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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(4S)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C33H33ClN4O4S
2-[(4S)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— (2S)-1-(3-methylphenoxy)-3-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanyl]propan-2-ol —— C21H23N3O2S
(2S)-1-(3-methylphenoxy)-3-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanyl]propan-2-ol
—— 2-[(4R)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C31H29ClN4O3S
2-[(4R)-3-(4-chlorophenyl)-4-(2-methoxyphenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— (2S)-1-[(5-cyclohexyl-1-phenyl-1,2,4-triazol-3-yl)sulfanyl]-3-morpholin-4-ium-4-ylpropan-2-ol —— C21H31N4O2S+
(2S)-1-[(5-cyclohexyl-1-phenyl-1,2,4-triazol-3-yl)sulfanyl]-3-morpholin-4-ium-4-ylpropan-2-ol
—— N-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]-5-(2-fluoro-4-methoxyphenyl)-1-methylpyrazole-3-carboxamide —— C19H22FN3O2
N-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]-5-(2-fluoro-4-methoxyphenyl)-1-methylpyrazole-3-carboxamide
—— N-[[5-(2,4-difluorophenoxy)-3-ethyl-1-(4-methoxyphenyl)pyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]thiophene-2-carboxamide —— C29H29F2N3O4S
N-[[5-(2,4-difluorophenoxy)-3-ethyl-1-(4-methoxyphenyl)pyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]thiophene-2-carboxamide
—— 3-tert-butyl-1-[[5-(2,4-difluorophenoxy)-3-ethyl-1-(4-methoxyphenyl)pyrazol-4-yl]methyl]-1-[[(2S)-oxolan-2-yl]methyl]urea —— C29H36F2N4O4
3-tert-butyl-1-[[5-(2,4-difluorophenoxy)-3-ethyl-1-(4-methoxyphenyl)pyrazol-4-yl]methyl]-1-[[(2S)-oxolan-2-yl]methyl]urea
—— (2S)-3-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanyl-2-methylpropanenitrile —— C13H15N5S
(2S)-3-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanyl-2-methylpropanenitrile
—— 2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C28H26Cl2N4O3S2
2-[(4S)-1-(2-chlorophenyl)-4-(3-chlorophenyl)-7-oxo-3-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— (5S,7S)-N-(2-adamantyl)-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C23H32N4O
(5S,7S)-N-(2-adamantyl)-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— (3R,4R)-4-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanyl-1,1-dioxothiolan-3-ol —— C13H16N4O3S2
(3R,4R)-4-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanyl-1,1-dioxothiolan-3-ol
—— (2S)-1-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-3-morpholin-4-ylpropan-2-ol —— C18H23FN4O2S
(2S)-1-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-3-morpholin-4-ylpropan-2-ol
—— (5R,7R)-N-[(1R)-1-(1-adamantyl)ethyl]-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C25H36N4O
(5R,7R)-N-[(1R)-1-(1-adamantyl)ethyl]-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— (4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H27ClN4O3S2
(4S)-3-(4-chlorophenyl)-1-(4-methylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— N-[[5-(2,4-difluorophenoxy)-3-ethyl-1-(4-methoxyphenyl)pyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]furan-2-carboxamide —— C29H29F2N3O5
N-[[5-(2,4-difluorophenoxy)-3-ethyl-1-(4-methoxyphenyl)pyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]furan-2-carboxamide
—— (2R)-2-[[5-(4-chlorophenyl)-4-(2-methoxyethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]pentanedinitrile —— C17H18ClN5OS
(2R)-2-[[5-(4-chlorophenyl)-4-(2-methoxyethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]pentanedinitrile
—— (2S)-2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]pentanedinitrile —— C17H16FN5S
(2S)-2-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]pentanedinitrile
—— (3S,4R)-4-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-1,1-dioxothiolan-3-ol —— C15H16FN3O3S2
(3S,4R)-4-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-1,1-dioxothiolan-3-ol
—— (3R,4R)-4-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-1,1-dioxothiolan-3-ol —— C15H16FN3O3S2
(3R,4R)-4-[[4-cyclopropyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-1,1-dioxothiolan-3-ol
—— (2R)-1-[(1S)-1-(4-chlorophenyl)ethoxy]-3-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanylpropan-2-ol —— C20H23ClN4O2S
(2R)-1-[(1S)-1-(4-chlorophenyl)ethoxy]-3-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanylpropan-2-ol
—— ethyl 4-[[2-[(5R,7R)-3-bromo-1-adamantyl]acetyl]oxymethyl]-1,3-thiazole-2-carboxylate —— C19H24BrNO4S
ethyl 4-[[2-[(5R,7R)-3-bromo-1-adamantyl]acetyl]oxymethyl]-1,3-thiazole-2-carboxylate
—— (2S)-1-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanyl-3-naphthalen-1-yloxypropan-2-ol —— C22H22N4O2S
(2S)-1-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanyl-3-naphthalen-1-yloxypropan-2-ol
—— (2R)-1-(1,3-benzodioxol-5-ylmethoxy)-3-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanylpropan-2-ol —— C20H22N4O4S
(2R)-1-(1,3-benzodioxol-5-ylmethoxy)-3-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanylpropan-2-ol
—— (2S)-3-[[4-benzyl-5-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-methylpropanenitrile —— C19H17FN4S
(2S)-3-[[4-benzyl-5-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-methylpropanenitrile
—— (2R)-1-[[3-ethyl-5-(2-methoxyphenoxy)-1-phenylpyrazol-4-yl]methyl-(2-methoxyethyl)amino]-3-phenylmethoxypropan-2-ol —— C32H39N3O5
(2R)-1-[[3-ethyl-5-(2-methoxyphenoxy)-1-phenylpyrazol-4-yl]methyl-(2-methoxyethyl)amino]-3-phenylmethoxypropan-2-ol
—— ethyl 4-[[2-[(5S,7S)-3-bromo-1-adamantyl]acetyl]oxymethyl]-1,3-thiazole-2-carboxylate —— C19H24BrNO4S
ethyl 4-[[2-[(5S,7S)-3-bromo-1-adamantyl]acetyl]oxymethyl]-1,3-thiazole-2-carboxylate
—— (2S)-1-[[3-ethyl-5-(2-methoxyphenoxy)-1-phenylpyrazol-4-yl]methyl-(2-methoxyethyl)amino]-3-phenylmethoxypropan-2-ol —— C32H39N3O5
(2S)-1-[[3-ethyl-5-(2-methoxyphenoxy)-1-phenylpyrazol-4-yl]methyl-(2-methoxyethyl)amino]-3-phenylmethoxypropan-2-ol
—— (2R)-2-chloro-1-[4-[6-[(4-methylphenyl)methyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-1-yl]-2-phenylethanone —— C32H31ClN6O
(2R)-2-chloro-1-[4-[6-[(4-methylphenyl)methyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-1-yl]-2-phenylethanone
—— N-[[(1R,2R,4S)-2-bicyclo[2.2.1]hept-5-enyl]methyl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)aniline —— C17H20N4
N-[[(1R,2R,4S)-2-bicyclo[2.2.1]hept-5-enyl]methyl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)aniline
—— N-[[(1R,2S,4S)-2-bicyclo[2.2.1]hept-5-enyl]methyl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)aniline —— C17H20N4
N-[[(1R,2S,4S)-2-bicyclo[2.2.1]hept-5-enyl]methyl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)aniline
—— (2S)-1-[[5-(4-chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-3-(2-methylphenoxy)propan-2-ol —— C19H20ClN3O2S
(2S)-1-[[5-(4-chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-3-(2-methylphenoxy)propan-2-ol
—— (2S)-1-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-3-(2,3,6-trimethylphenoxy)propan-2-ol —— C21H24FN3O2S
(2S)-1-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-3-(2,3,6-trimethylphenoxy)propan-2-ol
—— (2S)-1-(2,6-dimethylphenoxy)-3-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylpropan-2-ol —— C20H24N4O2S
(2S)-1-(2,6-dimethylphenoxy)-3-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylpropan-2-ol
—— (2S)-2-chloro-1-[4-[6-[(4-methylphenyl)methyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-1-yl]-2-phenylethanone —— C32H31ClN6O
(2S)-2-chloro-1-[4-[6-[(4-methylphenyl)methyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-1-yl]-2-phenylethanone
—— (2R)-2-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]pentanedinitrile —— C15H14FN5S
(2R)-2-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]pentanedinitrile
—— 3-[[5-(2-Fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C12H13FN4OS
3-[[5-(2-Fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 2-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]-N-[5-tert-butyl-2-(4-fluorophenyl)pyrazol-3-yl]acetamide —— C23H25FN4O3
2-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]-N-[5-tert-butyl-2-(4-fluorophenyl)pyrazol-3-yl]acetamide
—— (2S)-1-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanyl-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]oxy]propan-2-ol —— C22H26N4O2S
(2S)-1-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanyl-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]oxy]propan-2-ol
—— (2S)-1-(2,6-dimethylphenoxy)-3-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]propan-2-ol —— C20H22FN3O2S
(2S)-1-(2,6-dimethylphenoxy)-3-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]propan-2-ol
—— (2S)-2-[[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]pentanedinitrile —— C15H16N6S
(2S)-2-[[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]pentanedinitrile
—— (2R)-1-(3,5-dimethylphenoxy)-3-[[5-(4-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]propan-2-ol —— C20H22FN3O2S
(2R)-1-(3,5-dimethylphenoxy)-3-[[5-(4-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]propan-2-ol
—— (2S)-1-[[5-(4-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-3-(4-methylphenoxy)propan-2-ol —— C19H20FN3O2S
(2S)-1-[[5-(4-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-3-(4-methylphenoxy)propan-2-ol
—— 2-[(3aS,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]-N-[5-tert-butyl-2-(4-fluorophenyl)pyrazol-3-yl]acetamide —— C23H25FN4O3
2-[(3aS,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]-N-[5-tert-butyl-2-(4-fluorophenyl)pyrazol-3-yl]acetamide
—— 2-[(4R)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C33H27F2N5O3S
2-[(4R)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 2-[(4S)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C33H27F2N5O3S
2-[(4S)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— (2R)-1-(2,6-dimethylphenoxy)-3-[[5-(4-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]propan-2-ol —— C20H22FN3O2S
(2R)-1-(2,6-dimethylphenoxy)-3-[[5-(4-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]propan-2-ol
—— (2S)-3-[[4-cyclohexyl-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-methylpropanenitrile —— C21H28N4O3S
(2S)-3-[[4-cyclohexyl-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-methylpropanenitrile
—— N-ethyl-3-ethynyl-N-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)methyl]aniline —— C20H20N4
N-ethyl-3-ethynyl-N-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)methyl]aniline
—— (2R)-1-[1-(2-methylphenyl)tetrazol-5-yl]sulfanyl-3-naphthalen-1-yloxypropan-2-ol —— C21H20N4O2S
(2R)-1-[1-(2-methylphenyl)tetrazol-5-yl]sulfanyl-3-naphthalen-1-yloxypropan-2-ol
—— 2-[[4-Methyl-5-(trifluoromethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-5-phenyl-1,3-oxazole —— C14H11F3N4OS
2-[[4-Methyl-5-(trifluoromethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-5-phenyl-1,3-oxazole