyl)-5-(5H-[1,2,4]triazino[5,6-b]indol-3-ylsulfanylmethyl)-1,2,4-oxadiazole
—— 3-(2-morpholin-4-ylethyl)-2-oxo-5-phenyl-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-1-(thiophen-2-ylmethyl)imidazole-4-carboxamide —— C31H34N4O3S
3-(2-morpholin-4-ylethyl)-2-oxo-5-phenyl-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-1-(thiophen-2-ylmethyl)imidazole-4-carboxamide
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C33H33ClN4O4S
2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— (1R,2R,4R)-N-[3-(4-ethyl-1,2,4-triazol-3-yl)phenyl]bicyclo[2.2.1]heptane-2-carboxamide —— C18H22N4O
(1R,2R,4R)-N-[3-(4-ethyl-1,2,4-triazol-3-yl)phenyl]bicyclo[2.2.1]heptane-2-carboxamide
—— 2-[(4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C30H26ClFN4O2S
2-[(4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— 3-(2-morpholin-4-ylethyl)-2-oxo-5-phenyl-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]-1-(thiophen-2-ylmethyl)imidazole-4-carboxamide —— C31H34N4O3S
3-(2-morpholin-4-ylethyl)-2-oxo-5-phenyl-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]-1-(thiophen-2-ylmethyl)imidazole-4-carboxamide
—— 2-[[4-amino-5-(3-bromophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2S)-3-methylbutan-2-yl]acetamide —— C15H20BrN5OS
2-[[4-amino-5-(3-bromophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2S)-3-methylbutan-2-yl]acetamide
—— 1-[(1S,4S)-7,7-dimethyl-2-oxo-1-bicyclo[2.2.1]heptanyl]-N-[2-(3,5-dimethylpyrazol-1-yl)phenyl]methanesulfonamide —— C21H27N3O3S
1-[(1S,4S)-7,7-dimethyl-2-oxo-1-bicyclo[2.2.1]heptanyl]-N-[2-(3,5-dimethylpyrazol-1-yl)phenyl]methanesulfonamide
—— ethyl (4S)-6-[[(Z)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C27H24ClFN4O5
ethyl (4S)-6-[[(Z)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C32H31ClN4O4S
(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[[4-(4-chlorophenyl)-5-[(1S)-1-piperidin-1-ylethyl]-1,2,4-triazol-3-yl]sulfanyl]-1-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethanone —— C27H38ClN5OS
2-[[4-(4-chlorophenyl)-5-[(1S)-1-piperidin-1-ylethyl]-1,2,4-triazol-3-yl]sulfanyl]-1-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethanone
—— N-[(2R)-butan-2-yl]-2-[(4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C31H30ClFN4O2S
N-[(2R)-butan-2-yl]-2-[(4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— [(2S)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] (2S,3R)-1-(4-methylphenyl)-5-oxo-2-thiophen-2-ylpyrrolidine-3-carboxylate —— C30H30N4O5S
[(2S)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] (2S,3R)-1-(4-methylphenyl)-5-oxo-2-thiophen-2-ylpyrrolidine-3-carboxylate
—— [5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 2,5-dimethylfuran-3-carboxylate —— C17H14ClNO4
[5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 2,5-dimethylfuran-3-carboxylate
—— (2S)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]nonan-2-amine —— C14H26N2S
(2S)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]nonan-2-amine
—— 2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C33H33ClN4O4S
2-[(4R)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— N-[2-[[4-amino-5-(3-bromophenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]acetamide —— C12H14BrN5OS
N-[2-[[4-amino-5-(3-bromophenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]acetamide
—— (3aS)-3a-[(Z)-2-[4-[3-(3-chloro-4-methoxyphenyl)-1-phenylpyrazol-4-yl]phenyl]ethenyl]-4,4-dimethyl-1,3-dihydroimidazo[1,2-a]indol-2-one —— C36H31ClN4O2
(3aS)-3a-[(Z)-2-[4-[3-(3-chloro-4-methoxyphenyl)-1-phenylpyrazol-4-yl]phenyl]ethenyl]-4,4-dimethyl-1,3-dihydroimidazo[1,2-a]indol-2-one
—— 2-[(4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C30H28ClFN4O2S
2-[(4R)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C31H30ClFN4O3S
2-[(4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— (4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C32H31ClN4O4S
(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[[4-(4-fluorophenyl)-5-[(1S)-1-piperidin-1-ylethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[2-(4-sulfamoylphenyl)ethyl]acetamide —— C25H31FN6O3S2
2-[[4-(4-fluorophenyl)-5-[(1S)-1-piperidin-1-ylethyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[2-(4-sulfamoylphenyl)ethyl]acetamide
—— [(2S)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] (2R,3S)-1-(4-methylphenyl)-5-oxo-2-thiophen-2-ylpyrrolidine-3-carboxylate —— C30H30N4O5S
[(2S)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] (2R,3S)-1-(4-methylphenyl)-5-oxo-2-thiophen-2-ylpyrrolidine-3-carboxylate
—— N-[(2R)-butan-2-yl]-2-[(4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C31H30ClFN4O2S
N-[(2R)-butan-2-yl]-2-[(4S)-3-(4-chlorophenyl)-4-(4-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— (E)-2-cyano-3-[3-(2-methoxyphenyl)-1-phenylpyrazol-4-yl]-N-prop-2-enylprop-2-enamide —— C23H20N4O2
(E)-2-cyano-3-[3-(2-methoxyphenyl)-1-phenylpyrazol-4-yl]-N-prop-2-enylprop-2-enamide
—— 2-[[4-amino-5-(3-bromophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-propan-2-ylacetamide —— C13H16BrN5OS
2-[[4-amino-5-(3-bromophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-propan-2-ylacetamide
—— 2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C33H33ClN4O4S
2-[(4S)-3-(4-chlorophenyl)-1-(4-methoxyphenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide