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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C34H26F2N4O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C32H29FN4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-[5-(4-ethylphenyl)tetrazol-2-yl]-N-[2-(2-fluorophenyl)ethyl]acetamide —— C19H20FN5O
2-[5-(4-ethylphenyl)tetrazol-2-yl]-N-[2-(2-fluorophenyl)ethyl]acetamide
—— N-[3-(dimethylsulfamoyl)phenyl]-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide —— C19H22N6O3S
N-[3-(dimethylsulfamoyl)phenyl]-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C32H29FN4O5S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— N-cyclopentyl-N-[(3S)-1,1-dioxothiolan-3-yl]-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide —— C20H27N5O3S
N-cyclopentyl-N-[(3S)-1,1-dioxothiolan-3-yl]-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide
—— 2-[(4R)-3-tert-butyl-1-(2-chlorophenyl)-4-(2,5-dimethoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C29H35ClN4O5S
2-[(4R)-3-tert-butyl-1-(2-chlorophenyl)-4-(2,5-dimethoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— [2-[(3R)-5-naphthalen-2-yl-3-phenyl-3,4-dihydropyrazol-2-yl]-2-oxoethyl] 5-chloro-3-methyl-1-phenylpyrazole-4-carboxylate —— C32H25ClN4O3
[2-[(3R)-5-naphthalen-2-yl-3-phenyl-3,4-dihydropyrazol-2-yl]-2-oxoethyl] 5-chloro-3-methyl-1-phenylpyrazole-4-carboxylate
—— N-(3-ethylphenyl)-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide —— C19H21N5O
N-(3-ethylphenyl)-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide
—— (4S)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C32H34N4O5S2
(4S)-3-(2,6-dimethoxyphenyl)-1-(2,3-dimethylphenyl)-8-(2-morpholin-4-yl-2-oxoethyl)-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— [3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl (1R,5S)-9-oxobicyclo[3.3.1]nonane-3-carboxylate —— C20H22N2O5
[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl (1R,5S)-9-oxobicyclo[3.3.1]nonane-3-carboxylate
—— N-(2,4-dimethylphenyl)-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide —— C19H21N5O
N-(2,4-dimethylphenyl)-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide
—— 2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C33H34ClFN4O2S
2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C33H26FN5O4S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4R)-1-tert-butyl-4-(2,5-dimethoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C30H38N4O5S
2-[(4R)-1-tert-butyl-4-(2,5-dimethoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— 2-[5-(4-ethylphenyl)tetrazol-2-yl]-N-methyl-N-(thiophen-3-ylmethyl)acetamide —— C17H19N5OS
2-[5-(4-ethylphenyl)tetrazol-2-yl]-N-methyl-N-(thiophen-3-ylmethyl)acetamide
—— Ethyl 1-[2-[5-(4-ethylphenyl)tetrazol-2-yl]acetyl]piperidine-4-carboxylate —— C19H25N5O3
Ethyl 1-[2-[5-(4-ethylphenyl)tetrazol-2-yl]acetyl]piperidine-4-carboxylate
—— 2-[3-(4-methoxyphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]-N-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]acetamide —— C21H26N4O2S
2-[3-(4-methoxyphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]-N-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]acetamide
—— N-[2-[(2S)-butan-2-yl]phenyl]-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide —— C21H25N5O
N-[2-[(2S)-butan-2-yl]phenyl]-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide
—— 2-[5-(4-ethylphenyl)tetrazol-2-yl]-N-[2-(thiophen-2-ylmethylsulfanyl)ethyl]acetamide —— C18H21N5OS2
2-[5-(4-ethylphenyl)tetrazol-2-yl]-N-[2-(thiophen-2-ylmethylsulfanyl)ethyl]acetamide
—— N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide —— C22H23N7O2
N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide
—— 2-[(4S)-3-tert-butyl-1-(2-chlorophenyl)-4-(2,5-dimethoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C30H37ClN4O5S
2-[(4S)-3-tert-butyl-1-(2-chlorophenyl)-4-(2,5-dimethoxyphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— N-(2,6-difluorophenyl)-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide —— C17H15F2N5O
N-(2,6-difluorophenyl)-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide
—— 5-(4-Ethylphenyl)-2-[(2-fluorophenyl)methyl]tetrazole —— C16H15FN4
5-(4-Ethylphenyl)-2-[(2-fluorophenyl)methyl]tetrazole
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C34H26F2N4O4S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— N-(3-acetamidophenyl)-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide —— C19H20N6O2
N-(3-acetamidophenyl)-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide
—— 2-[5-(4-ethylphenyl)tetrazol-2-yl]-N-(furan-2-ylmethyl)-N-methylacetamide —— C17H19N5O2
2-[5-(4-ethylphenyl)tetrazol-2-yl]-N-(furan-2-ylmethyl)-N-methylacetamide
—— N-[(4-chlorophenyl)methyl]-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide —— C18H18ClN5O
N-[(4-chlorophenyl)methyl]-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide
—— 1-(2-methoxyethyl)-3-[(Z)-[3-(2-methoxyphenyl)-1-phenylpyrazol-4-yl]methylideneamino]thiourea —— C21H23N5O2S
1-(2-methoxyethyl)-3-[(Z)-[3-(2-methoxyphenyl)-1-phenylpyrazol-4-yl]methylideneamino]thiourea
—— N-[2-(cyanomethylsulfanyl)phenyl]-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide —— C19H18N6OS
N-[2-(cyanomethylsulfanyl)phenyl]-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide
—— N-(3-chloro-4-fluorophenyl)-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide —— C17H15ClFN5O
N-(3-chloro-4-fluorophenyl)-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide
—— 2-[5-(4-ethylphenyl)tetrazol-2-yl]-N-(2-methoxy-4-nitrophenyl)acetamide —— C18H18N6O4
2-[5-(4-ethylphenyl)tetrazol-2-yl]-N-(2-methoxy-4-nitrophenyl)acetamide
—— N-(2-bromophenyl)-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide —— C17H16BrN5O
N-(2-bromophenyl)-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide
—— N-[(3,4-dimethoxyphenyl)methyl]-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide —— C20H23N5O3
N-[(3,4-dimethoxyphenyl)methyl]-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide
—— N-[2-(2-chloroanilino)-2-oxoethyl]-2-[5-(4-ethylphenyl)tetrazol-2-yl]-N-methylacetamide —— C20H21ClN6O2
N-[2-(2-chloroanilino)-2-oxoethyl]-2-[5-(4-ethylphenyl)tetrazol-2-yl]-N-methylacetamide
—— N-[(4-ethylphenyl)methyl]-2-[5-(4-ethylphenyl)tetrazol-2-yl]-N-methylacetamide —— C21H25N5O
N-[(4-ethylphenyl)methyl]-2-[5-(4-ethylphenyl)tetrazol-2-yl]-N-methylacetamide
—— N-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide —— C20H21N5O3
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide
—— 2-[5-(4-ethylphenyl)tetrazol-2-yl]-N-[4-(trifluoromethoxy)phenyl]acetamide —— C18H16F3N5O2
2-[5-(4-ethylphenyl)tetrazol-2-yl]-N-[4-(trifluoromethoxy)phenyl]acetamide
—— N-(2-chlorophenyl)-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide —— C17H16ClN5O
N-(2-chlorophenyl)-2-[5-(4-ethylphenyl)tetrazol-2-yl]acetamide
—— N-methyl-3-(3-methylphenyl)-1-phenylpyrazole-4-carboxamide —— C18H17N3O
N-methyl-3-(3-methylphenyl)-1-phenylpyrazole-4-carboxamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C32H29FN4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— [2-oxo-2-[(4-phenyl-1,3-thiazol-2-yl)-prop-2-enylamino]ethyl] (Z)-3-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)prop-2-enoate —— C28H25ClN4O3S
[2-oxo-2-[(4-phenyl-1,3-thiazol-2-yl)-prop-2-enylamino]ethyl] (Z)-3-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)prop-2-enoate
—— [(2S)-1-[4-chloro-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)sulfamoyl]anilino]-1-oxopropan-2-yl] 3,5-dimethyl-1,2-oxazole-4-carboxylate —— C26H26ClN5O7S
[(2S)-1-[4-chloro-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)sulfamoyl]anilino]-1-oxopropan-2-yl] 3,5-dimethyl-1,2-oxazole-4-carboxylate
—— 2-chloro-N-[[3-ethyl-5-(2-fluorophenoxy)-1-phenylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide —— C30H29ClFN3O3
2-chloro-N-[[3-ethyl-5-(2-fluorophenoxy)-1-phenylpyrazol-4-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]benzamide
—— 1-[(Z)-[1-benzyl-3-(3-methylphenyl)pyrazol-4-yl]methylideneamino]-3-(2-methoxyethyl)thiourea —— C22H25N5OS
1-[(Z)-[1-benzyl-3-(3-methylphenyl)pyrazol-4-yl]methylideneamino]-3-(2-methoxyethyl)thiourea
—— 2-[5-(4-ethylphenyl)tetrazol-2-yl]-N-(4-fluorophenyl)acetamide —— C17H16FN5O
2-[5-(4-ethylphenyl)tetrazol-2-yl]-N-(4-fluorophenyl)acetamide
—— 2-chloro-N-[[3-ethyl-5-(2-fluorophenoxy)-1-phenylpyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide —— C30H29ClFN3O3
2-chloro-N-[[3-ethyl-5-(2-fluorophenoxy)-1-phenylpyrazol-4-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]benzamide
—— 4-[[5-(4-Ethylphenyl)tetrazol-2-yl]methyl]benzonitrile —— C17H15N5
4-[[5-(4-Ethylphenyl)tetrazol-2-yl]methyl]benzonitrile
—— 3-(3,4-dimethylphenyl)-1-phenyl-N-(1,3-thiazol-2-yl)pyrazole-4-carboxamide —— C21H18N4OS
3-(3,4-dimethylphenyl)-1-phenyl-N-(1,3-thiazol-2-yl)pyrazole-4-carboxamide
—— 5-chloro-3-methyl-1-(2-methylpropyl)-N-(1,3-thiazol-2-yl)pyrazole-4-carboxamide —— C12H15ClN4OS
5-chloro-3-methyl-1-(2-methylpropyl)-N-(1,3-thiazol-2-yl)pyrazole-4-carboxamide