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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-2-[[4-amino-5-(2-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2-methoxyphenyl)methyl]propanamide —— C19H20ClN5O2S
(2R)-2-[[4-amino-5-(2-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(2-methoxyphenyl)methyl]propanamide
—— (4Z,5S)-5-(2,3-dimethoxyphenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(3-morpholin-4-ylpropyl)pyrrolidine-2,3-dione —— C30H34N4O6
(4Z,5S)-5-(2,3-dimethoxyphenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(3-morpholin-4-ylpropyl)pyrrolidine-2,3-dione
—— 3-[4-benzyl-5-[(2R)-1-(2-methyl-1H-indol-3-yl)-1-oxopropan-2-yl]sulfanyl-1,2,4-triazol-3-yl]-N,N-diethylbenzenesulfonamide —— C31H33N5O3S2
3-[4-benzyl-5-[(2R)-1-(2-methyl-1H-indol-3-yl)-1-oxopropan-2-yl]sulfanyl-1,2,4-triazol-3-yl]-N,N-diethylbenzenesulfonamide
—— [3-(2-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 3-fluorobenzoate —— C17H13FN2O4
[3-(2-Methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 3-fluorobenzoate
—— 3-[4-benzyl-5-[(2S)-1-(2-methyl-1H-indol-3-yl)-1-oxopropan-2-yl]sulfanyl-1,2,4-triazol-3-yl]-N,N-diethylbenzenesulfonamide —— C31H33N5O3S2
3-[4-benzyl-5-[(2S)-1-(2-methyl-1H-indol-3-yl)-1-oxopropan-2-yl]sulfanyl-1,2,4-triazol-3-yl]-N,N-diethylbenzenesulfonamide
—— (4Z,5R)-1-[3-(dimethylamino)propyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-phenylpyrrolidine-2,3-dione —— C26H28N4O3
(4Z,5R)-1-[3-(dimethylamino)propyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-phenylpyrrolidine-2,3-dione
—— 3-[4-benzyl-5-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]-N,N-diethylbenzenesulfonamide —— C27H35N5O3S2
3-[4-benzyl-5-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]-N,N-diethylbenzenesulfonamide
—— [5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 5-methylpyrazine-2-carboxylate —— C16H12ClN3O3
[5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 5-methylpyrazine-2-carboxylate
—— (3S)-1-[5-(4-hydroxybut-1-ynyl)-1,3-thiazol-2-yl]-3-methylpyrrolidine-2,5-dione —— C12H12N2O3S
(3S)-1-[5-(4-hydroxybut-1-ynyl)-1,3-thiazol-2-yl]-3-methylpyrrolidine-2,5-dione
—— (4Z,5R)-1-[3-(dimethylamino)propyl]-5-(3-fluorophenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]pyrrolidine-2,3-dione —— C26H27FN4O3
(4Z,5R)-1-[3-(dimethylamino)propyl]-5-(3-fluorophenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]pyrrolidine-2,3-dione
—— 3-[4-benzyl-5-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]-N,N-diethylbenzenesulfonamide —— C27H35N5O3S2
3-[4-benzyl-5-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]sulfanyl-1,2,4-triazol-3-yl]-N,N-diethylbenzenesulfonamide
—— 2-[[4-amino-5-[3-(diethylsulfamoyl)phenyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(3S)-1,1-dioxothiolan-3-yl]-N-ethylacetamide —— C20H30N6O5S3
2-[[4-amino-5-[3-(diethylsulfamoyl)phenyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(3S)-1,1-dioxothiolan-3-yl]-N-ethylacetamide
—— (3R)-1-[5-(3-aminoprop-1-ynyl)-1,3-thiazol-2-yl]-3-methylpyrrolidine-2,5-dione —— C11H11N3O2S
(3R)-1-[5-(3-aminoprop-1-ynyl)-1,3-thiazol-2-yl]-3-methylpyrrolidine-2,5-dione
—— (2R)-N-[4-chloro-3-(trifluoromethyl)phenyl]-2-[(3-oxo-4-phenyl-4,5,7,9-tetrazatricyclo[7.5.0.02,6]tetradeca-1,5,7-trien-8-yl)sulfanyl]-2-phenylacetamide —— C31H25ClF3N5O2S
(2R)-N-[4-chloro-3-(trifluoromethyl)phenyl]-2-[(3-oxo-4-phenyl-4,5,7,9-tetrazatricyclo[7.5.0.02,6]tetradeca-1,5,7-trien-8-yl)sulfanyl]-2-phenylacetamide
—— (2S)-2-[[4-amino-5-(2-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,5-dimethylphenyl)propanamide —— C19H20ClN5OS
(2S)-2-[[4-amino-5-(2-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,5-dimethylphenyl)propanamide
—— 2-[(4R)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C31H30F2N4O4S
