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中文名称 英文名称 CAS号 化学式 结构式图片
—— (4Z,5S)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)-5-phenylpyrrolidine-2,3-dione —— C27H28N4O4
(4Z,5S)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)-5-phenylpyrrolidine-2,3-dione
—— (4Z,5S)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-phenylpyrrolidine-2,3-dione —— C25H26N4O3
(4Z,5S)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-phenylpyrrolidine-2,3-dione
—— [2-[[(2R)-2-cyano-3-methylbutan-2-yl]amino]-2-oxoethyl] 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate —— C18H18ClN3O3S
[2-[[(2R)-2-cyano-3-methylbutan-2-yl]amino]-2-oxoethyl] 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate
—— (4Z,5R)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-(3,4,5-trimethoxyphenyl)pyrrolidine-2,3-dione —— C28H32N4O6
(4Z,5R)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-(3,4,5-trimethoxyphenyl)pyrrolidine-2,3-dione
—— [(2S)-1-oxo-1-[(4-phenyl-1,3-thiazol-2-yl)amino]propan-2-yl] (Z)-3-[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C30H23FN4O3S
[(2S)-1-oxo-1-[(4-phenyl-1,3-thiazol-2-yl)amino]propan-2-yl] (Z)-3-[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [2-oxo-2-(4-sulfamoylanilino)ethyl] (Z)-3-[3-(1-benzofuran-2-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C28H22N4O6S
[2-oxo-2-(4-sulfamoylanilino)ethyl] (Z)-3-[3-(1-benzofuran-2-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [2-[2,5-dimethyl-1-[[(2S)-oxolan-2-yl]methyl]pyrrol-3-yl]-2-oxoethyl] (Z)-3-[3-(1-benzofuran-2-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C33H31N3O5
[2-[2,5-dimethyl-1-[[(2S)-oxolan-2-yl]methyl]pyrrol-3-yl]-2-oxoethyl] (Z)-3-[3-(1-benzofuran-2-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [2-oxo-2-[4-(trifluoromethoxy)anilino]ethyl] (Z)-3-[3-(3,4-dimethoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C29H24F3N3O6
[2-oxo-2-[4-(trifluoromethoxy)anilino]ethyl] (Z)-3-[3-(3,4-dimethoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [(1S)-2-(4-methyl-2-nitroanilino)-2-oxo-1-phenylethyl] (E)-3-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C34H28N4O6
[(1S)-2-(4-methyl-2-nitroanilino)-2-oxo-1-phenylethyl] (E)-3-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— (4Z,5S)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-(3,4,5-trimethoxyphenyl)pyrrolidine-2,3-dione —— C28H32N4O6
(4Z,5S)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-(3,4,5-trimethoxyphenyl)pyrrolidine-2,3-dione
—— (2-Thiophen-2-yl-1,3-oxazol-4-yl)methyl 2-(2-chloro-6-fluorophenyl)acetate —— C16H11ClFNO3S
(2-Thiophen-2-yl-1,3-oxazol-4-yl)methyl 2-(2-chloro-6-fluorophenyl)acetate
—— [2-[2-(3,4-dimethoxyphenyl)ethylamino]-2-oxoethyl] (Z)-3-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C33H29N3O7
[2-[2-(3,4-dimethoxyphenyl)ethylamino]-2-oxoethyl] (Z)-3-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— 1-[(1-phenylpyrazol-4-yl)methyl]-3-[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]urea —— C21H26N4O
1-[(1-phenylpyrazol-4-yl)methyl]-3-[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]urea
—— [2-oxo-2-(2,3,4-trifluoroanilino)ethyl] (Z)-3-[3-(3,4-dimethoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C28H22F3N3O5
[2-oxo-2-(2,3,4-trifluoroanilino)ethyl] (Z)-3-[3-(3,4-dimethoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [3-(2-Methylphenyl)-1,2,4-oxadiazol-5-yl]methyl 2-(2-chloro-6-fluorophenyl)acetate —— C18H14ClFN2O3
[3-(2-Methylphenyl)-1,2,4-oxadiazol-5-yl]methyl 2-(2-chloro-6-fluorophenyl)acetate
—— [2-[2,5-dimethyl-1-[[(2R)-oxolan-2-yl]methyl]pyrrol-3-yl]-2-oxoethyl] (Z)-3-[3-(1-benzofuran-2-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C33H31N3O5
[2-[2,5-dimethyl-1-[[(2R)-oxolan-2-yl]methyl]pyrrol-3-yl]-2-oxoethyl] (Z)-3-[3-(1-benzofuran-2-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [2-(Furan-2-ylmethylamino)-2-oxoethyl] 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate —— C17H13ClN2O4S
