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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C31H33FN4O3S
2-[(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide —— C29H35ClN4O3S
2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(2-methoxyethyl)acetamide
—— 2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide —— C29H33ClN4O2S
2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-cyclopropylacetamide
—— 1-(3-Ethylphenyl)-3-[[2-(2-methyl-1,3-thiazol-4-yl)acetyl]amino]thiourea —— C15H18N4OS2
1-(3-Ethylphenyl)-3-[[2-(2-methyl-1,3-thiazol-4-yl)acetyl]amino]thiourea
—— 2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C32H34ClN5O2S
2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— (5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 2-(3-methylbutylamino)-1,3-thiazole-4-carboxylate —— C18H20N4O3S
(5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 2-(3-methylbutylamino)-1,3-thiazole-4-carboxylate
—— 2-[[4-(3-methylphenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]sulfanylmethyl]-N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-1,3-thiazole-4-carboxamide —— C27H32N6OS3
2-[[4-(3-methylphenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]sulfanylmethyl]-N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-1,3-thiazole-4-carboxamide
—— 2-[(4S)-1-(2,3-dimethylphenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C35H30F2N4O2S
2-[(4S)-1-(2,3-dimethylphenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— (1R,2R)-N-benzyl-N-[2-[[2-(4-fluorophenyl)-5-phenylpyrazol-3-yl]amino]-2-oxoethyl]-2-phenylcyclopropane-1-carboxamide —— C34H29FN4O2
(1R,2R)-N-benzyl-N-[2-[[2-(4-fluorophenyl)-5-phenylpyrazol-3-yl]amino]-2-oxoethyl]-2-phenylcyclopropane-1-carboxamide
—— 2-[[4-(3-methylphenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]sulfanylmethyl]-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]-1,3-thiazole-4-carboxamide —— C27H32N6OS3
2-[[4-(3-methylphenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]sulfanylmethyl]-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]-1,3-thiazole-4-carboxamide
—— 1-(2-Ethylphenyl)-3-[[2-(2-methyl-1,3-thiazol-4-yl)acetyl]amino]thiourea —— C15H18N4OS2
1-(2-Ethylphenyl)-3-[[2-(2-methyl-1,3-thiazol-4-yl)acetyl]amino]thiourea
—— 1-(3-Ethylphenyl)-3-[(4-methyl-2-morpholin-4-yl-1,3-thiazole-5-carbonyl)amino]thiourea —— C18H23N5O2S2
1-(3-Ethylphenyl)-3-[(4-methyl-2-morpholin-4-yl-1,3-thiazole-5-carbonyl)amino]thiourea
—— [2-(Cyclopentylamino)-2-oxoethyl] 2-(3-methylbutylamino)-1,3-thiazole-4-carboxylate —— C16H25N3O3S
[2-(Cyclopentylamino)-2-oxoethyl] 2-(3-methylbutylamino)-1,3-thiazole-4-carboxylate
—— 2-[(4R)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C34H32N4O6S
2-[(4R)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 2-[(4S)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C34H32N4O6S
2-[(4S)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C34H30N4O5S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide —— C34H30N4O5S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(furan-2-ylmethyl)acetamide
—— N-[(E)-[(2R)-2-methylcyclohexylidene]amino]-2-[3-(trifluoromethyl)pyrazol-1-yl]acetamide —— C13H17F3N4O
N-[(E)-[(2R)-2-methylcyclohexylidene]amino]-2-[3-(trifluoromethyl)pyrazol-1-yl]acetamide
—— (Z,1S,4R)-N-[(Z)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine —— C21H25ClN4
(Z,1S,4R)-N-[(Z)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine
—— 1-[(2S)-2-ethylhexyl]-3-[[2-(5-phenyltetrazol-2-yl)acetyl]amino]thiourea —— C18H27N7OS
1-[(2S)-2-ethylhexyl]-3-[[2-(5-phenyltetrazol-2-yl)acetyl]amino]thiourea
—— 2-[(4S)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C33H27F2N5O3S
2-[(4S)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C35H31N5O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— (Z,1R,4S)-N-[(Z)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine —— C21H25ClN4
(Z,1R,4S)-N-[(Z)-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine
—— (Z)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-methoxy-N-methylprop-2-enamide —— C12H15N3O2S
(Z)-3-(2,6-dimethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-methoxy-N-methylprop-2-enamide
—— 2-[(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C33H37N5O2S
2-[(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— (3aS,7aS)-2-[[4-[[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]methyl]-3a,4,5,6,7,7a-hexahydroisoindole-1,3-dione —— C23H29N5O4
(3aS,7aS)-2-[[4-[[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]methyl]-3a,4,5,6,7,7a-hexahydroisoindole-1,3-dione
—— N-[2-[(2R)-2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]-N-(2-methoxyethyl)octanamide —— C26H37ClN4O4
N-[2-[(2R)-2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]-N-(2-methoxyethyl)octanamide
—— N-[2-[(2S)-2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]-N-(2-methoxyethyl)octanamide —— C26H37ClN4O4
N-[2-[(2S)-2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]-N-(2-methoxyethyl)octanamide
—— (2R)-1-[cyclopropylmethyl-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]amino]-3-phenylmethoxypropan-2-ol —— C31H33F2N3O3
(2R)-1-[cyclopropylmethyl-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]amino]-3-phenylmethoxypropan-2-ol
—— (2S)-1-[cyclopropylmethyl-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]amino]-3-phenylmethoxypropan-2-ol —— C31H33F2N3O3
(2S)-1-[cyclopropylmethyl-[[5-(2,4-difluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methyl]amino]-3-phenylmethoxypropan-2-ol
—— 2-[(4R)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C33H27F2N5O3S
2-[(4R)-4-(2,4-difluorophenyl)-1-(4-methoxyphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4R)-1-(2,3-dimethylphenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C35H30F2N4O2S
2-[(4R)-1-(2,3-dimethylphenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— N-[(E)-[(2S)-2-methylcyclohexylidene]amino]-2-[3-(trifluoromethyl)pyrazol-1-yl]acetamide —— C13H17F3N4O
N-[(E)-[(2S)-2-methylcyclohexylidene]amino]-2-[3-(trifluoromethyl)pyrazol-1-yl]acetamide
—— 2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C33H37N5O2S
2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4-chlorophenyl)sulfonyl-[[(2R)-oxolan-2-yl]methyl]amino]-N-[1-(3,4-dimethoxyphenyl)-4-phenylimidazol-2-yl]acetamide —— C30H31ClN4O6S
2-[(4-chlorophenyl)sulfonyl-[[(2R)-oxolan-2-yl]methyl]amino]-N-[1-(3,4-dimethoxyphenyl)-4-phenylimidazol-2-yl]acetamide
—— N-benzyl-N-[2-[(2R)-2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]-2-(4-fluorophenyl)acetamide —— C30H28ClFN4O3
N-benzyl-N-[2-[(2R)-2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]-2-(4-fluorophenyl)acetamide
—— 2-[(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide —— C31H33FN4O2S2
2-[(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-[(4-fluorophenyl)methyl]acetamide
—— 1-[(2R)-2-ethylhexyl]-3-[[2-(2-methyl-1,3-thiazol-4-yl)acetyl]amino]thiourea —— C15H26N4OS2
1-[(2R)-2-ethylhexyl]-3-[[2-(2-methyl-1,3-thiazol-4-yl)acetyl]amino]thiourea
—— [2-(4-ethoxycarbonyl-3,5-dimethyl-1H-pyrrol-2-yl)-2-oxoethyl] 2-(3-methylbutylamino)-1,3-thiazole-4-carboxylate —— C20H27N3O5S
[2-(4-ethoxycarbonyl-3,5-dimethyl-1H-pyrrol-2-yl)-2-oxoethyl] 2-(3-methylbutylamino)-1,3-thiazole-4-carboxylate
—— [2-[2-(4-Fluorophenyl)ethylamino]-2-oxoethyl] 2-(3-methylbutylamino)-1,3-thiazole-4-carboxylate —— C19H24FN3O3S
[2-[2-(4-Fluorophenyl)ethylamino]-2-oxoethyl] 2-(3-methylbutylamino)-1,3-thiazole-4-carboxylate
—— 1-(3-Ethylphenyl)-3-[(4-phenyl-1,3-thiazol-2-yl)amino]thiourea —— C18H18N4S2
1-(3-Ethylphenyl)-3-[(4-phenyl-1,3-thiazol-2-yl)amino]thiourea
—— 1-[(4-Fluorophenyl)methyl]-3-[[2-(5-phenyltetrazol-2-yl)acetyl]amino]thiourea —— C17H16FN7OS
1-[(4-Fluorophenyl)methyl]-3-[[2-(5-phenyltetrazol-2-yl)acetyl]amino]thiourea
—— methyl (E)-3-[1-benzyl-3-(2-methoxyphenyl)pyrazol-4-yl]-2-cyanoprop-2-enoate —— C22H19N3O3
methyl (E)-3-[1-benzyl-3-(2-methoxyphenyl)pyrazol-4-yl]-2-cyanoprop-2-enoate
—— 1-(2-Ethylphenyl)-3-[(2-imidazo[2,1-b][1,3]thiazol-6-ylacetyl)amino]thiourea —— C16H17N5OS2
1-(2-Ethylphenyl)-3-[(2-imidazo[2,1-b][1,3]thiazol-6-ylacetyl)amino]thiourea
—— (4S)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C35H38N4O5S
(4S)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— N-[(3S)-2,5-dioxopyrrolidin-3-yl]-N-ethyl-4-(5-methylpyrazol-1-yl)benzamide —— C17H18N4O3
N-[(3S)-2,5-dioxopyrrolidin-3-yl]-N-ethyl-4-(5-methylpyrazol-1-yl)benzamide
—— (3aS,7aR)-2-[[4-[[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]methyl]-3a,4,5,6,7,7a-hexahydroisoindole-1,3-dione —— C23H29N5O4
(3aS,7aR)-2-[[4-[[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]methyl]-3a,4,5,6,7,7a-hexahydroisoindole-1,3-dione
—— prop-2-enyl (E)-3-[1-benzyl-3-(2-methoxyphenyl)pyrazol-4-yl]-2-cyanoprop-2-enoate —— C24H21N3O3
prop-2-enyl (E)-3-[1-benzyl-3-(2-methoxyphenyl)pyrazol-4-yl]-2-cyanoprop-2-enoate
—— (4R)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C35H38N4O5S
(4R)-4-(2,5-dimethoxyphenyl)-1-(4-methoxyphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— N-benzyl-N-[2-[(2S)-2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]-2-(4-fluorophenyl)acetamide —— C30H28ClFN4O3
N-benzyl-N-[2-[(2S)-2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-oxoethyl]-2-(4-fluorophenyl)acetamide