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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(4R)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C31H34N4O5S2
2-[(4R)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— 2-(2,5-Dimethylfuran-3-yl)-5-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3,4-oxadiazole —— C18H16FN5O2S
2-(2,5-Dimethylfuran-3-yl)-5-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3,4-oxadiazole
—— (Z)-N-[(4R)-3,4-dihydro-2H-chromen-4-yl]-3-(furan-2-yl)-2-(5-phenyltetrazol-1-yl)prop-2-enamide —— C23H19N5O3
(Z)-N-[(4R)-3,4-dihydro-2H-chromen-4-yl]-3-(furan-2-yl)-2-(5-phenyltetrazol-1-yl)prop-2-enamide
—— 2-[(4S)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide —— C28H27ClN4O2S2
2-[(4S)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide
—— N-[(2R)-butan-2-yl]-2-[(4S)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C29H29ClN4O2S2
N-[(2R)-butan-2-yl]-2-[(4S)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— 2-[(4S)-4-(2-chlorophenyl)-3-(2,6-dimethoxyphenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C33H35ClN4O4S
2-[(4S)-4-(2-chlorophenyl)-3-(2,6-dimethoxyphenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— N-[(2-methoxyphenyl)methyl]-2-[5-(3-methoxyphenyl)tetrazol-2-yl]-N-methylacetamide —— C19H21N5O3
N-[(2-methoxyphenyl)methyl]-2-[5-(3-methoxyphenyl)tetrazol-2-yl]-N-methylacetamide
—— 2-[(4R)-4-(2-chlorophenyl)-3-(2,6-dimethoxyphenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C33H35ClN4O4S
2-[(4R)-4-(2-chlorophenyl)-3-(2,6-dimethoxyphenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— (4S)-4-(3-chlorophenyl)-1-(2-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H27ClN4O2S2
(4S)-4-(3-chlorophenyl)-1-(2-methylphenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 5-[[(1S)-2,2-dichlorocyclopropyl]methylsulfanyl]-1-(2,5-dimethylphenyl)tetrazole —— C13H14Cl2N4S
5-[[(1S)-2,2-dichlorocyclopropyl]methylsulfanyl]-1-(2,5-dimethylphenyl)tetrazole
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2-chlorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C32H25ClN4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2-chlorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 2-[(4S)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C30H29ClN4O3S2
2-[(4S)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-[(4R)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C30H29ClN4O3S2
2-[(4R)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— N-cyclopropyl-2-[(4S)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C31H32N4O4S2
N-cyclopropyl-2-[(4S)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— N-cyclopropyl-2-[(4R)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C31H32N4O4S2
N-cyclopropyl-2-[(4R)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— 2-[(4S)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C30H29ClN4O3S2
2-[(4S)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-[(4R)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C28H25ClN4O2S2
2-[(4R)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— N-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]-5-(3,4-difluorophenyl)-1-ethylpyrazole-3-carboxamide —— C19H21F2N3O
N-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]-5-(3,4-difluorophenyl)-1-ethylpyrazole-3-carboxamide
—— (4S)-4-(3-chlorophenyl)-1-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H27ClN4O3S2
(4S)-4-(3-chlorophenyl)-1-(2-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(2-chlorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C32H25ClN4O5S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(2-chlorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— N-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]-1-ethyl-5-[3-(trifluoromethyl)phenyl]pyrazole-3-carboxamide —— C20H22F3N3O
N-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]-1-ethyl-5-[3-(trifluoromethyl)phenyl]pyrazole-3-carboxamide
—— 2-[(4R)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide —— C28H27ClN4O2S2
2-[(4R)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propan-2-ylacetamide
—— 2-[(4S)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C31H34N4O5S2
2-[(4S)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]acetamide —— C20H20N4O3S
N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]acetamide
—— N-[(2R)-butan-2-yl]-2-[(4R)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C29H29ClN4O2S2
N-[(2R)-butan-2-yl]-2-[(4R)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— N-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]-5-(3,4-difluorophenyl)-1-ethylpyrazole-3-carboxamide —— C19H21F2N3O
N-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]-5-(3,4-difluorophenyl)-1-ethylpyrazole-3-carboxamide
—— 3-(2-Methoxyphenyl)-5-([1,2,4]triazolo[4,3-a]pyridin-3-ylsulfanylmethyl)-1,2,4-oxadiazole —— C16H13N5O2S
3-(2-Methoxyphenyl)-5-([1,2,4]triazolo[4,3-a]pyridin-3-ylsulfanylmethyl)-1,2,4-oxadiazole
—— 3-(4-Fluorophenyl)-5-(7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9,11-tetraen-12-ylsulfanylmethyl)-1,2,4-oxadiazole —— C18H13FN4OS2
3-(4-Fluorophenyl)-5-(7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9,11-tetraen-12-ylsulfanylmethyl)-1,2,4-oxadiazole
—— N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C20H20N4O4S
N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-2-[[5-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— 5-(4-Chlorophenyl)-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylsulfanylmethyl)-1,3-oxazole —— C16H11ClN4OS
5-(4-Chlorophenyl)-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylsulfanylmethyl)-1,3-oxazole
—— (E)-3-(3-methoxy-4-propan-2-yloxyphenyl)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]prop-2-enenitrile —— C22H21N3O3
(E)-3-(3-methoxy-4-propan-2-yloxyphenyl)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]prop-2-enenitrile
—— (E)-3-(4-bromothiophen-2-yl)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]prop-2-enenitrile —— C16H10BrN3OS
(E)-3-(4-bromothiophen-2-yl)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]prop-2-enenitrile
—— (E)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-3-(3-methylthiophen-2-yl)prop-2-enenitrile —— C17H13N3OS
(E)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-3-(3-methylthiophen-2-yl)prop-2-enenitrile
—— (E)-3-[5-(1,3-benzothiazol-2-yl)furan-2-yl]-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]prop-2-enenitrile —— C23H14N4O2S
(E)-3-[5-(1,3-benzothiazol-2-yl)furan-2-yl]-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]prop-2-enenitrile
—— [4-[(E)-2-cyano-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethenyl]-2-methoxyphenyl] cyclopropanecarboxylate —— C23H19N3O4
[4-[(E)-2-cyano-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethenyl]-2-methoxyphenyl] cyclopropanecarboxylate
—— (E)-3-(3-chloro-5-ethoxy-4-methoxyphenyl)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]prop-2-enenitrile —— C21H18ClN3O3
(E)-3-(3-chloro-5-ethoxy-4-methoxyphenyl)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]prop-2-enenitrile
—— (E)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-3-naphthalen-2-ylprop-2-enenitrile —— C22H15N3O
(E)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-3-naphthalen-2-ylprop-2-enenitrile
—— (E)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-3-(3,4,5-trimethoxyphenyl)prop-2-enenitrile —— C21H19N3O4
(E)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-3-(3,4,5-trimethoxyphenyl)prop-2-enenitrile
—— 2-[4-[(E)-2-cyano-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethenyl]-2-methoxyphenoxy]-N-ethylacetamide —— C23H22N4O4
2-[4-[(E)-2-cyano-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethenyl]-2-methoxyphenoxy]-N-ethylacetamide
—— (E)-3-(3-bromophenyl)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]prop-2-enenitrile —— C18H12BrN3O
(E)-3-(3-bromophenyl)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]prop-2-enenitrile
—— (E)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-3-thiophen-3-ylprop-2-enenitrile —— C16H11N3OS
(E)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-3-thiophen-3-ylprop-2-enenitrile
—— 5-[[5-(4-Fluorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanylmethyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C18H14FN5OS2
5-[[5-(4-Fluorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanylmethyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— 3-(4-nitro-phenyl)-2-(<i>p</i>-tolyl-[1,2,4]oxadiazol-5-yl)-acrylonitrile —— C18H12N4O3
3-(4-nitro-phenyl)-2-(<i>p</i>-tolyl-[1,2,4]oxadiazol-5-yl)-acrylonitrile
—— (E)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-3-pyridin-3-ylprop-2-enenitrile —— C17H12N4O
(E)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-3-pyridin-3-ylprop-2-enenitrile
—— (E)-3-(2,3-dimethoxyphenyl)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]prop-2-enenitrile —— C20H17N3O3
(E)-3-(2,3-dimethoxyphenyl)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]prop-2-enenitrile
—— (E)-3-(2-chloro-6-methoxyquinolin-3-yl)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]prop-2-enenitrile —— C22H15ClN4O2
(E)-3-(2-chloro-6-methoxyquinolin-3-yl)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]prop-2-enenitrile
—— 2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C32H31F3N4O3S
2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— (E)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-3-pyridin-4-ylprop-2-enenitrile —— C17H12N4O
(E)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-3-pyridin-4-ylprop-2-enenitrile
—— prop-2-enyl (E)-3-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]-2-cyanoprop-2-enoate —— C16H11ClN2O2S
prop-2-enyl (E)-3-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]-2-cyanoprop-2-enoate
—— 2-[(4S)-4-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-phenylacetamide —— C35H32N4O5S
2-[(4S)-4-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-phenylacetamide