2-[(4R)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— (4Z,5S)-1-[3-(dimethylamino)propyl]-5-(3-fluorophenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]pyrrolidine-2,3-dione —— C26H27FN4O3
(4Z,5S)-1-[3-(dimethylamino)propyl]-5-(3-fluorophenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]pyrrolidine-2,3-dione
—— (2S)-N-[4-chloro-3-(trifluoromethyl)phenyl]-2-[(3-oxo-4-phenyl-4,5,7,9-tetrazatricyclo[7.5.0.02,6]tetradeca-1,5,7-trien-8-yl)sulfanyl]-2-phenylacetamide —— C31H25ClF3N5O2S
(2S)-N-[4-chloro-3-(trifluoromethyl)phenyl]-2-[(3-oxo-4-phenyl-4,5,7,9-tetrazatricyclo[7.5.0.02,6]tetradeca-1,5,7-trien-8-yl)sulfanyl]-2-phenylacetamide
—— 2-[[4-amino-5-[3-(diethylsulfamoyl)phenyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(3R)-1,1-dioxothiolan-3-yl]-N-ethylacetamide —— C20H30N6O5S3
2-[[4-amino-5-[3-(diethylsulfamoyl)phenyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[(3R)-1,1-dioxothiolan-3-yl]-N-ethylacetamide
—— (2S)-2-[(3-oxo-4-phenyl-4,5,7,9-tetrazatricyclo[7.5.0.02,6]tetradeca-1,5,7-trien-8-yl)sulfanyl]-N-[3-(trifluoromethyl)phenyl]propanamide —— C26H24F3N5O2S
(2S)-2-[(3-oxo-4-phenyl-4,5,7,9-tetrazatricyclo[7.5.0.02,6]tetradeca-1,5,7-trien-8-yl)sulfanyl]-N-[3-(trifluoromethyl)phenyl]propanamide
—— (2R)-2-[[4-amino-5-(2-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(3-fluorophenyl)propanamide —— C17H15ClFN5OS
(2R)-2-[[4-amino-5-(2-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(3-fluorophenyl)propanamide
—— methyl 2-[(2R,3Z)-3-[(4-fluorophenyl)-hydroxymethylidene]-2-(furan-2-yl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C21H15FN2O6S
methyl 2-[(2R,3Z)-3-[(4-fluorophenyl)-hydroxymethylidene]-2-(furan-2-yl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— (2S)-2-[[4-amino-5-(2-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(thiophen-2-ylmethyl)propanamide —— C16H16ClN5OS2
(2S)-2-[[4-amino-5-(2-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(thiophen-2-ylmethyl)propanamide
—— (2S)-2-[[5-(4-chlorophenyl)-4-(2-ethoxyethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-ethoxyphenyl)-2-phenylacetamide —— C28H29ClN4O3S
(2S)-2-[[5-(4-chlorophenyl)-4-(2-ethoxyethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-ethoxyphenyl)-2-phenylacetamide
—— (2R)-2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(1-cyanocyclohexyl)propanamide —— C20H26N6O2S
(2R)-2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(1-cyanocyclohexyl)propanamide
—— 1-methyl-5-[(3S)-3-methyl-2,5-dioxopyrrolidin-1-yl]pyrazole-4-carboxylic acid —— C10H11N3O4
1-methyl-5-[(3S)-3-methyl-2,5-dioxopyrrolidin-1-yl]pyrazole-4-carboxylic acid
—— ethyl (3S)-1-[2-[6-[1-(2,5-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C29H33N5O4S
ethyl (3S)-1-[2-[6-[1-(2,5-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[2-[6-[1-(2,5-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C29H33N5O4S
ethyl (3R)-1-[2-[6-[1-(2,5-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate
—— 2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-benzyl-N-propan-2-ylacetamide —— C22H27N5O2S
2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-benzyl-N-propan-2-ylacetamide
—— (2S)-2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,4,6-trimethylphenyl)propanamide —— C22H27N5O2S
(2S)-2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2,4,6-trimethylphenyl)propanamide
—— ethyl (3S)-1-[2-[6-[1-(2-ethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C29H33N5O4S
ethyl (3S)-1-[2-[6-[1-(2-ethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate
—— (1S,2S,3R,4S)-3-(3-pyrazol-1-ylpropylcarbamoyl)bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C15H19N3O3
(1S,2S,3R,4S)-3-(3-pyrazol-1-ylpropylcarbamoyl)bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— 2-[(4-Fluorophenoxy)methyl]-4-[[1-(2-methylphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-thiazole —— C19H16FN5OS2
2-[(4-Fluorophenoxy)methyl]-4-[[1-(2-methylphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-thiazole
—— ethyl (3S)-1-[2-[6-[1-(2,4-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C29H33N5O4S
ethyl (3S)-1-[2-[6-[1-(2,4-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate
—— 2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(2R,6R)-2,6-dimethylmorpholin-4-yl]ethanone —— C18H25N5O3S
2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(2R,6R)-2,6-dimethylmorpholin-4-yl]ethanone
—— [(1R,2R,5R)-5-methyl-2-propan-2-ylcyclohexyl] 2-[[4-(2,2-dimethoxyethyl)-5-[3-(dimethylsulfamoyl)phenyl]-1,2,4-triazol-3-yl]sulfanyl]acetate —— C26H40N4O6S2
[(1R,2R,5R)-5-methyl-2-propan-2-ylcyclohexyl] 2-[[4-(2,2-dimethoxyethyl)-5-[3-(dimethylsulfamoyl)phenyl]-1,2,4-triazol-3-yl]sulfanyl]acetate
—— N-[2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]acetamide —— C14H19N5O2S
N-[2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]acetamide
—— N-cycloheptyl-2-[[5-(3-morpholin-4-ylsulfonylphenyl)-4-[(1R)-1-phenylethyl]-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C29H37N5O4S2
N-cycloheptyl-2-[[5-(3-morpholin-4-ylsulfonylphenyl)-4-[(1R)-1-phenylethyl]-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— (1S,2S,3S,4S)-3-[(1,3,5-trimethylpyrazol-4-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C16H21N3O3
(1S,2S,3S,4S)-3-[(1,3,5-trimethylpyrazol-4-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— (1S,2S,3S,4S)-3-[(1-methylpyrazol-4-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C14H17N3O3
(1S,2S,3S,4S)-3-[(1-methylpyrazol-4-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— N-benzyl-2-[[4-(2,4-dimethylphenyl)-5-(naphthalen-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(3R)-1,1-dioxothiolan-3-yl]acetamide —— C34H34N4O3S2
N-benzyl-2-[[4-(2,4-dimethylphenyl)-5-(naphthalen-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(3R)-1,1-dioxothiolan-3-yl]acetamide
—— (1S,2S,3R,4R)-3-[(1-methylpyrazol-4-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C14H17N3O3
(1S,2S,3R,4R)-3-[(1-methylpyrazol-4-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— (1S,2S,3R,4S)-3-[(1,3,5-trimethylpyrazol-4-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C16H21N3O3
(1S,2S,3R,4S)-3-[(1,3,5-trimethylpyrazol-4-yl)methylcarbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— (1S,2S,3R,4S)-3-[[(1S)-1-(1-ethyl-3-methylpyrazol-4-yl)ethyl]carbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C17H23N3O3
(1S,2S,3R,4S)-3-[[(1S)-1-(1-ethyl-3-methylpyrazol-4-yl)ethyl]carbamoyl]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— (1S,2S,3S,4R)-3-(3-pyrazol-1-ylpropylcarbamoyl)bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C15H19N3O3
(1S,2S,3S,4R)-3-(3-pyrazol-1-ylpropylcarbamoyl)bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— (2R)-N-(4-chloro-2-methoxy-5-methylphenyl)-2-[1-(2-methylphenyl)tetrazol-5-yl]sulfanylpropanamide —— C19H20ClN5O2S
(2R)-N-(4-chloro-2-methoxy-5-methylphenyl)-2-[1-(2-methylphenyl)tetrazol-5-yl]sulfanylpropanamide
—— [3-(4-Fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl 2-(3,4-dichlorophenyl)acetate —— C17H11Cl2FN2O3
[3-(4-Fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl 2-(3,4-dichlorophenyl)acetate
—— N-[2-(3-fluorophenyl)ethyl]-3-(2-methoxyphenyl)-1-phenylpyrazole-4-carboxamide —— C25H22FN3O2
N-[2-(3-fluorophenyl)ethyl]-3-(2-methoxyphenyl)-1-phenylpyrazole-4-carboxamide
—— [3-(4-Fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl 2,3-dichlorobenzoate —— C16H9Cl2FN2O3
[3-(4-Fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl 2,3-dichlorobenzoate
—— ethyl (3R)-1-[2-[6-[1-(2,4-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C29H33N5O4S
ethyl (3R)-1-[2-[6-[1-(2,4-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate