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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(4S)-1-(2-chlorophenyl)-4-(2-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C29H24ClFN4O2S
2-[(4S)-1-(2-chlorophenyl)-4-(2-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— N-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-4-methoxy-N-[[(2S)-oxolan-2-yl]methyl]benzenesulfonamide —— C29H29F2N3O5S
N-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-4-methoxy-N-[[(2S)-oxolan-2-yl]methyl]benzenesulfonamide
—— 2-[(4S)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C29H30N4O2S2
2-[(4S)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— (4S)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H27FN4O4S
(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H31ClN4O4S
(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— N-[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]-2-[[5-(ethylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]acetamide —— C18H22N6OS2
N-[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]-2-[[5-(ethylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C30H25FN4O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— (4R)-1-(2-chlorophenyl)-4-(2-fluorophenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C30H26ClFN4O2S
(4R)-1-(2-chlorophenyl)-4-(2-fluorophenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-1-(2-chlorophenyl)-4-(2-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C29H24ClFN4O2S
2-[(4R)-1-(2-chlorophenyl)-4-(2-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— 2-[(4R)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide —— C29H30N4O2S2
2-[(4R)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-propylacetamide
—— 2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C32H32F2N4O2S
2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 2-[(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C31H33FN4O2S2
2-[(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C31H29F3N4O2S
2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 2-[(4S)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C31H29F3N4O2S
2-[(4S)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 2-chloro-N-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide —— C29H26ClF2N3O3
2-chloro-N-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide
—— N-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-3-methoxy-N-[[(2S)-oxolan-2-yl]methyl]benzamide —— C30H29F2N3O4
N-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-3-methoxy-N-[[(2S)-oxolan-2-yl]methyl]benzamide
—— N-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-4-methoxy-N-[[(2R)-oxolan-2-yl]methyl]benzenesulfonamide —— C29H29F2N3O5S
N-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-4-methoxy-N-[[(2R)-oxolan-2-yl]methyl]benzenesulfonamide
—— 2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C32H31F3N4O2S
2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— N-[[4-(dimethylamino)phenyl]methyl]-2-[1-(4-propan-2-ylphenyl)tetrazol-5-yl]sulfanylacetamide —— C21H26N6OS
N-[[4-(dimethylamino)phenyl]methyl]-2-[1-(4-propan-2-ylphenyl)tetrazol-5-yl]sulfanylacetamide
—— (5S)-5-(3,5-dimethyl-1-phenylpyrazol-4-yl)-3-(4-methoxyphenyl)-2-sulfanylideneimidazolidin-4-one —— C21H20N4O2S
(5S)-5-(3,5-dimethyl-1-phenylpyrazol-4-yl)-3-(4-methoxyphenyl)-2-sulfanylideneimidazolidin-4-one
—— (4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C29H31ClN4O5S
(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(2-chlorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[6-[1-(2,5-difluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2R)-4-phenylbutan-2-yl]acetamide —— C29H27F2N5O2S
2-[6-[1-(2,5-difluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2R)-4-phenylbutan-2-yl]acetamide
—— 2-[6-[1-(3,4-dichlorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2R)-4-phenylbutan-2-yl]acetamide —— C29H27Cl2N5O2S
2-[6-[1-(3,4-dichlorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2R)-4-phenylbutan-2-yl]acetamide
—— 2-[6-[1-(3-fluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2R)-4-phenylbutan-2-yl]acetamide —— C29H28FN5O2S
2-[6-[1-(3-fluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2R)-4-phenylbutan-2-yl]acetamide
—— 2-imidazo[2,1-b][1,3]thiazol-6-yl-N-[(E)-(2-oxo-3,3a,4,5,5a,6,7,8,8a,8b-decahydroacenaphthylen-1-ylidene)amino]acetamide —— C19H22N4O2S
2-imidazo[2,1-b][1,3]thiazol-6-yl-N-[(E)-(2-oxo-3,3a,4,5,5a,6,7,8,8a,8b-decahydroacenaphthylen-1-ylidene)amino]acetamide
—— N-[2-[[1-(3,4-dimethoxyphenyl)-4-phenylimidazol-2-yl]amino]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]-1,3-benzodioxole-5-carboxamide —— C32H32N4O7
N-[2-[[1-(3,4-dimethoxyphenyl)-4-phenylimidazol-2-yl]amino]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]-1,3-benzodioxole-5-carboxamide
—— N-[2-[[1-(3,4-dimethoxyphenyl)-4-phenylimidazol-2-yl]amino]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]-1,3-benzodioxole-5-carboxamide —— C32H32N4O7
N-[2-[[1-(3,4-dimethoxyphenyl)-4-phenylimidazol-2-yl]amino]-2-oxoethyl]-N-[[(2S)-oxolan-2-yl]methyl]-1,3-benzodioxole-5-carboxamide
—— (4S)-1-(2-chlorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C28H25ClN4O3S2
(4S)-1-(2-chlorophenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C32H31F3N4O2S
2-[(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 2-[(4-chlorophenyl)sulfonyl-[[(2S)-oxolan-2-yl]methyl]amino]-N-[4-(4-methoxyphenyl)-1-(4-methylphenyl)imidazol-2-yl]acetamide —— C30H31ClN4O5S
2-[(4-chlorophenyl)sulfonyl-[[(2S)-oxolan-2-yl]methyl]amino]-N-[4-(4-methoxyphenyl)-1-(4-methylphenyl)imidazol-2-yl]acetamide
—— N-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-3-methoxy-N-[[(2R)-oxolan-2-yl]methyl]benzamide —— C30H29F2N3O4
N-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-3-methoxy-N-[[(2R)-oxolan-2-yl]methyl]benzamide
—— 3-[(4S)-4-(3,5-dimethyl-1-phenylpyrazol-4-yl)-5-oxo-2-sulfanylideneimidazolidin-1-yl]propyl-dimethylazanium —— C19H26N5OS+
3-[(4S)-4-(3,5-dimethyl-1-phenylpyrazol-4-yl)-5-oxo-2-sulfanylideneimidazolidin-1-yl]propyl-dimethylazanium
—— 2-[6-[1-(3,4-dichlorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2S)-4-phenylbutan-2-yl]acetamide —— C29H27Cl2N5O2S
2-[6-[1-(3,4-dichlorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2S)-4-phenylbutan-2-yl]acetamide
—— (5R)-5-(3,5-dimethyl-1-phenylpyrazol-4-yl)-3-(4-ethoxyphenyl)-2-sulfanylideneimidazolidin-4-one —— C22H22N4O2S
(5R)-5-(3,5-dimethyl-1-phenylpyrazol-4-yl)-3-(4-ethoxyphenyl)-2-sulfanylideneimidazolidin-4-one
—— 1-(4-fluorophenyl)-N-[(1R)-1-(furan-2-yl)ethyl]-3-methylthieno[2,3-c]pyrazole-5-carboxamide —— C19H16FN3O2S
1-(4-fluorophenyl)-N-[(1R)-1-(furan-2-yl)ethyl]-3-methylthieno[2,3-c]pyrazole-5-carboxamide
—— 2-chloro-N-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide —— C29H26ClF2N3O3
2-chloro-N-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide
—— N-[(Z)-[4-[2-hydroxyethyl(methyl)amino]phenyl]methylideneamino]-2-(5-phenyltetrazol-2-yl)acetamide —— C19H21N7O2
N-[(Z)-[4-[2-hydroxyethyl(methyl)amino]phenyl]methylideneamino]-2-(5-phenyltetrazol-2-yl)acetamide
—— 2-[6-[1-(2,3-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2R)-4-phenylbutan-2-yl]acetamide —— C31H33N5O2S
2-[6-[1-(2,3-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2R)-4-phenylbutan-2-yl]acetamide
—— 2-[6-[1-(2,5-difluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2S)-4-phenylbutan-2-yl]acetamide —— C29H27F2N5O2S
2-[6-[1-(2,5-difluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2S)-4-phenylbutan-2-yl]acetamide
—— 2-[1-(4-propan-2-ylphenyl)tetrazol-5-yl]sulfanyl-N-(4-pyrrolidin-1-ylphenyl)acetamide —— C22H26N6OS
2-[1-(4-propan-2-ylphenyl)tetrazol-5-yl]sulfanyl-N-(4-pyrrolidin-1-ylphenyl)acetamide
—— 2-[6-[1-(3-fluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2S)-4-phenylbutan-2-yl]acetamide —— C29H28FN5O2S
2-[6-[1-(3-fluorophenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2S)-4-phenylbutan-2-yl]acetamide
—— N-[(Z)-1-[4-(dimethylamino)phenyl]ethylideneamino]-2-(5-phenyltetrazol-2-yl)acetamide —— C19H21N7O
N-[(Z)-1-[4-(dimethylamino)phenyl]ethylideneamino]-2-(5-phenyltetrazol-2-yl)acetamide
—— 2-[(4S)-4-(2,5-dimethoxyphenyl)-1-methyl-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C30H29FN4O4S
2-[(4S)-4-(2,5-dimethoxyphenyl)-1-methyl-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 2-[6-[1-(2,3-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2S)-4-phenylbutan-2-yl]acetamide —— C31H33N5O2S
2-[6-[1-(2,3-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]-N-[(2S)-4-phenylbutan-2-yl]acetamide
—— 2-[[4-amino-5-(2-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C20H26ClN5OS
2-[[4-amino-5-(2-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— (4R)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C31H27FN4O4S
(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-8-(2-oxo-2-pyrrolidin-1-ylethyl)-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— 2-[[4-amino-5-(2,4-dichlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide —— C20H25Cl2N5OS
2-[[4-amino-5-(2,4-dichlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]acetamide
—— N-[(Z)-[4-[2-cyanoethyl(ethyl)amino]-2-methylphenyl]methylideneamino]-2-(5-phenyltetrazol-2-yl)acetamide —— C22H24N8O
N-[(Z)-[4-[2-cyanoethyl(ethyl)amino]-2-methylphenyl]methylideneamino]-2-(5-phenyltetrazol-2-yl)acetamide
—— N-[2-[6-(2,5-dimethoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]ethyl]-3,5-dimethoxy-N-[[(2R)-oxolan-2-yl]methyl]benzamide —— C29H33N3O6S
N-[2-[6-(2,5-dimethoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]ethyl]-3,5-dimethoxy-N-[[(2R)-oxolan-2-yl]methyl]benzamide
—— (5S)-3-(2,5-dimethylphenyl)-5-(3,5-dimethyl-1-phenylpyrazol-4-yl)-2-sulfanylideneimidazolidin-4-one —— C22H22N4OS
(5S)-3-(2,5-dimethylphenyl)-5-(3,5-dimethyl-1-phenylpyrazol-4-yl)-2-sulfanylideneimidazolidin-4-one