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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(4R)-4-(2,5-dimethoxyphenyl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C35H34N4O5S
2-[(4R)-4-(2,5-dimethoxyphenyl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 4-fluoro-N-[[5-(3-fluorophenoxy)-1-phenyl-3-propan-2-ylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide —— C31H31F2N3O3
4-fluoro-N-[[5-(3-fluorophenoxy)-1-phenyl-3-propan-2-ylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide
—— 4-chloro-N-[[5-(4-methoxyphenoxy)-1-methyl-3-phenylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide —— C30H30ClN3O4
4-chloro-N-[[5-(4-methoxyphenoxy)-1-methyl-3-phenylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide
—— (Z)-N-[2-[(5E)-2,4-dioxo-5-(pyridin-3-ylmethylidene)-1,3-thiazolidin-3-yl]ethyl]-3-[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]prop-2-enamide —— C29H22FN5O3S
(Z)-N-[2-[(5E)-2,4-dioxo-5-(pyridin-3-ylmethylidene)-1,3-thiazolidin-3-yl]ethyl]-3-[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]prop-2-enamide
—— N-[[5-(2-chlorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-3-methoxy-N-[[(2S)-oxolan-2-yl]methyl]benzamide —— C30H30ClN3O4
N-[[5-(2-chlorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-3-methoxy-N-[[(2S)-oxolan-2-yl]methyl]benzamide
—— N-[2-[(5E)-2,4-dioxo-5-[(3,4,5-trimethoxyphenyl)methylidene]-1,3-thiazolidin-3-yl]ethyl]-3-methyl-1-phenylthieno[2,3-c]pyrazole-5-carboxamide —— C28H26N4O6S2
N-[2-[(5E)-2,4-dioxo-5-[(3,4,5-trimethoxyphenyl)methylidene]-1,3-thiazolidin-3-yl]ethyl]-3-methyl-1-phenylthieno[2,3-c]pyrazole-5-carboxamide
—— N-[[5-(2-chlorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-3-methoxy-N-[[(2R)-oxolan-2-yl]methyl]benzamide —— C30H30ClN3O4
N-[[5-(2-chlorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-3-methoxy-N-[[(2R)-oxolan-2-yl]methyl]benzamide
—— (Z)-3-[3-(3,4-dimethoxyphenyl)-1-phenylpyrazol-4-yl]-N-[2-[(5E)-5-[(4-fluorophenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]prop-2-enamide —— C32H27FN4O5S
(Z)-3-[3-(3,4-dimethoxyphenyl)-1-phenylpyrazol-4-yl]-N-[2-[(5E)-5-[(4-fluorophenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]prop-2-enamide
—— 2-chloro-N-[[5-(4-methoxyphenoxy)-1-methyl-3-phenylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide —— C30H30ClN3O4
2-chloro-N-[[5-(4-methoxyphenoxy)-1-methyl-3-phenylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide
—— N-[[1-(4-chlorophenyl)-5-(2-methoxyphenoxy)-3-methylpyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]thiophene-2-carboxamide —— C28H28ClN3O4S
N-[[1-(4-chlorophenyl)-5-(2-methoxyphenoxy)-3-methylpyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]thiophene-2-carboxamide
—— (Z)-N-[2-[(5E)-5-[(4-fluorophenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]-3-[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]prop-2-enamide —— C30H22F2N4O3S
(Z)-N-[2-[(5E)-5-[(4-fluorophenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]-3-[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]prop-2-enamide
—— [2-[[(3S)-1,1-dioxothiolan-3-yl]-ethylamino]-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate —— C18H21N3O5S
[2-[[(3S)-1,1-dioxothiolan-3-yl]-ethylamino]-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate
—— N-[[5-(4-chlorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]-4-(trifluoromethyl)benzamide —— C30H27ClF3N3O3
N-[[5-(4-chlorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]-4-(trifluoromethyl)benzamide
—— [2-(2,5-dimethylanilino)-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate —— C20H19N3O3
[2-(2,5-dimethylanilino)-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate
—— (Z)-3-[3-(3,4-dimethoxyphenyl)-1-phenylpyrazol-4-yl]-N-[2-[(5Z)-5-[(4-fluorophenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]prop-2-enamide —— C32H27FN4O5S
(Z)-3-[3-(3,4-dimethoxyphenyl)-1-phenylpyrazol-4-yl]-N-[2-[(5Z)-5-[(4-fluorophenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]prop-2-enamide
—— methyl 2-[2-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-6-oxo-1H-pyrimidin-4-yl]acetate —— C17H16N4O4S
methyl 2-[2-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-6-oxo-1H-pyrimidin-4-yl]acetate
—— [(2S)-1-[(1-cyanocyclohexyl)amino]-1-oxopropan-2-yl] 3-phenyl-1H-pyrazole-5-carboxylate —— C20H22N4O3
[(2S)-1-[(1-cyanocyclohexyl)amino]-1-oxopropan-2-yl] 3-phenyl-1H-pyrazole-5-carboxylate
—— [2-[[(3S)-3-methyl-1,1-dioxothiolan-3-yl]amino]-2-oxoethyl] 1-benzyl-3,5-dimethylpyrazole-4-carboxylate —— C20H25N3O5S
[2-[[(3S)-3-methyl-1,1-dioxothiolan-3-yl]amino]-2-oxoethyl] 1-benzyl-3,5-dimethylpyrazole-4-carboxylate
—— [2-[[(3S)-1,1-dioxothiolan-3-yl]-methylamino]-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate —— C17H19N3O5S
[2-[[(3S)-1,1-dioxothiolan-3-yl]-methylamino]-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate
—— [2-(2-ethylanilino)-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate —— C20H19N3O3
[2-(2-ethylanilino)-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate
—— [2-(3-chloro-4-methoxyanilino)-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate —— C19H16ClN3O4
[2-(3-chloro-4-methoxyanilino)-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate
—— 2-chloro-N-[[5-(4-chlorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide —— C29H27Cl2N3O3
2-chloro-N-[[5-(4-chlorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide
—— [2-[(3-Methoxyphenyl)methyl-methylamino]-2-oxoethyl] 1-benzyl-3,5-dimethylpyrazole-4-carboxylate —— C24H27N3O4
[2-[(3-Methoxyphenyl)methyl-methylamino]-2-oxoethyl] 1-benzyl-3,5-dimethylpyrazole-4-carboxylate
—— [(2S)-1-oxo-1-[4-(trifluoromethyl)anilino]propan-2-yl] 3-phenyl-1H-pyrazole-5-carboxylate —— C20H16F3N3O3
[(2S)-1-oxo-1-[4-(trifluoromethyl)anilino]propan-2-yl] 3-phenyl-1H-pyrazole-5-carboxylate
—— (3-methoxycarbonylphenyl)methyl 3-phenyl-1H-pyrazole-5-carboxylate —— C19H16N2O4
(3-methoxycarbonylphenyl)methyl 3-phenyl-1H-pyrazole-5-carboxylate
—— [2-(5-chloro-2-methylanilino)-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate —— C19H16ClN3O3
[2-(5-chloro-2-methylanilino)-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate
—— [(3Z)-3-cyano-3-(3-methyl-1H-benzimidazol-2-ylidene)-2-oxopropyl] 3-phenyl-1H-pyrazole-5-carboxylate —— C22H17N5O3
[(3Z)-3-cyano-3-(3-methyl-1H-benzimidazol-2-ylidene)-2-oxopropyl] 3-phenyl-1H-pyrazole-5-carboxylate
—— [2-oxo-2-[[(1S)-1-thiophen-2-ylethyl]amino]ethyl] 1-benzyl-3,5-dimethylpyrazole-4-carboxylate —— C21H23N3O3S
[2-oxo-2-[[(1S)-1-thiophen-2-ylethyl]amino]ethyl] 1-benzyl-3,5-dimethylpyrazole-4-carboxylate
—— [2-(5-methylthiophen-2-yl)-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate —— C17H14N2O3S
[2-(5-methylthiophen-2-yl)-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate
—— [(2S)-1-(naphthalen-1-ylamino)-1-oxopropan-2-yl] 3-phenyl-1H-pyrazole-5-carboxylate —— C23H19N3O3
[(2S)-1-(naphthalen-1-ylamino)-1-oxopropan-2-yl] 3-phenyl-1H-pyrazole-5-carboxylate
—— [(3R)-3-cyano-3-(4-methyl-1,3-thiazol-2-yl)-2-oxopropyl] 3-phenyl-1H-pyrazole-5-carboxylate —— C18H14N4O3S
[(3R)-3-cyano-3-(4-methyl-1,3-thiazol-2-yl)-2-oxopropyl] 3-phenyl-1H-pyrazole-5-carboxylate
—— [2-[[2-(2-ethylanilino)-2-oxoethyl]-methylamino]-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate —— C23H24N4O4
[2-[[2-(2-ethylanilino)-2-oxoethyl]-methylamino]-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate
—— (4-methoxycarbonyl-5-methylfuran-2-yl)methyl 3-phenyl-1H-pyrazole-5-carboxylate —— C18H16N2O5
(4-methoxycarbonyl-5-methylfuran-2-yl)methyl 3-phenyl-1H-pyrazole-5-carboxylate
—— (Z)-N-[2-[(5Z)-2,4-dioxo-5-(pyridin-3-ylmethylidene)-1,3-thiazolidin-3-yl]ethyl]-3-[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]prop-2-enamide —— C29H22FN5O3S
(Z)-N-[2-[(5Z)-2,4-dioxo-5-(pyridin-3-ylmethylidene)-1,3-thiazolidin-3-yl]ethyl]-3-[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]prop-2-enamide
—— [2-(N-ethyl-4-fluoroanilino)-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate —— C20H18FN3O3
[2-(N-ethyl-4-fluoroanilino)-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate
—— (2-methylphenyl)methyl 3-phenyl-1H-pyrazole-5-carboxylate —— C18H16N2O2
(2-methylphenyl)methyl 3-phenyl-1H-pyrazole-5-carboxylate
—— 4-chloro-N-[[5-(2-methoxyphenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide —— C30H30ClN3O4
4-chloro-N-[[5-(2-methoxyphenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide
—— [2-[(3-Cyanothiophen-2-yl)amino]-2-oxoethyl] 1-benzyl-3,5-dimethylpyrazole-4-carboxylate —— C20H18N4O3S
[2-[(3-Cyanothiophen-2-yl)amino]-2-oxoethyl] 1-benzyl-3,5-dimethylpyrazole-4-carboxylate
—— [2-(4,5-dimethyl-2-nitroanilino)-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate —— C20H18N4O5
[2-(4,5-dimethyl-2-nitroanilino)-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate
—— 2-chloro-N-[[5-(4-methoxyphenoxy)-1-methyl-3-phenylpyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide —— C30H30ClN3O4
2-chloro-N-[[5-(4-methoxyphenoxy)-1-methyl-3-phenylpyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide
—— [2-(2-Acetylhydrazinyl)-2-oxoethyl] 1-benzyl-3,5-dimethylpyrazole-4-carboxylate —— C17H20N4O4
[2-(2-Acetylhydrazinyl)-2-oxoethyl] 1-benzyl-3,5-dimethylpyrazole-4-carboxylate
—— [2-[[(2S)-butan-2-yl]amino]-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate —— C16H19N3O3
[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl] 3-phenyl-1H-pyrazole-5-carboxylate
—— [(2S)-1-(4-fluoroanilino)-1-oxopropan-2-yl] 3-phenyl-1H-pyrazole-5-carboxylate —— C19H16FN3O3
[(2S)-1-(4-fluoroanilino)-1-oxopropan-2-yl] 3-phenyl-1H-pyrazole-5-carboxylate
—— 2-[(4S)-4-(2,5-dimethoxyphenyl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C35H34N4O5S
2-[(4S)-4-(2,5-dimethoxyphenyl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— N-[[3-benzyl-2-[(2-fluorophenyl)methylsulfonyl]imidazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]furan-2-carboxamide —— C28H28FN3O5S
N-[[3-benzyl-2-[(2-fluorophenyl)methylsulfonyl]imidazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]furan-2-carboxamide
—— 1-[(1R,2S)-2-methylcyclohexyl]-3-[[2-(4-methyl-1,3-thiazol-2-yl)acetyl]amino]thiourea —— C14H22N4OS2
1-[(1R,2S)-2-methylcyclohexyl]-3-[[2-(4-methyl-1,3-thiazol-2-yl)acetyl]amino]thiourea
—— 2-[[(Z)-3-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]prop-2-enoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C29H26N4O4S
2-[[(Z)-3-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]prop-2-enoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 1-Cyclopropyl-3-[[2-(4-methyl-1,3-thiazol-2-yl)acetyl]amino]thiourea —— C10H14N4OS2
1-Cyclopropyl-3-[[2-(4-methyl-1,3-thiazol-2-yl)acetyl]amino]thiourea
—— 1-[(1S,2R)-2-methylcyclohexyl]-3-[[2-(4-methyl-1,3-thiazol-2-yl)acetyl]amino]thiourea —— C14H22N4OS2
1-[(1S,2R)-2-methylcyclohexyl]-3-[[2-(4-methyl-1,3-thiazol-2-yl)acetyl]amino]thiourea
—— Methyl 4-[[1-(4-fluorophenyl)-4-oxopyrazolo[3,4-d]pyrimidin-5-yl]methyl]benzoate —— C20H15FN4O3
Methyl 4-[[1-(4-fluorophenyl)-4-oxopyrazolo[3,4-d]pyrimidin-5-yl]methyl]benzoate