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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-1-(2,3-dimethylphenyl)-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C27H31N5O7S
5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-1-(2,3-dimethylphenyl)-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 2-[[4-Amino-5-(3-bromophenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]benzonitrile —— C16H12BrN5S
2-[[4-Amino-5-(3-bromophenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]benzonitrile
—— [3-(2,4-Dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 5-chloro-1-benzofuran-2-carboxylate —— C20H15ClN2O6
[3-(2,4-Dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 5-chloro-1-benzofuran-2-carboxylate
—— [(2R)-oxolan-2-yl]-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone —— C18H21N3O3
[(2R)-oxolan-2-yl]-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone
—— 5-[(2,5-Dimethoxyphenyl)methylsulfanyl]-1-(2,6-dimethylphenyl)tetrazole —— C18H20N4O2S
5-[(2,5-Dimethoxyphenyl)methylsulfanyl]-1-(2,6-dimethylphenyl)tetrazole
—— 2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-(3-propan-2-yloxypropyl)acetamide —— C17H25N5O2S
2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-(3-propan-2-yloxypropyl)acetamide
—— [4-[[6-(1-benzothiophen-2-yl)-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1S,3R)-3-methoxycyclohexyl]methanone —— C34H35ClN4O2S
[4-[[6-(1-benzothiophen-2-yl)-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1S,3R)-3-methoxycyclohexyl]methanone
—— 5-[2-(tert-butylsulfamoyl)-4-[[(2S)-2-methylbutanoyl]amino]phenoxy]-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxylic acid —— C27H34N4O7S
5-[2-(tert-butylsulfamoyl)-4-[[(2S)-2-methylbutanoyl]amino]phenoxy]-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxylic acid
—— N-(1,3-benzodioxol-5-ylmethyl)-2-[[4-[(2S)-1-methoxypropan-2-yl]-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]benzamide —— C29H30N4O4S
N-(1,3-benzodioxol-5-ylmethyl)-2-[[4-[(2S)-1-methoxypropan-2-yl]-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]benzamide
—— (Z)-N-(3-pyrazol-1-ylpropyl)-3-thiophen-2-ylprop-2-enamide —— C13H15N3OS
(Z)-N-(3-pyrazol-1-ylpropyl)-3-thiophen-2-ylprop-2-enamide
—— 5-[4-(cyclopentanecarbonylamino)-2-(propylsulfamoyl)phenoxy]-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxylic acid —— C27H32N4O7S
5-[4-(cyclopentanecarbonylamino)-2-(propylsulfamoyl)phenoxy]-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxylic acid
—— [3-(3,4-Dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 5-chloro-1-benzofuran-2-carboxylate —— C20H15ClN2O6
[3-(3,4-Dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 5-chloro-1-benzofuran-2-carboxylate
—— (Z)-N-[(2S)-3,3-dimethylbutan-2-yl]-N-methyl-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide —— C16H27N3O
(Z)-N-[(2S)-3,3-dimethylbutan-2-yl]-N-methyl-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide
—— [4-[[6-(1-benzothiophen-2-yl)-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1R,3R)-3-methoxycyclohexyl]methanone —— C34H35ClN4O2S
[4-[[6-(1-benzothiophen-2-yl)-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1R,3R)-3-methoxycyclohexyl]methanone
—— 5-[4-(cyclobutanecarbonylamino)-2-morpholin-4-ylsulfonylphenoxy]-1-(2,3-dimethylphenyl)-4-methylpyrazole-3-carboxylic acid —— C28H32N4O7S
5-[4-(cyclobutanecarbonylamino)-2-morpholin-4-ylsulfonylphenoxy]-1-(2,3-dimethylphenyl)-4-methylpyrazole-3-carboxylic acid
—— 2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-[(4-methylphenyl)methyl]-N-propylacetamide —— C22H27N5OS
2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-[(4-methylphenyl)methyl]-N-propylacetamide
—— (3-Phenyl-1,2,4-oxadiazol-5-yl)methyl 5-chloro-1-benzofuran-2-carboxylate —— C18H11ClN2O4
(3-Phenyl-1,2,4-oxadiazol-5-yl)methyl 5-chloro-1-benzofuran-2-carboxylate
—— N'-(5-chlorothiophen-2-yl)sulfonyl-2-(2-methyl-1,3-thiazol-4-yl)acetohydrazide —— C10H10ClN3O3S3
N'-(5-chlorothiophen-2-yl)sulfonyl-2-(2-methyl-1,3-thiazol-4-yl)acetohydrazide
—— 2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-[2-(2-methylphenyl)ethyl]acetamide —— C20H23N5OS
2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-[2-(2-methylphenyl)ethyl]acetamide
—— [(2S)-oxolan-2-yl]-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone —— C18H21N3O3
[(2S)-oxolan-2-yl]-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone
—— (Z)-N-[(2R)-3,3-dimethylbutan-2-yl]-N-methyl-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide —— C16H27N3O
(Z)-N-[(2R)-3,3-dimethylbutan-2-yl]-N-methyl-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide
—— 5-[2-(tert-butylsulfamoyl)-4-[[(2R)-2-methylbutanoyl]amino]phenoxy]-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxylic acid —— C27H34N4O7S
5-[2-(tert-butylsulfamoyl)-4-[[(2R)-2-methylbutanoyl]amino]phenoxy]-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxylic acid
—— 1-(3-fluorophenyl)-5-[2-(furan-2-ylmethylsulfamoyl)-4-[[(2S)-2-methylbutanoyl]amino]phenoxy]-4-methylpyrazole-3-carboxylic acid —— C27H27FN4O7S
1-(3-fluorophenyl)-5-[2-(furan-2-ylmethylsulfamoyl)-4-[[(2S)-2-methylbutanoyl]amino]phenoxy]-4-methylpyrazole-3-carboxylic acid
—— 1-(3-Fluoro-4-methylphenyl)-3-[(4-hydroxy-1-phenylpyrazole-3-carbonyl)amino]thiourea —— C18H16FN5O2S
1-(3-Fluoro-4-methylphenyl)-3-[(4-hydroxy-1-phenylpyrazole-3-carbonyl)amino]thiourea
—— 1-(3-fluorophenyl)-4-methyl-5-[4-[[(2R)-2-methylbutanoyl]amino]-2-(propylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid —— C25H29FN4O6S
1-(3-fluorophenyl)-4-methyl-5-[4-[[(2R)-2-methylbutanoyl]amino]-2-(propylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid
—— 1-(3-fluorophenyl)-5-[2-(furan-2-ylmethylsulfamoyl)-4-[[(2R)-2-methylbutanoyl]amino]phenoxy]-4-methylpyrazole-3-carboxylic acid —— C27H27FN4O7S
1-(3-fluorophenyl)-5-[2-(furan-2-ylmethylsulfamoyl)-4-[[(2R)-2-methylbutanoyl]amino]phenoxy]-4-methylpyrazole-3-carboxylic acid
—— 1-(3-fluorophenyl)-4-methyl-5-[4-[[(2S)-2-methylbutanoyl]amino]-2-(propylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid —— C25H29FN4O6S
1-(3-fluorophenyl)-4-methyl-5-[4-[[(2S)-2-methylbutanoyl]amino]-2-(propylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid
—— N-[(1R)-1-phenylethyl]-4-(trifluoromethyl)-N-[2-[3-(3,4,5-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl]benzamide —— C29H28F3N3O5
N-[(1R)-1-phenylethyl]-4-(trifluoromethyl)-N-[2-[3-(3,4,5-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl]benzamide
—— 5-(4-Fluorophenyl)-3-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]thieno[2,3-d]pyrimidin-4-one —— C21H13FN4O2S
5-(4-Fluorophenyl)-3-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]thieno[2,3-d]pyrimidin-4-one
—— 2-[(5S,7S)-3-bromo-1-adamantyl]-N-[5-[1-(difluoromethyl)imidazol-2-yl]-4-methyl-1,3-thiazol-2-yl]acetamide —— C20H23BrF2N4OS
2-[(5S,7S)-3-bromo-1-adamantyl]-N-[5-[1-(difluoromethyl)imidazol-2-yl]-4-methyl-1,3-thiazol-2-yl]acetamide
—— N-[(1S)-1-phenylethyl]-4-(trifluoromethyl)-N-[2-[3-(3,4,5-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl]benzamide —— C29H28F3N3O5
N-[(1S)-1-phenylethyl]-4-(trifluoromethyl)-N-[2-[3-(3,4,5-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl]benzamide
—— 1-(3-Ethylphenyl)-3-[(4-methyl-2-phenyl-1,3-thiazole-5-carbonyl)amino]thiourea —— C20H20N4OS2
1-(3-Ethylphenyl)-3-[(4-methyl-2-phenyl-1,3-thiazole-5-carbonyl)amino]thiourea
—— [2-[(1,5-Dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-amino-4-fluorobenzoate —— C20H19FN4O4
[2-[(1,5-Dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-amino-4-fluorobenzoate
—— 1-[(2S)-2-ethylhexyl]-3-[[4-(tetrazol-1-yl)benzoyl]amino]thiourea —— C17H25N7OS
1-[(2S)-2-ethylhexyl]-3-[[4-(tetrazol-1-yl)benzoyl]amino]thiourea
—— 2-[(4R)-4-(2,4-difluorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C33H32F2N4O3S
2-[(4R)-4-(2,4-difluorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— [2-[2-(benzylamino)-2-oxoethyl]-1,3-thiazol-4-yl]methyl (5S,7S)-3-chloroadamantane-1-carboxylate —— C24H27ClN2O3S
[2-[2-(benzylamino)-2-oxoethyl]-1,3-thiazol-4-yl]methyl (5S,7S)-3-chloroadamantane-1-carboxylate
—— [3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl 2-[(5R,7R)-3-bromo-1-adamantyl]acetate —— C19H27BrN2O3
[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl 2-[(5R,7R)-3-bromo-1-adamantyl]acetate
—— (1R,2R,4S)-N-[[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]methyl]-N-methylbicyclo[2.2.1]hept-5-ene-2-carboxamide —— C25H24ClN3O
(1R,2R,4S)-N-[[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]methyl]-N-methylbicyclo[2.2.1]hept-5-ene-2-carboxamide
—— [4-[[6-(1-benzothiophen-2-yl)-2-phenylimidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1S,3R)-3-methoxycyclohexyl]methanone —— C34H36N4O2S
[4-[[6-(1-benzothiophen-2-yl)-2-phenylimidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1S,3R)-3-methoxycyclohexyl]methanone
—— [4-[[6-(1-benzothiophen-2-yl)-2-phenylimidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1S,3S)-3-methoxycyclohexyl]methanone —— C34H36N4O2S
[4-[[6-(1-benzothiophen-2-yl)-2-phenylimidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1S,3S)-3-methoxycyclohexyl]methanone
—— (1R,2S,4S)-N-[[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]methyl]-N-methylbicyclo[2.2.1]hept-5-ene-2-carboxamide —— C25H24ClN3O
(1R,2S,4S)-N-[[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]methyl]-N-methylbicyclo[2.2.1]hept-5-ene-2-carboxamide
—— (Z)-N-[(2-methoxypyridin-3-yl)methyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C19H18N4O2
(Z)-N-[(2-methoxypyridin-3-yl)methyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— 1-[[3-benzyl-2-[(4-fluorophenyl)methylsulfonyl]imidazol-4-yl]methyl]-3-tert-butyl-1-[[(2S)-oxolan-2-yl]methyl]urea —— C28H35FN4O4S
1-[[3-benzyl-2-[(4-fluorophenyl)methylsulfonyl]imidazol-4-yl]methyl]-3-tert-butyl-1-[[(2S)-oxolan-2-yl]methyl]urea
—— N-[[3-ethyl-5-(3-methoxyphenoxy)-1-phenylpyrazol-4-yl]methyl]-4-methoxy-N-[[(2R)-oxolan-2-yl]methyl]benzenesulfonamide —— C31H35N3O6S
N-[[3-ethyl-5-(3-methoxyphenoxy)-1-phenylpyrazol-4-yl]methyl]-4-methoxy-N-[[(2R)-oxolan-2-yl]methyl]benzenesulfonamide
—— 2-[(4S)-4-(2,4-difluorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C33H32F2N4O3S
2-[(4S)-4-(2,4-difluorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— [4-[[6-(1-benzothiophen-2-yl)-2-phenylimidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1R,3S)-3-methoxycyclohexyl]methanone —— C34H36N4O2S
[4-[[6-(1-benzothiophen-2-yl)-2-phenylimidazo[1,2-a]pyridin-3-yl]methyl]piperazin-1-yl]-[(1R,3S)-3-methoxycyclohexyl]methanone
—— [2-[2-(benzylamino)-2-oxoethyl]-1,3-thiazol-4-yl]methyl (5R,7R)-3-chloroadamantane-1-carboxylate —— C24H27ClN2O3S
[2-[2-(benzylamino)-2-oxoethyl]-1,3-thiazol-4-yl]methyl (5R,7R)-3-chloroadamantane-1-carboxylate
—— [3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl 2-[(5S,7S)-3-bromo-1-adamantyl]acetate —— C19H27BrN2O3
[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl 2-[(5S,7S)-3-bromo-1-adamantyl]acetate
—— N-[2-[[4-(4-chlorophenyl)-1-(3,4-dimethylphenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]thiophene-2-carboxamide —— C29H29ClN4O3S
N-[2-[[4-(4-chlorophenyl)-1-(3,4-dimethylphenyl)imidazol-2-yl]amino]-2-oxoethyl]-N-[[(2R)-oxolan-2-yl]methyl]thiophene-2-carboxamide
—— 1-[[3-benzyl-2-[(4-fluorophenyl)methylsulfonyl]imidazol-4-yl]methyl]-3-tert-butyl-1-[[(2R)-oxolan-2-yl]methyl]urea —— C28H35FN4O4S
1-[[3-benzyl-2-[(4-fluorophenyl)methylsulfonyl]imidazol-4-yl]methyl]-3-tert-butyl-1-[[(2R)-oxolan-2-yl]methyl]urea