[2-(Furan-2-ylmethylamino)-2-oxoethyl] 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate
—— [(2R)-1-(3-morpholin-4-ylsulfonylanilino)-1-oxopropan-2-yl] 3-(4-fluorophenyl)-1-phenylpyrazole-4-carboxylate —— C29H27FN4O6S
[(2R)-1-(3-morpholin-4-ylsulfonylanilino)-1-oxopropan-2-yl] 3-(4-fluorophenyl)-1-phenylpyrazole-4-carboxylate
—— [2-[[(3S)-1,1-dioxothiolan-3-yl]amino]-2-oxoethyl] (Z)-3-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C27H23N3O7S
[2-[[(3S)-1,1-dioxothiolan-3-yl]amino]-2-oxoethyl] (Z)-3-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— (4Z,5R)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-phenylpyrrolidine-2,3-dione —— C25H26N4O3
(4Z,5R)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-phenylpyrrolidine-2,3-dione
—— (4Z,5R)-5-(4-chlorophenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione —— C27H27ClN4O4
(4Z,5R)-5-(4-chlorophenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione
—— [2-[3-(dimethylsulfamoyl)anilino]-2-oxoethyl] (Z)-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enoate —— C26H24N4O5S2
[2-[3-(dimethylsulfamoyl)anilino]-2-oxoethyl] (Z)-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enoate
—— [2-(2-methoxy-4-nitroanilino)-2-oxoethyl] (Z)-3-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C30H22N4O8
[2-(2-methoxy-4-nitroanilino)-2-oxoethyl] (Z)-3-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [2-[[(3R)-1,1-dioxothiolan-3-yl]-ethylamino]-2-oxoethyl] (Z)-3-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C29H27N3O7S
[2-[[(3R)-1,1-dioxothiolan-3-yl]-ethylamino]-2-oxoethyl] (Z)-3-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [(1S)-2-(4-chloro-3-nitroanilino)-2-oxo-1-phenylethyl] (E)-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enoate —— C30H21ClN4O5S
[(1S)-2-(4-chloro-3-nitroanilino)-2-oxo-1-phenylethyl] (E)-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enoate
—— ethyl 4-cyclopropyl-2-[[2-[(Z)-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enoyl]oxyacetyl]amino]thiophene-3-carboxylate —— C28H25N3O5S2
ethyl 4-cyclopropyl-2-[[2-[(Z)-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enoyl]oxyacetyl]amino]thiophene-3-carboxylate
—— [2-[3-(dimethylsulfamoyl)anilino]-2-oxoethyl] (Z)-3-[3-(5-methylfuran-2-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C27H26N4O6S
[2-[3-(dimethylsulfamoyl)anilino]-2-oxoethyl] (Z)-3-[3-(5-methylfuran-2-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— (4Z,5S)-5-(4-chlorophenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione —— C27H27ClN4O4
(4Z,5S)-5-(4-chlorophenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione
—— [2-[[(3S)-1,1-dioxothiolan-3-yl]-ethylamino]-2-oxoethyl] (Z)-3-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C29H27N3O7S
[2-[[(3S)-1,1-dioxothiolan-3-yl]-ethylamino]-2-oxoethyl] (Z)-3-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— (4Z,5R)-4-[(4-chlorophenyl)-hydroxymethylidene]-1-(4,5-dimethyl-1,3-thiazol-2-yl)-5-(furan-2-yl)pyrrolidine-2,3-dione —— C20H15ClN2O4S
(4Z,5R)-4-[(4-chlorophenyl)-hydroxymethylidene]-1-(4,5-dimethyl-1,3-thiazol-2-yl)-5-(furan-2-yl)pyrrolidine-2,3-dione
—— (4Z,5S)-4-[(4-chlorophenyl)-hydroxymethylidene]-1-(4,5-dimethyl-1,3-thiazol-2-yl)-5-(furan-2-yl)pyrrolidine-2,3-dione —— C20H15ClN2O4S
(4Z,5S)-4-[(4-chlorophenyl)-hydroxymethylidene]-1-(4,5-dimethyl-1,3-thiazol-2-yl)-5-(furan-2-yl)pyrrolidine-2,3-dione
—— [(2S)-1-(dimethylamino)-1-oxopropan-2-yl] 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate —— C15H15ClN2O3S
[(2S)-1-(dimethylamino)-1-oxopropan-2-yl] 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate
—— [(1R)-2-(4-chloro-3-nitroanilino)-2-oxo-1-phenylethyl] (Z)-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enoate —— C30H21ClN4O5S
