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中文名称 英文名称 CAS号 化学式 结构式图片
—— (1R,2S,4S)-N-(1H-pyrazol-4-ylmethyl)bicyclo[2.2.1]hept-5-ene-2-carboxamide —— C12H15N3O
(1R,2S,4S)-N-(1H-pyrazol-4-ylmethyl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
—— N-[(1S)-1-(furan-2-yl)ethyl]-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]acetamide —— C17H18N4O2S
N-[(1S)-1-(furan-2-yl)ethyl]-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]acetamide
—— N-(2-methoxyethyl)-2-[(4S)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C28H28N4O4S2
N-(2-methoxyethyl)-2-[(4S)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— (1R,2R,4S)-N-(1H-pyrazol-4-ylmethyl)bicyclo[2.2.1]hept-5-ene-2-carboxamide —— C12H15N3O
(1R,2R,4S)-N-(1H-pyrazol-4-ylmethyl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
—— 2-[[5-(furan-2-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-(3-propan-2-yloxypropyl)acetamide —— C20H24N4O3S
2-[[5-(furan-2-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-(3-propan-2-yloxypropyl)acetamide
—— N-(2-methoxyethyl)-2-[(4R)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide —— C28H28N4O4S2
N-(2-methoxyethyl)-2-[(4R)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]acetamide
—— N'-(7-chloro-1,3-benzodioxole-5-carbonyl)-3-phenyl-1H-pyrazole-5-carbohydrazide —— C18H13ClN4O4
N'-(7-chloro-1,3-benzodioxole-5-carbonyl)-3-phenyl-1H-pyrazole-5-carbohydrazide
—— [(2S)-1-(benzylamino)-1-oxopropan-2-yl] 2-(3-chlorophenyl)-5-methyltriazole-4-carboxylate —— C20H19ClN4O3
[(2S)-1-(benzylamino)-1-oxopropan-2-yl] 2-(3-chlorophenyl)-5-methyltriazole-4-carboxylate
—— [(2S)-1-(cyclopropylamino)-1-oxopropan-2-yl] 2-(3-chlorophenyl)-5-methyltriazole-4-carboxylate —— C16H17ClN4O3
[(2S)-1-(cyclopropylamino)-1-oxopropan-2-yl] 2-(3-chlorophenyl)-5-methyltriazole-4-carboxylate
—— 2-[(4R)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C29H30N4O4S2
2-[(4R)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— (1R,2S,3R,4R)-3-[(4-methyl-1,2,4-triazol-3-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C13H16N4O3
(1R,2S,3R,4R)-3-[(4-methyl-1,2,4-triazol-3-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— (1R,2S,3S,4R)-3-[(4-methyl-1,2,4-triazol-3-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C13H16N4O3
(1R,2S,3S,4R)-3-[(4-methyl-1,2,4-triazol-3-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— 2-[[5-(furan-2-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[2-(2-methylphenyl)ethyl]acetamide —— C23H22N4O2S
2-[[5-(furan-2-yl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]-N-[2-(2-methylphenyl)ethyl]acetamide
—— 2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-pentylacetamide —— C18H23FN4OS
2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-pentylacetamide
—— 2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(3-propan-2-yloxypropyl)acetamide —— C19H25FN4O2S
2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(3-propan-2-yloxypropyl)acetamide
—— 2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2R)-2-ethylhexyl]acetamide —— C21H29FN4OS
2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2R)-2-ethylhexyl]acetamide
—— 1-(Azocan-1-yl)-2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]ethanone —— C20H25FN4OS
1-(Azocan-1-yl)-2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]ethanone
—— 3-[(2,5-Dimethoxyphenyl)methylsulfanyl]-5-(4-methoxyphenyl)-1,2,4-triazol-4-amine —— C18H20N4O3S
3-[(2,5-Dimethoxyphenyl)methylsulfanyl]-5-(4-methoxyphenyl)-1,2,4-triazol-4-amine
—— (E)-3-[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-4-(3-hydroxy-4-methoxyphenyl)but-3-enoic acid —— C21H20N2O7
(E)-3-[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-4-(3-hydroxy-4-methoxyphenyl)but-3-enoic acid
—— 2-[[4-amino-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[2-(2-methylphenyl)ethyl]acetamide —— C20H23N5O2S
2-[[4-amino-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[2-(2-methylphenyl)ethyl]acetamide
—— (2S)-N-[(1R)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(3-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C21H28N4O2S
(2S)-N-[(1R)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(3-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— (2R)-N-[(1S)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(3-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C21H28N4O2S
(2R)-N-[(1S)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(3-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 1-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-2-[[4-(4-fluorophenyl)-5-[(1S)-1-piperidin-1-ylethyl]-1,2,4-triazol-3-yl]sulfanyl]ethanone —— C26H36FN5OS
1-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-2-[[4-(4-fluorophenyl)-5-[(1S)-1-piperidin-1-ylethyl]-1,2,4-triazol-3-yl]sulfanyl]ethanone
—— (3R)-1,1-dioxo-N-[(Z)-1-[3-(tetrazol-1-yl)phenyl]ethylideneamino]thiolane-3-carboxamide —— C14H16N6O3S
(3R)-1,1-dioxo-N-[(Z)-1-[3-(tetrazol-1-yl)phenyl]ethylideneamino]thiolane-3-carboxamide
—— 1-[(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-2-[[4-(4-fluorophenyl)-5-[(1S)-1-piperidin-1-ylethyl]-1,2,4-triazol-3-yl]sulfanyl]ethanone —— C26H36FN5OS
1-[(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-2-[[4-(4-fluorophenyl)-5-[(1S)-1-piperidin-1-ylethyl]-1,2,4-triazol-3-yl]sulfanyl]ethanone
—— (2S)-N-[(1S)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(3-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C21H28N4O2S
(2S)-N-[(1S)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-[[4-(3-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 2-[(4R)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H26ClN5O2S2
2-[(4R)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4S)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C31H26ClN5O2S2
2-[(4S)-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 1-(2-Methoxyethyl)-3-[[4-(2-methyl-1,3-thiazol-4-yl)phenyl]methyl]thiourea —— C15H19N3OS2
1-(2-Methoxyethyl)-3-[[4-(2-methyl-1,3-thiazol-4-yl)phenyl]methyl]thiourea
—— (E)-4-(4-chlorophenyl)-3-[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]but-3-enoic acid —— C20H17ClN2O5
(E)-4-(4-chlorophenyl)-3-[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]but-3-enoic acid
—— (3S)-1,1-dioxo-N-[(Z)-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)methylideneamino]thiolane-3-carboxamide —— C19H18N4O3S2
(3S)-1,1-dioxo-N-[(Z)-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)methylideneamino]thiolane-3-carboxamide
—— 1-(3,5-Dichlorophenyl)-3-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]thiourea —— C19H18Cl2N4S
1-(3,5-Dichlorophenyl)-3-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]thiourea
—— (E)-4-(3-chlorophenyl)-3-[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]but-3-enoate —— C20H16ClN2O5-
(E)-4-(3-chlorophenyl)-3-[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]but-3-enoate
—— N-[(Z)-1-(2-chloro-4-fluorophenyl)ethylideneamino]-2-(4-methyl-1,3-thiazol-2-yl)acetamide —— C14H13ClFN3OS
N-[(Z)-1-(2-chloro-4-fluorophenyl)ethylideneamino]-2-(4-methyl-1,3-thiazol-2-yl)acetamide
—— (1Z,3S)-3-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-1-(1,3,3-trimethylindol-2-ylidene)butan-2-one —— C24H25FN4OS
(1Z,3S)-3-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-1-(1,3,3-trimethylindol-2-ylidene)butan-2-one
—— (2S)-2-[[5-[(1S)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(2S,6S)-2,6-dimethylpiperidin-1-yl]propan-1-one —— C22H32FN5OS
(2S)-2-[[5-[(1S)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(2S,6S)-2,6-dimethylpiperidin-1-yl]propan-1-one
—— 4-methyl-6-oxo-3-[(E)-2-(1-phenylpyrazol-4-yl)ethenyl]-1H-pyridazine-5-carbonitrile —— C17H13N5O
4-methyl-6-oxo-3-[(E)-2-(1-phenylpyrazol-4-yl)ethenyl]-1H-pyridazine-5-carbonitrile
—— (3R)-N-[(Z)-[3-(furan-2-yl)-1-phenylpyrazol-4-yl]methylideneamino]-1,1-dioxothiolane-3-carboxamide —— C19H18N4O4S
(3R)-N-[(Z)-[3-(furan-2-yl)-1-phenylpyrazol-4-yl]methylideneamino]-1,1-dioxothiolane-3-carboxamide
—— (3S)-1,1-dioxo-N-[(Z)-1-[3-(tetrazol-1-yl)phenyl]ethylideneamino]thiolane-3-carboxamide —— C14H16N6O3S
(3S)-1,1-dioxo-N-[(Z)-1-[3-(tetrazol-1-yl)phenyl]ethylideneamino]thiolane-3-carboxamide
—— (1Z,3S)-3-[[4-ethyl-5-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-(1,3,3-trimethylindol-2-ylidene)butan-2-one —— C26H30N4O2S
(1Z,3S)-3-[[4-ethyl-5-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-(1,3,3-trimethylindol-2-ylidene)butan-2-one
—— (2R)-2-[[5-[(1S)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(2S,6S)-2,6-dimethylpiperidin-1-yl]propan-1-one —— C22H32FN5OS
(2R)-2-[[5-[(1S)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(2S,6S)-2,6-dimethylpiperidin-1-yl]propan-1-one
—— (2S)-1-[cyclopropylmethyl-[[3-ethyl-5-(2-methoxyphenoxy)-1-phenylpyrazol-4-yl]methyl]amino]-3-phenylmethoxypropan-2-ol —— C33H39N3O4
(2S)-1-[cyclopropylmethyl-[[3-ethyl-5-(2-methoxyphenoxy)-1-phenylpyrazol-4-yl]methyl]amino]-3-phenylmethoxypropan-2-ol
—— 1-[[4-(2-Methyl-1,3-thiazol-4-yl)phenyl]methyl]-3-(2-morpholin-4-ium-4-ylethyl)thiourea —— C18H25N4OS2+
1-[[4-(2-Methyl-1,3-thiazol-4-yl)phenyl]methyl]-3-(2-morpholin-4-ium-4-ylethyl)thiourea
—— (3S)-N-[(Z)-(3,5-dimethyl-1-phenylpyrazol-4-yl)methylideneamino]-1,1-dioxothiolane-3-carboxamide —— C17H20N4O3S
(3S)-N-[(Z)-(3,5-dimethyl-1-phenylpyrazol-4-yl)methylideneamino]-1,1-dioxothiolane-3-carboxamide
—— (3R)-N-[(Z)-[5-chloro-1-(2-chlorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-1,1-dioxothiolane-3-carboxamide —— C16H16Cl2N4O3S
(3R)-N-[(Z)-[5-chloro-1-(2-chlorophenyl)-3-methylpyrazol-4-yl]methylideneamino]-1,1-dioxothiolane-3-carboxamide
—— (1Z,3S)-3-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-(1,3,3-trimethylindol-2-ylidene)butan-2-one —— C25H28N4OS
(1Z,3S)-3-[[4-methyl-5-(2-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-(1,3,3-trimethylindol-2-ylidene)butan-2-one
—— (E)-3-[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-4-(4-ethylphenyl)but-3-enoic acid —— C22H22N2O5
(E)-3-[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-4-(4-ethylphenyl)but-3-enoic acid
—— (2S)-2-[[5-[(1R)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(2S,6S)-2,6-dimethylpiperidin-1-yl]propan-1-one —— C22H32FN5OS
(2S)-2-[[5-[(1R)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(2S,6S)-2,6-dimethylpiperidin-1-yl]propan-1-one
—— 3-[(E)-2-[1-benzyl-3-(3,4-dimethylphenyl)pyrazol-4-yl]ethenyl]-4-methyl-6-oxo-1H-pyridazine-5-carbonitrile —— C26H23N5O
3-[(E)-2-[1-benzyl-3-(3,4-dimethylphenyl)pyrazol-4-yl]ethenyl]-4-methyl-6-oxo-1H-pyridazine-5-carbonitrile
—— (3R)-1,1-dioxo-N-[(Z)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethylideneamino]thiolane-3-carboxamide —— C15H17N5O3S
(3R)-1,1-dioxo-N-[(Z)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethylideneamino]thiolane-3-carboxamide