[(1R)-2-(4-chloro-3-nitroanilino)-2-oxo-1-phenylethyl] (Z)-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)prop-2-enoate
—— (4-Oxo-4-thiophen-2-ylbutyl) 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate —— C18H14ClNO3S2
(4-Oxo-4-thiophen-2-ylbutyl) 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate
—— [(2S)-1-(3-morpholin-4-ylsulfonylanilino)-1-oxopropan-2-yl] 3-(4-fluorophenyl)-1-phenylpyrazole-4-carboxylate —— C29H27FN4O6S
[(2S)-1-(3-morpholin-4-ylsulfonylanilino)-1-oxopropan-2-yl] 3-(4-fluorophenyl)-1-phenylpyrazole-4-carboxylate
—— [2-[[(3R)-1,1-dioxothiolan-3-yl]-methylamino]-2-oxoethyl] (Z)-3-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C28H25N3O7S
[2-[[(3R)-1,1-dioxothiolan-3-yl]-methylamino]-2-oxoethyl] (Z)-3-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— (4Z,5S)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-thiophen-2-ylpyrrolidine-2,3-dione —— C23H24N4O3S
(4Z,5S)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-thiophen-2-ylpyrrolidine-2,3-dione
—— 1-[(1-phenylpyrazol-4-yl)methyl]-3-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]urea —— C21H26N4O
1-[(1-phenylpyrazol-4-yl)methyl]-3-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]urea
—— (4Z,5R)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-thiophen-2-ylpyrrolidine-2,3-dione —— C23H24N4O3S
(4Z,5R)-1-[2-(dimethylamino)ethyl]-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-5-thiophen-2-ylpyrrolidine-2,3-dione
—— ethyl (4R)-6-[[3-(4-fluorophenyl)-1-phenylpyrazole-4-carbonyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C30H25FN4O5
ethyl (4R)-6-[[3-(4-fluorophenyl)-1-phenylpyrazole-4-carbonyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— [(1R)-1-(5-phenyl-1,3,4-oxadiazol-2-yl)ethyl] 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate —— C20H14ClN3O3S
[(1R)-1-(5-phenyl-1,3,4-oxadiazol-2-yl)ethyl] 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate
—— [2-[[(3S)-1,1-dioxothiolan-3-yl]-methylamino]-2-oxoethyl] (Z)-3-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C28H25N3O7S
[2-[[(3S)-1,1-dioxothiolan-3-yl]-methylamino]-2-oxoethyl] (Z)-3-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— 1-[(1S)-1-(4-imidazol-1-ylphenyl)ethyl]-3-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]urea —— C22H28N4O
1-[(1S)-1-(4-imidazol-1-ylphenyl)ethyl]-3-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]urea
—— 1-[(1S)-1-(4-imidazol-1-ylphenyl)ethyl]-3-[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]urea —— C22H28N4O
1-[(1S)-1-(4-imidazol-1-ylphenyl)ethyl]-3-[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]urea
—— 1-[(1R)-1-(4-imidazol-1-ylphenyl)ethyl]-3-[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]urea —— C22H28N4O
1-[(1R)-1-(4-imidazol-1-ylphenyl)ethyl]-3-[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]urea
—— [2-[(1-Cyanocyclopentyl)amino]-2-oxoethyl] 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate —— C18H16ClN3O3S
[2-[(1-Cyanocyclopentyl)amino]-2-oxoethyl] 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate
—— [2-Oxo-2-(propan-2-ylamino)ethyl] 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate —— C15H15ClN2O3S
[2-Oxo-2-(propan-2-ylamino)ethyl] 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate
—— [2-(Cyclopropylamino)-2-oxoethyl] 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate —— C15H13ClN2O3S
[2-(Cyclopropylamino)-2-oxoethyl] 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate
—— 1-[(1R)-1-(4-imidazol-1-ylphenyl)ethyl]-3-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]urea —— C22H28N4O
1-[(1R)-1-(4-imidazol-1-ylphenyl)ethyl]-3-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]urea
—— (4Z,5S)-5-(4-bromophenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione —— C27H27BrN4O4
(4Z,5S)-5-(4-bromophenyl)-4-[hydroxy-(5-methyl-1-phenylpyrazol-4-yl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione